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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 199 / 252
Proguanil Approved DB01131
small molecule | CAS: 500-92-5

Proguanil is a prophylactic antimalarial drug, which works by stopping the malaria parasite, _Plasmodium falciparum_ and _Plasmodium vivax_, from reproducing once it is in the red blood cells. It does this by inhibiting the enzyme, dihydrofolate reductase, wh…

Kategori:
AmidinesAnti-Infective AgentsAntimalarials +15
Target Protein:
Dihydrofolate reductasePeptide deformylase, mitochondrialBifunctional dihydrofolate reductase-thymidylate synthase
Gen Terkait:
CYP2C19 CYP2C19
Waktu ParuhApproximately 20 ho…
Vol. Distribusi-
Klirens-
Genetik 2 Varian
biotech | CAS: 67422-14-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolease-r-hFSH DB05826
biotech

Prolease-r-hFSH is a recombinant human follicle stimulating hormone (r-hFSH) with Alkermes' ProLease injectable sustained release drug delivery technology. It provides patients with long term therapeutic benefit from a single administration rather than multip…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolectin-M DB16521
small molecule

Prolectin-M is a (1-6)-alpha-D-mannopyranose[L31338] and acts as an antagonist of galectin.[L31343] It is being investigated in the clinical trial NCT04512027 (Prolectin-M in COVID-19 Patients Having Mild to Moderate Symptoms Not Requiring Oxygen Support. (Pr…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolgolimab DB16740
biotech | CAS: 2093956-19-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates +2
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proline DB00172
small molecule | CAS: 147-85-3

Proline is one of the twenty amino acids used in living organisms as the building blocks of proteins. Proline is sometimes called an imino acid, although the IUPAC definition of an imine requires a carbon-nitrogen double bond. Proline is a non-essential amino…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +4
Target Protein:
Peptidyl-prolyl cis-trans isomerase BPeptidyl-prolyl cis-trans isomerase APyrroline-5-carboxylate reductase 1, mitochondrial +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolintane DB13438
small molecule | CAS: 493-92-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System AgentsCentral Nervous System StimulantsNervous System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promazine Approved DB00420
small molecule | CAS: 58-40-2

A phenothiazine with actions similar to chlorpromazine but with less antipsychotic activity. It is primarily used in short-term treatment of disturbed behavior and as an antiemetic. It is currently not approved for use in the United States.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +49
Target Protein:
D(2) dopamine receptorMuscarinic acetylcholine receptor M55-hydroxytryptamine receptor 2A +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promegestone DB13602
small molecule | CAS: 34184-77-5

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promethazine Approved DB01069
small molecule | CAS: 60-87-7

Promethazine, originally known as 3,277 R.P., is an N-dimethylaminopropyl derivative of [phenothiazine] that was developed in France in 1946.[A189901] Promethazine antagonizes a variety of receptors, allowing it to be used for a number of indications includin…

Kategori:
Acid ReducersAgents producing tachycardiaAgents that reduce seizure threshold +44
Target Protein:
Histamine H1 receptorD(2) dopamine receptorMuscarinic acetylcholine receptor M1 +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe intravenous cle…
Genetik -
Propacetamol DB09288
small molecule | CAS: 66532-85-2

Propacetamol is a non-opioid analgesic devoid of the major contraindications.[A32051] It is a derivative of [acetaminophen], or paracetamol, with the molecular formula glycine, N, N-diethyl-,4-(acetylamino)phenyl ester. Propacetamol is a parenteral formulatio…

Kategori:
Acetaminophen and ProdrugsAcetanilidesAgents causing hyperkalemia +37
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Transient receptor potential cation channel subfamily V member 1 +1
Waktu ParuhThe half-life of pr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Propafenone Approved DB01182
small molecule | CAS: 54063-53-5

An antiarrhythmia agent that is particularly effective in ventricular arrhythmias. It also has weak beta-blocking activity. The drug is generally well tolerated.

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +25
Target Protein:
Sodium channel protein type 5 subunit alphaVoltage-gated inwardly rectifying potassium channel KCNH2Beta-1 adrenergic receptor +1
Waktu Paruh2-10 hours
Vol. Distribusi* 252 L
Klirens-
Genetik -
Propagermanium DB17608
small molecule | CAS: 12758-40-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntineoplastic AgentsElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propamidine DB13296
small molecule | CAS: 104-32-5

Deskripsi belum tersedia.

Kategori:
AmidinesAnti-Infective AgentsAntiparasitic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propantheline Approved DB00782
small molecule | CAS: 298-50-0

A muscarinic antagonist used as an antispasmodic, in rhinitis, in urinary incontinence, and in the treatment of ulcers. At high doses it has nicotinic effects resulting in neuromuscular blocking.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +13
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proparacaine Approved DB00807
small molecule | CAS: 499-67-2

Proparacaine is a topical anesthetic drug of the amino ester group. It is found in ophthalmic solutions at a concentration of 0.5% as the hydrochloride salt.

Kategori:
Acids, CarbocyclicAminobenzoatesAnesthetics +18
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2921-92-8

Deskripsi belum tersedia.

Kategori:
AlcoholsAntianginal AgentsCardiac Therapy +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propentofylline DB06479
small molecule | CAS: 55242-55-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnti-Ulcer AgentsCentral Nervous System Agents +12
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propicillin DB13660
small molecule | CAS: 551-27-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propidium DB02166
small molecule | CAS: 36015-30-2

Quaternary ammonium analog of ethidium; an intercalating dye with a specific affinity to certain forms of DNA and, used as diiodide, to separate them in density gradients; also forms fluorescent complexes with cholinesterase which it inhibits. [PubChem]

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household settingHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiolactone Approved DB09348
small molecule | CAS: 57-57-8

Propiolactone is a lactone compound with a four-membered ring. It is a colorless liquid with a pungent slightly sweet odor. Propiolactone is a disinfectant used for the sterilization of blood plasma, vaccines, tissue grafts, surgical instruments, and enzymes.…

Kategori:
Anti-Infective AgentsCompounds used in a research, industrial, or household settingDisinfectants +1
Target Protein:
DNA
Waktu ParuhThe half-life of pr…
Vol. Distribusi-
Klirens-
Genetik -
Propiomazine Approved DB00777
small molecule | CAS: 362-29-8

Propiomazine, an atypical antipsychotic agent, is used to treat both negative and positive symptoms of schizophrenia, acute mania with bipolar disorder, agitation, and psychotic symptoms in dementia. Future uses may include the treatment of obsessive-compulsi…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +20
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptorAlpha-1A adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propionamide DB04161
small molecule | CAS: 79-05-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiopromazine DB11540
small molecule | CAS: 3568-24-9

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiverine Approved DB12278
small molecule | CAS: 60569-19-9

Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB) [A32576]. Overactive bladder (OAB) is a chronic condition of the lower urinary tract characterized by urinary…

Kategori:
Acids, CarbocyclicAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +4
Waktu ParuhIn three studies in…
Vol. DistribusiIn one study, the v…
KlirensMean total clearanc…
Genetik -
Propofol Approved DB00818
small molecule | CAS: 2078-54-8

Propofol is an intravenous anaesthetic agent used for induction and maintenance of general anaesthesia. IV administration of propfol is used to induce unconsciousness after which anaesthesia may be maintained using a combination of medications. Recovery from …

Kategori:
Agents Causing Muscle ToxicityAgents that produce hypertensionAgents that reduce seizure threshold +32
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit beta-3GABA(A) Receptor +2
Waktu ParuhInitial distributio…
Vol. Distribusi* 60 L/kg [healthy …
Klirens* 23 - 50 mL/kg/min…
Genetik -
small molecule | CAS: 184869-48-5

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, General
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propolis wax Approved DB11355
small molecule

Propolis wax is naturally produced by honeybees by mixing the resin or exudate collected from tree buds, sap flows, or other botanical sources with beeswax that contains fatty acids and bee enzymes. Propolis itself contains various chemical compounds includin…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propoxycaine Approved DB09342
small molecule | CAS: 86-43-1

Propoxycaine is a local anesthetic of the ester type that has a rapid onset of action and a longer duration of action than procaine hydrochloride [L1588]. This drug was removed from the US market in 1996. Although no longer available in the United States,…

Kategori:
Acids, CarbocyclicAminobenzoatesAnesthetics +11
Target Protein:
Voltage-gated sodium channel alpha subunit
Waktu Paruh-
Vol. Distribusi-
KlirensVia the kidneys, pr…
Genetik -
Propranolol Approved DB00571
small molecule | CAS: 525-66-6

Propranolol is a racemic mixture of 2 enantiomers where the S(-)-enantiomer has approximately 100 times the binding affinity for beta adrenergic receptors.[L6904] Propranolol is used to treat a number of conditions but most commonly is used for hypertension.[…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +37
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of pr…
Genetik -
Propyl alcohol Approved DB03175
small molecule | CAS: 71-23-8

A colorless liquid made by oxidation of aliphatic hydrocarbons that is used as a solvent and chemical intermediate.

Kategori:
AlcoholsAntiseptics and DisinfectantsDermatologicals +1
Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propyl Gallate DB12450
small molecule | CAS: 121-79-9

Propyl Gallate is under investigation in clinical trial NCT01450098 (A Study of LY2484595 in Healthy Subjects).

Kategori:
Acids, CarbocyclicAntioxidantsBenzene Derivatives +7
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propylene glycol Approved DB01839
small molecule | CAS: 57-55-6

A clear, colorless, viscous organic solvent and diluent used in pharmaceutical preparations.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingDrug Delivery Systems +7
Target Protein:
B12-independent glycerol dehydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propyliodone Approved DB09366
small molecule | CAS: 587-61-1

Radiopaque medium usually in oil; used in bronchography.

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propylthiouracil Approved DB00550
small molecule | CAS: 51-52-5

A thiourea antithyroid agent. Propythiouracil inhibits the synthesis of thyroxine and inhibits the peripheral conversion of throxine to tri-iodothyronine. It is used in the treatment of hyperthyroidism. (From Martindale, The Extra Pharmacopeoia, 30th ed, p534)

Kategori:
Agents Causing Muscle ToxicityAntimetabolitesAntithyroid agents +14
Target Protein:
Type I iodothyronine deiodinaseThyroid peroxidase
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Propyphenazone DB13524
small molecule | CAS: 479-92-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proquazone DB13649
small molecule | CAS: 22760-18-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prosopis velutina seed Approved DB15510
biotech

Prosopis velutina seed allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13367-85-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 41598-07-6

The principal cyclooxygenase metabolite of arachidonic acid. It is released upon activation of mast cells and is also synthesized by alveolar macrophages. Among its many biological actions, the most important are its bronchoconstrictor, platelet-activating-fa…

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Target Protein:
Prostaglandin D2 receptorProstaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtype +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prostalene DB11454
small molecule | CAS: 54120-61-5

Analog of prostaglandin F2 alpha.

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protamine sulfate Approved DB09141
biotech | CAS: 9009-65-8

Since it's earliest discovery in salmon rine sperm heads in the late 1800's to its formal introduction via US FDA approval in 1939, protamine sulfate has occupied an important therapeutic niche as perhaps the only viable option for reversing the anticoagulant…

Kategori:
Amino Acids, Peptides, and ProteinsAntiheparin AgentsHematologic Agents +5
Waktu ParuhThe half-life of pr…
Vol. DistribusiIn a study group of…
KlirensIn a study group of…
Genetik -
Protein hydrolysate Approved DB09356
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsProtein HydrolysatesProteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protein S human Approved DB13149
biotech

Protein S human is a vitamin K-dependent plasma glycoprotein which has antcoagulant properties [A19561]. It serves as a negative feedback mechanism in the coagulation cascade.

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBiological Factors +8
Target Protein:
Coagulation factor VCoagulation factor XVitamin K-dependent protein C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prothipendyl DB12958
small molecule | CAS: 303-69-5

Prothipendyl has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsNervous System +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protiofate DB13632
small molecule | CAS: 58416-00-5

Deskripsi belum tersedia.

Kategori:
Genito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protirelin Approved DB09421
small molecule | CAS: 24305-27-9

Protirelin is the pharmaceutically available synthetic analogue of the endogenous peptide thyrotropin-releasing hormone (TRH). It is a tri-peptide tropic hormone, released by the hypothalamus, that stimulates the release of Thyroid Stimulating Hormone (TSH) a…

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +12
Target Protein:
Thyrotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 139-85-5

Also known as protocatechuic aldehyde, protocatechualdehyde is a naturally-occuring phenolic aldehyde that is found in barley, green cavendish bananas, grapevine leaves and root of the herb S. miltiorrhiza [A27224]. Protocatechualdehyde possesses antiprolifer…

Kategori:
AldehydesAnticoagulantsBenzene Derivatives +2
Target Protein:
Amine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protoporphyrin DB02285
small molecule | CAS: 553-12-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsDermatologicalsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Hematopoietic prostaglandin D synthaseFerritin light chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9901–9950 dari 12560
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