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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

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Hasil Pencarian (16004)

Halaman 196 / 321
small molecule

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 2Beta-lactamase OXA-10UDP-N-acetylmuramoylalanine--D-glutamate ligase +16
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Lysozyme DB13260
biotech | CAS: 12650-88-3

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseDermatologicals +6
Waktu Paruh-
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LYT-200 DB18179
biotech

LYT-200 is a fully human IgG4 monoclonal antibody directed against galectin-9.

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Genetik -
small molecule | CAS: 156021-12-4

Deskripsi belum tersedia.

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetylcholinesterase
Waktu Paruh-
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M-032 DB17258
biotech

Deskripsi belum tersedia.

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M-2698 DB15431
small molecule | CAS: 1379545-95-5

M-2698 is under investigation in clinical trial NCT01971515 (First-in-Human Dose Escalation Trial in Subjects With Advanced Malignancies).

Target Protein:
RAC-alpha serine/threonine-protein kinaseRAC-gamma serine/threonine-protein kinaseRibosomal protein S6 kinase beta-1
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M-701 DB17504
biotech

M-701 is a recombinant anti-EpCAM/CD3 bispecific antibody.

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small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamaseBeta-lactamase
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small molecule | CAS: 6640-24-0

m-Chlorophenylpiperazine has been used in trials studying the treatment of Alcoholism.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNeurotransmitter Agents +7
Target Protein:
5-hydroxytryptamine receptor 1E5-hydroxytryptamine receptor 75-hydroxytryptamine receptor 6 +4
Waktu Paruh-
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M-Cresol DB01776
small molecule | CAS: 108-39-4

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesPhenols
Target Protein:
Insulin
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Genetik -
small molecule | CAS: 1637-75-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzamides and benzamide derivatives +3
Target Protein:
Kynureninase
Waktu Paruh-
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M0002 DB05091
small molecule

M0002 is an orally-active selective vasopressin antagonist that inhibits water re-absorption from the kidneys. It is a vasopressin 2 antagonist and represents a new class of compounds – aquaretics – that produce profound diuresis without loss of electrolytes.…

Target Protein:
Vasopressin V2 receptor
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M1-c6v1 DB18596
biotech

M1-c6v1 is a recombinant oncolytic virus.

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MaaT013 DB18648
biotech

MaaT013 is an allogeneic fecal microbiota therapy. It is being investigated for the treatment of Graft-Versus-Host Disease.

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Macadamia oil DB14330
biotech

Macadamia oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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biotech

Macadamia seed oil glycereth-8 esters is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Macelignan DB14129
small molecule | CAS: 107534-93-0

Macelignan is an NSAID with antioxidant, free radical scavenging, and neuroprotective activities.

Kategori:
Benzene DerivativesBenzyl Compounds
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Macimorelin Approved DB13074
small molecule | CAS: 381231-18-1

Macimorelin, a novel and orally active ghrelin mimetic that stimulates GH secretion, is used in the diagnosis of adult GH deficiency (AGHD). More specifically, macimorelin is a peptidomimetic growth hormone secretagogue (GHS) that acts as an agonist of GH sec…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +11
Target Protein:
Growth hormone secretagogue receptor type 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Macitentan Approved DB08932
small molecule | CAS: 441798-33-0

Macitentan is a dual endothelin receptor antagonist used in the treatment of pulmonary arterial hypertension (PAH).[L35890] It was first approved by the FDA in 2013. Macitentan differs from its predecessor [bosentan] in part due to its lower risk of hepatotox…

Kategori:
AmidesAntihypertensive AgentsAntihypertensives for Pulmonary Arterial Hypertension +13
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu ParuhThe half-life of el…
Vol. DistribusiMacitentan has an a…
KlirensClearance data was …
Genetik -
biotech

Maclura tricuspidata whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Macozinone DB14821
small molecule | CAS: 1377239-83-2

Macozinone is under investigation in clinical trial NCT03036163 (Phase 1 Study of PBTZ169).

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsDrugs for Treatment of Tuberculosis +1
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Madecassic acid DB14037
small molecule | CAS: 18449-41-7

Deskripsi belum tersedia.

Kategori:
Terpenes
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Madecassoside DB15532
small molecule | CAS: 34540-22-2

Deskripsi belum tersedia.

Kategori:
Terpenes
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Maduramicin DB11525
small molecule | CAS: 84878-61-5

Maduramicin is an antiprotozoal agent used in veterinary medicine as prophylaxis against coccidiosis. It is a naturally occurring compound which was first isolated from the actinomycete, Actinomadura rubra.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsIonophores
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Mafenide Approved DB06795
small molecule | CAS: 138-39-6

Mafenide is a sulfonamide-type antimicrobial agent used to treat severe burns. It acts by reducing the bacterial population present in the burn tissue and promotes healing of deep burns.[L36773] In 1998, mafenide acetate was approved under the FDA’s accelerat…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 12Carbonic anhydrase 14 +2
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Mafosfamide DB12083
small molecule | CAS: 88859-04-5

Mafosfamide has been used in trials studying the treatment of Lymphoma, Leukemia, Meningeal Neoplasm, and Brain and Central Nervous System Tumors.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsHydrocarbons, Halogenated +6
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Maftivimab Approved DB15899
biotech | CAS: 2135632-36-7

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhMaftivimab administ…
Vol. DistribusiMaftivimab administ…
KlirensMaftivimab administ…
Genetik -
Magaldrate Approved DB08938
small molecule | CAS: 74978-16-8

Magaldrate is an antacid drug used for the treatment of esophagitis, duodenal and gastric ulcers, and gastroesophageal reflux. Magaldrate has been discontinued in the US market.

Kategori:
Alimentary Tract and MetabolismAlkaliesAluminium Compounds +13
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Magnesium Approved DB14513
small molecule | CAS: 7439-95-4

Magnesium is classified as an alkaline earth metal and has 2 hydration shells.[A19349] The element can be found in abundance in the hydrosphere and in mineral salts such as dolomite and magnesium carbonate.[A19349] Common dietary sources of magnesium incl…

Kategori:
ElementsLaxativesMagnesium Compounds +6
Waktu ParuhMagnesiums biologic…
Vol. DistribusiAccording to a phar…
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Magnesium acetate Approved DB13996
small molecule | CAS: 142-72-3

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAgents that produce neuromuscular block (indirect)Fatty Acids +3
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
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small molecule | CAS: 16674-78-5

Magnesium acetate tetrahydrate is a hydrated form of anhydrous magnesium acetate salt with the chemical formula of Mg(CH3COO)2 • 4H2O. As a salt form of magnesium, magnesium acetate is one of the bioavailable forms of magnesium and forms a very water soluble …

Kategori:
Agents that produce neuromuscular block (indirect)Laxatives
Target Protein:
Glutamate (NMDA) receptor
Waktu ParuhElimination half-li…
Vol. DistribusiMagnesium ions disp…
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Magnesium Aluminum Silicate Approved DB11230
small molecule | CAS: 1327-43-1

Magnesium aluminum silicate is a naturally occurring mineral obtained from silicate ores of the montmorillonite group [A32782]. It is refined to a powder for use in cosmetic and pharmaceutical applications as an absorbent, anticaking agent, opacifying agent, …

Kategori:
Agents that produce neuromuscular block (indirect)MineralsPharmaceutic Aids +1
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Magnesium ascorbate Approved DB14484
small molecule | CAS: 15431-40-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntioxidantsBiological Factors +10
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small molecule | CAS: 7018-07-7

Magnesium aspartate is a magnesium salt of aspartic acid that is commonly used as a mineral supplement. It displays high oral bioavailability and water solubiltiy compared to other magnesium salts such as magnesium citrate, magnesium carbonate and magnesium o…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAmino Acids +8
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small molecule | CAS: 28184-71-6

Deskripsi belum tersedia.

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Magnesium carbonate Approved DB09481
small molecule | CAS: 546-93-0

Magnesium carbonate, also known as magnesite, is a common over the counter remedy for heartburn and upset stomach caused by overproduction of acid in the stomach [FDA Label].

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAluminum and magnesium containing antacids +20
Target Protein:
Glutamate (NMDA) receptor
Waktu ParuhHalf life of 27.7 h…
Vol. DistribusiVd for magnesium is…
KlirensMaximum magnesium c…
Genetik -
Magnesium cation Approved DB01378
small molecule | CAS: 22537-22-0

Magnesium hydroxide is used primarily in "Milk of Magnesia", a white aqueous, mildly alkaline suspension of magnesium hydroxide formulated at about 8%w/v. Milk of magnesia is primarily used to alleviate constipation, but can also be used to relieve indigestio…

Kategori:
Agents that produce neuromuscular block (indirect)Calculi Dissolution AgentIncreased Large Intestinal Motility +9
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
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Magnesium chloride Approved DB09407
small molecule | CAS: 7786-30-3

Magnesium chloride salts are highly soluble in water and the hydrated form of magnesium chloride can be extracted from brine or sea water.

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismBlood and Blood Forming Organs +12
Waktu ParuhElimination half-li…
Vol. DistribusiBone (50% to 60%); …
KlirensMaximum magnesium c…
Genetik -
Magnesium citrate Approved DB11110
small molecule | CAS: 3344-18-1

Magnesium citrate is a low volume and osmotic cathartic agent. The cathartic action works primarily through the high osmolarity of the solution which draws large amounts of fluid into space where is used.[T215] Magnesium citrate is considered by the FDA as an…

Kategori:
Acids, AcyclicAgents that produce neuromuscular block (indirect)Alimentary Tract and Metabolism +15
Waktu ParuhThe study of the ha…
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Magnesium gluconate Approved DB13749
small molecule | CAS: 59625-89-7

Magnesium gluconate is a magnesium salt of gluconate. It demonstrates the highest oral bioavailability of magnesium salts [L2608] and is used as a mineral supplement. Magnesium is ubiquitous in the human body, and is naturally present in many foods, added to …

Kategori:
Acids, AcyclicAgents that produce neuromuscular block (indirect)Alimentary Tract and Metabolism +7
Waktu Paruh-
Vol. DistribusiAbout 60% of the ma…
KlirensThe kidney plays a …
Genetik -
Magnesium glycinate Approved DB11189
small molecule | CAS: 14783-68-7

Magnesium glycinate is a magnesium salt of glycine that is available as dietary supplements as a source of magnesium. It is used in the treatment of magnesium deficiency.

Kategori:
Agents that produce neuromuscular block (indirect)Laxatives
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Magnesium hydroxide Approved DB09104
small molecule | CAS: 1309-42-8

Magnesium hydroxide is an inorganic compound. It is naturally found as the mineral brucite. Magnesium hydroxide can be used as an antacid or a laxative in either an oral liquid suspension or chewable tablet form. Additionally, magnesium hydroxide has smoke …

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAlkalies +22
Waktu ParuhN/A
Vol. DistribusiThe peak action and…
KlirensMagnesium hydroxide…
Genetik -
small molecule | CAS: 18917-93-6

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismMagnesium CompoundsMetal cations +2
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh-
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small molecule | CAS: 58505-81-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismEnzyme InhibitorsKeto Acids +4
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh-
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Magnesium malate Approved DB15555
small molecule | CAS: 869-06-7

Deskripsi belum tersedia.

Waktu Paruh-
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small molecule | CAS: 83918-60-9

Deskripsi belum tersedia.

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small molecule | CAS: 34717-03-8

Magnesium orotate is a magnesium salt of orotic acid and is poorly soluble in water. It is a source of magnesium and is used as a mineral supplement to treat Mg deficiency. Orotic acid acts as a transporter that carries magnesium into the cells. It also exhib…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismMagnesium Compounds +5
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Magnesium oxide Approved DB01377
small molecule | CAS: 1309-48-4

Magnesium oxide is an inorganic compound that occurs in nature as the mineral periclase. In aqueous media combines quickly with water to form magnesium hydroxide. It is used as an antacid and mild laxative and has many nonmedicinal uses.

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAluminum and magnesium containing antacids +16
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small molecule | CAS: 14452-57-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAluminum and magnesium containing antacidsAnions +15
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