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11778

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8554 (72.6%)
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6383 (54.2%)
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11778 (100.0%)

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Halaman 198 / 236
small molecule | CAS: 89-73-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Infective AgentsAntifungal Agents +3
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Salicylic acid Approved DB00936
small molecule | CAS: 69-72-7

A compound obtained from the bark of the white willow and wintergreen leaves, and also prepared synthetically. It has bacteriostatic, fungicidal, and keratolytic actions. Its salts, the salicylates, are used as analgesics.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +35
Target Protein:
Carbonic anhydrase 6Carbonic anhydrase 12Carbonic anhydrase 2 +5
Waktu Paruh-
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Salix alba bark Approved DB14274
biotech

Salix alba bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Herbs and Natural Products
Waktu Paruh-
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Salix discolor pollen Approved DB10753
biotech

Salix discolor pollen is the pollen of the Salix discolor plant. Salix discolor pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Salix lasiolepis pollen Approved DB10752
biotech

Salix lasiolepis pollen is the pollen of the Salix lasiolepis plant. Salix lasiolepis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Salmeterol Approved DB00938
small molecule | CAS: 89365-50-4

Salmeterol is a long-acting beta-2 adrenergic receptor agonist drug that is currently prescribed for the treatment of asthma and chronic obstructive pulmonary disease COPD.[L11545,L11548,L11551,L11554,L11557] It has a longer duration of action than the short-…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +35
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhThe half life of sa…
Vol. DistribusiIn asthmatic patien…
KlirensThe average clearan…
Genetik -
Salmon calcitonin Approved DB00017
biotech | CAS: 47931-85-1

Synthetic peptide, 32 residues long formulated as a nasal spray.

Kategori:
Amino Acids, Peptides, and ProteinsBone Density Conservation AgentsBone Density, drug effects +15
Target Protein:
Calcitonin receptor
Waktu ParuhHalf-life eliminati…
Vol. Distribusi0.15 to 0.3 L/kg
Klirens-
Genetik -
biotech

Salvia miltiorrhiza root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +15
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 96574-01-5

Salvianolic acid A is under investigation in clinical trial NCT03908242 (Phase I Study of Continuous Administration of Salvianolic Acid A Tablet).

Kategori:
Acids, CarbocyclicAntineoplastic AgentsCinnamates +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 121521-90-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAldehyde ReductaseAldehyde Reductase, antagonists & inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Salvinorin A DB12327
small molecule | CAS: 83729-01-5

Salvinorin A has been investigated for the basic science of Pharmaceutical Preparations.

Kategori:
AlkaloidsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
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Samalizumab DB12636
biotech | CAS: 1073059-33-2

Samalizumab has been used in trials studying the treatment of Multiple Myeloma and B-cell Chronic Lymphocytic Leukemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Samarium DB12403
small molecule | CAS: 7440-19-9

Samarium has been used in trials studying the treatment and prevention of Pain, Cancer, Metastasis, Prostate Cancer, and Metastatic Osteosarcoma, among others.

Kategori:
ElementsLanthanoid Series ElementsMetals +1
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Samarium (153Sm) lexidronam Approved DB05273
small molecule | CAS: 122575-21-7

Samarium Sm 153 lexidronam is a radioactive medication used to treat pain caused by cancer that has spread to the bone. It is a radiopharmaceutical. Radiopharmaceuticals are radioactive agents that may be used to diagnose some diseases by studying the functio…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticCentral Nervous System Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samarium Sm-153 DB12905
small molecule | CAS: 15766-00-4

Samarium 153 has been used in trials studying the supportive care of Pain, Lung Cancer, Breast Cancer, Prostate Cancer, and Metastatic Cancer.

Kategori:
ElementsIsotopesLanthanoid Series Elements +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Samatasvir DB12660
small molecule | CAS: 1312547-19-5

Samatasvir has been used in trials studying the treatment of Hepatitis C, Chronic, Chronic Hepatitis C Virus, and Chronic Hepatitis C Infection.

Kategori:
Acids, AcyclicHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

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Samuraciclib DB16061
small molecule | CAS: 1805833-75-3

Samuraciclib is under investigation in clinical trial NCT03363893 (Modular Study to Evaluate CT7001 Alone in Cancer Patients With Advanced Malignancies).

Target Protein:
Cyclin-dependent kinase 7
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 141646-08-4

Sanfetrinem cilexetil is under investigation in clinical trial NCT05388448 (EBA, Safety and Tolerability of Sanfetrinem Cilexetil).

Kategori:
Amides
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Santonin DB19377
small molecule

Santonin is a anthelmintic drug that was previously approved in the US to treat certain parasitic infections.

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sapablursen DB18608
biotech | CAS: 2273007-95-5

Sapablursen is a synthetic 2'-O-(2-methoxyethyl)-modified antisense oligonucleotide linked to a tri-antennary cluster of N-acetyl galactosamine (GalNAc3) sugars targeting transmembrane protease, serine 6 messenger ribonucleic acid

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Saposin C DB17380
biotech

Saposin C is a lysosomal protein. Recombinant, non-glycosylated Saposin C is an active ingredient of BXQ-350, which is a novel, investigational anti-neoplastic therapy. BXQ-350 consists of Saposin C and the phospholipid dioleoylphosphatidyl-serine (DOPS), a p…

Kategori:
CoenzymesEnzymes and CoenzymesSphingolipid Activator Proteins
Waktu Paruh-
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Genetik -
Saprisartan DB01347
small molecule | CAS: 146623-69-0

Saprisartan is an AT1 receptor antagonist. It is based on medications of losartan's prototypical chemical structure. The mode of (functional) AT1 receptor antagonism has been characterized as insurmountable/noncompetitive for saprisartan. It is very likely t…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +6
Target Protein:
Type-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sapropterin Approved DB00360
small molecule | CAS: 62989-33-7

Sapropterin (tetrahydrobiopterin or BH4) is a cofactor in the synthesis of nitric oxide. It is also essential in the conversion of phenylalanine to tyrosine by the enzyme phenylalanine-4-hydroxylase; the conversion of tyrosine to L-dopa by the enzyme tyrosine…

Kategori:
Alimentary Tract and MetabolismAminesBCRP/ABCG2 Inhibitors +15
Target Protein:
Phenylalanine-4-hydroxylaseNitric oxide synthase 3Tyrosine 3-monooxygenase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Saquinavir Approved DB01232
small molecule | CAS: 127779-20-8

Saquinavir is an HIV-1 protease inhibitor used in combination with [ritonavir] and other antiretrovirals for the treatment of human immunodeficiency virus-1 (HIV-1) infection. In 1995 it became the first protease inhibitor approved by the FDA, followed shortl…

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +44
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh-
Vol. DistribusiThe steady-state vo…
KlirensThe systemic cleara…
Genetik -
SAR-125844 DB15382
small molecule | CAS: 1116743-46-4

SAR-125844 is under investigation in clinical trial NCT01391533 (Study of SAR125844 Single Agent Administered as Slow Intravenous Infusion in Adult Patients With Advanced Malignant Solid Tumors).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfur Compounds +1
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR-405838 DB12541
small molecule | CAS: 1303607-60-4

SAR405838 has been used in trials studying the treatment of Neoplasm Malignant.

Kategori:
Heterocyclic Compounds, Fused-RingP-glycoprotein substrates
Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
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SAR-439459 DB17864
biotech | CAS: 2114339-57-8

SAR-439459 is a pan-transforming Growth Factor-beta (TGF?) neutralizing antibody.[A259862] Developed by Sanofi, it is being investigated for the treatment of cancers and Osteogenesis Imperfecta.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
SAR421869 DB17909
biotech

SAR421869 is a Lentiviral Vector Containing The Human My07A Gene currently being investigated for the treatment of retinitis pigmentosa associated with Usher syndrome 1B gene defect.

Waktu Paruh-
Vol. Distribusi-
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SAR422459 DB17908
biotech

SAR422459 is a Lentiviral Vector Containing The Human Abca4 Gene that is currently being investigated to treat Stargardt disease.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
SAR443122 DB16492
small molecule | CAS: 2125450-76-0

SAR443122, was investigated in several clinical trials to evaluate its safety and efficacy. NCT04469621 was studied in severe COVID-19 patients, while NCT05588843 is currently recruiting participants with ulcerative colitis. Additionally, NCT04781816, which w…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Receptor-interacting serine/threonine-protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
SAR445136 DB17708
biotech

SAR445136 is an investigational zinc finger nuclease gene-edited cell therapy. It consists of autologous CD34+ hematopoietic stem precursor cells (HSPC) modified ex vivo by zinc finger nucleases (ZFN) that target the BCL11A gene erythroid-specific enhancer (E…

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Vol. Distribusi-
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Genetik -
small molecule | CAS: 110880-55-2

Sar9, Met (O2)11-Substance P is a neurokinin-1 receptor agonist. It is an analog of the naturally occurring human neuropeptide Substance P, which can be found throughout the body, including in the airways of humans and many other species.

Kategori:
Amino Acids, Peptides, and ProteinsAutacoidsBiological Factors +11
Waktu Paruh-
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Saracatinib DB11805
small molecule | CAS: 379231-04-6

Saracatinib has been investigated for the treatment of Cancer, Osteosarcoma, Ovarian Cancer, Fallopian Tube Cancer, and Primary Peritoneal Cancer.

Kategori:
Antineoplastic AgentsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +6
Target Protein:
Proto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase ABL1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Saralasin DB06763
small molecule | CAS: 34273-10-4

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAgents that produce hypertension +8
Target Protein:
Type-2 angiotensin II receptorType-1 angiotensin II receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Sarcobatus vermiculatus pollen is the pollen of the Sarcobatus vermiculatus plant. Sarcobatus vermiculatus pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Sarconeos DB16457
small molecule

Sarconeos is an activator of the MAS receptor.

Kategori:
Experimental Unapproved Treatments for COVID-19
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Genetik -
Sarcosine DB12519
small molecule | CAS: 107-97-1

Sarcosine has been investigated for the treatment of Schizophrenia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsN-substituted Glycines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Sarecycline Approved DB12035
small molecule | CAS: 1035654-66-0

Sarecycline is a semi-synthetic derivative of tetracycline that was initially discovered by Paratek Pharmaceuticals from Boston, MA but then licensed to Warner Chilcott of Rockaway, NJ in July of 2007 [A40005]. After completing various phase-II and phase-III …

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Systemic UseAnti-Bacterial Agents +7
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent o…
Genetik -
Sargramostim Approved DB00020
biotech | CAS: 123774-72-1

Sargramostim is a human recombinant granulocyte macrophage colony-stimulating factor (GM-CSF) expressed in yeast. It is a glycoprotein that is 127 residues. Substitution of Leu23 leads to a difference from native protein.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaInterleukin-3 receptor subunit alphaCytokine receptor common subunit beta +2
Waktu Paruh-
Vol. Distribusi-
Klirens* 420 mL/min/m2 [No…
Genetik -
Sarilumab Approved DB11767
biotech | CAS: 1189541-98-7

Sarilumab is a fully human anti-interleukin 6 (IL-6) receptor monoclonal IgG1 antibody that binds to both membrane-bound and soluble IL-6 receptor forms, thus blocking the cis- and trans-inflammatory signalling cascades of IL-6.[A27262] Sarilumab was develope…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +22
Target Protein:
Interleukin-6 receptor subunit alphaHigh affinity immunoglobulin gamma Fc receptor ILow affinity immunoglobulin gamma Fc region receptor II-a +3
Waktu ParuhThe half-life will …
Vol. DistribusiIn patients with rh…
KlirensSarilumab is not el…
Genetik -
Sarpogrelate DB12163
small molecule | CAS: 125926-17-2

Sarpogrelate has been investigated for the treatment of Diabetes Mellitus, Diabetic Nephropathy, Coronary Artery Disease, and Renal Insufficiency, Chronic.

Kategori:
Acids, AcyclicAntidepressive AgentsAntiplatelet agents +8
Target Protein:
5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The University of Queensland (UQ), in partnership with The Coalition for Epidemic Preparedeness Inovations (CEPI) and CSL has developed a COVID-19 candidate, SARS-CoV-2 Sclamp. The vaccine was developed using UQ’s rapid response ‘molecular clamp’ vaccine plat…

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Genetik -
biotech

Bimervax is an adjuvanted non-mRNA COVID-19 vaccine utilizing a SARS-CoV-2 recombinant spike (S) protein receptor binding domain (RBD) fusion heterodimer.[L48902] It is intended to elicit protection against Omicron XBB.1.5, one of the dominant circulating SAR…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
Waktu Paruh-
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Genetik -
Saruparib DB18982
small molecule | CAS: 2589531-76-8

Saruparib is under investigation in clinical trial NCT06380751 (Saruparib (AZD5305) Plus Camizestrant Compared With CDK4/6 Inhibitor Plus Endocrine Therapy or Plus Camizestrant in Hr-positive, Her2-negative (IHC 0, 1+, 2+/ ISH Non-amplified), BRCA1, BRCA2, or…

Kategori:
Heterocyclic Compounds, Fused-Ring
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Sasanlimab DB18849
biotech | CAS: 2206792-50-7

Sasanlimab is under investigation in clinical trial NCT06218069 (Immuno-pet Imaging Responses Administered Immune Checkpoint Inhibitor).

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Satavaptan DB14923
small molecule | CAS: 185913-78-4

Satavaptan is under investigation in clinical trial NCT00359437 (Satavaptan in the Prevention of Ascites Recurrence in Patients With Ascites Due to Cirrhosis of the Liver).

Kategori:
Antidiuretic Hormone Receptor AntagonistsNatriuretic AgentsOxazines
Target Protein:
Vasopressin V2 receptor
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Vol. Distribusi-
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Genetik -
small molecule | CAS: 1039726-31-2

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 1638746-88-9

Deskripsi belum tersedia.

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Satralizumab Approved DB15762
biotech | CAS: 1535963-91-7

Satralizumab is a recombinant humanized monoclonal antibody targeted against human interleukin-6 (IL-6) receptors, similar to [tocilizumab], which is produced in Chinese hamster ovary cells and based on an IgG2 framework.[L15536] Satralizumab is used in the t…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Interleukin-6 receptor subunit alpha
Waktu ParuhThe terminal half-l…
Vol. DistribusiSatralizumab is sub…
KlirensThe total clearance…
Genetik -
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