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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 199 / 236
Savolitinib DB12048
small molecule | CAS: 1313725-88-0

Savolitinib has been used in trials studying the treatment and health services research of Tumor, Food Effect, Gastric Cancer, Health Subjects, and Colorectal Cancer, among others.

Kategori:
Tyrosine Kinase Inhibitors
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saxagliptin Approved DB06335
small molecule | CAS: 361442-04-8

Saxagliptin (rINN) is an orally active hypoglycemic (anti-diabetic drug) of the new dipeptidyl peptidase-4 (DPP-4) inhibitor class of drugs. FDA approved on July 31, 2009.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismAmino Acids, Peptides, and Proteins +20
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhSaxagliptin = 2.5 h…
Vol. Distribusi151 L
KlirensRenal clearance, si…
Genetik -
SB 11285 DB17511
small molecule

SB 11285 is a second-generation Stimulator of Interferon Genes (STING) agonist.[L45123] SB 11285 is under investigation in clinical trial NCT04096638 (Evaluating Safety and Efficacy of SB 11285 Alone and in Combination With Atezolizumab in Patients With Advan…

Waktu Paruh-
Vol. Distribusi-
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SB 224289 DB17052
small molecule | CAS: 180083-23-2

SB-224289 is a small molecule with a high affinity for human 5-HT1B receptors.[A253122]

Kategori:
Piperidines
Target Protein:
5-hydroxytryptamine receptor 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-1578 DB15294
small molecule | CAS: 937273-04-6

SB-1578 is under investigation in clinical trial NCT01235871 (A Single and Multiple-Dose Study of SB1578).

Kategori:
fms-Like Tyrosine Kinase 3, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingJanus Kinase 2, antagonists & inhibitors +1
Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-218078 DB17051
small molecule | CAS: 135897-06-2

SB-218078 is a specific inhibitor of CHK1.[A253117]

Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-269970 DB13988
small molecule | CAS: 201038-74-6

SB-269970 is an experimental drug developed by GlaxoSmithKline. In the studies performed with this agent, it has been suggested that SB-269970 acts either as a selective antagonist or inverse agonist of the serotonin receptor 7 (5-HT7).[A31816,A31817]

Kategori:
AmidesBenzene DerivativesSulfones +1
Target Protein:
5-hydroxytryptamine receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-409513 DB01793
small molecule

Deskripsi belum tersedia.

Target Protein:
Glycogen synthase kinase-3 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-509 DB05579
small molecule

SB-509 is under investigation in multiple clinical trials for the treatment of Diabetic Neuropathy.

Waktu Paruh-
Vol. Distribusi-
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SB-705498 DB11883
small molecule | CAS: 501951-42-4

SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.

Kategori:
AmidesTRPV Cation Channels, antagonists & inhibitors
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-743921 DB05546
small molecule | CAS: 618430-39-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SB-773812 DB16042
small molecule | CAS: 630407-66-8

SB-773812 is under investigation in clinical trial NCT00259870 (SB-773812 Administered in Adults With Schizophrenia).

Waktu Paruh-
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SB719125 DB16753
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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SBT-100 DB17215
biotech

SBT-100 is an anti-signal transducer and activator of transcription 3 (STAT3) B VHH13 single-domain antibody (sdAb). It was granted orphan drug designation by the FDA for the treatment of pancreatic cancer and osteosarcoma.[L44131,L44136]

Waktu Paruh-
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SBT-272 DB18037
small molecule | CAS: 2356106-71-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
SC 41930 DB17101
small molecule | CAS: 120072-59-5

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +9
Target Protein:
Leukotriene B4 receptor 1Leukotriene B4 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SC-236 DB14059
small molecule | CAS: 170569-86-5

SC-236 is a potent, selective, orally active inhibitor of cyclooxygenase-2 (COX-2) [L2964] that has been studied in cancer therapy [A33375], lower back pain [A33376], and inflammation [A33373], [A33374],[L2962], [A33377].

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +14
Target Protein:
Cyclooxygenase 2Prostaglandin G/H synthase 2Nuclear factor NF-kappa-B complex
Waktu ParuhLong plasma half-li…
Vol. Distribusi-
Klirens-
Genetik -
SC-74020 DB01630
small molecule

Deskripsi belum tersedia.

Kategori:
AmidesAminesHydroxy Acids +3
Target Protein:
72 kDa type IV collagenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SC12267 DB05125
small molecule

SC12267 is a novel, small molecule agent from the class of DMARDs (disease modifying anti-rheumatic drug) for the therapy of autoimmune diseases such as rheumatoid arthritis or multiple sclerosis. Through highly selective inhibition of pyrimidine biosynthesis…

Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SC45647 DB04778
small molecule

Deskripsi belum tersedia.

Kategori:
AmidinesSweetening Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
scAAV9.U7.ACCA DB18582
biotech

scAAV9.U7.ACCA is a non-replicating recombinant adeno-associated virus vector containing 4 antisense sequences designed to target exon 2 in the human DMD gene under the control of U7 small nuclear non-coding RNA. Developed by Nationwide Children’s Hospital, i…

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Vol. Distribusi-
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SCH-486757 DB12782
small molecule | CAS: 524019-25-8

Sch 486757 has been used in trials studying the treatment of Cough.

Kategori:
Aza Compounds
Waktu Paruh-
Vol. Distribusi-
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Genetik -
SCH-58500 DB17416
biotech

SCH-58500 is a recombinant replication-deficient adenovirus vector carrying the human p53 gene.

Waktu Paruh-
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SCH-900271 DB12433
small molecule | CAS: 915210-50-3

Sch 900271 has been used in trials studying the treatment of Mixed Hyperlipidemia and Primary Hypercholesterolemia.

Target Protein:
Hydroxycarboxylic acid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Scopolamine Approved DB00747
small molecule | CAS: 51-34-3

Scopolamine is a tropane alkaloid isolated from members of the _Solanaceae_ family of plants, similar to [atropine] and [hyoscyamine], all of which structurally mimic the natural neurotransmitter [acetylcholine].[A228423, A228763] Scopolamine was first synthe…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents producing tachycardia +30
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +5
Waktu ParuhThe half-life of sc…
Vol. DistribusiThe volume of distr…
KlirensIV infusion of 0.5 …
Genetik -
biotech

Centruroides (scorpion) Immune F(ab')2 (equine) is a purified preparation of immune globulin F(ab’)2 fragments that are derived from plasma of the horses immunized with venom of *C. noxius*, *C. l. limpidus*, *C. l. tecomanus*, and *C. s. suffusus*. It is int…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Waktu Paruh159 ± 57 h [FDA lab…
Vol. DistribusiSteady state: 13.6 …
Klirens83.5 ± 38.4 ml/Hr […
Genetik -
Scriptaid DB17053
small molecule | CAS: 287383-59-9

Scriptaid is a histone deacetylase (HDAC) inhibitor researched for its anti-tumor properties.[A253127]

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
Histone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SCY-635 DB12451
small molecule | CAS: 210759-10-7

SCY-635 has been investigated for the treatment of Chronic Hepatitis C and Hepatitis C Infection.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic
Target Protein:
Guided entry of tail-anchored proteins factor CAMLG
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
scyllo-inositol DB03106
small molecule | CAS: 488-59-5

An isomer of glucose that has traditionally been considered to be a B vitamin although it has an uncertain status as a vitamin and a deficiency syndrome has not been identified in man. (From Martindale, The Extra Pharmacopoeia, 30th ed, p1379) Inositol phosph…

Kategori:
AlcoholsCarbohydratesStereoisomerism +1
Target Protein:
Lysosomal acid glucosylceramidase1-phosphatidylinositol phosphodiesteraseCDP-diacylglycerol--inositol 3-phosphatidyltransferase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD-0006 DB07943
small molecule | CAS: 271576-80-8

Deskripsi belum tersedia.

Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD118 DB05207
small molecule

SD118 was previously under investigation in Japan for a different indication and now, following re-profiling and evaluation in experimental animal models, has demonstrated its potential as a new oral therapy for neuropathic pain.

Target Protein:
Tumor necrosis factorInterleukin-1 receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SD146 DB02729
small molecule | CAS: 183854-21-9

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SEA-CD70 DB17555
biotech

SEA-CD70 is an investigational humanized, non-fucosylated monoclonal antibody targeting CD70. SEA-CD70 is under investigation in clinical trial NCT04227847 (A Safety Study of SEA-CD70 in Patients With Myeloid Malignancies).

Waktu Paruh-
Vol. Distribusi-
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Sebacic acid DB07645
small molecule | CAS: 111-20-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsLipids
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sebelipase alfa Approved DB11563
biotech | CAS: 1276027-63-4

The lysosomal acid lipase (LAL) enzyme is found in lysosomes and is primarily responsible for the metabolism of lipids, and its absence or deficiency results in the accumulation of lipids in various organs. This lipid accumulation can lead to end-organ damage…

Kategori:
Alimentary Tract and MetabolismCarboxylic Ester HydrolasesCholesterol Ester Storage Disease, drug therapy +7
Waktu ParuhThe mean half-life …
Vol. DistribusiIn patients 4-11 ye…
KlirensAcross all age grou…
Genetik -
Secalciferol DB18406
small molecule | CAS: 55721-11-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secale cereale pollen Approved DB10717
biotech

Secale cereale pollen is the pollen of the Secale cereale plant. Secale cereale pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seclidemstat DB17117
small molecule | CAS: 1423715-37-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysine-specific histone demethylase 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secnidazole Approved DB12834
small molecule | CAS: 3366-95-8

Secnidazole is a second-generation 5-nitroimidazole antimicrobial agent. It is structurally related to other 5-nitroimidazoles, including [DB00916] and [DB00911], but displays improved oral absorption and a longer terminal elimination half-life than other dru…

Kategori:
Anti-Infective AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +18
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensThe total body clea…
Genetik -
Secobarbital Approved DB00418
small molecule | CAS: 76-73-3

Secobarbital (marketed by Eli Lilly and Company under the brand names Seconal and Tuinal) is a barbiturate derivative drug with anaesthetic, anticonvulsant, sedative and hypnotic properties. It is commonly known as quinalbarbitone in the United Kingdom.

Kategori:
AdjuvantsAdjuvants, AnesthesiaAnticholinergic Agents +27
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-4 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 29388-59-8

Secoisolariciresinol has been used in trials studying the prevention of Breast Cancer.

Kategori:
AlcoholsBenzene DerivativesBenzyl Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secretin human Approved DB09532
biotech | CAS: 108153-74-8

Human secretin is a gastrointestinal peptide hormone that regulates secretions in the stomach, pancreas, and liver. The hormone is produced from the enterochromaffin cells in the duodenum in response to the duodenal content with the pH less than 4.5 [L1875]. …

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGastrointestinal Agents +11
Target Protein:
Secretin receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of sy…
Genetik -
Secretin porcine Approved DB09527
biotech | CAS: 17034-35-4

Secretin porcine stimulates pancreatic and gastric secretions to aid in the diagnosis of pancreatic exocrine dysfunction and the diagnosis of gastrinoma.

Kategori:
Gastrointestinal AgentsSecretin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Secukinumab Approved DB09029
biotech | CAS: 1229022-83-6

Secukinumab is a fully human monoclonal IgG1/? antibody against interleukin-17A (IL-17A), a proinflammatory cytokine implicated in various chronic immune-mediated inflammatory disorders, such as plaque psoriasis.[L39600] By blocking the actions of IL-17A, sec…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAntibodies +14
Target Protein:
Interleukin-17A
Waktu ParuhThe half-life range…
Vol. DistribusiThe mean volume of …
KlirensThe mean systemic c…
Genetik -
Segesterone DB14584
small molecule | CAS: 7690-08-6

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesProgestins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Segesterone acetate Approved DB14583
small molecule | CAS: 7759-35-5

Segesterone acetate is a steroidal progestin or synthetic progesterone and a 19-norprogesterone derivative with no CH3 group radical in position 6 [A37048]. In animal studies, segesterone acetate was shown to be one of the most potent progestins [A37090]. It …

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +24
Target Protein:
Progesterone receptorAndrogen receptorGlucocorticoid receptor
Waktu ParuhThe mean (SD) half …
Vol. DistribusiThe volume of distr…
KlirensNo pharmacokinetic …
Genetik -
small molecule | CAS: 1609522-33-9

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 19Cyclin-dependent kinase 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Seladelpar Approved DB12390
small molecule | CAS: 851528-79-5

Seladelpar is a peroxisome proliferator-activated receptor (PPAR)-delta (?) agonist. Seladelpar is a single enantiomer of the R-configuration.[L51149] On August 14, 2024, seladelpar was granted accelerated approval by the FDA for the treatment of primary bili…

Kategori:
Acids, AcyclicAntimetabolitesBCRP/ABCG2 Substrates +13
Target Protein:
Peroxisome proliferator-activated receptor delta
Waktu ParuhFollowing administr…
Vol. DistribusiSeladelpar steady s…
KlirensThe apparent oral c…
Genetik -
Selamectin DB11459
small molecule | CAS: 220119-17-5

Selamectin is a topical parasiticide and antihelminthic used on dogs and cats to treat and prevent infections of heartworms, fleas, ear mites, sarcoptic mange, and certain types of ticks in dogs as well as prevent heartworms, fleas, ear mites, hookworms, and …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Selatogrel DB15163
small molecule | CAS: 1159500-34-1

Selatogrel is under investigation in clinical trial NCT03814200 (A Study to Investigate the Effect of Rifampicin on the Uptake and Breakdown of ACT-246475 in Healthy Subjects).

Kategori:
Organophosphorus Compounds
Target Protein:
P2Y purinoceptor 12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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