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72

Total database: 17430
Struktur (SMILES)
71 (98.6%)
Target
56 (77.8%)
Genomik
1 (1.4%)
Referensi
72 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (72)

Halaman 2 / 2
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase pim-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
RAC-beta serine/threonine-protein kinaseGlycogen synthase kinase-3 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase B-raf
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nedometinib DB18102
small molecule | CAS: 2252314-46-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olanzapine Approved DB00334
small molecule | CAS: 132539-06-1

Olanzapine is a thienobenzodiazepine classified as an atypical or second-generation antipsychotic agent.[A176996] The second-generation antipsychotics were introduced in the 90s and quickly gained traction due to their impressive efficacy, reduced risk for ex…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +50
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorD(1A) dopamine receptor +17
Gen Terkait:
HTR1A
Waktu ParuhOlanzapine presents…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik 1 Varian
Osugacestat DB12006
small molecule | CAS: 1401066-79-2

Osugacestat (BMS-906024) has been used in trials studying the treatment of Cancer, Lymphoblastic Leukemia, Acute T-cell, and Precursor T-Cell Lymphoblastic Lymphoma.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Phenaglycodol DB19373
small molecule | CAS: 79-93-6

Deskripsi belum tersedia.

Kategori:
AlcoholsGlycols
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirenzepine Approved DB00670
small molecule | CAS: 28797-61-7

An antimuscarinic agent that inhibits gastric secretion at lower doses than are required to affect gastrointestinal motility, salivary, central nervous system, cardiovascular, ocular, and urinary function. It promotes the healing of duodenal ulcers and due to…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Ulcer Agents +10
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirmitegravir DB18974
small molecule | CAS: 2245231-10-9

Pirmitegravir is under investigation in clinical trial NCT05869643 (A Clinical Trial of STP0404 in Treatment-naïve Adults With HIV-1 Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PLX-4720 DB06999
small molecule | CAS: 918505-84-7

Deskripsi belum tersedia.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Vascular endothelial growth factor receptor 2Serine/threonine-protein kinase B-raf
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Quinoline DB18050
small molecule | CAS: 91-22-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sonrotoclax DB18753
small molecule | CAS: 2383086-06-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Urokinase-type plasminogen activatorSerine protease 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tofisopam DB08811
small molecule | CAS: 22345-47-7

Tofisopam (marketed under brand names Emandaxin and Grandaxin) is a 2,3-benzodiazepine drug which is a benzodiazepine derivative. In contrast to classical 1,4-benzodiazepines, the compound does not bind to the benzodiazepine binding site of the gamma-aminobut…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsBenzazepines +12
Target Protein:
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A3',5'-cyclic-AMP phosphodiesterase 4AcGMP-dependent 3',5'-cyclic phosphodiesterase +1
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
VAD-044 DB17697
small molecule

VAD-044 is an allosteric AKT inhibitor developed by Vaderis Therapeutics AG. It is being investigated for the treatment of Hereditary Hemorrhagic Telangiectasia.[L46098]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Venetoclax Approved DB11581
small molecule | CAS: 1257044-40-8

Venetoclax is a BCL-2 inhibitor that was initially approved by the FDA in April 2016 [FDA label]. Proteins in the B cell CLL/lymphoma 2 (BCL-2) family are important regulators of the apoptotic (programmed cell death) process [A18565], [A18566]. Venetoclax is…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Apoptosis regulator Bcl-2
Waktu ParuhThe half-life of ve…
Vol. DistribusiThe population esti…
KlirensMainly hepatic [FDA…
Genetik -
Zilucoplan Approved DB15636
small molecule | CAS: 1841136-73-9

Zilucoplan is a 15 amino-acid, synthetic macrocyclic peptide. It is a complement inhibitor that works to prevent the activation of C5, which is a complement protein involved in the innate immune system to initiate inflammatory responses.[A261841] On October 1…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBlood Proteins +5
Target Protein:
Complement C5
Waktu ParuhThe mean plasma ter…
Vol. DistribusiThe mean volume of …
KlirensNo information is a…
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase Sgk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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