Hasil Filter

17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (17430)

Halaman 199 / 349
small molecule | CAS: 998-06-1

Deskripsi belum tersedia.

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +3
Target Protein:
Phosphatidylcholine transfer protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Eflornithine DB03856
small molecule | CAS: 66640-93-5

Deskripsi belum tersedia.

Target Protein:
Ornithine decarboxylase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 6779-87-9

7,8-Dihydrobiopterin is an inhibitor of the enzyme dihydroneopterin aldolase (DHNA), which catalyzes the conversion of 7,8-Dihydrobiopterin to 6-hydroxymethyl-7,8-dihydropterin and glycolaldehyde.

Kategori:
CoenzymesEnzymes and CoenzymesHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Nitric oxide synthase, inducibleTyrosine 3-monooxygenasePhenylalanine-4-hydroxylase +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
L-Gluconic Acid DB04304
small molecule | CAS: 526-97-6

Deskripsi belum tersedia.

Target Protein:
Beta-glucosidase A
Waktu Paruh-
Vol. Distribusi-
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Genetik -
L-Glutamine Approved DB00130
small molecule | CAS: 56-85-9

A non-essential amino acid present abundantly throughout the body and is involved in many metabolic processes. It is synthesized from glutamic acid and ammonia. It is the principal carrier of nitrogen in the body and is an important energy source for many cel…

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids and Derivatives +8
Target Protein:
CTP synthase 1AmidophosphoribosyltransferaseGlutamine synthetase
Waktu ParuhThe half life of el…
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesMonosaccharides
Target Protein:
Ferrichrome-iron receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
3-keto-L-gulonate-6-phosphate decarboxylase UlaD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Hut operon positive regulatory protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 25679-93-0

Deskripsi belum tersedia.

Target Protein:
Histidinol-phosphate aminotransferaseHistidinol-phosphate aminotransferase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
L-homoarginine DB03974
small molecule | CAS: 156-86-5

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +2
Target Protein:
Nitric oxide synthase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Homoserine DB04193
small molecule | CAS: 672-15-1

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
L-Lactic acid Approved DB14475
small molecule | CAS: 79-33-4

Deskripsi belum tersedia.

Kategori:
Hydroxy AcidsLactates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Thermolysin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 120484-65-3

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
small molecule | CAS: 29586-66-1

L-lysyl-l-arginine is under investigation in clinical trial NCT03972488 (Study to Evaluate the Efficacy and Safety of Lutathera in Patients With Grade 2 and Grade 3 Advanced GEP-NET).

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Genetik -
small molecule | CAS: 62697-73-8

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Target Protein:
Thymidylate synthaseAmyloid-beta precursor proteinCatalase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Thymidylate synthasePossible cellulase CelA1 (Endoglucanase) (Endo-1,4-beta-glucanase) (FI-cmcase) (Carboxymethyl cellulase)Ras-related protein Rab-5A +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 7314-32-1

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins +2
Target Protein:
Catalase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Inositol monophosphatase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase 3Nitric oxide synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Nitric oxide synthase 3Nitric oxide synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Subtilisin Carlsberg
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 80875-98-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 6152-89-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiomarkers
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 3182-95-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Pyruvate kinase PKM
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 471-87-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +1
Target Protein:
Glycine betaine-binding periplasmic protein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
L-Rhamnitol DB02399
small molecule | CAS: 488-28-8

Deskripsi belum tersedia.

Target Protein:
L-rhamnose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Saccharopine DB04207
small molecule | CAS: 997-68-2

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +1
Target Protein:
Alpha-aminoadipic semialdehyde synthase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 626-69-7

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, NeutralAmino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
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Genetik -
L-tartaric acid DB09459
small molecule | CAS: 87-69-4

Tartaric acid is a white crystalline organic acid that occurs naturally in many plants, most notably in grapes.Tartaric is an alpha-hydroxy-carboxylic acid, is diprotic and aldaric in acid characteristics, and is a dihydroxyl derivative of succinic acid.

Kategori:
Acids, AcyclicCarbohydratesChelating Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-thioproline DB02846
small molecule | CAS: 2756-91-4

Deskripsi belum tersedia.

Target Protein:
Annexin A5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-threonic acid DB11192
small molecule | CAS: 7306-96-9

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Threoninol DB01724
small molecule | CAS: 3228-51-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
3-keto-L-gulonate-6-phosphate decarboxylase UlaD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-tyrosinamide DB03380
small molecule | CAS: 4985-46-0

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Pro-neuropeptide YValacyclovir hydrolase
Waktu Paruh-
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Genetik -
L-valinol DB04383
small molecule | CAS: 2026-48-4

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 64913-51-5

Deskripsi belum tersedia.

Kategori:
CarbohydratesSugar Phosphates
Target Protein:
3-keto-L-gulonate-6-phosphate decarboxylase UlaD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
L-Xylopyranose DB03911
small molecule

Deskripsi belum tersedia.

Target Protein:
Xylose isomerase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 60802-29-1

Deskripsi belum tersedia.

Target Protein:
3-keto-L-gulonate-6-phosphate decarboxylase UlaD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxypeptidase A1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
L523S DB06498
biotech

According to Nemunaitis J., et al, "L523S is an immunogenic lung cancer antigen that has demonstrated preclinical safety when the gene is injected intramuscularly as an expressive plasmid (pVAX/L523S) and when delivered following incorporation into an E1B-del…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Labetalol Approved DB00598
small molecule | CAS: 36894-69-6

Labetalol is a racemic mixture of 2 diastereoisomers where dilevalol, the R,R' stereoisomer, makes up 25% of the mixture.[L7730] Labetalol is formulated as an injection or tablets to treat hypertension.[L7727,L7730] Labetalol was granted FDA approval on 1 …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +35
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorAlpha-1 adrenergic receptors
Waktu ParuhLabetalol has a hal…
Vol. DistribusiIn normotensive pat…
KlirensLabetalol has a pla…
Genetik -
Labetuzumab DB05097
biotech | CAS: 219649-07-7

Labetuzumab is a humanized monoclonal antibody to carcinoembryonic antigen that inhibits tumor growth. It is used in radioimmunotherapy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Cell adhesion molecule CEACAM5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1469876-18-3

Labetuzumab govitecan has been used in trials studying the treatment of Colon Cancer, Rectal Cancer, and Metastatic Colorectal Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Labradimil DB06549
small molecule | CAS: 159768-75-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAutacoidsBiological Factors +8
Target Protein:
B2 bradykinin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lacidipine Approved DB09236
small molecule | CAS: 103890-78-4

Lacidipine is a lipophilic dihydropyridine calcium antagonist with an intrinsically slow onset of activity. Due to its long duration of action, lacidipine does not lead to reflex tachycardia [A31536]. It displays specificity in the vascular smooth muscle, whe…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +16
Target Protein:
Voltage-dependent L-type calcium channel
Waktu ParuhThe average termina…
Vol. Distribusi-
Klirens-
Genetik -
Lacnotuzumab DB14928
biotech | CAS: 1831128-32-5

Lacnotuzumab is under investigation in clinical trial NCT01643850 (MCS110 in Patients With Pigmented Villonodular Synovitis (PVNS)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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