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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Halaman 198 / 272
Orilanolimab DB15312
biotech | CAS: 2066544-85-0

Orilanolimab is under investigation in clinical trial NCT03075878 (A Safety Study of SYNT001 in Subjects With Chronic, Stable Warm Autoimmune Hemolytic Anemia (WAIHA)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orismilast DB19042
small molecule | CAS: 1353546-86-7

Orismilast is under investigation in clinical trial NCT05190419 (Study to Assess the Efficacy and Safety of Orismilast in Psoriasis).

Waktu Paruh-
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Oritavancin Approved DB04911
small molecule | CAS: 171099-57-3

Oritavancin is a glycopeptide antibiotic used for the treatment of skin infections. It was developed by The Medicines Company (acquired by Novartis).[L12858] Oritavancin was initially approved by the FDA in 2014 and formulated to combat susceptible gram-posit…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +24
Target Protein:
Dihydropteroate synthasePeptidoglycan precursorsBacterial cell wall peptide bridging segments +1
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of or…
Genetik -
Orlistat Approved DB01083
small molecule | CAS: 96829-58-2

The global prevalence of obesity is increasing rapidly. Obesity-related complications lead to significant personal and economic burden by reducing quality of life and increasing the cost of healthcare. In some individuals, diet and exercise are insufficient …

Kategori:
Alimentary Tract and MetabolismAnti-Obesity AgentsAntiobesity Preparations, Excl. Diet Products +11
Target Protein:
Pancreatic triacylglycerol lipaseCannabinoid receptor 1Gastric triacylglycerol lipase +1
Waktu ParuhThe half-life of or…
Vol. DistribusiVolume of distribut…
Klirens-
Genetik -
ORM-13070 C-11 DB15324
small molecule | CAS: 1227170-74-2

ORM-13070 C-11 is under investigation in clinical trial NCT00735774 (Suitability of 11C-ORM-13070 as a PET Tracer).

Kategori:
Carbon Radioisotopes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ormeloxifene DB13310
small molecule | CAS: 31477-60-8

Ormeloxifene is a third-generation selective estrogen receptor (ER) modulator. In India, ormeloxifene has been marketed since the 1990s as a non-hormonal, non-steroidal oral contraceptive taken once a week,[A251450] and it was later introduced for the treatme…

Kategori:
Adrenal Cortex HormonesBenzopyransChromans +13
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu ParuhIn healthy, non-lac…
Vol. DistribusiIn healthy women, t…
KlirensIn healthy, non-lac…
Genetik -
Ornidazole DB13026
small molecule | CAS: 16773-42-5

Ornidazole has been used in trials studying the prevention of Elective Colorectal Surgery.

Kategori:
AmebicidesAnti-Infective AgentsAntibacterials for Systemic Use +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ornipressin DB13464
biotech | CAS: 3397-23-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsCoagulants +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ornithine Approved DB00129
small molecule | CAS: 70-26-8

Produced during the urea cycle, ornithine is an amino acid produced from the splitting off of urea from arginine. L-Ornithine allows for the disposal of excess nitrogen and acts as a precursor of citrulline and arginine.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Basic +9
Target Protein:
Ornithine aminotransferase, mitochondrialOrnithine transcarbamylase, mitochondrialArginase-1 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orotic acid DB02262
small molecule | CAS: 65-86-1

Deskripsi belum tersedia.

Kategori:
PyrimidinesPyrimidinones
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialOrotate phosphoribosyltransferaseDihydroorotate dehydrogenase (quinone), mitochondrial +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ORP-101 DB16072
small molecule | CAS: 1820753-68-1

ORP-101 is under investigation in clinical trial NCT04129619 (A Comparison of the Effects of ORP-101 Versus Placebo in Adult Patients With Irritable Bowel Syndrome With Diarrhea (IBS-D)).

Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orphenadrine Approved DB01173
small molecule | CAS: 83-98-7

A muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.

Kategori:
Agents producing tachycardiaAminesAnti-Dyskinesia Agents +41
Target Protein:
Glutamate receptor ionotropic, NMDA 2DGlutamate receptor ionotropic, NMDA 1Glutamate receptor ionotropic, NMDA 3B +4
Waktu Paruh13-20 hours
Vol. Distribusi-
Klirens-
Genetik -
Orris Approved DB10413
biotech

Orris allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ortataxel DB11669
small molecule | CAS: 186348-23-2

Ortataxel has been used in trials studying the treatment of Lymphoma, Lung Cancer, Glioblastoma, and Kidney Cancer.

Kategori:
Antineoplastic AgentsCyclodecanesCycloparaffins +3
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orteronel DB12066
small molecule | CAS: 566939-85-3

Orteronel has been investigated for the treatment of Prostate Cancer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Orthosiphon aristatus leaf Approved DB15838
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Orticumab DB16653
biotech | CAS: 1314241-10-5

Orticumab is under investigation in clinical trial NCT04776629 (A Proof-of-activity Study With Orticumab in Subjects With Psoriasis and Cardiometabolic Risk Factors).

Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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ORY-1001 DB16848
small molecule | CAS: 1401966-39-9

Deskripsi belum tersedia.

Kategori:
AminesCycloparaffinsPolyamines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OS2966 DB17207
biotech

OS2966 is a humanized integrin ?1 (CD29) blocking antibody currently evaluated for the treatment of acute myeloid leukemia, glioblastoma and ovarian cancer.[A254561, L47351]

Waktu Paruh-
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Osalmid DB16273
small molecule | CAS: 526-18-1

Osalmid is under investigation in clinical trial NCT03670173 (Safety and Efficacy Assessments of Osalmid in Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
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Osanetant DB04872
small molecule | CAS: 160492-56-8

Developed by Sanofi-Aventis (formerly Sanofi-Synthelabo), osanetant (SR-142801) is an NK3 receptor antagonist which was under development for the treatment of schizophrenia and other Central Nervous System (CNS) disorders. In a review of its R&D portfolio, th…

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Neuromedin-K receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osbond acid DB14088
small molecule | CAS: 25182-74-5

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oseltamivir Approved DB00198
small molecule | CAS: 196618-13-0

Oseltamivir (marketed as the product Tamiflu?), is an antiviral neuraminidase inhibitor used for the treatment and prophylaxis of infection with influenza viruses A (including pandemic H1N1) and B. Oseltamivir exerts its antiviral activity by inhibiting the a…

Kategori:
AcetamidesAcetatesAmides +8
Target Protein:
NeuraminidaseSialidase-1Sialidase-2
Waktu ParuhPlasma concentratio…
Vol. DistribusiThe mean volume of …
KlirensRenal clearance (18…
Genetik -
Osemitamab DB18219
biotech | CAS: 2460539-61-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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OSI-027 DB12387
small molecule | CAS: 936890-98-1

OSI-027 has been used in trials studying the treatment of Any Solid Tumor or Lymphoma.

Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSI-7836 DB05837
small molecule

OSI-7836 is a member of the nucleoside class of cytotoxic drugs of which gemcitabine is the market leader. OSI Pharmaceuticals develops OSI-7836 as a next-generation gemcitabine. The anti-tumor activity of OSI-7836 appeares to be less schedule dependent than …

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSI-930 DB05913
small molecule | CAS: 728033-96-3

OSI-930 is an orally active inhibitor of two clinically validated targets: c-Kit and the vascular endothelial growth factor receptor-2 (VEGFR-2). OSI-930 is designed to target both cancer cell proliferation and blood vessel growth (angiogenesis) in selected t…

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor KitVascular endothelial growth factor receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osilodrostat Approved DB11837
small molecule | CAS: 928134-65-0

Osilodrostat is an inhibitor of 11?-hydroxylase (also referred to as CYP11B1), the enzyme that catalyzes the final step in the biosynthesis of endogenous cortisol.[L12123] It is used to lower circulating cortisol levels in the treatment of Cushing's disease, …

Kategori:
Antiadrenal PreparationsAnticorticosteroidsCortisol Synthesis Inhibitors +32
Target Protein:
Cytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial
Waktu ParuhThe elimination hal…
Vol. DistribusiThe median apparent…
KlirensData regarding the …
Genetik -
Osimertinib Approved DB09330
small molecule | CAS: 1421373-65-0

Osimertinib is an oral, third-generation epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) drug developed by AstraZeneca Pharmaceuticals.[A7926,L43453] Its use is indicated for the treatment of metastatic non-small cell lung cancer (NSCL…

Kategori:
Acids, AcyclicAcrylatesAmides +29
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe population esti…
Vol. DistribusiThe mean volume of …
KlirensOral clearance is 1…
Genetik -
Osivelotor DB18071
small molecule | CAS: 2417955-18-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Osocimab DB14818
biotech | CAS: 2056878-75-0

Osocimab is under investigation in clinical trial NCT03276143 (Factor XIa inhibition for the prevention of venous Thromboembolism in Patients Undergoing Total Knee Arthroplasty).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osoresnontrine DB16274
small molecule | CAS: 1189767-28-9

Osoresnontrine is under investigation in clinical trial NCT02281773 (A Study to Investigate the Efficacy, Safety and Tolerability of Four Different Doses of BI 409306 Compared to Placebo Given for 12 Weeks in Patients With Schizophrenia on Stable Antipsychoti…

Kategori:
Enzyme InhibitorsPhosphodiesterase Inhibitors
Target Protein:
High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ospemifene Approved DB04938
small molecule | CAS: 128607-22-7

Ospemifene is a new selective non-hormonal estrogen receptor modulator (SERM) that is used for the treatment of moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause. FDA approved on February 26, 2013.

Kategori:
Benzene DerivativesBenzylidene CompoundsCytochrome P-450 CYP2B6 Substrates +14
Target Protein:
Estrogen receptor
Waktu ParuhTerminal half-life …
Vol. Distribusi448 L
KlirensTotal body clearanc…
Genetik -
OSSM-007 DB18553
biotech

OSSM-007 consists of interferon-gamma primed allogeneic mesenchymal stem cells.

Waktu Paruh-
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Ostabolin-C DB05536
small molecule | CAS: 188899-65-2

Ostabolin C was under investigation in clinical trial NCT00787358 (A Proof-of-Concept Study Investigating the Safety and Efficacy of ZT-031 on Hip Fracture Healing in Men and Postmenopausal Women (SHIFT)).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OSU-6162 DB19178
small molecule | CAS: 146798-66-5

OSU-6162 is under investigation in clinical trial NCT05641623 (OSU6162 as Add-on in Ssri/snri-resistant Depression).

Kategori:
Dopamine AgentsDopamine AntagonistsDopamine D2 Receptor Antagonists +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Osugacestat DB12006
small molecule | CAS: 1401066-79-2

Osugacestat (BMS-906024) has been used in trials studying the treatment of Cancer, Lymphoblastic Leukemia, Acute T-cell, and Precursor T-Cell Lymphoblastic Lymphoma.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OT-730 DB16112
small molecule | CAS: 870809-51-1

OT-730 is under investigation in clinical trial NCT00753168 (Phase 1-2 Evaluation of OT-730 Eye Drops in Reducing the Intraocular Pressure in Patients With Ocular Hypertension or Open-angle Glaucoma).

Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otamixaban DB06635
small molecule | CAS: 193153-04-7

Otamixaban is a novel direct Factor Xa (FXa) inhibitor. It is currently being developed by the French pharmaceutical company Sanofi-Aventis as a treatment for acute coronary syndrome.

Kategori:
AnticoagulantsAntithrombinsEnzyme Inhibitors +4
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otelixizumab DB05496
biotech | CAS: 881191-44-2

Otelixizumab is a monoclonal antibody that binds to a receptor found on all T cells called CD3, which is involved in normal T cell signaling. Otelixizumab is believed to inhibit the function of autoreactive T cells, which are important in propagating autoimmu…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otenabant DB11745
small molecule | CAS: 686344-29-6

Otenabant has been investigated for the treatment of Obesity.

Kategori:
Cannabinoid Receptor AntagonistsCannabinoids and similarsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oteracil Approved DB03209
small molecule | CAS: 937-13-3

Oteracil is an adjunct to antineoplastic therapy, used to reduce the toxic side effects associated with chemotherapy. Approved by the European Medicines Agency (EMA) in March 2011, Oteracil is available in combination with [DB09257] and [DB09256] within the c…

Kategori:
Triazines
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Oteseconazole Approved DB13055
small molecule | CAS: 1340593-59-0

Oteseconazole is an azole metalloenzyme inhibitor that targets fungal CYP51.[L41635] CYP51, also known as 14? demethylase, participates in the formation of ergosterol, a compound that plays a vital role in the integrity of cell membranes.[L41635,A247020] By b…

Kategori:
14-alpha Demethylase InhibitorsAntifungal AgentsAntiinfectives for Systemic Use +5
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe median terminal…
Vol. DistribusiOn average, the vol…
KlirensClinical phase I st…
Genetik -
OTI-030 DB05648
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Otilimab DB06303
biotech | CAS: 1638332-55-4

Investigated for the treatment of osteoarthritis and rheumatoid arthritis (RA).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otilonium DB13500
small molecule | CAS: 105360-89-2

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents producing tachycardiaAlimentary Tract and Metabolism +26
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OTL-102 DB18642
biotech

OTL-102 consists of autologous CD34+ enriched cells that contain hematopoietic stem and progenitor cells transduced ex vivo using a lentiviral vector encoding the human gp91phox gene. It is being investigated for the treatment of X-linked chronic granulomatou…

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OTL-103 DB17593
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
OTL-201 DB17652
biotech

OTL-201 is an investigational hematopoietic stem cell (HSC) gene therapy being developed by Orchard Therapeutics for the treatment of mucopolysaccharidosis type IIIA (MPS-IIIA). It consists of a lentiviral vector to insert a functional copy of the human N-Sul…

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