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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 202 / 321
Metahexamide DB13675
small molecule | CAS: 565-33-3

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAmidesBlood Glucose Lowering Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metamfetamine Approved DB01577
small molecule | CAS: 537-46-2

Metamfetamine (methamphetamine) is a psychostimulant and sympathomimetic drug, and a member of the amphetamine group of sympathomimetic amines. Methamphetamine can induce effects such as euphoria, increased alertness and energy, and enhanced self-esteem. It i…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +33
Target Protein:
D(2) dopamine receptorAlpha-1B adrenergic receptorSodium-dependent dopamine transporter +10
Gen Terkait:
PICK1
Waktu ParuhThe biological half…
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Metamizole Approved DB04817
small molecule | CAS: 50567-35-6

Metamizole (dipyrone) is a pyrazolone derivative that belongs to the group of nonacid nonopioids. It is considered a potent analgesic and antipyretic with favourable gastrointestinal tolerability.[A251885] Metamizole was formerly marketed in the US as Dimetho…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAminopyrine +16
Target Protein:
Prostaglandin G/H synthase 1
Waktu Paruh_In vitro_, the hal…
Vol. DistribusiMetamizole is quick…
KlirensThe clearance of 4-…
Genetik -
Metampicillin DB13836
small molecule | CAS: 6489-97-0

Metampicillin is a penicillin antibiotic prepared by the reaction of ampicillin with formaldehyde. It is hydrolysed in aqueous solution to form ampicillin. Hydrolysis is rapid under acid conditions like the stomach.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metandienone DB13586
small molecule | CAS: 72-63-9

Metandienone is an orally active anabolic androgenic steroid. It was introduced to the market in the 1960s but later discontinued and withdrawn from the market. Although it is prohibited in and outside competition by the World Anti-Doping Agency, metandienone…

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Heat-labile enterotoxin B chainCholera enterotoxin subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metaraminol Approved DB00610
small molecule | CAS: 54-49-9

An adrenergic agonist that acts predominantly at alpha adrenergic receptors and also stimulates the release of norepinephrine. It has been used primarily as a vasoconstrictor in the treatment of hypotension.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +17
Target Protein:
D(2) dopamine receptorAlpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metavert DB17306
small molecule | CAS: 1841125-91-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metaxalone Approved DB00660
small molecule | CAS: 1665-48-1

Metaxalone is a moderate to strong muscle relaxant used in the symptomatic treatment of musculoskeletal pain caused by strains, sprains, and other musculoskeletal conditions. It is marketed by King Pharmaceuticals under the brand name Skelaxin®. Its main mech…

Kategori:
Central Nervous System DepressantsCentrally-mediated Muscle RelaxationDrugs that are Mainly Renally Excreted +5
Waktu Paruh9.2 (+/- 4.8) hours
Vol. Distribusi* 800 L
Klirens* 68 +/- 50 L/h [Su…
Genetik -
Metelimumab DB18695
biotech | CAS: 272780-74-2

Metelimumab (CAT-192) is a monoclonal antibody targeted against transforming growth factor (TGF) beta-1.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metenkefalin DB12668
small molecule | CAS: 58569-55-4

Metenkefalin is an endogenous opioid and beta-endorphin.[A203225] It has been shown to reduce chromosomal abberations in patients with multiple sclerosis.[A203210] Metenkefalin, along with [tridecactide], are under investigation as an immunomodulatory therap…

Kategori:
Amino Acids, Peptides, and ProteinsEnkephalin, MethionineEnkephalins +9
Target Protein:
Delta-type opioid receptorMu-type opioid receptor
Waktu ParuhThe half life of me…
Vol. Distribusi-
Klirens-
Genetik -
Metenolone DB13710
small molecule | CAS: 153-00-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metergoline Approved DB13520
small molecule | CAS: 17692-51-2

Metergoline is an ergot-derived psychoactive drug that acts as a ligand for serotonin and dopamine receptors. Metergoline is an antagonist at various 5-HT receptor subtypes at a relatively low concentration and agonist at dopamine receptors.[A27181] Its use h…

Kategori:
Agents that produce hypertensionAlkaloidsAntidepressive Agents +18
Target Protein:
5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1E +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metformin Approved DB00331
small molecule | CAS: 657-24-9

Metformin is a biguanide antihyperglycemic agent and first-line pharmacotherapy used in the management of type II diabetes.[L12207,A176173] Metformin is considered an antihyperglycemic drug because it lowers blood glucose concentrations in type II diabete…

Kategori:
Alimentary Tract and MetabolismAmidinesBiguanides +11
Target Protein:
Multidrug and toxin extrusion protein 1Acetyl-CoA carboxylase 2Electron transfer flavoprotein-ubiquinone oxidoreductase, mitochondrial +2
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensRenal clearance is …
Genetik -
Metformin C-11 DB15181
small molecule

Metformin c-11 is under investigation in clinical trial NCT03122769 (Cardiac Uptake of Metformin, Visualized by Positron Emission Tomography).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 72156-70-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methacholine Approved DB06709
small molecule | CAS: 55-92-5

Asthma is a complex condition associated with phenomena such as airway hyperresponsiveness (AHR), in which the smooth muscle in the airways (ASM) excessively contracts in response to stimuli, reducing pulmonary function and causing symptoms such as difficulty…

Kategori:
AminesAmmonium CompoundsAutonomic Agents +17
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6008-91-9

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Isobutyryl-CoA dehydrogenase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methadone Approved DB00333
small molecule | CAS: 76-99-3

Methadone is a potent synthetic analgesic that works as a full µ-opioid receptor (MOR) agonist and N-methyl-d-aspartate (NMDA) receptor antagonist. As a full MOR agonist, methadone mimics the natural effects of the body's opioids, endorphins, and enkephalins …

Kategori:
AnalgesicsAnticholinergic AgentsAntidepressive Agents +50
Target Protein:
Mu-type opioid receptorNMDA receptorDelta-type opioid receptor +5
Waktu ParuhDue to interindivid…
Vol. DistribusiDue to interindivid…
KlirensDue to interindivid…
Genetik -
small molecule | CAS: 509-74-0

A narcotic analgesic with a long onset and duration of action. It is used mainly in the treatment of narcotic dependence.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methallenestril DB13143
small molecule | CAS: 517-18-0

Deskripsi belum tersedia.

Kategori:
EstrogensGenito Urinary System and Sex HormonesSex Hormones and Modulators of the Genital System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methamidophos DB14972
small molecule | CAS: 10265-92-6

Methamidophos is under investigation in clinical trial NCT03223753 (Web-Based Physical Activity Intervention in Improving Long Term Health in Children and Adolescents With Newly Diagnosed Acute Lymphoblastic Leukemia in First Remission).

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsecticides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methane DB15994
small molecule | CAS: 74-82-8

Deskripsi belum tersedia.

Kategori:
AlkanesHydrocarbons, Acyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 558-25-8

Methanesulfonyl Fluoride has been used in trials studying the treatment of Safety.

Kategori:
Cholinergic AgentsCholinesterase InhibitorsEnzyme Inhibitors +2
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methantheline Approved DB00940
small molecule | CAS: 5818-17-7

Methantheline is a synthetic antispasmodic. Antispasmodics are used to relieve cramps or spasms of the stomach, intestines, and bladder. Methantheline is used to treat intestine or stomach ulcers (peptic ulcer disease), intestine problems (irritable bowel syn…

Kategori:
Acid ReducersAgents producing tachycardiaAlimentary Tract and Metabolism +12
Target Protein:
Histamine H2 receptorMuscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M2 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methapyrilene DB04819
small molecule | CAS: 91-80-5

Methapyrilene, formerly marketed in many drug products, was shown to be a potent carcinogen. Manufacturers voluntarily withdrew methapyriline drug products from the market in May and June 1979.

Kategori:
AminesAminopyridinesAnti-Allergic Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methaqualone DB04833
small molecule | CAS: 72-44-6

Methaqualone is a sedative-hypnotic drug that is similar in effect to barbiturates, a general central nervous system depressant. The sedative-hypnotic activity was first noted by Indian researchers in the 1950s and in 1962 methaqualone itself was patented in …

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP3A Substrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metharbital DB00463
small molecule | CAS: 50-11-3

Metharbital is a barbiturate anticonvulsant, similar to phenobarbital, marketed as Gemonil by Abbott Laboratories. It was patented in 1905 by Emil Fischer of Merck.

Kategori:
Anticholinergic AgentsAnticonvulsantsBarbiturates and Derivatives +5
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-3 +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methazolamide Approved DB00703
small molecule | CAS: 554-57-4

A carbonic anhydrase inhibitor that is used as a diuretic and in the treatment of glaucoma.

Kategori:
Antiglaucoma Preparations and MioticsCarbonic Anhydrase InhibitorsCardiovascular Agents +15
Target Protein:
Carbonic anhydrase 1Carbonic anhydrase 4Carbonic anhydrase 2 +2
Waktu Paruh14 hours
Vol. Distribusi* 17 to 23 L
Klirens-
Genetik -
Methcathinone DB15339
small molecule | CAS: 5650-44-2

Methcathinone is under investigation in clinical trial NCT02617862 (PCI Imaging System in Pediatric Ophthalmology).

Kategori:
Ketones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methdilazine Approved DB00902
small molecule | CAS: 1982-37-2

Methdilazine is a phenothiazine compound with antihistaminic activity. It is used in the treatment of various dermatoses to relieve pruritus.

Kategori:
Agents that reduce seizure thresholdAntihistamines for Systemic UseHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methenamine Approved DB06799
small molecule | CAS: 100-97-0

Methenamine is a heterocyclic organic compound with a cage-like structure similar to adamantane. In salt form it is used for the treatment of urinary tract infection (Example: methenamine hippurate which is the hippuric acid salt of methenamine).

Kategori:
Acids, CarbocyclicAmidesAmines +14
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens70-90% of a single…
Genetik -
Methfuroxam DB16231
small molecule | CAS: 28730-17-8

Methfuroxam is under investigation in clinical trial NCT01213407 (Dendritic Cell Cancer Vaccine for High-grade Glioma).

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactam-inducible penicillin-binding protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 26403-67-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methimazole Approved DB00763
small molecule | CAS: 60-56-0

Methimazole is a thionamide antithyroid agent that inhibits the synthesis of thyroid hormones.[A184559,A184733,A184694] It was first introduced as an antithyroid agent in 1949[A184502] and is now commonly used in the management of hyperthyroidism, particularl…

Kategori:
Antithyroid agentsCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +30
Target Protein:
Thyroid peroxidase
Waktu ParuhFollowing a single …
Vol. DistribusiThe apparent volume…
KlirensFollowing a single …
Genetik -
Methiodal DB13321
small molecule | CAS: 143-47-5

Deskripsi belum tersedia.

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methionine Approved DB00134
small molecule | CAS: 63-68-3

A sulfur containing essential amino acid that is important in many body functions. It is a chelating agent for heavy metals.

Kategori:
Amino AcidsAmino Acids, EssentialAmino Acids, Neutral +7
Target Protein:
Methionine synthase reductaseMethionine synthaseMethionine aminopeptidase 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methionine C-11 DB17147
small molecule | CAS: 60305-58-0

Deskripsi belum tersedia.

Kategori:
Diagnostic RadiopharmaceuticalsTumour Detection
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 15985-39-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 21752-32-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methocarbamol Approved DB00423
small molecule | CAS: 532-03-6

Methocarbamol was developed in the early 1950s as a treatment for muscle spasticity and the associated pain.[A178441,A178450] It is a guaiacol glyceryl ether.[A178450] Methocarbamol tablets and intramuscular injections are prescription medicines indicated …

Kategori:
Acids, AcyclicBenzene DerivativesCarbamates +14
Target Protein:
Carbonic anhydrase 1
Waktu ParuhThe elimination hal…
Vol. DistribusiVolume of distribut…
Klirens0.2-0.8L/h/kg.[L626…
Genetik -
Methohexital Approved DB00474
small molecule | CAS: 151-83-7

An intravenous anesthetic with a short duration of action that may be used for induction of anesthesia.

Kategori:
AnestheticsAnesthetics, GeneralAnesthetics, Intravenous +10
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh5.6 ± 2.7 mi…
Vol. Distribusi-
Klirens-
Genetik -
Methopterin DB16620
small molecule | CAS: 2410-93-7

Methopterin is thought to have effects on osteoclasts and to inhibit inflammatory bone destruction.[A229843]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methoserpidine DB13631
small molecule | CAS: 865-04-3

Deskripsi belum tersedia.

Kategori:
Antiadrenergic Agents, Centrally ActingAntihypertensive AgentsSecologanin Tryptamine Alkaloids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methotrexate Approved DB00563
small molecule | CAS: 59-05-2

Methotrexate is a folate derivative that inhibits several enzymes responsible for nucleotide synthesis.[A180322] This inhibition leads to suppression of inflammation as well as prevention of cell division.[A180322] Because of these effects, methotrexate is of…

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAgents Causing Muscle Toxicity +42
Target Protein:
Thymidylate synthaseReduced folate transporterProton-coupled folate transporter +2
Gen Terkait:
ABCC2 MTHFR
Waktu ParuhThe half life of lo…
Vol. DistribusiThe volume of distr…
KlirensMethotrexate cleara…
Genetik 2 Varian
Methotrimeprazine Approved DB01403
small molecule | CAS: 60-99-1

A phenothiazine with pharmacological activity similar to that of both chlorpromazine and promethazine. It has the histamine-antagonist properties of the antihistamines together with central nervous system effects resembling those of chlorpromazine. (From Mart…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +46
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor +16
Waktu ParuhApproximately 20 ho…
Vol. Distribusi-
Klirens-
Genetik -
Methoxamine Approved DB00723
small molecule | CAS: 390-28-3

An alpha-adrenergic agonist that causes prolonged peripheral vasoconstriction. It has little if any direct effect on the central nervous system.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +19
Target Protein:
Alpha-1A adrenergic receptorAlpha-1D adrenergic receptorAlpha-1B adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methoxsalen Approved DB00553
small molecule | CAS: 298-81-7

A naturally occurring furocoumarin compound found in several species of plants, including Psoralea corylifolia. It is a photoactive substance that forms DNA adducts in the presence of ultraviolet A irradiation.

Kategori:
AntipsoriaticsAntipsoriatics for Systemic UseAntipsoriatics for Topical Use +24
Target Protein:
DNACytochrome P450 2A6
Waktu ParuhApproximately 2 hou…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 180509-15-3

Methoxy arachidonyl fluorophosphonate, commonly referred as MAFP, is an irreversible active site-directed enzyme inhibitor that inhibits nearly all serine hydrolases and serine proteases. It inhibits phospholipase A2 and fatty acid amide hydrolase with specia…

Kategori:
EicosanoidsEnzyme InhibitorsFatty Acids +5
Target Protein:
Fatty-acid amide hydrolase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 10051–10100 dari 16004
Sebelumnya Halaman 202 / 321 Berikutnya