Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 206 / 236
SR 140333 DB05790
small molecule

SR 140333 is tachykinin antagonist which has potential to treat diarrhoea due to food allergy or inflammatory bowel disease.

Kategori:
Stereoisomerism
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SR-123781A DB05361
biotech | CAS: 232602-93-6

SR-123781A is a synthetic hexadecasaccharide Factor IIa and Xa antagonist. It is under investigation by Sanofi-Aventis and Organon for the treatment of thrombosis and acute coronary syndromes (ACS).

Kategori:
AnticoagulantsCarbohydratesHeparin and similars
Target Protein:
Coagulation factor XProthrombinAntithrombin-III +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SR-9009 DB14013
small molecule | CAS: 1379686-30-2

SR-9009 is a REV-ERB agonist. SR-9011 has been demonstrated that it is specifically lethal to cancer cells and oncogene-induced senescent cells, including melanocytic naevi, and has no effect on the viability of normal cells or tissues [A32628].

Kategori:
Sulfur Compounds
Target Protein:
Nuclear receptor subfamily 1 group D member 1Nuclear receptor subfamily 1 group D member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SR-9011 DB14014
small molecule | CAS: 1379686-29-9

SR-9011 is a REV-ERB agonist. SR-9011 has been demonstrated that it is specifically lethal to cancer cells and oncogene-induced senescent cells, including melanocytic naevi, and has no effect on the viability of normal cells or tissues [A32628].

Kategori:
Sulfur Compounds
Target Protein:
Nuclear receptor subfamily 1 group D member 2Nuclear receptor subfamily 1 group D member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRA-737 DB16876
small molecule | CAS: 1489389-18-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRP-6004 DB16998
biotech

A recombinant AAVrh74 gene therapy expressing the dysferlin transgene under control of a muscle-specific promoter (rAAVrh74.MHCK7.DYSF.DV).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRP-9005 DB17958
biotech

SRP-9005 is a rAAVrh74 vector containing a codon-optimized human SGCG transgene. Developed by the Kurt+Peter Foundation and Sarepta Therapeutics, it is being investigated for the treatment of Limb-girdle muscular dystrophy (LGMD) type 2C/R5.[A260142]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRT-1720 DB17057
small molecule | CAS: 925434-55-5

SRT-1720 is an activator of NAD(+)-dependent histone deacetylase SIRT1.[A253147]

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRX-1177 DB17126
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SRX-246 DB16968
small molecule | CAS: 512784-93-9

Deskripsi belum tersedia.

Kategori:
Antidiuretic Hormone Receptor AntagonistsAzetinesNatriuretic Agents
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SS1(dsFv)-PE38 DB17579
biotech

SS1(dsFv)-PE38 is a recombinant anti-mesothelin immunotoxin. SS1(dsFv)-PE38 is under investigation in clinical trial NCT01051934 (A Phase I Trial of SS1 (Dsfv) PE38 With Paclitaxel, Carboplatin, and Bevacizumab in Subjects With Unresectable Non-small Cell Lun…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SSR-126517E DB05362
small molecule

SSR-126517E is a second generation synthetic pentasaccharide that binds antithrombin with such high affinity that it assumes a plasma half-life of 80 hours.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ST-003 DB18197
biotech | CAS: 143896-17-7

ST-003 is a novel galanin receptor inhibitor being investigated for the treatment of primary sclerosing cholangitis.

Kategori:
Amino Acids, Peptides, and ProteinsNerve Tissue ProteinsNeuropeptides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ST-101 DB12621
biotech | CAS: 887603-94-3

ST-101 is a small peptide antagonist of C/EBP? and T-type calcium channel activator. ST101 has been used in trials studying the treatment of Essential Tremor and Alzheimer's Disease.[A260411]

Kategori:
Indenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ST-36 DB17275
biotech

ST-36 is a cell-penetrating dominant-negative form of activating transcription factor 5. In 2017, it received orphan drug designation by the FDA for the treatment of glioma.[L47341]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ST101 peptide DB17272
biotech

ST101 is a cell-penetrating peptide that disrupts the protein-protein interactions driving ATF5-regulated gene transcription.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stachybotrys chartarum Approved DB10847
biotech

Stachybotrys chartarum is a fungus which can provoke allergic reactions. Stachybotrys chartarum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stachyose DB19276
small molecule | CAS: 470-55-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stamulumab DB05915
biotech | CAS: 705287-60-1

MYO-029 is a human anti-GDF-8 monoclonal antibody, which is being developed to treat muscle-wasting diseases including muscular dystrophy and age-related sarcopenia.

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Target Protein:
Growth/differentiation factor 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stannous chloride Approved DB11056
small molecule | CAS: 7772-99-8

Stannous chloride is used as a source of tin in radiopharmaceutical kits. Tin reduces technetium-99m, the active radiological agent, allowing it to form a complex with phosphate-containing moeities [A32700]. These complexes localize primarily in bone (40-50%)…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stannous fluoride Approved DB11092
small molecule | CAS: 7783-47-3

Stannous Fluoride, or Tn(II) Fluoride, is a compound commonly used in toothpastes for the prevention of gingivitis, dental infections, cavities, and to relieve dental hypersensitivity. Although similar in function and activity to Sodium Fluoride (NaF), the co…

Kategori:
Alimentary Tract and MetabolismCaries Prophylactic AgentsCariostatic Agents +6
Waktu ParuhThe half-life for t…
Vol. DistribusiStannous fluoride i…
KlirensStimulated and nons…
Genetik -
Stanolone DB02901
small molecule | CAS: 521-18-6

A potent androgenic metabolite of testosterone. Dihydrotestosterone (DHT) is generated by a 5-alpha reduction of testosterone. Unlike testosterone, DHT cannot be aromatized to estradiol therefore DHT is considered a pure androgenic steroid.

Kategori:
5-Androstanon (3) DerivativesAlimentary Tract and MetabolismAnabolic Agents for Systemic Use +17
Target Protein:
Androgen receptorEstrogen receptorMineralocorticoid receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stanozolol Approved DB06718
small molecule | CAS: 10418-03-8

Stanozolol is a synthetic anabolic steroid with therapeutic uses in treating hereditary angioedema. Stanozolol is derived from testosterone, and has been abused by several high profile professional athletes.

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +10
Target Protein:
Androgen receptorGlucocorticoid binding proteins
Waktu Paruh24 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stapokibart DB18990
biotech | CAS: 2734715-10-5

Stapokibart is under investigation in clinical trial NCT06424470 (Study on the Treatment of Prurigo Nodularis With Stapokibart Injection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stapuldencel DB19275
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Starch, corn Approved DB11599
small molecule | CAS: 9005-25-8

Corn starch refers to the starch extracted from the corn grain that is commonly used as a food ingredient and chemical additive. Starch is any of a group of polysaccharides of the general formula (C6-H10-O5)n, composed of a long-chain polymer of glucose in th…

Kategori:
BiopolymersCarbohydratesCompounds used in a research, industrial, or household setting +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Staurosporine DB02010
small molecule | CAS: 62996-74-1

An indolocarbazole that is a potent protein kinase C inhibitor which enhances cAMP-mediated responses in human neuroblastoma cells. (Biochem Biophys Res Commun 1995;214(3):1114-20)

Kategori:
AlkaloidsCarbazolesEnzyme Inhibitors +6
Target Protein:
Inhibitor of nuclear factor kappa-B kinase subunit betaMuscarinic acetylcholine receptor M1Tyrosine-protein kinase Lck +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stavudine Approved DB00649
small molecule | CAS: 3056-17-5

A dideoxynucleoside analog that inhibits reverse transcriptase and has in vitro activity against HIV.

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +23
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh0.8-1.5 hours (in a…
Vol. Distribusi* 46 ± 21 L
Klirens* Renal cl=272 mL/m…
Genetik -
small molecule | CAS: 26194-89-8

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesDeoxyribonucleotidesDideoxynucleosides +6
Target Protein:
Nucleoside diphosphate kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
STC3141 DB16475
small molecule

STC3141, was investigated in clinical trial NCT04880694 to evaluate its safety and effect in subjects with severe COVID-19 pneumonia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stearic acid Approved DB03193
small molecule | CAS: 57-11-4

Stearic acid (IUPAC systematic name: octadecanoic acid) is one of the useful types of saturated fatty acids that comes from many animal and vegetable fats and oils. It is a waxy solid.

Kategori:
Fatty AcidsLipidsStearic Acids
Target Protein:
Peroxisome proliferator-activated receptor alphaGroup IID secretory phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stem bromelain Approved DB12249
biotech | CAS: 37189-34-7

The primary therapeutic use for which stem bromelain is currently and formally indicated is as a burn wound eschar debridement agent that has been approved by the EMA since 2012 and marketed under the brand name Nexobrid [FDA Label]. Bromelain itself belon…

Kategori:
Cysteine EndopeptidasesCysteine ProteasesEndopeptidases +4
Waktu ParuhThe estimated plasm…
Vol. DistribusiNo readily accessib…
KlirensNo readily accessib…
Genetik -
biotech

Mesenchymal stem cells (MSCs) exert their therapeutic effects through multiple modalities, including paracrine factors such as exosomes. Exosomes are nanometer-sized, membrane-bound vesicles secreted for the purpose of cell-cell communication. Once secreted i…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stemphylium sarciniforme Approved DB10702
biotech

Stemphylium sarciniforme is a fungus which can provoke allergic reactions. Stemphylium sarciniforme extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stepronin DB01423
small molecule | CAS: 72324-18-6

Strepronin is a mucolytic drug. A mucolytic agent is any agent which dissolves thick mucus usually used to help relieve respiratory difficulties. The viscosity of mucous secretions in the lungs is dependent upon the concentrations of mucoprotein as well as th…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAnions +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stevioside DB16882
small molecule | CAS: 57817-89-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsCarbohydratesCompounds used in a research, industrial, or household setting +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
STF-31 DB16761
small molecule | CAS: 724741-75-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
STG-001 DB16734
small molecule

STG-001 is under investigation in clinical trial NCT04489511 (Study of STG-001 in Subjects With Stargardt Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
STI-1499 DB16487
biotech

STI-1499 (COVI-GUARD was under investigation in clinical trial NCT04454398 to evaluate its safety and efficacy in patients with moderate COVID-19.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Stiripentol Approved DB09118
small molecule | CAS: 49763-96-4

Stiripentol is an antiepileptic agent that is an aromatic allylic alcohol drug, which makes it structurally unique from other antiepileptic drugs.[A19740, A250825] The clinical development and marketing of stiripentol were first delayed due to the drug's pote…

Kategori:
AnticonvulsantsBCRP/ABCG2 InhibitorsCentral Nervous System Agents +37
Target Protein:
GABA(A) ReceptorGamma-aminobutyric acid receptor subunit gamma-3L-lactate dehydrogenase A chain +1
Waktu ParuhThe elimination hal…
Vol. DistribusiThe average volume …
KlirensPlasma clearance de…
Genetik -
STM-217 DB17358
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
STP-707 DB18499
biotech

STP-707 is a small interfering RNA (siRNA) targeting TGF-Beta1 and COX-2 mRNA.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Strawberry Approved DB10571
biotech

Strawberry allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Streptococcus pneumoniae type 1 capsular polysaccharide diphtheria CRM197 protein conjugate antigen is a sterile vaccine that contains saccharides of the capsular antigens of *Streptococcus pneumoniae* serotype 1 individually conjugated to the CRM197 protein,…

Kategori:
Actively Acquired ImmunityInactivated Pneumococcal Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Streptococcus pneumoniae type 10A capsular polysaccharide diphtheria CRM197 protein conjugate antigen is a sterile vaccine that contains saccharides of the capsular antigens of *Streptococcus pneumoniae* serotype 10A individually conjugated to the CRM197 prot…

Kategori:
Inactivated Pneumococcal Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Streptococcus pneumoniae type 11A capsular polysaccharide diphtheria CRM197 protein conjugate antigen is a sterile vaccine that contains saccharides of the capsular antigens of *Streptococcus pneumoniae* serotype 11A individually conjugated to the CRM197 prot…

Kategori:
Inactivated Pneumococcal Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Streptococcus pneumoniae type 12F capsular polysaccharide diphtheria CRM197 protein conjugate antigen is a sterile vaccine that contains saccharides of the capsular antigens of *Streptococcus pneumoniae* serotype 12F individually conjugated to the CRM197 prot…

Kategori:
Inactivated Pneumococcal Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Streptococcus pneumoniae type 14 capsular polysaccharide diphtheria CRM197 protein conjugate antigen is a sterile vaccine that contains saccharides of the capsular antigens of *Streptococcus pneumoniae* serotype 14 individually conjugated to the CRM197 protei…

Kategori:
Actively Acquired ImmunityInactivated Pneumococcal Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Streptococcus pneumoniae type 15A capsular polysaccharide diphtheria CRM197 protein conjugate antigen is a sterile vaccine that contains saccharides of the capsular antigens of _Streptococcus pneumoniae_ serotype 15A individually conjugated to the CRM197 prot…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10251–10300 dari 11778
Sebelumnya Halaman 206 / 236 Berikutnya