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63

Total database: 17430
Struktur (SMILES)
62 (98.4%)
Target
52 (82.5%)
Genomik
0 (0%)
Referensi
63 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (63)

Halaman 2 / 2
small molecule

Deskripsi belum tersedia.

Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nemtabrutinib DB18866
small molecule | CAS: 2095393-15-8

Nemtabrutinib is under investigation in clinical trial NCT05624554 (A Study of Nemtabrutinib vs Chemoimmunotherapy for Participants With Previously Untreated Chronic Lymphocytic Leukemia/small Lymphocytic Lymphoma (CLL/SLL) Without TP53 Aberrations (MK-1026-0…

Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Repotrectinib Approved DB16826
small molecule | CAS: 1802220-02-5

Repotrectinib is a next-generation tyrosine kinase inhibitor (TKI) specifically designed to address resistance in the treatment of non-small cell lung cancer (NSCLC), specifically due to mutations in the ROS1 gene.[A262056] ROS1 mutations are one of the defin…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +28
Target Protein:
Proto-oncogene tyrosine-protein kinase ROSHigh affinity nerve growth factor receptorBDNF/NT-3 growth factors receptor +1
Waktu ParuhThe repotrectinib m…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Ropsacitinib DB18709
small molecule | CAS: 2127109-84-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selpercatinib Approved DB15685
small molecule | CAS: 2152628-33-4

Selpercatinib is a kinase inhibitor with enhanced specificity for RET tyrosine kinase receptors (RTKs) over other RTK classes.[A202055, A202052, L13604] Enhanced RET (Rearranged during transfection) oncogene expression is a hallmark of many cancers. Although …

Kategori:
Agents that produce hypertensionAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +19
Target Protein:
Proto-oncogene tyrosine-protein kinase receptor RetVascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 3 +3
Waktu ParuhSelpercatinib has a…
Vol. DistribusiSelpercatinib has a…
KlirensSelpercatinib has a…
Genetik -
small molecule | CAS: 667931-25-1

Deskripsi belum tersedia.

Kategori:
Receptors, Calcium-Sensing, antagonists & inhibitors
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tildacerfont DB18545
small molecule | CAS: 1014983-00-6

Tildacerfont is a corticotropin-releasing factor receptor-1 antagonist containing an unfused thiazole ring

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tomivosertib DB15219
small molecule | CAS: 1849590-01-7

Tomivosertib is under investigation in clinical trial NCT03318562 (A PD Study of Oral eFT508 in Subjects With Advanced TNBC and HCC).

Target Protein:
MAP kinase-interacting serine/threonine-protein kinase 1MAP kinase-interacting serine/threonine-protein kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tovinontrine DB16193
small molecule | CAS: 2062661-53-2

Tovinontrine is an orally administered, highly selective phosphodiesterase 9 (PDE9) small molecule inhibitor. Tovinontrine is under investigation in clinical trial NCT04474314 (A Study of IMR-687 in Subjects With Sickle Cell Disease).

Target Protein:
High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tuvusertib DB18790
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vactosertib DB15310
small molecule | CAS: 1352608-82-2

Vactosertib is under investigation in clinical trial NCT03724851 (Vactosertib in Combination With Pembrolizumab in Metastatic Colorectal or Gastric Cancer).

Kategori:
AminesEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
TGF-beta receptor type-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zaleplon Approved DB00962
small molecule | CAS: 151319-34-5

Zaleplon is a sedative/hypnotic, mainly used for insomnia. It is known as a nonbenzodiazepine hypnotic. Zaleplon interacts with the GABA receptor complex and shares some of the pharmacological properties of the benzodiazepines. Zaleplon is a schedule IV drug …

Kategori:
AcetatesAcids, AcyclicAmides +22
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
Waktu ParuhApproximately 1 hour
Vol. Distribusi* 1.4 L/kg
Klirens* 1 L/h/kg
Genetik -
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