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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 206 / 321
Midazolam Approved DB00683
small molecule | CAS: 59467-70-8

Midazolam is a short-acting hypnotic-sedative drug with anxiolytic, muscle relaxant, anticonvulsant, sedative, hypnotic, and amnesic properties.[A173842] It belongs to a class of drugs called _benzodiazepines_. This drug is unique from others in this class du…

Kategori:
Adjuvants, AnesthesiaAnestheticsAnti-Anxiety Agents +27
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site +1
Waktu Paruh**Intravenous**: …
Vol. DistribusiFemale gender, old …
Klirens**Intramuscular** …
Genetik -
Midecamycin DB13456
small molecule | CAS: 35457-80-8

Midecamycin is a naturally occurring 16-membered macrolide[A33072] that fits under the category of acetoxy-substituted macrolide antibiotics. In this molecule, an acetoxy group is substituted on the position 9 of the 16-member ring and on position 4 of the te…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +12
Waktu ParuhThe half-life of mi…
Vol. DistribusiThe reported appare…
KlirensMidecamycin present…
Genetik -
Midodrine Approved DB00211
small molecule | CAS: 42794-76-3

An ethanolamine derivative that is an adrenergic alpha agonist. It is used as a vasoconstrictor agent in the treatment of hypotension.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +19
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor
Waktu ParuhThe metabolites dis…
Vol. Distribusi-
Klirens* Renal cl=385 mL/m…
Genetik -
Midomafetamine DB01454
small molecule | CAS: 42542-10-9

An N-substituted amphetamine analog. It is a widely abused drug classified as a hallucinogen and causes marked, long-lasting changes in brain serotonergic systems. It is commonly referred to as MDMA or ecstasy. It is a widely abused drug classified as a hallu…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +20
Target Protein:
Synaptic vesicular amine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter +4
Waktu Paruh6–10 (though durati…
Vol. Distribusi-
Klirens-
Genetik -
Midostaurin Approved DB06595
small molecule | CAS: 120685-11-2

Midostaurin (as Rydapt) is a multitarget kinase inhibitor for the treatment for adult patients with newly diagnosed acute myeloid leukemia (AML) who have a specific genetic mutation called FLT3. It was initially characterized as a potential broad-spectrum ant…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +53
Target Protein:
Protein kinase C gamma typeProtein kinase C alpha typeVascular endothelial growth factor receptor 2 +4
Waktu ParuhElimination half li…
Vol. DistribusiThe Vd of midostaur…
KlirensThe clearance value…
Genetik -
Mifamurtide Approved DB13615
small molecule | CAS: 83461-56-7

Mifamurtide is an immunomodulator with antitumor activity via activation of macrophages and monocytes. Also called L-MTP-PE, mifamurtide may be a liposomal form of of the active ingredient MTP-PE, which is a synthetic, less pyrogenic, and longer-acting deriva…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAmino Sugars +15
Target Protein:
Toll-like receptor 4Nucleotide-binding oligomerization domain-containing protein 2
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe mean volume of …
KlirensThe clearance from …
Genetik -
Mifepristone Approved DB00834
small molecule | CAS: 84371-65-3

Mifepristone is a progestational and glucocorticoid hormone antagonist. Its inhibition of progesterone induces bleeding during the luteal phase and in early pregnancy by releasing endogenous prostaglandins from the endometrium or decidua. As a glucocorticoid …

Kategori:
Abortifacient AgentsAbortifacient Agents, SteroidalAdrenal Cortex Hormones +49
Target Protein:
Progesterone receptorGlucocorticoid receptorProstate-specific antigen +1
Waktu Paruh18 hours
Vol. Distribusi-
Klirens-
Genetik -
Migalastat Approved DB05018
small molecule | CAS: 108147-54-2

Fabry disease is a rare, progressive genetic disorder characterized by a defective GLA gene that causes a deficiency in the enzyme alpha-Galactosidase A (alpha-Gal A). This enzyme is responsible for breaking down glycosphingolipid substrate that, when deficie…

Kategori:
Alimentary Tract and MetabolismAlkaloidsAlpha-Galactosidase A (alpha-Gal A) Pharmacological Chaperones +6
Target Protein:
Alpha-galactosidase A
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn healthy voluntee…
KlirensFollowing ascending…
Genetik -
Miglitol Approved DB00491
small molecule | CAS: 72432-03-2

Miglitol inhibits the breakdown complex carbohydrates into glucose. It is primarily used in diabetes mellitus type 2 for establishing greater glycemic control by preventing the digestion of carbohydrates (such as disaccharides, oligosaccharides, and polysacch…

Kategori:
Alimentary Tract and MetabolismAlkaloidsBlood Glucose Lowering Agents +10
Target Protein:
Lysosomal alpha-glucosidaseNeutral alpha-glucosidase ABNeutral alpha-glucosidase C +1
Waktu ParuhThe elimination hal…
Vol. Distribusi* 0.18 L/kg
Klirens-
Genetik -
Miglustat Approved DB00419
small molecule | CAS: 72599-27-0

Miglustat, commonly marketed under the trade name Zavesca, is a drug used to treat Gaucher disease. It inhibits the enzyme glucosylceramide synthase, an essential enzyme for the synthesis of most glycosphingolipids. It is only used for patients who cannot be …

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnti-HIV Agents +14
Target Protein:
Ceramide glucosyltransferase
Waktu ParuhThe effective half-…
Vol. Distribusi-
Klirens-
Genetik -
Milademetan DB15257
small molecule | CAS: 1398568-47-2

Milademetan is under investigation in clinical trial NCT02319369 (Safety, Tolerability and Pharmacokinetics of Milademetan Alone and With 5-Azacitidine (AZA) in Acute Myelogenous Leukemia (AML) or High-Risk Myelodysplastic Syndrome (MDS)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Coagulation factor VIII
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milataxel DB12334
small molecule | CAS: 352425-37-7

Milataxel has been used in trials studying the treatment of Mesothelioma.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Target Protein:
Tubulin beta-1 chainTubulin beta chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milatuzumab DB12943
biotech | CAS: 899796-83-9

Milatuzumab has been used in trials studying the treatment of Lupus Nephritis, Multiple Myeloma (MM), GVHD (Acute or Chronic), Myelodysplastic Syndrome, and Chronic Lymphocytic Leukemia, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 129496-10-2

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 802539-81-7

Milciclib Maleate is under investigation in clinical trial NCT01301391 (Study of Oral PHA-848125AC in Patients With Malignant Thymoma Previously Treated With Multiple Lines of Chemotherapy).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Cyclin-dependent kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milk thistle Approved DB14375
biotech | CAS: 65666-07-1

Milk thistle is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milnacipran Approved DB04896
small molecule | CAS: 92623-85-3

Milnacipran is a selective serotonin and norepinephrine reuptake inhibitor (SNRI) and like many agents in this category was originally developed for and continues to be approved and indicated for the treatment of depression [F3928, F3934, A175786, A175951]. F…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +30
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterNMDA receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThe total plasma cl…
Genetik -
Milrinone Approved DB00235
small molecule | CAS: 78415-72-2

Heart failure is a multifactorial condition that affects roughly 1-2% of the adult population. Often the result of long-term myocardial ischemia, cardiomyopathy, or other cardiac insults, heart failure results from an inability of the heart to perfuse periphe…

Kategori:
AminesAminopyridinesCardiac Stimulants Excl. Cardiac Glycosides +12
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu ParuhMilrinone administe…
Vol. DistribusiMilrinone administe…
KlirensMilrinone administe…
Genetik -
Miltefosine Approved DB09031
small molecule | CAS: 58066-85-6

Miltefosine is a broad spectrum antimicrobial, anti-leishmanial, phospholipid drug that was originally developed in the 1980s as an anti-cancer agent. It is currently the only recognized oral agent used to treat visceral, cutaneous, and mucosal forms of leish…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAminesAnti-Infective Agents +9
Target Protein:
Phospholipase A2ATP-dependent translocase ABCB1
Waktu ParuhThe primary elimina…
Vol. DistribusiRadioactivity studi…
KlirensPlasma clearance is…
Genetik -
Milvexian DB16233
small molecule | CAS: 1802425-99-5

Milvexian is under investigation in clinical trial NCT03766581 (A Study on BMS-986177 for the Prevention of a Stroke in Patients Receiving Aspirin and Clopidogrel).

Target Protein:
Coagulation factor XI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mimopezil DB05520
small molecule | CAS: 180694-97-7

Mimopezil is an acetylcholinesterase (AChE) inhibitor that has demonstrated potential use in the treatment of Alzheimer's disease. Mimopezil is a pro-drug that is rapidly absorbed and converted into huperzine A.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mimosine DB01055
small molecule | CAS: 500-44-7

Mimosine is an antineoplastic alanine-substituted pyridine derivative isolated from _Leucena glauca_.

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +2
Target Protein:
Serine hydroxymethyltransferase, cytosolicC-C motif chemokine 2Tyrosinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minaprine Approved DB00805
small molecule | CAS: 25905-77-5

Minaprine is a psychotropic drug which has proved to be effective in the treatment of various depressive states. Like most antidepressants minaprine antagonizes behavioral despair. Minaprine is an amino-phenylpyridazine antidepressant reported to be relative…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +17
Target Protein:
Amine oxidase [flavin-containing] A5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2A +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mineral oil Approved DB11057
small molecule | CAS: 8042-47-5

Mineral oil, or paraffin oil, is a mixture of higher alkanes from a mineral source, such as petroleum. Petroleum mineral oil is manufactured from crude oils by vacuum distillation to produce several distillates and a residual oil that are then further refined…

Kategori:
Alimentary Tract and MetabolismBasic Ointments and ProtectantsDermatologicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minigastrin DB19196
biotech | CAS: 101212-63-9

Minigastrin is under investigation in clinical trial NCT06155994 (68ga-dota-mgs5 PET/CT in Patients With Advanced Neuroendocrine Tumours).

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minnelide DB17309
small molecule | CAS: 1254702-87-8

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +6
Target Protein:
Heat shock 70 kDa protein 1BHeat shock 70 kDa protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1254885-39-6

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minocycline Approved DB01017
small molecule | CAS: 10118-90-8

Minocycline was first described in the literacture in 1966.[A190681] It is a second generation tetracycline antibiotic that is active against gram-negative and gram-positive bacteria.[A190723] Like other semisynthetic tetracyclines, minocycline has modificati…

Kategori:
Agents Causing Muscle ToxicityAgents that produce neuromuscular block (indirect)Alimentary Tract and Metabolism +16
Target Protein:
30S ribosomal protein S930S ribosomal protein S416S ribosomal RNA +9
Waktu ParuhThe half life of mi…
Vol. DistribusiThe volume of distr…
KlirensIntravenous minocyc…
Genetik -
Minodronic acid DB06548
small molecule | CAS: 180064-38-4

Deskripsi belum tersedia.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Target Protein:
Farnesyl pyrophosphate synthaseGeranylgeranyl pyrophosphate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minoxidil Approved DB00350
small molecule | CAS: 38304-91-5

A potent direct-acting peripheral vasodilator (vasodilator agents) that reduces peripheral resistance and produces a fall in blood pressure.

Kategori:
Antihypertensive AgentsAntihypertensive Agents Indicated for HypertensionArteriolar Smooth Muscle, Agents Acting On +13
Target Protein:
ATP-sensitive inward rectifier potassium channel 1ReninProstaglandin G/H synthase 1
Waktu Paruh4.2 hours
Vol. Distribusi-
Klirens-
Genetik -
Minretumomab DB15470
biotech | CAS: 195189-17-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minzasolmin DB18961
small molecule | CAS: 1802518-92-8

Minzasolmin is under investigation in clinical trial NCT05543252 (An Extension Study to Evaluate the Long-term Efficacy, Safety and Tolerability of Minzasolmin (UCB0599) in Study Participants With Parkinson's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miocamycin Approved DB13287
biotech | CAS: 55881-07-7

Miocamycin is a macrolide type antimicrobial [A176170]. This drug may be marketed in Japan for clinical use as it is listed in the Japanese pharmacopeia [L5737]. It has shown to be effective against several gram-positive and gram-negative microbes and may be …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MIP-1095 I-123 DB12994
small molecule | CAS: 949575-25-1

123 I Mip 1095 is under investigation in clinical trial NCT00712829 (Study to Evaluate the Safety, Pharmacokinetics, Tissue Distribution, Metabolism and Dosimetry of Two Prostate Cancer Imaging Agents).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MIP-1095 I-131 DB14978
small molecule | CAS: 1258980-67-4

MIP-1095 I-131 is under investigation in clinical trial NCT03030885 (Use of an Experimental Radiopharmaceutical (131I-MIP-1095) in Men With Metastatic Castration-Resistant Prostate Cancer (mCRPC)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mipicoledine DB15075
small molecule | CAS: 942149-56-6

Mipicoledine is under investigation in clinical trial NCT01048008 (Study of 4-Demethylcholesteryloxycarbonylpenclomedine (DM-CHOC-PEN) in Patients With Advanced Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mipomersen Approved DB05528
biotech | CAS: 1000120-98-8

Mipomersen sodium, which was known as the investigational drug, isis-301012, is the salt form of a synthetic phosphorothioate oligonucleotide. Mipomersen sodium prevents the formation of apo B-100, resulting in a decrease in the levels of apolipoprotein B (ap…

Kategori:
Anticholesteremic AgentsAntisense Elements (Genetics)Antisense Oligonucleotides +20
Target Protein:
Apolipoprotein B-100mRNA of ApoB-100
Waktu ParuhMipomersem has a ve…
Vol. DistribusiThe volume of distr…
KlirensClearance of mipome…
Genetik -
Mipsagargin DB11813
small molecule | CAS: 1245732-48-2

Mipsagargin has been used in trials studying the treatment of Prostate Cancer, Prostatic Neoplasms, Advanced Solid Tumors, Glioblastoma Multiforme, and Hepatocellular Carcinoma, among others.

Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirabegron Approved DB08893
small molecule | CAS: 223673-61-8

Mirabegron is a sympathomimetic beta-3 adrenergic receptor agonist used to relax the smooth muscle of the bladder in the treatment of urinary frequency and incontinence. It is unique amongst overactive bladder treatment options in that, unlike other treatment…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-3 Receptor Agonists +32
Target Protein:
Beta-3 adrenergic receptorBeta-1 adrenergic receptor
Waktu ParuhThe mean terminal e…
Vol. DistribusiFollowing intraveno…
KlirensTotal plasma cleara…
Genetik -
Miramistin ion DB19386
small molecule | CAS: 91481-38-8

Miramistin ion is under investigation in clinical trial NCT05561816 (Efficacy and Safety of Dioxidin Versus Miramistin in Superficial Pyoderma).

Kategori:
AminesBenzylammonium CompoundsOnium Compounds +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miransertib DB14982
small molecule | CAS: 1313881-70-7

Miransertib is under investigation in clinical trial NCT01473095 (Phase 1 Dose Escalation Study of ARQ 092 in Adult Subjects With Advanced Solid Tumors and Recurrent Malignant Lymphoma).

Kategori:
AminesPyridines
Target Protein:
RAC-gamma serine/threonine-protein kinaseRAC-alpha serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miravirsen DB12851
biotech | CAS: 1072874-90-8

Miravirsen has been investigated for the treatment of Hepatitis C and Hepatitis C, Chronic.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirdametinib DB07101
small molecule | CAS: 391210-10-9

PD-0325901 has been used in trials studying the treatment and basic science of Melanoma, Solid Tumour, Solid Tumors, Advanced Cancer, and Breast Neoplasms, among others.

Kategori:
Acids, CarbocyclicAmidesAmines +3
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirfentanil DB09175
small molecule | CAS: 117523-47-4

Mirfentanil is a derivative of fentanyl that presents high selectivity for the mu opioid receptor. At lower doses, it antagonizes the analgesic effects of alfentanil and substitutes for naloxone in morphine-treated monkeys; however, it also reverses naloxone-…

Kategori:
Piperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miricorilant DB16234
small molecule | CAS: 1400902-13-7

Miricorilant is under investigation in clinical trial NCT03818256 (Study Evaluating the Safety, Efficacy, and Pharmacokinetics of Miricorilant (CORT118335) in Obese Adult Patients With Schizophrenia and Recent Weight Gain While Taking Antipsychotic Medication…

Kategori:
PyrimidinesPyrimidinones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miridesap DB13087
small molecule | CAS: 224624-80-0

Miridesap has been used in trials studying the prevention of HIV and treatment of AL amyloidosis.

Target Protein:
Serum amyloid P-component
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirikizumab Approved DB14910
biotech | CAS: 1884201-71-1

Mirikizumab is a monoclonal antibody developed by Eli Lilly intended to treat ulcerative colitis. It inhibits the actions of interleukin-23 (IL-23), a pro-inflammatory cytokine that activates pathways contributing to the development of inflammatory diseases.[…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnti-Inflammatory Agents +16
Target Protein:
Interleukin-23 subunit alpha
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Mirococept DB06492
biotech | CAS: 507453-82-9

Mirococept (APT070) is a complement inhibitor currently under development for treatment of rheumatoid arthritis and I/RI. It is a truncated form of the human Complement Receptor 1 (CR1) linked to a unique Prodaptin™ construct that regulates the over-productio…

Target Protein:
Complement C3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirodenafil DB11792
small molecule | CAS: 862189-95-5

Mirodenafil has been used in trials studying the treatment and supportive care of Kidney Diseases, Urologic Diseases, Renal Insufficiency, Erectile Dysfunction, and Male Erectile Dysfunction.

Kategori:
AmidesEnzyme InhibitorsPhosphodiesterase 5 Inhibitors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mirogabalin DB11825
small molecule | CAS: 1138245-13-2

Mirogabalin has been used in trials studying the treatment of Post-herpetic Neuralgia, Pain Associated With Fibromyalgia, and Diabetic peripheral neuropathic pain.

Kategori:
AnalgesicsBridged-Ring CompoundsGabapentinoids +1
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10251–10300 dari 16004
Sebelumnya Halaman 206 / 321 Berikutnya