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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 199 / 321
Mdl-29951 DB04175
small molecule | CAS: 101861-63-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Fructose-1,6-bisphosphatase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MDL72527 DB04188
small molecule | CAS: 99207-33-7

Deskripsi belum tersedia.

Kategori:
AminesBiogenic AminesBiogenic Polyamines +3
Target Protein:
Spermine oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MDR-101 DB18513
biotech

MDR-101 is a CD34+ hematopoietic stem and progenitor cells with CD3+ T-cells

Waktu Paruh-
Vol. Distribusi-
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Genetik -
MDX-018 DB05484
small molecule

MDX-018, also known as HuMax-Inflam, is a fully human antibody that is directed to IL-8 (interleukin-8) and may have potential application in oncology and inflammation. Trials will initially focus on studies to treat glioblastoma, a cancer of the central nerv…

Target Protein:
Interleukin-8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MDX-1097 DB18383
biotech

MDX-1097 is a chimeric monoclonal antibody directed against the kappa myeloma antigen (KMA).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
MDX-1303 DB05945
biotech | CAS: 915947-57-8

MDX-1303 is a fully human antibody against the inhalation anthrax, the most lethal form of illness in humans caused by the Bacillus anthracis bacterium, and targets a protein component of these lethal toxins known as the anthrax protective antigen.

Target Protein:
Anthrax toxin receptor 2Anthrax toxin receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MDX-1379 DB05329
biotech

MDX-1379 vaccine consists of two gp100 melanoma peptides. This drug is underinvestigation to treat malignant melanoma.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MDX-210 DB17250
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MDX-214 DB06110
small molecule

MDX-214 consists of recombinant human epidermal growth factor (EGF) genetically linked to a fully human antibody fragment that is designed to activate cytotoxic killing of cancer cells by immune effector cells. It is developed for the treatment of EGF-R overe…

Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ME-344 DB13062
small molecule | CAS: 1374524-68-1

ME-344 has been used in trials studying the treatment of Solid Tumors.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Me-4(18F)DG DB19207
small molecule | CAS: 915776-36-2

Me-4(18F)DG is under investigation in clinical trial NCT05558904 (An Investigational Scan (Me-4fdg PET/CT) for the Detection of Sodium-glucose Transport for Early Diagnosis of Lung Cancer).

Kategori:
CarbohydratesFluorine RadioisotopesGlycosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 153065-40-8

Meadowfoam seed oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesLipids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebanazine DB09248
small molecule | CAS: 65-64-5

Mebanazine, also known as _Actomol_, is a monoamine oxidase inhibitor (MAOI) belonging to the _hydrazine_ class of chemicals. It was used in the past as an antidepressant in the 1960s, but has since been discontinued because of its hepatotoxic potential.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebendazole Approved DB00643
small molecule | CAS: 31431-39-7

A benzimidazole that acts by interfering with carbohydrate metabolism and inhibiting polymerization of microtubules. [PubChem]

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +11
Target Protein:
Tubulin alpha-1A chainTubulin beta-4B chain
Waktu Paruh2.5 to 5.5 hours (r…
Vol. Distribusi-
Klirens-
Genetik -
Mebenil DB14728
small molecule | CAS: 7055-03-0

An obsolete fungicide used to control various pathogens on cereals and seed potatoes.

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebeverine Approved DB12554
small molecule | CAS: 3625-06-7

Mebeverine has been investigated for the treatment of Irritable Bowel Syndrome and Post-cholecystectomy Gastrointestinal Spasms.

Kategori:
Agents Causing Muscle ToxicityAgents producing tachycardiaAlimentary Tract and Metabolism +10
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebhydrolin DB13808
small molecule | CAS: 524-81-2

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic UseHeterocyclic Compounds, Fused-RingIndole Alkaloids +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebicar DB13522
small molecule | CAS: 10095-06-4

Deskripsi belum tersedia.

Kategori:
AmidesAnalgesicsAnti-Anxiety Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebrofenin Approved DB15779
small molecule | CAS: 78266-06-5

Deskripsi belum tersedia.

Kategori:
AminesAmino AcidsAmino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebutamate Approved DB06797
small molecule | CAS: 64-55-1

Mebutamate is a sedative and anxiolytic drug with anti-hypertensive (blood pressure lowering) effects comparable to those of other barbiturates but is only around 1/3rd the potency of secobarbital as a sedative. Side effects include dizziness and headaches.

Kategori:
Anti-Anxiety AgentsCarbamatesCentral Nervous System Depressants +2
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mebutizide DB13430
small molecule | CAS: 3568-00-1

Deskripsi belum tersedia.

Kategori:
DiureticsHeterocyclic Compounds, Fused-RingHyperglycemia-Associated Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mecamylamine Approved DB00657
small molecule | CAS: 60-40-2

A nicotinic antagonist that is well absorbed from the gastrointestinal tract and crosses the blood-brain barrier. Mecamylamine has been used as a ganglionic blocker in treating hypertension, but, like most ganglionic blockers, is more often used now as a rese…

Kategori:
Agents that produce neuromuscular block (indirect)Antiadrenergic Agents, Ganglion-BlockingAnticholinergic Agents +15
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-4 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1570067-55-8

Mecapegfilgrastim is under investigation in clinical trial NCT05463601 (Mecapegfilgrastim for the Prevention of Dalpiciclib -Induced Neutropenia in Advanced Breast Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mecasermin Approved DB01277
biotech | CAS: 68562-41-4

Mecasermin contains recombinant-DNA-engineered human insulin-like growth factor-1 (rhIGF-1)[FDA Label]. IGF-1 consists of 70 amino acids in a single chain with three intramolecular disulfide bridges and a molecular weight of 7649 daltons. The amino acid seque…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesBiological Factors +15
Target Protein:
Insulin-like growth factor 1 receptorInsulin-like growth factor-binding protein 3Insulin receptor +1
Waktu ParuhMean half life of 5…
Vol. Distribusi* 0.257 ± 0.073 L/k…
KlirensClearance of Mecase…
Genetik -
Mecasermin rinfabate Approved DB14751
biotech | CAS: 478166-15-3

Mecasermin rinfabate is approved for severe primary insulin-like growth factor (IGF) deficiency or in patients with GH gene deletion who have developed antibodies to growth hormone (GH)[A176020]. Mecasermin rinfabate is similar to [DB01277] in that both drugs…

Kategori:
Anterior Pituitary Lobe Hormones and AnaloguesPituitary and Hypothalamic Hormones and AnaloguesSomatropin and Somatropin Agonists +1
Target Protein:
Insulin-like growth factor 1 receptorInsulin receptorCation-independent mannose-6-phosphate receptor
Waktu ParuhHalf life ranges fr…
Vol. DistribusiApproximately 1000m…
KlirensClearance ranges fr…
Genetik -
biotech | CAS: 2460400-64-8

Mecbotamab vedotin is an anti-Axl humanized monoclonal antibody conjugated to monomethyl auristatin E using a cleavable linker (CAB-Axl-ADC).[A255212]

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mechlorethamine Approved DB00888
small molecule | CAS: 51-75-2

A vesicant and necrotizing irritant destructive to mucous membranes, mechlorethamine is an alkylating drug. It was formerly used as a war gas. The hydrochloride is used as an antineoplastic in Hodgkin's disease and lymphomas. It causes severe gastrointestinal…

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +16
Target Protein:
DNA
Waktu Paruh15 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meclinertant DB06455
small molecule | CAS: 146362-70-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Neurotensin, antagonists & inhibitors
Target Protein:
Neurotensin receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meclizine Approved DB00737
small molecule | CAS: 569-65-3

Meclizine is a histamine H1 antagonist with antiemetic and antivertigo properties. It is used in the symptomatic treatment of motion sickness and control of vertigo associated with vestibular system diseases. It also exhibits anticholinergic, central nervous …

Kategori:
Anti-Allergic AgentsAnticholinergic AgentsAntiemetics +19
Target Protein:
Histamine H1 receptorNuclear receptor subfamily 1 group I member 3
Waktu ParuhMeclizine has a pla…
Vol. DistribusiThe volume of distr…
KlirensThere is limited da…
Genetik -
Meclocycline DB13092
small molecule | CAS: 2013-58-3

Meclocycline is under investigation in clinical trial NCT00385515 (Efficacy of SNX-1012 in the Treatment of Oral Mucositis) [L797].

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Bacterial Agents +5
Target Protein:
30S ribosomal protein S7
Waktu ParuhHalf life estimated…
Vol. DistribusiEstimated Vd of 121…
Klirens-
Genetik -
Meclofenamic acid Approved DB00939
small molecule | CAS: 644-62-2

A non-steroidal anti-inflammatory agent with antipyretic and antigranulation activities. It also inhibits prostaglandin biosynthesis.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +25
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Polyunsaturated fatty acid 5-lipoxygenase +2
Waktu ParuhIn a study in 10 he…
Vol. Distribusi* 9.1 to 43.2 L
Klirens* Oral cl=206 mL/min
Genetik -
Meclofenoxate DB13758
small molecule | CAS: 51-68-3

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicCentral Nervous System Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mecloxamine DB15790
small molecule | CAS: 5668-06-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mecobalamin Approved DB03614
small molecule | CAS: 13422-55-4

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansCorrinoids +4
Target Protein:
Methionine synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medazepam DB13437
small molecule | CAS: 2898-12-6

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsAnticonvulsantsBenzazepines +17
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medetomidine DB11428
small molecule | CAS: 86347-14-0

Medetomidine is a synthetic compound used as a surgical anesthetic and analgesic. It is normally found as its hydrochloride salt, medetomidine hydrochloride. Medetomidine is an intravenously available alpha-2 adrenergic agonist. The drug has been developed by…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +12
Target Protein:
Alpha-2A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI-491 DB17859
biotech

MEDI-491 is a recombinant human parvovirus B19 vaccine composed of the VP1 and VP2 capsid proteins.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI-547 DB18360
biotech

MEDI-547 is an anti-EphA1 monoclonal antibody conjugated to mcMMAF

Kategori:
Acids, CarbocyclicAmino Acids, Peptides, and ProteinsAntibodies +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI-6469 DB15306
biotech | CAS: 1715924-11-0

MEDI-6469 is a monoclonal antibody under investigation in clinical trial NCT02205333 (A Phase 1b/2 Safety and Tolerability of MEDI6469 in Combination With Therapeutic Immune Agents or Monoclonal Antibodies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI3506 DB16473
biotech | CAS: 2376858-66-9

Tozorakimab (MEDI3506), developed by AstraZeneca, was investigated in multiple clinical trials to evaluate its safety, tolerability, efficacy, and pharmacokinetics across various conditions. These trials include NCT03096795 (completed; healthy participants, C…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Interleukin-33
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEDI6012 DB14833
biotech

Recombinant human lecithin:cholesterol acyltransferase is under investigation in clinical trial NCT03578809 (A Study to Evaluate the Safety and Efficacy of MEDI6012 in Acute ST Elevation Myocardial Infarction).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 84082-36-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Medical air Approved DB09337
small molecule | CAS: 132259-10-0

Medical air is supplied by a special air compressor to patient care areas using clean outside air.

Kategori:
Medical GasesOther Miscellaneous Therapeutic Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The use of the plant species _Cannabis sativa_ and _Cannabis indica_, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical conditions as a wave of legalization in North America has changed public …

Kategori:
Agents producing tachycardiaBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Inducers +51
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +38
Waktu ParuhThe half life of TH…
Vol. DistribusiAs a very lipophili…
KlirensOne study reported …
Genetik -
Medifoxamine Approved DB13219
small molecule | CAS: 32359-34-5

Medifoxamine was marketed as an atypical antidepressant, with anxiolyitc properties in France, Spain, and Morrocco in the 1990s but was later withdrawn from the market due to it causing cases of hepatotoxicity [L5461, A174976].

Kategori:
AminesAntidepressive AgentsCentral Nervous System Depressants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medium-chain triglycerides Approved DB13959
small molecule | CAS: 438544-49-1

Medium-chain triglycerides (MCTs) are triglycerides made up of a glycerol backbone and three fatty acids with an aliphatic tail of six to 12 carbon atoms. MCTs are found in natural foods, such as coconut oil, palm kernel oil, and raw coconut meat. In the body…

Kategori:
LipidsOilsParenteral Nutrition Solutions +1
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of me…
Genetik -
Medrogestone Approved DB09124
small molecule | CAS: 977-79-7

Medrogestone (INN), also known as 6,17?-dimethyl-6-dehydroprogesterone, is a progestational agent derived from 17-methylprogesterone. It was conceived as an alternative for an orally effective contraceptive option.[A31526] It was developed by Ayerst, approved…

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Target Protein:
Progesterone receptor
Waktu ParuhThe half-life of me…
Vol. Distribusi-
Klirens-
Genetik -
Medronic acid Approved DB14078
small molecule | CAS: 1984-15-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Medroxyprogesterone acetate Approved DB00603
small molecule | CAS: 71-58-9

Medroxyprogesterone acetate (MPA) is a [progesterone] derivative that is more resistant to metabolism for improved pharmacokinetic properties.[A14848] MPA can be use to treat secondary amenorrhea, endometrial hyperplasia, abnormal uterine bleeding, osteoporos…

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +46
Target Protein:
Progesterone receptorEstrogen receptorATP-dependent translocase ABCB1 +1
Waktu ParuhOral medroxyprogest…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Medrysone Approved DB00253
small molecule | CAS: 2668-66-8

Medrysone is a corticosteroid used in ophthalmology.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +24
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9901–9950 dari 16004
Sebelumnya Halaman 199 / 321 Berikutnya