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12560

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9109 (72.5%)
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6912 (55.0%)
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12560 (100.0%)

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Halaman 204 / 252
RAPA-501-Allo DB15890
biotech

RAPA-501-ALLO is composed of T-cells extracted from healthy volunteers; these cells are then reprogrammed _ex vivo_ in a process that involves de-differentiation and re-differentiation.[L16483]

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Rapacuronium Approved DB04834
small molecule | CAS: 465499-11-0

Rapacuronium was withdrawn in 2001 in many countries due to risk of fatal bronchospasm.

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +9
Target Protein:
Muscarinic acetylcholine receptor M2
Waktu Paruh141 minutes (mean)
Vol. Distribusi-
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Raphanus sativus Approved DB10650
biotech

Radish allergenic extract is used in allergenic testing.

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Rasagiline Approved DB01367
small molecule | CAS: 136236-51-6

Rasagiline is an irreversible inhibitor of monoamine oxidase and is used as a monotherapy in early Parkinson's disease or as an adjunct therapy in more advanced cases.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Parkinson Drugs +19
Target Protein:
Amine oxidase [flavin-containing] BApoptosis regulator Bcl-2
Waktu ParuhRasagiline has a me…
Vol. Distribusi* 87 L
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Rasburicase Approved DB00049
biotech | CAS: 134774-45-1

Rasburicase is a recombinant urate-oxidase enzyme produced by a genetically modified <i>Saccharomyces cerevisiae</i> strain. The cDNA coding for rasburicase was cloned from a strain of _Aspergillus flavus_.

Kategori:
Antigout PreparationsDetoxifying Agents for Antineoplastic TreatmentEnzymes +7
Target Protein:
Uric acid
Waktu Paruh18 hours
Vol. Distribusi* 110 to 127 mL/kg …
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biotech | CAS: 1587257-96-2

Rasdegafusp alfa is under investigation in clinical trial NCT03206047 (Atezolizumab, Guadecitabine, and CDX-1401 Vaccine in Treating Patients With Recurrent Ovarian, Fallopian Tube, or Primary Peritoneal Cancer).

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Raubasine DB15949
small molecule | CAS: 483-04-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Beta-1 adrenergic receptor
Waktu Paruh-
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small molecule | CAS: 8063-17-0

Rauwolfia (Rauwolfia serpentina), also spelled _ravolphia_, is a medicinal plant in the milkweed family. The root of the plant is ground into a powder or sold in tablets or capsules. It is a compound commonly used in Asian medicine, which includes traditional…

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +6
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhAfter oral ingestio…
Vol. Distribusi-
KlirensHepatically and ren…
Genetik -
RAV12 DB05140
biotech

RAV12 is investigated for use/treatment in solid tumors. RAV12 is a solid. RAV12 is a chimeric antibody that recognizes RAAG12, an N-linked carbohydrate antigen found on gastric, colon, pancreatic, prostate, ovarian, breast, and kidney cancer cells.

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Ravagalimab DB16676
biotech | CAS: 2050816-56-1

Ravagalimab is under investigation in clinical trial NCT03695185 (A Study to Investigate How Well Ravagalimab (ABBV-323) Works and How Safe It Is in Participants With Moderate to Severe Ulcerative Colitis Who Failed Prior Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
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Ravidasvir DB15652
small molecule | CAS: 1242087-93-9

Ravidasvir is under investigation in clinical trial NCT02961426 (Sofosbuvir Plus Ravidasvir for the Treatment of HCV Chronic Infection).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +6
Target Protein:
Genome polyprotein
Waktu Paruh-
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Ravoxertinib DB15281
small molecule | CAS: 1453848-26-4

Ravoxertinib is under investigation in clinical trial NCT01875705 (A Dose-Escalation Study of GDC-0994 in Patients With Locally Advanced or Metastatic Solid Tumors).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors +1
Target Protein:
Mitogen-activated protein kinase 3Mitogen-activated protein kinase 1
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Ravulizumab Approved DB11580
biotech | CAS: 1803171-55-2

Ravulizumab is a potent and selective complement 5 (C5) inhibitor. It is a humanized monoclonal IgG2/4 kappa antibody produced in Chinese hamster ovary (CHO) cells.[L39690] Ravulizumab was engineered from [eculizumab], another complement inhibitor, to increas…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Complement C5
Waktu ParuhThe mean (%CV) term…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean (%CV) clea…
Genetik -
Raxibacumab Approved DB08902
biotech | CAS: 565451-13-0

Raxibacumab is a human IgG1? monoclonal antibody that binds the protective antigen (PA) component of B. anthracis toxin. Raxibacumab has a molecular weight of approximately 146 kilodaltons. Raxibacumab is produced by recombinant DNA technology in a murine cel…

Kategori:
Amino Acids, Peptides, and ProteinsAnthrax Protective Antigen-directed AntibodyAnthrax Protective Antigen-directed Antibody Interactions +12
Target Protein:
Protective antigen
Waktu ParuhMean terminal elimi…
Vol. DistribusiSteady state volume…
KlirensClearance values we…
Genetik -
Raxtozinameran Approved DB18228
biotech

Deskripsi belum tersedia.

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Razupenem DB12587
small molecule | CAS: 426253-04-5

Razupenem has been used in trials studying the treatment of Skin Infections.

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
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Razuprotafib DB16353
small molecule | CAS: 1008510-37-9

Razuprotafib, also known as AKB-9778, is a small-molecule inhibitor restoring Tie2 activation by inhibiting VE-PTP.[L27171,L27176] In investigations against diabetes and COVID-19, razuprotafib is self-administered by patients through subcutaneous injection.

Kategori:
AcidsAcids, NoncarboxylicAmines +2
Target Protein:
Receptor-type tyrosine-protein phosphatase betaAngiopoietin-1 receptor
Waktu Paruh-
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RBIO-101 DB18425
biotech

RBIO-101 is a recombinant adeno-associated virus vector encoding human CYP4V2 protein.

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RCT1100 DB18830
biotech

RCT1100 is an investigational mRNA-based therapeutic that aims to treat primary ciliary dyskinesia caused by pathogenic mutations in DNAI1.[L50788]

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RDEA806 DB05228
small molecule

RDEA806 is a new HIV non-nucleoside reverse transcriptase inhibitor (NNRTI) with a high genetic barrier to resistance and a broad spectrum of activity.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
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RDP58 DB06566
small molecule

RDP58 (NH2-arg-norleucine (nle)-nle-arg-nle-nle-nle-gly-tyr-CONH2) (Sangstat Corp., Fremont, California) is a novel synthetic peptide that inhibits early signal transduction pathways for the expression of inflammatory cytokines.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +3
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small molecule

Deskripsi belum tersedia.

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Rebamipide Approved DB11656
small molecule | CAS: 90098-04-7

Rebamipide has been investigated for the treatment of Stomach Ulcer, Keratoconjunctivitis Sicca, and Gastric Adenoma and Early Gastric Cancer.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Peptides, and Proteins +11
Target Protein:
fMet-Leu-Phe receptor
Waktu Paruh-
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Rebastinib DB13005
small molecule | CAS: 1020172-07-9

Rebastinib has been used in trials studying the treatment of Chronic Myeloid Leukemia. It is an inhibitor of Tie2 tyrosine kinase receptor and an antineoplastic agent.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Tyrosine-protein kinase ABL1Angiopoietin-1 receptor
Waktu Paruh-
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Rebaudioside A DB15136
small molecule | CAS: 58543-16-1

Rebaudioside A is under investigation in clinical trial NCT03510624 (Acute Effect of Rebaudioside A on Glucose Excursion During an Oral Glucose Tolerance Test in Type 2 Diabetes Mellitus).

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +2
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Rebimastat DB06573
small molecule | CAS: 259188-38-0

Deskripsi belum tersedia.

Kategori:
Matrix Metalloproteinases
Waktu Paruh-
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biotech | CAS: 1966978-67-5

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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REC-994 DB15616
small molecule

REC-994 was cleared by the FDA in July, 2018 for a phase I trial for the treatment of cerebral cavernous malformation (CCM).

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Recanaclotide DB15417
biotech | CAS: 1667762-62-0

Recanaclotide is under investigation in clinical trial NCT01712412 (Phase 2a Study of IW-9179 to Treat Functional Dyspepsia).

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Recaticimab DB19302
biotech | CAS: 2361290-85-7

Recaticimab is under investigation in clinical trial NCT06467617 (Adebrelimab Plus Chemo and Recaticimab Perioperative Treatment for Resectable NSCLC).

Waktu Paruh-
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biotech

Receptor binding domain SARS-CoV-2 Hepatitis B surface antigen virus-like particle vaccine (RBD SARS-CoV-2 HBsAg VLP vaccine), is a virus-like particle vaccine candidate where the RBD antigen is conjugated to the hepatitis B surface antigen[A226593]. Virus-li…

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Recoflavone DB12058
small molecule | CAS: 203191-10-0

Recoflavone has been used in trials studying the treatment of Acute Gastritis, Dry Eye Syndrome, and Chronic Gastritis.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Nuclear factor NF-kappa-B p105 subunitTranscription factor RelBNuclear factor NF-kappa-B p100 subunit +2
Waktu Paruh-
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Genetik -
biotech

Alpha 1-antitrypsin is a glycoprotein primarily produced by hepatocytes, and to a lesser extent, immune system cells. Recombinant alpha 1-antitrypsin (rAAT) is produced from yeast, which unlike commercially available forms of plasma-derived AAT, eliminates th…

Target Protein:
Alpha-1-antitrypsin
Waktu Paruh-
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biotech | CAS: 122320-05-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsPeptides +4
Waktu Paruh-
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biotech

B38-CAP is structured as a carboxypeptidase and derived from _Paenibacillus sp._ The molecule, an Angiotensin Converting Enzyme 2 (ACE2)-like enzyme, shares structural similarities to the mammalian ACE2. B38-CAP is an ACE2-like enzyme which decreases angioten…

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biotech

Recombinant CD40-ligand is under investigation in clinical trial NCT00053391 (Vaccine Therapy in Treating Patients With Stage III or Stage IV Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +8
Waktu Paruh-
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biotech | CAS: 389069-73-2

Recombinant human kallikrein-1 is under investigation in clinical trial NCT01845064 (A Study to Evaluate the Safety and Effectiveness of DM199 in Healthy Subjects and Type 2 Diabetes Patients).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +9
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biotech

Deskripsi belum tersedia.

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biotech

Plasma gelsolin (pGSN) is a protein found in the blood of healthy individuals which scavenges compounds left over from damaged tissues.

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersCalcium-Binding Proteins +9
Waktu Paruh-
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biotech

Recombinant human thrombopoietin is a full-length glycosylated cytokine produced by Chinese hamster ovary cells and is used to promote the generation of megakaryocytes and platelets.[A225691, A225696] This drug is used in the treatment of thrombocytopenia.

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biotech

Deskripsi belum tersedia.

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biotech

The Recombinant SARS-CoV-2 Vaccine was created by inserting genes of the SARS-CoV-2 spike protein’s receptor-binding domain into a baculovirus expression system[F4738, A226853]. In pre-clinical trial testing on mice, rabbits, and non-human primates, the candi…

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biotech

Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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biotech

Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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biotech

Recombinant super-compound interferon (rSIFN-co) is a recombinant version of interferon alpha with modified spatial configuration. This interferon has antiviral and antitumor activity.

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Red king crab Approved DB10526
biotech

Crab allergenic extract is used in allergenic testing.

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Red pepper Approved DB14759
biotech

Red pepper allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Redaporfin DB17219
small molecule | CAS: 1224104-08-8

Deskripsi belum tersedia.

Kategori:
AmidesBiological FactorsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
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Redasemtide DB19121
biotech | CAS: 1606186-88-2

Redasemtide is under investigation in clinical trial NCT05953480 (A Phase 2b, Randomized, Double-blind Study of Redasemtide (S-005151) in Adult Participants With Acute Ischemic Stroke).

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Refametinib DB06309
small molecule | CAS: 923032-37-5

Deskripsi belum tersedia.

Kategori:
AmidesAminesAniline Compounds +2
Waktu Paruh-
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