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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 206 / 252
Reslizumab Approved DB06602
biotech | CAS: 241473-69-8

Reslizumab is a humanized interleukin-5 (IL-5) antagonist monoclonal antibody (IgG4 kappa) that is produced by recombinant DNA technology in murine myeloma non-secreting 0 (NS0) cells. IL-5 is a pro-inflammatory cytokine that is responsible for the growth and…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +12
Target Protein:
Interleukin-5
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe approximate vol…
KlirensReslizumab clearanc…
Genetik -
Resmetirom Approved DB12914
small molecule | CAS: 920509-32-6

Resmetirom is a thyroid hormone receptor-beta (THR-beta) agonist. On March 14, 2024, it was approved by the FDA as the first treatment of liver fibrosis due to noncirrhotic non-alcoholic steatohepatitis (NASH), which is a form of non-alcoholic fatty liver dis…

Kategori:
BCRP/ABCG2 InhibitorsBCRP/ABCG2 SubstratesBSEP/ABCB11 Inhibitors +15
Target Protein:
Thyroid hormone receptor beta
Waktu ParuhThe median terminal…
Vol. DistribusiResmetirom apparent…
KlirensThe steady state ap…
Genetik -
Resolvin E1 DB13105
small molecule | CAS: 552830-51-0

Resolvin E1 (RX 10001) is under investigation in clinical trial NCT00941018 (Single and Multiple Ascending Oral Dose Study of Resolvin E1 in Healthy Volunteers).

Kategori:
Dietary FatsDietary Fats, UnsaturatedEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Resorcinol Approved DB11085
small molecule | CAS: 108-46-3

Resorcinol is a 1,3-isomer (or meta-isomer) of benzenediol with the formula C6H4(OH)2. It is used as an antiseptic and disinfectant in topical pharmaceutical products in the treatment of skin disorders and infections such as acne, seborrheic dermatitis, eczem…

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Infective Agents +8
Target Protein:
Carbonic anhydrase 12Carbonic anhydrase 2Carbonic anhydrase 14 +2
Waktu ParuhSpecific data regar…
Vol. DistribusiSpecific data regar…
KlirensSpecific data regar…
Genetik -
Resorcinol monoacetate Approved DB15480
small molecule | CAS: 102-29-4

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesPhenols
Waktu Paruh-
Vol. Distribusi-
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Genetik -
RESP301 DB16497
small molecule

RESP301 was under investigation in clinical trials for various conditions. It was studied in community patients at risk of viral infections, including SARS-CoV-2, in a terminated trial (NCT04858451) and adults with rifampicin-susceptible pulmonary tuberculosi…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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Respigam DB17765
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Arexvy (respiratory syncytial virus vaccine, adjuvanted) is an adjuvanted vaccine developed by GlaxoSmithKline Biologicals. It comprises lyophilized recombinant respiratory syncytial virus glycoprotein F (RSVPreF3) stabilized in pre-fusion conformation as the…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
Waktu Paruh-
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Genetik -
Resveratrol DB02709
small molecule | CAS: 501-36-0

Resveratrol (3,5,4'-trihydroxystilbene) is a polyphenolic phytoalexin. It is a stilbenoid, a derivate of stilbene, and is produced in plants with the help of the enzyme stilbene synthase. It exists as cis-(Z) and trans-(E) isomers. The trans- form can undergo…

Kategori:
Angiogenesis InhibitorsAnticarcinogenic AgentsAntioxidants +33
Target Protein:
NAD-dependent protein deacetylase sirtuin-1Ribosyldihydronicotinamide dehydrogenase [quinone]Casein kinase II subunit alpha +23
Waktu Paruh-
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Retagliptin DB14898
small molecule | CAS: 1174122-54-3

Retagliptin is under investigation in clinical trial NCT02822534 (The Pharmacokinetics and Pharmacodynamics Study of Single and Multiple Dose of SP2086 in Type 2 Diabetes Patients).

Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
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Retapamulin Approved DB01256
small molecule | CAS: 224452-66-8

Retapamulin, marketed by GlaxoSmithKline as the ointment Altabax, is an antibiotic for skin infections like impetigo. It was approved by the FDA in April 2007.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics for Topical Use +6
Target Protein:
50S ribosomal protein L3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Retaspimycin DB05626
small molecule | CAS: 857402-23-4

Deskripsi belum tersedia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Retatrutide DB18993
biotech | CAS: 2381089-83-2

Retatrutide is under investigation in clinical trial NCT06354660 (Effect of Retatrutide Compared With Placebo in Adult Participants With Type 2 Diabetes and Inadequate Glycemic Control With Diet and Exercise Alone (TRANSCEND-T2D-1)).

Kategori:
Amino Acids, Peptides, and ProteinsLipids
Waktu Paruh-
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Reteplase Approved DB00015
biotech | CAS: 133652-38-7

Human tissue plasminogen activator, purified, glycosylated, 355 residues purified from CHO cells. Retavase is considered a "third-generation" thrombolytic agent, genetically engineered to retain and delete certain portions of human tPA. Retavase is a deletion…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +17
Target Protein:
PlasminogenFibrinogen alpha chainPlasminogen activator inhibitor 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Retifanlimab Approved DB15766
biotech | CAS: 2079108-44-2

Retifanlimab is a humanized IgG4 kappa monoclonal antibody that binds to the programmed death receptor-1 (PD-1), blocking PD-1 interaction with its ligands, programmed death-ligand 1 (PD-L1) and programmed death-ligand 2 (PD-L2). By blocking the PD-1/PD-L1/2 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +11
Target Protein:
Programmed cell death protein 1
Waktu ParuhAt steady-state, re…
Vol. DistribusiAt steady-state, re…
KlirensFollowing the first…
Genetik -
small molecule | CAS: 74193-17-2

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech | CAS: 2395839-91-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Retosiban DB11818
small molecule | CAS: 820957-38-8

Retosiban has been used in trials studying the treatment of Premature Labor and Obstetric Labour, Premature.

Target Protein:
Oxytocin receptor
Waktu Paruh-
Vol. Distribusi-
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REV131 DB05032
small molecule

rEV131 is in development for allergic rhinitis, asthma and several inflammatory eye diseases. It is a topically delivered small protein that acts as an anti-inflammatory agent.

Kategori:
Amino Acids, Peptides, and ProteinsProteins
Target Protein:
Histamine H4 receptor
Waktu ParuhApproximately 8 hou…
Vol. Distribusi-
Klirens-
Genetik -
Revamilast DB11838
small molecule | CAS: 893555-90-3

Revamilast has been used in trials studying the treatment of Asthma and Rheumatoid Arthritis.

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Revaprazan DB16308
small molecule | CAS: 199463-33-7

Revaprazan is under investigation in clinical trial NCT01750437 (Phase 2 Clinical Trial to Investigate the Safety, Tolerability and Efficacy of YH1885L in Patients With Non-erosive Reflux Disease(nerd)).

Kategori:
Heterocyclic Compounds, Fused-RingIsoquinolinesPyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Revefenacin Approved DB11855
small molecule | CAS: 864750-70-9

Revefenacin is a novel biphenyl carbamate tertiary amine agent that belongs to the family of the long-acting muscarinic antagonists (LAMA). The labile primary amide in the structure produces a "soft-drug" site that allows rapid systemic clearance and minimizi…

Kategori:
AmidesAnticholinergic AgentsBCRP/ABCG2 Substrates +9
Target Protein:
Muscarinic acetylcholine receptor
Waktu ParuhThe apparent termin…
Vol. DistribusiAfter intravenous a…
KlirensThe renal clearance…
Genetik -
biotech | CAS: 1446198-96-4

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Reversine DB07340
small molecule | CAS: 656820-32-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingOxazinesProtein Kinase Inhibitors
Target Protein:
Adenosine receptor A3Dual specificity mitogen-activated protein kinase kinase 1Aurora kinase B +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Reviparin Approved DB09259
small molecule | CAS: 9041-08-1

Reviparin is a low molecular weight heparin which seems to have a better safety profile than unfractionated heparin.[A32019] It is prepared from porcine intestinal mucosa by nitrous acid depolymerization. Reviparin has a molecular weight of 3.9 kDa.[A32021] I…

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Revumenib Approved DB18515
small molecule | CAS: 2169919-21-3

Abnormal gene rearrangements at chromosome locus 11q23, called KMT2A rearrangements or translocations, are present in 5%-10% of patients with acute leukemias and are the sole genetic aberration found in the majority of infant acute lymphoblastic leukemia case…

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +17
Target Protein:
Menin
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe the geometric m…
KlirensFollowing oral admi…
Genetik -
Revusiran DB16309
biotech | CAS: 1438322-82-7

Revusiran is under investigation in clinical trial NCT02319005 (ENDEAVOUR: Phase 3 Multicenter Study of Revusiran (ALN-TTRSC) in Patients With Transthyretin (TTR) Mediated Familial Amyloidotic Cardiomyopathy (FAC)).

Kategori:
Antisense Elements (Genetics)Molecular ProbesNucleic Acid Probes +5
Target Protein:
Transthyretin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rexin G DB16450
biotech | CAS: 1023923-93-4

Rexin-G is a tumor-targeted, injectable retroviral vector carrying a mutant form of the cyclin G1 gene. It is under development by Epeius Biotechnologies for the potential treatment of metastatic cancer. It is also being investigated for preventing SARSCOV-2 …

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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biotech | CAS: 2172954-10-6

Rexlemestrocel-L is an investigational human bone marrow-derived allogeneic mesenchymal precursor cell (MPC) product. It is being investigated in various cardiac conditions, such as chronic heart failure and acute myocardial infarction.

Waktu Paruh-
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Genetik -
biotech

Reynoutria multiflora root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Rezafungin Approved DB16310
small molecule | CAS: 1396640-59-7

Rezafungin is an echinocandin antifungal drug.[A258393,L45633] Unlike other echinocandins such as [caspofungin] and [micafungin], rezafungin has long?acting pharmacokinetics and a high stability that allows for it to have long dosing intervals maintaining hig…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +8
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu ParuhRezafungin has a te…
Vol. DistribusiRezafungin has a vo…
KlirensRezafungin has an e…
Genetik -
Rezatapopt DB18980
small molecule | CAS: 2636846-41-6

Rezatapopt is under investigation in clinical trial NCT04585750 (The Evaluation of PC14586 in Patients With Advanced Solid Tumors Harboring a TP53 Y220C Mutation (PYNNACLE)).

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biotech | CAS: 2641686-76-0

Rezpegaldesleukin is under investigation in clinical trial NCT04433585 (A Study of LY3471851 in Adults With Systemic Lupus Erythematosus (SLE)).

Waktu Paruh-
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Rezvilutamide DB19133
small molecule | CAS: 1572045-62-5

Rezvilutamide is under investigation in clinical trial NCT05956639 (Comparing a 6-month vs Long-term Course of Rezvilutamide With ADT Plus Chemotherapy in Mhspc).

Waktu Paruh-
Vol. Distribusi-
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RG-2833 DB16955
small molecule | CAS: 1215493-56-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAcids, CarbocyclicAmides +5
Target Protein:
Histone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RG-4733 DB11870
small molecule | CAS: 847925-91-1

Ro4929097 has been used in trials studying the treatment of Sarcoma, LYMPHOMA, Neoplasms, Wilm's Tumor, and OSTEOSARCOMA, among others.

Kategori:
Amyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme InhibitorsGamma Secretase Inhibitors and Modulators +3
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RG-7795 DB06329
small molecule | CAS: 892498-64-5

Deskripsi belum tersedia.

Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
RG2417 DB05055
small molecule

RG2417 is a proprietary formulation of uridine, a biological compound essential for the synthesis of DNA and RNA, the basic hereditary material found in all cells, and numerous other factors essential for cell metabolism. Uridine is synthesized by the mitocho…

Waktu Paruh-
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RGG0853 DB18669
biotech

RGG0853 is an E1A lipid complex, a repressor gene complexed with a cationic lipid vector.

Waktu Paruh-
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rGLP-1 DB05433
small molecule

rGLP-1 is a continuous infusion of glucagon-like peptide 1, or GLP-1, targeted for the treatment of congestive heart failure (CHF) in patients ineligible for transplant. GLP-1 is a naturally occurring hormone produced in the intestines in response to food int…

Kategori:
Gastrointestinal HormonesGlucagon-Like PeptidesHormones +3
Waktu Paruh-
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RGX-501 DB17639
biotech

RGX-501 is an adeno-associated virus vector 8 (AAV8)-mediated gene therapy that delivers a functional copy of the human low-density lipoprotein receptor (LDLR) gene to liver cells. It is being investigated for the treatment of homozygous familial hypercholest…

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RH-1 DB04090
small molecule | CAS: 221635-42-3

RH-1 has been used in trials studying the treatment of Advanced Solid Tumors and Non-Hodgkin's Lymphoma.

Target Protein:
NAD(P)H dehydrogenase [quinone] 1
Waktu Paruh-
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Rhamnose DB02961
small molecule | CAS: 3615-41-6

A methylpentose whose L- isomer is found naturally in many plant glycosides and some gram-negative bacterial lipopolysaccharides. [PubChem]

Kategori:
CarbohydratesDeoxy Sugars
Target Protein:
L-rhamnose isomerase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
RHCC10 DB18531
biotech

RHCC10 is a recombinant human Clara cell protein.

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Rheinanthrone DB13175
small molecule | CAS: 480-09-1

Rheinanthrone is the active metabolite of senna glycoside [DB11365] known for its laxative effect [A19235]. It is commonly produced by plants of the Rheum species [L772].

Kategori:
Anthracenes
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Genetik -
small molecule | CAS: 644961-22-8

Deskripsi belum tersedia.

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Rhenium re-186 DB19266
small molecule | CAS: 14998-63-1

Rhenium re-186 is under investigation in clinical trial NCT01906385 (Maximum Tolerated Dose, Safety, and Efficacy of Rhenium Nanoliposomes in Recurrent Glioma (Respect)).

Kategori:
ElementsIsotopesMetals +2
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Rhenium re-188 DB19267
small molecule | CAS: 14378-26-8

Rhenium re-188 is under investigation in clinical trial NCT03458559 (Rhenium-188-hedp vs. Radium-223-chloride in Patients With Advanced Prostate Cancer Refractory to Hormonal Therapy).

Kategori:
ElementsIsotopesMetals +2
Waktu Paruh-
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rhGAD65 DB04963
biotech

rhGAD65 (recombinant human glutamic acid decarboxylase) is a vaccine being developed to treat insulin dependent type 1 diabetes.

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rhIGFBP-3 DB05897
biotech

rhIGFBP-3 (recombinant human insulin-like growth factor binding protein-3) is Insmed’s proprietary anti-cancer compound that has demonstrated significant decreases in cancerous growth in several models of human. It is developed by Insmed and is currently unde…

Target Protein:
Insulin-like growth factor 1 receptor
Waktu Paruh-
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