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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 205 / 321
Metildigoxin DB13401
small molecule | CAS: 30685-43-9

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCarbohydratesCardanolides +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metipranolol Approved DB01214
small molecule | CAS: 22664-55-7

A beta-adrenergic antagonist effective for both beta-1 and beta-2 receptors. It is used as an antiarrhythmic, antihypertensive, and antiglaucoma agent.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metisazone DB13641
small molecule | CAS: 1910-68-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metixene Approved DB00340
small molecule | CAS: 4969-02-2

Metixene (or methixene) is a anticholinergic used as an antiparkinsonian agent.

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +6
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metizoline DB13614
small molecule | CAS: 17692-22-7

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoclopramide Approved DB01233
small molecule | CAS: 364-62-5

Diabetic gastroparesis is a condition that causes frequent nausea and vomiting, which has a negative impact on quality of life and poses a significant burden on the healthcare system.[A184934] Metoclopramide is a dopamine antagonist used to treat nausea and v…

Kategori:
Acids, CarbocyclicAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +35
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3AMuscarinic acetylcholine receptor M1 +1
Gen Terkait:
KCNH2 ADRA1D CYP2D6 +4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik 7 Varian
Metocurine Approved DB01336
small molecule | CAS: 5152-30-7

Dimethyltubocurarinium (INN) or metocurine (USAN), also known as dimethyltubocurarine, is a non-depolarizing muscle relaxant. Patients on chronic anticonvulsant drugs are relatively resistant to metocurine. [A2393]

Kategori:
Agents producing tachycardiaAlkaloidsAmines +18
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metocurine iodide Approved DB00416
small molecule | CAS: 7601-55-0

Metocurine iodide is a benzylisoquinolinium competitive nondepolarizing neuromuscular blocking agent. It is used as an anesthesia adjunct to induce skeletal muscle relaxation and to reduce the intensity of muscle contractions in convulsive therapy Metocurine …

Kategori:
AlkaloidsAminesAnticholinergic Agents +12
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit beta-2Neuronal acetylcholine receptor subunit alpha-2
Waktu Paruh3 to 4 hours
Vol. Distribusi-
Klirens-
Genetik -
Metolazone Approved DB00524
small molecule | CAS: 17560-51-9

A quinazoline-sulfonamide that is considered a thiazide-like diuretic which is long-acting so useful in chronic renal failure. It also tends to lower blood pressure and increase potassium loss.

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +21
Target Protein:
Solute carrier family 12 member 3
Waktu ParuhApproximately 14 ho…
Vol. Distribusi-
Klirens-
Genetik -
Metopimazine DB13591
small molecule | CAS: 14008-44-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntiemeticsAntiemetics and Antinauseants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoprine DB04655
small molecule | CAS: 7761-45-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsFolic Acid Antagonists +1
Target Protein:
Peptide deformylase, mitochondrialHistamine N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoprolol Approved DB00264
small molecule | CAS: 51384-51-1

Metoprolol is a selective beta-1 blocker commonly employed as the succinate and tartrate derivatives depending if the formulation is designed to be of immediate release or extended release.[A175159, L5530] The possibility of the generation of these formulatio…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta adrenergic receptor
Gen Terkait:
ADRB1 CYP2D6 ADRB1
Waktu ParuhThe immediate relea…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik 3 Varian
Metoserpate DB11530
small molecule | CAS: 1178-28-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIndole Alkaloids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metralindole DB09306
small molecule | CAS: 54188-38-4

Metralindole, also known as Inkazan, is similar in structure and pharmacology to pirlindole. It functions as a reversible inhibitor of monoamine oxidase A. In Russia, this drug was investigated for potential antidepressant activity.

Kategori:
Heterocyclic Compounds, Fused-RingIndole AlkaloidsIndoles +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metreleptin Approved DB09046
biotech | CAS: 186018-45-1

Metreleptin, a recombinant analog of the human hormone leptin, is an orphan drug used to treat complications of leptin deficiency in people with lipodystrophy. Lipodystrophies include a range of disorders characterized by the reduction, absence, or altered di…

Kategori:
AdipokinesAlimentary Tract and MetabolismAmino Acids and Derivatives +11
Target Protein:
Leptin receptor
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing intraveno…
KlirensThe clearance of me…
Genetik -
Metribolone DB02998
small molecule | CAS: 965-93-5

A synthetic non-aromatizable androgen and anabolic steroid. It binds strongly to the androgen receptor and has therefore also been used as an affinity label for this receptor in the prostate and in prostatic tumors.

Kategori:
EstranesEstrenesFused-Ring Compounds +1
Target Protein:
Progesterone receptorAndrogen receptorNuclear receptor coactivator 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrifonate DB11473
small molecule | CAS: 52-68-6

Metrifonate or trichlorfon is an irreversible organophosphate acetylcholinesterase inhibitor. It is a prodrug which is activated non-enzymatically into 2,2-dichlorovinyl dimethyl phosphate.

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizamide DB01578
small molecule | CAS: 31112-62-6

Metrizamide is a solute for density gradient centrifugation offering higher maximum solution density without the problems of increased viscosity. It is also used as a resorbable, non-ionic contrast medium.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizoic acid Approved DB09346
small molecule | CAS: 1949-45-7

Metrizoic acid is a molecule used as a contrast medium. It present a higher risk of allergic reactions due to its high osmolality. Its approval has been discontinued by the FDA. One study in 1976 demonstrated that metrizoic acid, when used for cardiac angiog…

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metronidazole Approved DB00916
small molecule | CAS: 443-48-1

Metronidazole is a commonly used antibiotic, belonging to the nitroimidazole class of antibiotics.[L3754] It is frequently used to treat gastrointestinal infections as well as trichomoniasis and giardiasis, and amebiasis which are parasitic infections.[A18103…

Kategori:
Agents that reduce seizure thresholdAlimentary Tract and MetabolismAnti-Bacterial Agents +38
Target Protein:
Oxygen-insensitive NADPH nitroreductaseAnaerobic bacterial DNAProtozoal DNA
Waktu ParuhThe elimination hal…
Vol. DistribusiMetronidazole is wi…
KlirensDose adjustments ma…
Genetik -
small molecule | CAS: 13182-89-3

Deskripsi belum tersedia.

Kategori:
ImidazolesNitro CompoundsNitroimidazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metyrapone Approved DB01011
small molecule | CAS: 54-36-4

An inhibitor of the enzyme steroid 11-beta-monooxygenase. It is used as a test of the feedback hypothalamic-pituitary mechanism in the diagnosis of cushing syndrome.

Kategori:
Cytochrome P-450 CYP2A6 InhibitorsCytochrome P-450 CYP2A6 Inhibitors (strength unknown)Cytochrome P-450 CYP2E1 Inhibitors +17
Target Protein:
Cytochrome P450 11B1, mitochondrialCamphor 5-monooxygenase
Waktu Paruh1.9 ±0.7 hou…
Vol. Distribusi-
Klirens-
Genetik -
Metyrosine Approved DB00765
small molecule | CAS: 672-87-7

An inhibitor of the enzyme tyrosine 3-monooxygenase, and consequently of the synthesis of catecholamines. It is used to control the symptoms of excessive sympathetic stimulation in patients with pheochromocytoma. (Martindale, The Extra Pharmacopoeia, 30th ed)

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +6
Target Protein:
Tyrosine 3-monooxygenase
Waktu Paruh3.4 to 3.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Mevalonic acid DB03518
small molecule | CAS: 150-97-0

Deskripsi belum tersedia.

Kategori:
Hydroxy Acids
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevastatin DB06693
small molecule | CAS: 73573-88-3

Mevastatin or compactin is a cholesterol-lowering agent isolated from <i>Penicillium citinium</i>. It was the first discovered agent belonging to the class of cholesterol-lowering medications known as statins. During a search for antibiotic compounds produced…

Kategori:
Agents Causing Muscle ToxicityAnti-Infective AgentsAnticholesteremic Agents +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevidalen DB19034
small molecule | CAS: 1638667-79-4

Mevidalen is under investigation in clinical trial NCT03305809 (A Study of LY3154207 in Participants With Dementia Due to Lewy Body Dementia (LBD) Associated With Idiopathic Parkinson's Disease (PD) or Dementia With Lewy Bodies (DLB)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75225-51-3

Deskripsi belum tersedia.

Kategori:
Naphthalenes
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevonlerbart DB19416
biotech | CAS: 2453195-99-6

Mevonlerbart is under investigation in clinical trial NCT06602726 (A Study to Demonstrate How Well REGN1908-1909 Works in Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Cat Allergy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mexazolam DB15489
small molecule | CAS: 31868-18-5

Mexazolam (CS-386) is a benzodiazepine indicated for the treatment of anxiety with or without psychoneurotic conditions.[A184910] Mexazolam's structure is similar to that of other benzodiazepines such as [oxazolam] and [cloxazolam].[A184910] The use of benzod…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +7
Target Protein:
GABA(A) Receptor Benzodiazepine Binding SiteGABA(A) Receptor
Waktu ParuhMexazolam follows a…
Vol. Distribusi-
Klirens-
Genetik -
Mexiletine Approved DB00379
small molecule | CAS: 31828-71-4

Antiarrhythmic agent pharmacologically similar to lidocaine. It may have some anticonvulsant properties.

Kategori:
AminesAntiarrhythmic agentsAntiarrhythmics, Class I +20
Target Protein:
Sodium channel protein type 5 subunit alphaAryl hydrocarbon receptor
Waktu Paruh10-12 hours
Vol. Distribusi* 5 to 7 L/lg
Klirens-
Genetik -
Mezagitamab DB16370
biotech | CAS: 2227490-52-8

Mezagitamab is under investigation in clinical trial NCT04278924 (Study to Evaluate Safety, Tolerability, and Efficacy of TAK-079 in Participants With Persistent/chronic Primary Immune Thrombocytopenia).

Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezigdomide DB17584
small molecule | CAS: 2259648-80-9

Mezigdomide is under investigation in clinical trial NCT05372354 (A Study to Evaluate Safety, Drug Levels and Effectiveness of CC-92480 (BMS-986348) in Combination With Other Treatments in Participants With Relapsed or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezlocillin Approved DB00948
small molecule | CAS: 51481-65-3

Semisynthetic ampicillin-derived acylureido penicillin. It has been proposed for infections with certain anaerobes and may be useful in inner ear, bile, and CNS infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1APeptidoglycan synthase FtsIPenicillin-binding protein 3 +1
Waktu Paruh1.3 to 4.4 hours
Vol. Distribusi-
Klirens-
Genetik -
MF101 DB05052
small molecule

MF101 is a novel estrogen receptor beta (ER?) selective agonist and unlike currently available hormone therapies, does not activate the estrogen receptor alpha (ER?), known to be implicated in tumor formation. MF101 is an oral drug designed for the treatment …

Target Protein:
Estrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MG-4101 DB18906
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MG-S-2525 DB18063
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MG98 DB06544
biotech

MG98, a second-generation antisense oligodeoxynucleotide inhibitor of human DNMT1, was investigated in the completed clinical trial NCT00003890 for treating patients with advanced solid tumors.

Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGB-BP-3 DB12892
small molecule | CAS: 1000277-08-6

Mgb Bp 3 is under investigation in clinical trial NCT02518607 (Safety, Blood Levels and Effects of MGB-BP-3).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGD-024 DB17265
biotech

MGD-024 is an anti-CD123/anti-CD3 bispecific DART molecule.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGN-4893 DB17338
biotech

MGN-4893 is an inhibitor of microRNA-451. In February 2011, it was granted FDA orphan designation for the treatment of polycythemia vera.[L47356]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mianserin Approved DB06148
small molecule | CAS: 24219-97-4

A tetracyclic compound with antidepressant effects. Mianserin was previously available internationally, however in most markets it has been phased out in favour of [mirtazapine].

Kategori:
Adrenergic AgentsAgents that produce hypertensionAntidepressive Agents +29
Target Protein:
Alpha-2A adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C +17
Waktu Paruh10-17 hours
Vol. Distribusi-
Klirens-
Genetik -
Mibampator DB12717
small molecule | CAS: 375345-95-2

Mibampator has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
AmidesBenzene DerivativesSulfones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibavademab DB16673
biotech | CAS: 2305770-44-7

Mibavademab is under investigation in clinical trial NCT04159415 (Study of REGN4461, a Leptin Receptor Agonist Antibody, in Patients With Generalized Lipodystrophy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibefradil DB01388
small molecule | CAS: 116644-53-2

Mibefradil was withdrawn from the market in 1998 because of potentially harmful interactions with other drugs.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +31
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1GVoltage-dependent T-type calcium channel subunit alpha-1HVoltage-dependent L-type calcium channel subunit alpha-1C +8
Waktu Paruh17 to 25 hours at s…
Vol. Distribusi-
Klirens-
Genetik -
Mibenratide DB15195
small molecule | CAS: 1239011-83-6

Mibenratide is under investigation in clinical trial NCT01798745 (A Study to Assess the Pharmacokinetics and Pharmacodynamics of JNJ-54452840 in Participants With Heart Failure and Anti-beta1-adrenergic Receptor Autoantibodies).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibolerone DB11429
small molecule | CAS: 3704-09-4

Mibolerone is a potent anabolic steroid which is both higher affinity and more selective for the androgen receptor than metribolone.

Kategori:
EstranesEstrenesFused-Ring Compounds +7
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Micafungin Approved DB01141
small molecule | CAS: 235114-32-6

Micafungin is an antifungal drug. It belongs to the antifungal class of compounds known as echinocandins and exerts its effect by inhibiting the synthesis of 1,3-beta-D-glucan, an integral component of the fungal cell wall.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +9
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu Paruh14-17 hours
Vol. Distribusi* 0.39 ± 0.11 L/kg …
Klirens* 0.359 +/- 0.179 m…
Genetik -
Miconazole Approved DB01110
small molecule | CAS: 22916-47-8

Miconazole is a broad-spectrum azole antifungal with some activity against Gram-positive bacteria as well.[A203636] It is widely used to treat mucosal yeast infections, including both oral and vaginal infections; although intravenous miconazole is no longer a…

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +41
Target Protein:
Lanosterol 14-alpha demethylaseNitric oxide synthase 3Nitric oxide synthase, inducible +5
Waktu ParuhMiconazole has a te…
Vol. DistribusiA 1200 mg miconazol…
Klirens-
Genetik -
Microcrystalline cellulose Approved DB14158
small molecule | CAS: 9004-34-6

A polysaccharide with glucose units linked as in CELLOBIOSE. It is the chief constituent of plant fibers, cotton being the purest natural form of the substance. As a raw material, it forms the basis for many derivatives used in chromatography, ion exchange ma…

Kategori:
BiopolymersCarbohydratesCellulose +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Micronomicin Approved DB13274
small molecule | CAS: 52093-21-7

Micronomicin is an aminoglycoside antibiotic which is marketed in Japan, and sold under the brand names Sagamicin and Luxomicina.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10201–10250 dari 16004
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