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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 197 / 282
biotech | CAS: 503621-56-5

Deskripsi belum tersedia.

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Nevanimibe DB16254
small molecule | CAS: 133825-80-6

Nevanimibe is under investigation in clinical trial NCT03053271 (A Study of ATR-101 for the Treatment of Endogenous Cushing's Syndrome).

Kategori:
AmidesBenzene Derivatives
Target Protein:
Sterol O-acyltransferase 1Sterol O-acyltransferase 2
Waktu Paruh-
Vol. Distribusi-
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Nevirapine Approved DB00238
small molecule | CAS: 129618-40-2

A potent, non-nucleoside reverse transcriptase inhibitor (NNRTI) used in combination with nucleoside analogues for treatment of Human Immunodeficiency Virus Type 1 (HIV-1) infection and AIDS. Structurally, nevirapine belongs to the dipyridodiazepinone chemica…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +39
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseH
Waktu Paruh45 hours
Vol. Distribusi* 1.21 ± 0.09 L/kg …
Klirens-
Genetik -
Nezastomig DB19061
biotech | CAS: 2657613-60-8

Nezastomig is under investigation in clinical trial NCT06085664 (A Pilot Presurgical Trial of REGN5678 (Anti-psma X CD28) in Patients With High-risk, Localized Prostate Cancer Followed by Radical Prostatectomy).

Waktu Paruh-
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NFS-02 DB18422
biotech

NFS-02 is a recombinant adeno-associated virus serotype 2 containing human mitochondrial ND1 codon optimized gene (rAAV2-ND1).

Waktu Paruh-
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NGD-4715 DB06027
small molecule | CAS: 476322-70-0

NGD-4715 is an investigational compound developed for the treatment of Obesity. NGD-4715 functions as a melanin-concentrating hormone receptor 1 antagonist.

Target Protein:
Melanin-concentrating hormone receptor 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NGGT-002 DB17881
biotech

NGGT-002 is a recombinant adeno-associated virus serotype 8 vector encoding human phenylalanine hydroxylase (PAH).

Waktu Paruh-
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NGN-401 DB18594
biotech

NGN-401 is a recombinant serotype 9 adeno-associated virus (AAV) encoding an intron encoding a miRNA generating sequence, complementary miRNA binding sites and a full-length human methyl cytosine binding protein 2 (MECP2). Developed by Neurogene Inc., it is b…

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NGX267 DB05152
small molecule | CAS: 503431-81-0

NGX267 is a muscarinic agonist. It is developed for the treatment of Alzheimer’s disease and has shown the potential to both reduce symptoms and slow disease progression.

Kategori:
Cholinergic AgentsCholinergic AgonistsMuscarinic Agonists +2
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Niacin Approved DB00627
small molecule | CAS: 59-67-6

Niacin is a B vitamin used to treat vitamin deficiencies as well as hyperlipidemia, dyslipidemia, hypertriglyceridemia, and to reduce the risk of myocardial infarctions.[L7550,L7553,L7556,L7559,L7562,L7565]

Kategori:
Agents Causing Muscle ToxicityCardiovascular AgentsCytochrome P-450 CYP2D6 Inhibitors +31
Target Protein:
Hydroxycarboxylic acid receptor 3Diacylglycerol O-acyltransferase 2Hydroxycarboxylic acid receptor 2 +2
Waktu ParuhThe half life of ni…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Nialamide Approved DB04820
small molecule | CAS: 51-12-7

Withdrawn from the Canadian, US, and UK markets in 1963 due to interactions with food products containing tyrosine.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] ACatechol O-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niaprazine DB13687
small molecule | CAS: 27367-90-4

Niaprazine is a selective brain catecholamine depletor.

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nicardipine Approved DB00622
small molecule | CAS: 55985-32-5

A potent calcium channel blockader with marked vasodilator action. It has antihypertensive properties and is effective in the treatment of angina and coronary spasms without showing cardiodepressant effects. It has also been used in the treatment of asthma an…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +48
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit beta-2Voltage-dependent calcium channel subunit alpha-2/delta-1 +16
Waktu Paruh8.6 hours
Vol. Distribusi* 8.3 L/kg
Klirens* 0.4 L/hr?kg [Foll…
Genetik -
Nicergoline Approved DB00699
small molecule | CAS: 27848-84-6

An ergot derivative that has been used as a cerebral vasodilator and in peripheral vascular disease. It has been suggested to ameliorate cognitive deficits in cerebrovascular disease.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +14
Target Protein:
Alpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nickel cation DB14204
small molecule | CAS: 14701-22-5

Deskripsi belum tersedia.

Waktu Paruh-
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Nicoboxil Approved DB12911
small molecule | CAS: 13912-80-6

Nicoboxil has been investigated for the treatment of Acute Low Back Pain, where it is typically considered an effective and safe therapeutic option. Nevertheless, it is predominantly found paired with nonivamide as a combination topical analgesic product wher…

Kategori:
Drugs that are Mainly Renally ExcretedPyridines
Waktu ParuhThe half-life of es…
Vol. DistribusiDespite the fact th…
KlirensThe elimination of …
Genetik -
Nicofuranose DB13422
small molecule | CAS: 15351-13-0

Deskripsi belum tersedia.

Kategori:
Cardiovascular AgentsLipid Modifying AgentsLipid Modifying Agents, Plain +4
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Nicorandil Approved DB09220
small molecule | CAS: 65141-46-0

Nicorandil is an orally efficacious vasodilatory drug and antianginal agent marketed in the UK, Australia, most of Europe, India, Philippines, Japan, South Korea, and Taiwan. It is not an approved drug by FDA. It is a niacinamide derivative that induces vasod…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +10
Target Protein:
ATP-binding cassette sub-family C member 9
Waktu ParuhThe elimination hal…
Vol. DistribusiAfter oral (and i.v…
KlirensThe total body clea…
Genetik -
Nicotinaldehyde DB15905
small molecule | CAS: 500-22-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Nicotinamide Approved DB02701
small molecule | CAS: 98-92-0

An important compound functioning as a component of the coenzyme NAD. Its primary significance is in the prevention and/or cure of blacktongue and pellagra. Most animals cannot manufacture this compound in amounts sufficient to prevent nutritional deficiency …

Kategori:
Alimentary Tract and MetabolismCytochrome P-450 CYP2D6 InhibitorsCytochrome P-450 CYP2D6 Inhibitors (strength unknown) +13
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2Exotoxin APoly [ADP-ribose] polymerase 1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
6-phosphogluconate dehydrogenase, decarboxylating
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

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small molecule | CAS: 53-59-8

Nicotinamide adenine dinucleotide phosphate. A coenzyme composed of ribosylnicotinamide 5'-phosphate (NMN) coupled by pyrophosphate linkage to the 5'-phosphate adenosine 2',5'-bisphosphate. It serves as an electron carrier in a number of react…

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +6
Target Protein:
Isocitrate dehydrogenase [NADP]Aldo-keto reductase family 1 member B1Glucose-6-phosphate 1-dehydrogenase +57
Waktu Paruh-
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Genetik -
small molecule

3-Carbamoyl-1-beta-D-ribofuranosyl pyridinium hydroxide-5'phosphate, inner salt. A nucleotide in which the nitrogenous base, nicotinamide, is in beta-N-glycosidic linkage with the C-1 position of D-ribose. Synonyms: Nicotinamide Ribonucleotide; NMN. [PubC…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesRibonucleotides
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 2Nicotinamide/nicotinic acid mononucleotide adenylyltransferase 1Nicotinamide/nicotinic acid mononucleotide adenylyltransferase 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1341-23-7

Nicotinamide riboside is under investigation in clinical trial NCT03432871 (Nicotinamide Riboside and Mitochondrial Biogenesis).

Kategori:
Nicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

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Nicotine Approved DB00184
small molecule | CAS: 54-11-5

Nicotine is highly toxic alkaloid. It is the prototypical agonist at nicotinic cholinergic receptors where it dramatically stimulates neurons and ultimately blocks synaptic transmission. Nicotine is also important medically because of its presence in tobacco …

Kategori:
Agents producing tachycardiaAlkaloidsAutonomic Agents +40
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit beta-2 +10
Waktu ParuhCotinine has a half…
Vol. Distribusi* 2 to 3 L/kg
Klirens* 1.2 L/min [health…
Genetik -
Nidufexor DB16255
small molecule | CAS: 1773489-72-7

Nidufexor is under investigation in clinical trial NCT03804879 (Safety, Tolerability and Efficacy of LMB763 in Patients With Diabetic Nephropathy).

Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifedipine Approved DB01115
small molecule | CAS: 21829-25-4

Nifedipine, or BAY a 1040, is a first generation dihydropyridine L-type calcium channel blocker, similar to [nicardipine].[A190210,A190273,A175390,L11383] Nifedipine was developed by Bayer and first described in the literature, along with other dihydropyridin…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +57
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DVoltage-dependent L-type calcium channel subunit beta-2 +5
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe steady state vo…
KlirensThe total body clea…
Genetik -
Nifekalant DB16008
small molecule | CAS: 130636-43-0

Nifekalant is under investigation in clinical trial NCT03855826 (Evaluation of the Efficacy and Safety of Nifekalant Hydrochloride (NIF) Injection).

Kategori:
Antiarrhythmic agentsCardiovascular AgentsPyrimidines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Nifenazone DB13407
small molecule | CAS: 2139-47-1

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niflumic acid DB04552
small molecule | CAS: 4394-00-7

Niflumic acid is an analgesic and anti-inflammatory agent used in the treatment of rheumatoid arthritis.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +25
Target Protein:
Phospholipase A2Prostaglandin G/H synthase 2Chloride channel protein ClC-Ka +3
Waktu Paruh2.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Nifuratel DB13724
small molecule | CAS: 4936-47-4

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiparasitic Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifuroxazide DB13855
small molecule | CAS: 965-52-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAnti-Infective Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifurtimox Approved DB11820
small molecule | CAS: 23256-30-6

Chagas disease, caused by a parasite known as Trypanosoma cruzi (T.cruzi), is a vector-transmitted disease affecting animals and humans in the Americas. It is commonly known as American Trypanosomiasis.[L15366] The CDC estimates that approximately 8 millio…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +11
Target Protein:
NitroreductasesGlyceraldehyde-3-phosphate dehydrogenase, glycosomal
Waktu ParuhThe elimination hal…
Vol. DistribusiNifurtimox crosses …
KlirensOne pharmacokinetic…
Genetik -
Nifurtoinol DB13730
small molecule | CAS: 1088-92-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nifurzide DB13325
small molecule | CAS: 39978-42-2

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntidiarrheals, Intestinal Antiinflammatory/antiinfective AgentsFurans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nigericin DB14056
small molecule | CAS: 28380-24-7

A polyether antibiotic which affects ion transport and ATPase activity in mitochondria. It is produced by Streptomyces hygroscopicus. (From Merck Index, 11th ed)

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Niguldipine DB09239
small molecule | CAS: 113165-32-5

Niguldipine is a calcium channel blocker drug (CCB) with a1-adrenergic antagonist properties.

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +17
Target Protein:
Alpha-1A adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nikethamide DB13655
small molecule | CAS: 59-26-7

Deskripsi belum tersedia.

Kategori:
Central Nervous System AgentsCentral Nervous System StimulantsConvulsants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nikkomycin Z DB12939
small molecule | CAS: 59456-70-1

Nikkomycin Z has been used in trials studying the treatment and basic science of Coccidioidomycosis.

Kategori:
Anti-Infective AgentsAntifungal AgentsCarbohydrates +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nilotinib Approved DB04868
small molecule | CAS: 641571-10-0

Nilotinib, also known as AMN107, is a tyrosine kinase inhibitor under investigation as a possible treatment for chronic myelogenous leukemia (CML). A Phase I clinical trial in 2006 showed that this drug was relatively safe and offered significant therapeutic …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBcr-Abl Tyrosine Kinase Inhibitors +39
Target Protein:
Tyrosine-protein kinase ABL1Mast/stem cell growth factor receptor Kit
Gen Terkait:
UGT1A1
Waktu Paruh15 hours
Vol. Distribusi-
Klirens-
Genetik 1 Varian
Niludipine DB09240
small molecule | CAS: 22609-73-0

Niludipine is a calcium channel blocker.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nilutamide Approved DB00665
small molecule | CAS: 63612-50-0

Nilutamide is an antineoplastic hormonal agent primarily used in the treatment of prostate cancer. Nilutamide is a pure, nonsteroidal anti-androgen with affinity for androgen receptors (but not for progestogen, estrogen, or glucocorticoid receptors). Conseque…

Kategori:
Androgen Receptor AntagonistsAndrogen Receptor InhibitorsAntiandrogens +18
Target Protein:
Androgen receptor
Waktu Paruh38.0-59.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Nilvadipine Approved DB06712
small molecule | CAS: 75530-68-6

Nilvadipine is a calcium channel blocker (CCB) for the treatment of hypertension.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +27
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimacimab DB15115
biotech | CAS: 2098636-09-8

Nimacimab is under investigation in clinical trial NCT03261739 (Safety Tolerability, and PK of RYI-018 After Repeat Dosing in Subjects With Non-Alcoholic Fatty Liver Disease (NAFLD)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimesulide Approved DB04743
small molecule | CAS: 51803-78-2

Nimesulide is a relatively COX-2 selective, non-steroidal anti-inflammatory drug (NSAID) with analgesic and antipyretic properties. Its approved indications are the treatment of acute pain, the symptomatic treatment of osteoarthritis and primary dysmenorrhoea…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +25
Target Protein:
Prostaglandin G/H synthase 2Tumor necrosis factor ligand superfamily member 10Lactotransferrin +1
Waktu Paruh1.8–4.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Nimodipine Approved DB00393
small molecule | CAS: 66085-59-4

Nimodipine is a 1,4-dihydropyridine calcium channel blocker. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium in smooth muscle cells, nim…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +19
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DVoltage-dependent L-type calcium channel subunit alpha-1F +7
Waktu Paruh1.7-9 hours
Vol. Distribusi-
Klirens-
Genetik -
Nimorazole DB12172
small molecule | CAS: 6506-37-2

Nimorazole has been used in trials studying the treatment of Hypoxia, Radiotherapy, Hypoxic Modification, Gene Profile, Gene Signature, and Head and Neck Squamous Cell Carcinoma, among others.

Kategori:
Anti-Infective AgentsAntiparasitic AgentsAntiparasitic Products, Insecticides and Repellents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Nimotuzumab DB06192
biotech | CAS: 780758-10-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9801–9850 dari 14063
Sebelumnya Halaman 197 / 282 Berikutnya