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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 207 / 321
Miromavimab DB17803
biotech | CAS: 2247163-73-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mirostipen DB06453
small molecule | CAS: 244130-01-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mirtazapine Approved DB00370
small molecule | CAS: 85650-52-8

Mirtazapine is a tetracyclic _piperazino-azepine_ antidepressant agent that was initially approved for the treatment of major depressive disorder (MDD) in the Netherlands in 1994.[A177946] This drug was first manufactured by Organon Inc., and received FDA app…

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +38
Target Protein:
5-hydroxytryptamine receptor 2A5HT3 serotonin receptorAlpha-2A adrenergic receptor +4
Waktu Paruh20-40 hours [FDA la…
Vol. DistribusiThe volume of distr…
KlirensTotal body clearanc…
Genetik -
Mirvetuximab DB16235
biotech | CAS: 1453084-36-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirvetuximab soravtansine Approved DB12489
biotech | CAS: 1453084-37-1

Mirvetuximab soravtansine-gynx (IMGN853) is an antibody-drug conjugate (ADC) formed by a monoclonal antibody (M9346A) that targets folate receptor alpha (FR?), covalently joined by a cleavable disulfide linker to the genotoxic compound DM4 (also known as sora…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Folate receptor alpha
Waktu ParuhAfter the first dos…
Vol. DistribusiMirvetuximab soravt…
KlirensThe total plasma cl…
Genetik -
Misetionamide DB18098
small molecule | CAS: 856785-75-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Misonidazole DB11716
small molecule | CAS: 13551-87-6

Misonidazole is under investigation in clinical trial NCT00038038 (Assessment of Head and Neck Tumor Hypoxia Using 18F-Fluoromisonidazole).

Kategori:
Anti-Infective AgentsAntineoplastic AgentsAntiparasitic Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Misoprostol Approved DB00929
small molecule | CAS: 59122-46-2

Misoprostol is a prostaglandin analog used to reduce the risk of NSAID related ulcers, manage miscarriages, prevent post partum hemorrhage, and also for first trimester abortions.[L7616,L7619,A181589,A181583,A181697] The stimulation of prostaglandin receptors…

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAlimentary Tract and Metabolism +24
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP2 subtype +2
Waktu ParuhThe half life of an…
Vol. DistribusiData regarding the …
KlirensBecause of the rapi…
Genetik -
Mitapivat Approved DB16236
small molecule | CAS: 1260075-17-9

Mitapivat is a novel, first-in-class pyruvate kinase activator. It works to increase the activity of erythrocyte pyruvate kinase, a key enzyme involved in the survival of red blood cells. Defects in the pyruvate kinase enzyme in various red blood cells disord…

Kategori:
Anemia, Hemolytic, Congenital, drug therapyBlood and Blood Forming OrgansCytochrome P-450 CYP1A2 Substrates +27
Target Protein:
Pyruvate kinase PKLRAromatase
Waktu ParuhIn patients with py…
Vol. DistribusiThe mean volume of …
KlirensPopulation pharmaco…
Genetik -
Mitazalimab DB15225
biotech | CAS: 2055640-86-1

Mitazalimab is under investigation in clinical trial NCT02379741 (ADC-1013 First-in-Human Study).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitemcinal DB06587
small molecule | CAS: 154738-42-8

Mitemcinal (GM-611) is a novel erythromycin-derived prokinetic agent that acts as an agonist at the motilin receptor.

Kategori:
Anti-Bacterial AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +5
Target Protein:
Motilin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitiglinide DB01252
small molecule | CAS: 145375-43-5

Mitiglinide is a drug for the treatment of type 2 diabetes. It may stimulate insulin secretion in beta-cells by closing off ATP dependant potassium ion channels.

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes +4
Target Protein:
ATP-binding cassette sub-family C member 8ATP-sensitive inward rectifier potassium channel 10Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitiperstat DB18963
small molecule | CAS: 1933460-19-5

Mitiperstat is under investigation in clinical trial NCT05492877 (An Efficacy and Safety Study of Mitiperstat (AZD4831) (MPO Inhibitor) vs Placebo in the Treatment of Moderate to Severe COPD.).

Target Protein:
Myeloperoxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mito-4509 DB05846
small molecule

Mito-4509 is a non-feminizing estrogen analog that could affect mitochondrial metabolic pathways. It is used to treat Parkinson's Disease, Alzheimer's Disease, Retinal Disorders and other neurologic Disorders.

Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitobronitol DB13543
small molecule | CAS: 488-41-5

Deskripsi belum tersedia.

Kategori:
AlcoholsAlkylating DrugsAntineoplastic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitoglitazone DB11721
small molecule | CAS: 146062-49-9

Mitoglitazone has been used in trials studying the treatment of Type 2 Diabetes and Alzheimer's Disease.

Kategori:
Sulfur CompoundsThiazoles
Target Protein:
Insulin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitoguazone DB12967
small molecule | CAS: 459-86-9

Mitoguazone has been used in trials studying the treatment of Lymphoma, HIV Infections, and Lymphoma, Non-Hodgkin.

Kategori:
AmidinesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +2
Target Protein:
S-adenosylmethionine decarboxylase proenzyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitolactol DB12916
small molecule | CAS: 10318-26-0

Mitolactol has been used in trials studying the treatment of Brain and Central Nervous System Tumors.

Kategori:
AlcoholsAlkylating DrugsAntineoplastic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitometh DB12117
small molecule | CAS: 107465-03-2

Mitometh is under investigation for the treatment of Adenocarcinoma, Oropharyngeal Neoplasms, Nasopharyngeal Carcinoma, Non-small Cell Lung Cancer, and Stage IV Non-small Cell Lung Cancer, among others. Mitometh has been investigated for the treatment of Lung…

Kategori:
Hydrocarbons, ChlorinatedHydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitomycin Approved DB00305
small molecule | CAS: 50-07-7

Mitomycin is an antineoplastic antibiotic first isolated by Japanese microbiologists in the 1950s from cultures of _Streptomyces caespitosus_.[L12867,A193419] It is an alkylating agent that inhibits DNA synthesis (and, at higher concentrations, RNA and protei…

Kategori:
Alkylating ActivityAlkylating DrugsAntibiotics, Antineoplastic +19
Target Protein:
DNA
Waktu Paruh8-48 min
Vol. Distribusi-
Klirens-
Genetik -
Mitomycin A DB19369
small molecule | CAS: 4055-39-4

Deskripsi belum tersedia.

Kategori:
AzirinesHeterocyclic Compounds, Fused-RingIndolequinones +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mitoquinone DB05063
small molecule | CAS: 444890-41-9

Mitoquinone is based on a novel technology, targeted lipophilic cations, that transport and concentrate antioxidants into the mitochondria -- organelles inside cells that provide energy for life processes -- where they accumulate up to a thousand fold. In 200…

Kategori:
BenzoquinonesCoenzymesEnzymes and Coenzymes +1
Waktu Paruh-
Vol. Distribusi-
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Mitotane Approved DB00648
small molecule | CAS: 53-19-0

Mitotane is an adrenolytic isomer of the insecticide dichlorodiphenyldichloroethane (DDD) - itself a metabolite of dichlorodiphenyltrichloroethane (DDT) - that inhibits cells of the adrenal cortex and their production of hormones. It has been in use since 195…

Kategori:
Adrenal Cytotoxic AgentsAntineoplastic AgentsAntineoplastic Agents, Hormonal +15
Target Protein:
Cytochrome P450 11B1, mitochondrialEstrogen receptorProgesterone receptor +2
Waktu ParuhThe plasma terminal…
Vol. DistribusiMitotane is extensi…
Klirens-
Genetik -
Mitoxantrone Approved DB01204
small molecule | CAS: 65271-80-9

An anthracenedione-derived antineoplastic agent.

Kategori:
AnalgesicsAnthracenesAnthracyclines and Related Substances +30
Target Protein:
DNA topoisomerase 2-betaDNADNA topoisomerase 2-alpha
Waktu Paruh75 hours
Vol. Distribusi* 1000 L/m2
Klirens* 21.3 L/hr/m2 [Eld…
Genetik -
Mitsugumin-53 DB16969
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Mitumomab DB06462
biotech | CAS: 216503-58-1

Mitumomab, an anti-BEC-2 monoclonal antibody derived from mice, was previously studied to treat small cell lung carcinoma in combination with BCG vaccination.

Waktu Paruh-
Vol. Distribusi-
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MIV-701 DB05736
small molecule

MIV-701 is a selective, potent inhibitor of the protease Cathepsin K. It is developed for the treatment of osteoporosis.

Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MIV-711 DB15599
small molecule

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsAntineoplastic AgentsAntirheumatic Agents
Target Protein:
Cathepsin K
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mivacurium Approved DB01226
small molecule | CAS: 133814-19-4

Mivacurium is a bisbenzylisoquinolinium based neuromuscular blocker or muscle relaxant. It binds competitively to cholinergic receptors on the motor end-plate to antagonize the action of acetylcholine, resulting in a block of neuromuscular transmission.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCentral Nervous System Depressants +13
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +1
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Mivavotinib DB16849
small molecule | CAS: 1312691-33-0

Deskripsi belum tersedia.

Target Protein:
Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mivelsiran DB19003
biotech | CAS: 2572991-83-2

Mivelsiran is under investigation in clinical trial NCT06393712 (A Phase 2 Trial of ALN-APP in Patients With Cerebral Amyloid Angiopathy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ATP-dependent dethiobiotin synthetase BioD 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mizagliflozin DB19036
small molecule | CAS: 666843-10-3

Mizagliflozin is under investigation in clinical trial NCT05721729 (Effect of Mizagliflozin Repeat Dosing on Adverse Events and Postprandial Glucose Excursions).

Kategori:
CarbohydratesGlycosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mizolastine Approved DB12523
small molecule | CAS: 108612-45-9

Mizolastine is under investigation in clinical trial NCT01928316 (A Bioequivalence Study of Domestic (Made in China) and Imported Mizolastine Tablets in Healthy Volunteers).

Kategori:
Antihistamines for Systemic UseCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +9
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mizoribine DB12617
small molecule | CAS: 50924-49-7

Mizoribine has been investigated for the treatment of Rheumatoid Arthritis.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Infective Agents +15
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0249 DB11910
small molecule | CAS: 1167574-41-5

MK0249 has been used in trials studying the treatment of Hypopnea Syndrome, Alzheimer's Disease, Paranoid Schizophrenia, Sleep Apnea, Obstructive, and Excessive Daytime Sleepiness, among others.

Kategori:
Heterocyclic Compounds, Fused-RingQuinazolines
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0354 DB05939
small molecule | CAS: 851776-28-8

MK-0354, is an orally administered drug candidate under development by Merck for the treatment of atherosclerosis and related disorders. It targets G protein-coupled receptor, or GPCR, that have the potential to regulate plasma lipid profiles, including HDL, …

Target Protein:
Hydroxycarboxylic acid receptor 2G-protein coupled estrogen receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0482 DB17453
biotech

MK-0482 is a novel humanized IgG4 monoclonal antibody targeting the immunoglobulin-like transcript (ILT) 3.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0533 DB15242
small molecule | CAS: 668455-28-5

MK-0533 is under investigation in clinical trial NCT00543959 (Efficacy and Tolerability of MK0533 in Patients With Type 2 Diabetes (0533-005)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0557 DB12168
small molecule | CAS: 328232-95-7

MK0557 has been investigated for the treatment of Schizophrenia and Paranoid Schizophrenia.

Kategori:
Cycloparaffins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0668 DB15791
small molecule | CAS: 865110-07-2

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Target Protein:
Integrin beta-1Integrin alpha-4VLA-4 (very late antigen-4)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0686 DB12563
small molecule | CAS: 578727-68-1

MK0686 has been used in trials studying the treatment of Osteoarthritis, Pain, Postoperative, and Neuralgia, Postherpetic.

Kategori:
AcetatesAcids, AcyclicAcids, Carbocyclic +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0731 DB08037
small molecule | CAS: 845256-65-7

MK-0731 is a kinesin spindle protein inhibitor and antineoplastic agent.

Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0736 DB15209
small molecule | CAS: 719272-79-4

MK-0736 is under investigation in clinical trial NCT00679055 (A Study of How MK-0736 Affects Arterial Plaque (0736-006)(TERMINATED)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0752 DB12852
small molecule | CAS: 471905-41-6

Mk 0752 is under investigation in clinical trial NCT00572182 (MK0752 in Treating Young Patients With Recurrent or Refractory CNS Cancer).

Kategori:
Acids, AcyclicAmyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme Inhibitors +5
Target Protein:
Gamma-secretase subunit PEN-2NicastrinGamma-secretase subunit APH-1B +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0767 DB12055
small molecule | CAS: 934017-32-0

MK0767 has been used in trials studying the treatment of Dyslipidemia, Diabetes Mellitus, Type 2 Diabetes Mellitus, Diabetes Mellitus, Type 2, and Diabetes Mellitus, Type II, among others.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0773 DB16244
small molecule | CAS: 606101-58-0

MK-0773 is under investigation in clinical trial NCT00529659 (A Study of the Safety and Efficacy of MK-0773 in Women With Sarcopenia (Loss of Muscle Mass)(mk-0773-005)).

Kategori:
Fused-Ring CompoundsSteroids
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0777 DB12238
small molecule | CAS: 252977-51-8

MK-0777 has been used in trials studying the treatment of Schizophrenia, Anxiety Disorder, and Generalized Anxiety Disorder.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0812 DB11990
small molecule | CAS: 624733-88-6

MK0812 has been used in trials studying the treatment of Relapsing-Remitting Multiple Sclerosis.

Target Protein:
C-C chemokine receptor type 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MK-0873 DB13029
small molecule | CAS: 500355-52-2

MK-0873 has been used in trials studying the treatment of Rheumatoid Arthritis.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +1
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10301–10350 dari 16004
Sebelumnya Halaman 207 / 321 Berikutnya