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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 205 / 236
Soticlestat DB16987
small molecule | CAS: 1429505-03-2

Deskripsi belum tersedia.

Kategori:
Cholesterol 24S-Hydroxylase Inhibitor
Target Protein:
Cholesterol 24-hydroxylase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sotigalimab DB16413
biotech | CAS: 2305607-45-6

Sotigalimab is under investigation in clinical trial NCT03123783 (CD40 Agonistic Antibody APX005M in Combination With Nivolumab).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Sotirimod DB05680
small molecule | CAS: 227318-75-4

Deskripsi belum tersedia.

Waktu Paruh-
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Sotorasib Approved DB15569
small molecule | CAS: 2252403-56-6

Sotorasib, also known as AMG-510, is an acrylamide-derived KRAS inhibitor developed by Amgen.[A187547,A187556] It is indicated in the treatment of adult patients with KRAS G12C mutant non-small cell lung cancer.[L34288] This mutation makes up >50% of all KRAS…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalAntineoplastic and Immunomodulating Agents +13
Target Protein:
GTPase KRas
Waktu ParuhSotorasib has a ter…
Vol. DistribusiThe volume of distr…
KlirensSotorasib has an ap…
Genetik -
Sotrastaurin DB12369
small molecule | CAS: 425637-18-9

Sotrastaurin has been used in trials studying the basic science and treatment of Uveal Melanoma, Richter Syndrome, Prolymphocytic Leukemia, Recurrent Mantle Cell Lymphoma, and Recurrent Small Lymphocytic Lymphoma, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Protein kinase C theta typeProtein kinase C beta typeProtein kinase C alpha type
Waktu Paruh-
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Sotrovimab Approved DB16355
biotech | CAS: 2423014-07-5

Sotrovimab (VIR-7831), also known as GSK4182136, is a monoclonal antibody that can neutralize the SARS-CoV-2 virus.[L34440] Sotrovimab was initially been granted emergency use authorization (EUA) to treat mild-to-moderate COVID-19 on May 26, 2021, based on in…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +13
Target Protein:
Spike glycoprotein
Waktu ParuhThis antibody has u…
Vol. DistribusiSotrovimab is an Fc…
Klirens-
Genetik -
Sovaprevir DB12069
small molecule | CAS: 1001667-23-7

Sovaprevir has been investigated for the treatment of Hepatitis C, Chronic.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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Sovleplenib DB17557
small molecule | CAS: 1415792-84-5

Sovleplenib is a novel, investigational, selective small molecule inhibitor for oral administration targeting spleen tyrosine kinase (Syk). It is under investigation in clinical trial NCT03483948 (Phase I Study of Hmpl-523+azacitidine in Elderly Patients With…

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Soybean oil Approved DB09422
biotech | CAS: 8001-22-7

Derived from soybeans, soybean oil is a common vegetable oil and a source of polyunsaturated and saturated fatty acids. It is a complex mixture of triglycerides where per 100 g, soybean oil has 16 g of saturated fat, 23 g of monounsaturated fat, and 58 g of p…

Kategori:
Biological ProductsCaloric AgentsComplex Mixtures +12
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. DistribusiAfter triglycerides…
KlirensThe elimination rat…
Genetik -
SP-101 DB18274
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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SP-420 DB16069
small molecule | CAS: 911714-45-9

SP-420 is under investigation in clinical trial NCT03801889 (SP-420 in Subjects With Transfusion-dependent Beta-thalassemia or Other Rare Anemias).

Kategori:
CyclohexanesCycloparaffinsKetones +1
Waktu Paruh-
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Sp-722 DB04503
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
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SP-8203 DB11670
small molecule | CAS: 1176758-04-5

SP-8203 has been used in trials studying the treatment of Ischemic Stroke.

Kategori:
AcetatesAcids, AcyclicAmides +5
Waktu Paruh-
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SP-876 DB03558
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
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SP1049C DB04978
small molecule

SP1049C is a novel anthracycline chemotherapeutic agent containing [doxorubicin] and two nonionic pluronic block copolymers.[A260416] It is designed to overcome drug resistance in a number of cancers. It has successfully completed Phase 1 trials. Phase 2 resu…

Kategori:
AlcoholsAnthracyclinesCarbohydrates +8
Target Protein:
DNA topoisomerase 2-alpha
Waktu Paruh-
Vol. Distribusi-
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SP2456 DB03957
small molecule

Deskripsi belum tersedia.

Target Protein:
Interleukin-2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Spaglumic acid DB08835
small molecule | CAS: 4910-46-7

Spaglumic acid is the ?-aspartyl isoform of N-Acetyl-l-aspartylglutamate (isospaglumic Acid is N-(N-Acetyl-l-?-aspartyl)-l-glutamic acid). In eye drops, spaglumic acid is either a magnesium or sodium salt of N-Acetyl-l-aspartylglutamate. Spaglumic acid is a m…

Kategori:
Antiallergic Agents, Excl. CorticosteroidsDecongestants and AntiallergicsMast Cell Stabilizers +3
Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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Sparfloxacin Approved DB01208
small molecule | CAS: 110871-86-8

Sparfloxacin is a fluoroquinolone antibiotic indicated for bacterial infections. Sparfloxacin exerts its antibacterial activity by inhibiting DNA gyrase, a bacterial topoisomerase. DNA gyrase is an essential enzyme which controls DNA topology and assists in D…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhMean terminal elimi…
Vol. Distribusi-
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Sparfosic acid DB03459
small molecule | CAS: 51321-79-0

Sparfosic acid is a solid. This compound belongs to the n-acyl-alpha amino acids. These are compounds containing an alpha amino acid which bears an acyl group at the terminal nitrogen atom. This substance is known to target aspartate carbamoyltransferase cata…

Kategori:
AcetatesAcids, AcyclicAmino Acids +12
Target Protein:
Aspartate carbamoyltransferase catalytic chainMultifunctional protein CAD
Waktu Paruh-
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Genetik -
Sparsentan Approved DB12548
small molecule | CAS: 254740-64-2

Sparsentan is a dual antagonist of the endothelin type A receptor (ET<sub>A</sub>R) and the angiotensin II (Ang II) type 1 receptor (AT<sub>1</sub>R) with a similar affinity for both (9.3 nM for ET<sub>A</sub>R and 0.8 nM for AT<sub>1</sub>R).[A257330,L45300]…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAmidesAngiotensin 2 Receptor Blocker +30
Target Protein:
Endothelin-1 receptorType-1 angiotensin II receptorType-2 angiotensin II receptor
Waktu ParuhSparsentan has an e…
Vol. DistribusiAt the approved rec…
KlirensSparsentan has a ti…
Genetik -
Sparsomycin DB04222
small molecule | CAS: 1404-64-4

An antitumor antibiotic produced by Streptomyces sparsogenes. It inhibits protein synthesis in 70S and 80S ribosomal systems. [PubChem]

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsEnzyme Inhibitors +3
Waktu Paruh-
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Spartalizumab DB14892
biotech | CAS: 1935694-88-4

Spartalizumab is under investigation in clinical trial NCT02605967 (Safety and Efficacy Study of PDR001 in Patients With Recurrent or Metastatic Nasopharyngeal Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
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Sparteine DB06727
small molecule | CAS: 90-39-1

Sparteine is a plant alkaloid derived from _Cytisus scoparius_ and _Lupinus mutabilis_ which may chelate calcium and magnesium. It is a sodium channel blocker, so it falls in the category of class 1a antiarrhythmic agents. Sparteine is not currently FDA-appro…

Kategori:
AlkaloidsAntiarrhythmic agentsAntiarrhythmics, Class I +13
Waktu Paruh-
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SPC2968 DB06351
biotech

SPC2968 is a synthetic antisense oligodeoxynucleotide targeting hypoxia-inducible factor-1alpha (HIF-1alpha). It was under investigation in clinical trial NCT02564614 (A Study of Hypoxia-inducible Factor 1a (HIF1A) Messenger Ribonucleic Acid (mRNA) Antagonist…

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Spebrutinib DB11764
small molecule | CAS: 1202757-89-8

Spebrutinib has been used in trials studying the treatment of Rheumatoid Arthritis, Lymphoma, Large B-Cell, Diffuse, and Leukemia Lymphocytic Chronic B-Cell.

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
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Spectinomycin Approved DB00919
small molecule | CAS: 1695-77-8

An antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +5
Target Protein:
30S ribosomal protein S12
Waktu Paruh1 to 3 hours in pat…
Vol. Distribusi-
Klirens-
Genetik -
Spermine DB00127
small molecule | CAS: 71-44-3

Spermine is a spermidine-derived biogenic polyamine found as a polycation at all pH values. Found in various tissues and organisms, it often acts as an essential growth factor in some bacterial species. Spermine is associated with nucleic acids, particularly …

Kategori:
AminesBiogenic AminesBiogenic Polyamines +4
Target Protein:
Spermine synthaseCarbonic anhydrase 4Glutamate receptor ionotropic, NMDA 1 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spesolimab Approved DB15626
biotech | CAS: 2097104-58-8

Spesolimab is an interleukin-36 (IL-36) receptor antagonist. It is a humanized monoclonal immunoglobulin G1 antibody that was produced in Chinese hamster ovary (CHO) cells by recombinant DNA technology. The biosimilar of the drug, spesolimab-sbzo, was first a…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-1 receptor-like 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiBased on the popula…
KlirensIn the linear dose …
Genetik -
SPG302 DB18103
small molecule | CAS: 2274723-90-7

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
SPG601 DB18742
small molecule

SPG601 is being investigated for the treatment of fragile X syndrome.

Waktu Paruh-
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SPH-3127 DB19108
small molecule | CAS: 1399849-02-5

SPH-3127 is under investigation in clinical trial NCT05359068 (Study to Evaluate the Efficacy and Safety of SPH3127 in Patients With Mild-moderate Essential Hypertension).

Kategori:
Oxazines
Waktu Paruh-
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Spheramine DB16979
biotech | CAS: 500604-72-8

Deskripsi belum tersedia.

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Sphingosine DB03203
small molecule | CAS: 123-78-4

An amino alcohol with a long unsaturated hydrocarbon chain. Sphingosine and its derivative sphinganine are the major bases of the sphingolipids in mammals. (Dorland, 28th ed)

Kategori:
AlcoholsAminesAmino Alcohols +2
Target Protein:
Choline-phosphate cytidylyltransferase BGenome polyproteinGenome polyprotein +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sphinxolide B DB04783
small molecule

Deskripsi belum tersedia.

Target Protein:
Actin, alpha skeletal muscle
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spiperone DB17056
small molecule | CAS: 749-02-0

Spiperone is a dopamine antagonist that binds dopamine and serotonin receptors.[A253142]

Kategori:
Antipsychotic AgentsButyrophenonesCentral Nervous System Agents +9
Target Protein:
Alpha-1A adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Spiradoline DB12704
small molecule | CAS: 87151-85-7

Spiradoline has been investigated for the basic science of Bipolar Depression.

Kategori:
AnalgesicsAntiarrhythmic agentsCardiovascular Agents +6
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Spiramycin Approved DB06145
small molecule | CAS: 24916-50-5

Spiramycin is a primarily bacteriostatic macrolide antimicrobial agent with activity against Gram-positive cocci and rods, Gram-negative cocci and also Legionellae, mycoplasmas, chlamydiae, some types of spirochetes, Toxoplasma gondii and Cryptosporidium. Sp…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +14
Target Protein:
50S ribosomal protein L3
Waktu ParuhIntravenous: Young…
Vol. DistribusiThe tissue distribu…
Klirens80% of the administ…
Genetik -
Spirapril Approved DB01348
small molecule | CAS: 83647-97-6

Spirapril is an ACE inhibitor antihypertensive drug used to treat hypertension. Spirapril is converted to the active spiraprilat after administration. ACE inhibitors are used primarily in treatment of hypertension and congestive heart failure.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +9
Target Protein:
Angiotensin-converting enzyme
Waktu Paruh30 to 35 hours
Vol. Distribusi-
Klirens-
Genetik -
Spironolactone Approved DB00421
small molecule | CAS: 52-01-7

Spironolactone is a potassium-sparing diuretic. It binds to mineralocorticoid receptors and functions as aldosterone antagonists.[A178192] It promotes sodium and water excretion and potassium retention.[A11837] Spironolactone was originally developed purely f…

Kategori:
Agents causing hyperkalemiaAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +19
Target Protein:
Mineralocorticoid receptorGlucocorticoid receptorAndrogen receptor +4
Waktu ParuhThe mean half-life …
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
SPK-1001 DB17973
biotech

Deskripsi belum tersedia.

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SPK-7001 DB18242
biotech

Deskripsi belum tersedia.

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SPL23-2 DB17866
biotech

SPL23-2 is an antisense oligonucleotide (ASO) targeting the W1282X nonsense mutation associated with a severe form of cystic fibrosis.[L46767]

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SPL84-23-1 DB18575
biotech

SPL84-23-1 is a sodium salt of 19-bp single-stranded RNA uniformly modified 2'-O-(2-methoxyethyl) phosphorothioate Antisense Oligonucleotide (ASO) consisting of 19 nucleotide residues with the sequence 5'-5MeC-5MeU-G-5MeC-A-A-5MeC-A-G-A-5MeU-G-G-A-A-G-A-5MeC-…

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Sporisorium cruentum Approved DB10873
biotech

Sporisorium cruentum is a fungus which can provoke allergic reactions. Sporisorium cruentum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Genetik -
SQ-109 DB05186
small molecule | CAS: 502487-67-4

SQ-109 is an orally active, small molecule antibiotic for treatment of pulmonary TB. Currently in Phase I clinical trials, SQ-109 could replace one or more drugs in the current first-line TB drug regimen, simplify therapy, and shorten the TB treatment regimen.

Kategori:
AminesBridged-Ring CompoundsCycloparaffins +2
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Squalamine DB06461
small molecule | CAS: 148717-90-2

Deskripsi belum tersedia.

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAnti-Bacterial Agents +11
Target Protein:
Vascular endothelial growth factor CVascular endothelial growth factor DFibroblast growth factor 2 +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 2892-62-8

Squaric acid dibutyl ester is under investigation in clinical trial NCT01971385 (Safety and Efficacy of Squaric Acid Dibutyl Ester for the Treatment of Herpes Labialis).

Kategori:
Adjuvants, ImmunologicAllergensAntigens +3
Waktu Paruh-
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Squash Approved DB10570
biotech

Squash allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Genetik -
Menampilkan 10201–10250 dari 11778
Sebelumnya Halaman 205 / 236 Berikutnya