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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 202 / 252
Quemliclustat DB19160
small molecule | CAS: 2105904-82-1

Quemliclustat is under investigation in clinical trial NCT05329766 (A Safety and Efficacy Study of Treatment Combinations With and Without Chemotherapy in Adult Participants With Advanced Upper Gastrointestinal Tract Malignancies).

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalImmune Checkpoint Inhibitors
Target Protein:
5'-nucleotidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quercetin DB04216
small molecule | CAS: 117-39-5

Quercetin is a flavonol widely distributed in plants. It is an antioxidant, like many other phenolic heterocyclic compounds. Glycosylated forms include RUTIN and quercetrin.

Kategori:
AntioxidantsBCRP/ABCG2 InhibitorsBenzopyrans +26
Target Protein:
Signal transducer and activator of transcription 3Lysophosphatidylcholine acyltransferase 2Lysophosphatidylcholine acyltransferase 1 +29
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quercus dumosa pollen Approved DB10952
biotech

Quercus dumosa pollen is the pollen of the Quercus dumosa plant. Quercus dumosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quercus virginiana pollen Approved DB10375
biotech

Quercus virginiana pollen is the pollen of the Quercus virginiana plant. Quercus virginiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quetiapine Approved DB01224
small molecule | CAS: 111974-69-7

Initially approved by the FDA in 1997, quetiapine is a second-generation atypical antipsychotic used in schizophrenia, major depression, and bipolar disorder.[L8546] Quetiapine demonstrates a high level of therapeutic efficacy and low risk of adverse effects …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +44
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +21
Waktu ParuhThe average termina…
Vol. DistribusiQuetiapine distribu…
KlirensThe clearance of qu…
Genetik -
Queuine DB14732
small molecule | CAS: 72496-59-4

Queuine is a derivative of [7-Deazaguanine]. Bacteria possess the exclusive ability to synthesize queuine, which is then salvaged and passed on to plants and animals. Quantities of queuine have been found in tomatoes, wheat, coconut water, and milk from human…

Kategori:
Heterocyclic Compounds, Fused-RingPurinesPurinones
Waktu ParuhData regarding the …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Quilizumab DB15176
biotech | CAS: 1228538-47-3

Quilizumab is under investigation in clinical trial NCT01160861 (A Study to Investigate the Safety, Tolerability, and Pharmacokinetics of MEMP1972A in Patients With Allergic Rhinitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quilseconazole DB17758
small molecule | CAS: 1340593-70-5

Deskripsi belum tersedia.

Target Protein:
Lanosterol 14-alpha demethylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinagolide Approved DB09097
small molecule | CAS: 87056-78-8

Quinagolide is a non-ergot-derived selective dopamine D2 receptor agonist used for the treatment of elevated levels of prolactin or hyperprolactinaemia. Hyperprolalctinaemia is associated with gonadal dysfunction, including infertility and reduced libido, as …

Kategori:
Dopamine AgentsDopamine AgonistsDopamine D2 Receptor Agonists +6
Target Protein:
D(2) dopamine receptorD(1) dopamine receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiApproximate volume …
Klirens-
Genetik -
Quinalizarin DB08660
small molecule | CAS: 81-61-8

Deskripsi belum tersedia.

Kategori:
AnthracenesQuinones
Target Protein:
Casein kinase II subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinapril Approved DB00881
small molecule | CAS: 85441-61-8

Quinapril is the ethyl ester prodrug of the non-sulfhydryl angiotensin converting enzyme inhibitor quinaprilat.[L8420,L8423] It is used to treat hypertension and heart failure.[L8420,L8423] ACE inhibitors are commonly used as a first line therapy in the treat…

Kategori:
ACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin SystemAgents causing angioedema +12
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhThe active metaboli…
Vol. DistribusiThe mean volume of …
KlirensThe clearance of qu…
Genetik -
Quinaprilat DB14217
small molecule | CAS: 82768-85-2

The active metabolite of the prodrug [quinapril].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinestrol Approved DB04575
small molecule | CAS: 152-43-2

The 3-cyclopentyl ether of ethinyl estradiol.

Kategori:
Estradiol CongenersEstrogenic Steroids, AlkylatedEstrogens +11
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinethazone Approved DB01325
small molecule | CAS: 73-49-4

Quinethazone, marketed as Hydromox, is a thiazide diuretic indicated for hypertension. Patients may experience adverse reactions such as dizziness, dry mouth, nausea, and hypokalemia.

Kategori:
AmidesCardiovascular AgentsDiuretics +10
Target Protein:
Solute carrier family 12 member 1Solute carrier family 12 member 2Solute carrier family 12 member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinfamide DB12780
small molecule | CAS: 62265-68-3

Quinfamide has been used in trials studying the treatment of Amoebiasis and Helminthiasis.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quingestanol DB13685
small molecule | CAS: 10592-65-1

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinidine Approved DB00908
small molecule | CAS: 56-54-2

Quinidine is a D-isomer of [quinine] present in the bark of the Cinchona tree and similar plant species. This alkaloid was first described in 1848 and has a long history as an antiarrhythmic medication.[A38016,A250050] Quinidine is considered the first antiar…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +81
Target Protein:
Sodium channel protein type 5 subunit alphaPotassium channel subfamily K member 1Potassium channel subfamily K member 6 +4
Waktu ParuhThe elimination hal…
Vol. DistribusiQuinidine has a vol…
KlirensThe clearance of qu…
Genetik -
Quinine Approved DB00468
small molecule | CAS: 130-95-0

An alkaloid derived from the bark of the cinchona tree. It is used as an antimalarial drug, and is the active ingredient in extracts of the cinchona that have been used for that purpose since before 1633. Quinine is also a mild antipyretic and analgesic and h…

Kategori:
Agents that produce neuromuscular block (indirect)Agents that reduce seizure thresholdAlkaloids +57
Target Protein:
Fe(II)-protoporphyrin IXPlatelet glycoprotein IXIntermediate conductance calcium-activated potassium channel protein 4
Waktu ParuhApproximately 18 ho…
Vol. Distribusi* 1.43 ± 0.18 L/kg …
Klirens* 0.17 L/h/kg [heal…
Genetik -
Quinoline DB18050
small molecule | CAS: 91-22-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 79647-29-3

Deskripsi belum tersedia.

Target Protein:
Phenylalanine-4-hydroxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinupramine Approved DB13246
small molecule | CAS: 31721-17-2

Quinupramine has been approved in France under the brand name Kinupril, as an antidepressant [A175003].

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinupristin Approved DB01369
small molecule | CAS: 120138-50-3

Quinupristin/dalfopristin is a combination of two antibiotics used to treat infections by staphylococci and by vancomycin-resistant Enterococcus faecium. Dalfopristin inhibits the early phase of protein synthesis in the bacterial ribosome and quinupristin inh…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
23S ribosomal RNA50S ribosomal protein L1050S ribosomal protein L22
Waktu Paruh3.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Quisinostat DB12985
small molecule | CAS: 875320-29-9

Quisinostat has been used in trials studying the treatment of Lymphoma, Neoplasms, Myelodysplastic Syndromes, and Advanced or Refractory Leukemia.

Kategori:
AminesHydroxy AcidsHydroxylamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quisovalimab DB16482
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quisqualic acid DB02999
small molecule | CAS: 52809-07-1

Quisqualic acid is an agonist at two subsets of excitatory amino acid receptors, ionotropic receptors that directly control membrane channels and metabotropic receptors that indirectly mediate calcium mobilization from intracellular stores. The compound is ob…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsExcitatory Amino Acid Agents +4
Target Protein:
Metabotropic glutamate receptor 1Glutamate receptor ionotropic, kainate 1Metabotropic glutamate receptor 2 +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quizartinib Approved DB12874
small molecule | CAS: 950769-58-1

Quizartinib is an oral and potent fms-like tyrosine kinase 3 (FLT3) inhibitor and it is the first drug developed specifically targeting FLT3, as other agents with FLT3 inhibition activities were investigated with other targets in mind.[A260641] Additionally, …

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean (SD) effec…
Vol. DistribusiVolume of distribut…
KlirensTotal body clearanc…
Genetik -
QXL138AM DB18552
biotech

QXL138AM is a masked immunocytokine (MIC) comprised of an anti-CD138 immunoglobulin G1 antibody fused to interferon alpha 2a. It binds the CD138 protein on the surface of the tumour cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 37571-78-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-1487 DB06518
small molecule | CAS: 449811-92-1

Deskripsi belum tersedia.

Kategori:
Mitogen-Activated Protein Kinase 14, antagonists & inhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-306465 DB12382
small molecule | CAS: 604769-01-9

R306465 has been used in trials studying the treatment of Neoplasms.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-348 DB06321
small molecule | CAS: 916742-11-5

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein kinase JAK3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-82913 DB08598
small molecule | CAS: 126347-69-1

Deskripsi belum tersedia.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +7
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-851 DB05747
small molecule

R-851 is part of the family of immune response modifier (IRM) and it acts in a novel way to stimulate the human body's immnune system to attack virus-infected cells and tumor cells. It is expected to be topical treatment for cervical displasia and cervical hi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14047-28-0

Deskripsi belum tersedia.

Target Protein:
Thymidine kinase, cytosolicThymidine kinaseThymidine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-95845 DB07327
small molecule | CAS: 163435-77-6

R-95845 is an inhibitor of HIV-1 reverse transcriptase.

Kategori:
AcetatesAcids, AcyclicAmides +1
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R-azabisabolene DB03985
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R048-8071 DB02016
small molecule | CAS: 161582-11-2

Deskripsi belum tersedia.

Target Protein:
Lanosterol synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R107474 DB06553
small molecule | CAS: 214548-46-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R112 DB06252
small molecule | CAS: 575474-82-7

R112 is an investigational compound developed to treat Allergic Rhinitis. It's mechanism of action is to inhibit SYK kinase.

Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R1204 DB05118
small molecule

R1204 is G-protein-coupled receptor modulator. It is developed for the treatment of depression.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R1295 DB05122
small molecule

R1295 is an integrin antagonist currently in clinical trials for the treatment of rheumatoid arthritis. Integrins are associated to the pathology seen in some of the autoimmune diseases such as rheumatoid arthritis.

Target Protein:
Integrin alpha-4Integrin beta-4Integrin beta-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R1626 DB05060
small molecule

R1626 is one of a new class of hepatitis C therapies called polymerase inhibitors. It achieves significant reductions in viral load in chronic hepatitis C patients infected with the difficult to treat genotype 1 virus. R1626 is very effective in inhibiting vi…

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides
Target Protein:
RNA-dependent RNA-polymerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R343 DB06316
small molecule | CAS: 575484-78-5

R343, was investigated in clinical trial NCT01591044 to evaluate its safety and efficacy in patients with mild to moderate asthma.

Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R411 DB05468
small molecule

R411 is a non-steroid oral medicine for the treatment of asthma. It is not immunosuppressive, but blocks the activation and recruitment of cells involved in respiratory inflammation. It is a dual-acting competitive integrin antagonist (as compared to previous…

Target Protein:
Integrin alpha-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R450 DB05469
small molecule

R450 is an alpha 1 antagonist that acts to tighten the muscle tone in the bladder. It is being considered for treatment of stress-related urinary incontinence. Phase IIa data for the drug show it reduced the number of incontinent episodes compared to placebo …

Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R673 DB05466
small molecule

R673 is a novel NK1 antagonist that penetrates the blood-brain barrier, has excellent safety and tolerability and shows low P450-based drug interaction potential. The phase II program for treatment of depression and anxiety is ongoing in the US and EU.It is n…

Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
R906289 DB19126
small molecule | CAS: 2602614-45-7

R906289 is under investigation in clinical trial NCT05308264 (Study of R289 in Participants With Lower-risk Myelodysplastic Syndromes (LR MDS)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
rAAV9-hNAGLU DB18415
biotech

rAAV9-hNAGLU consists of a recombinant AAV9 expressing human alpha-N-acetylglucosaminidase.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Rabacfosadine DB12762
small molecule | CAS: 859209-74-8

Rabacfosadine has been used in trials studying the treatment of Multiple Myeloma, Non-Hodgkin's Lymphoma, and Chronic Lymphocytic Leukemia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rabbit Approved DB10415
biotech

Rabbit allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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