Hasil Filter

17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (17430)

Halaman 195 / 349
Ivosidenib Approved DB14568
small molecule | CAS: 1448347-49-6

Ivosidenib is a first-in-class isocitrate dehydrogenase-1 (IDH1) inhibitor. IDH1 is an enzyme that is often mutated and overexpressed in some cancers, leading to aberrant cell growth and proliferation.[A248750] Ivosidenib inhibits mutated IDH1, blocking the e…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntineoplastic Agents +26
Target Protein:
Isocitrate dehydrogenase [NADP] cytoplasmic
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Ivospemin DB17988
small molecule | CAS: 748119-79-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IVT-8086 DB18381
biotech

IVT-8086 is a humanized secreted frizzled-related protein-2 monoclonal antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ivuxolimab DB16208
biotech | CAS: 2128729-41-7

Ivuxolimab is under investigation in clinical trial NCT02554812 (A Study of Avelumab in Combination With Other Cancer Immunotherapies in Advanced Malignancies (JAVELIN Medley)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ixabepilone Approved DB04845
small molecule | CAS: 219989-84-1

Ixabepilone is an epothilone B analog developed by Bristol-Myers Squibb as a cancer drug. It was FDA approved on October 16, 2007, for the treatment of unresponsive aggressive metastatic or locally advanced breast cancer. Ixabepilone is administered through i…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Tubulin beta-3 chain
Waktu Paruh52 hours
Vol. Distribusi-
Klirens-
Genetik -
Ixazomib Approved DB09570
small molecule | CAS: 1072833-77-2

Ixazomib is a reversible proteasome inhibitor. Because it is a modified peptide boronic acid with one chiral center,[A264329] it is considered a boronate proteasome inhibitor.[A7948] More than 99% of the drug compound is the R-enantiomer.[A264329] Ixazomib…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP1A2 Substrates +20
Target Protein:
Proteasome subunit beta type-5
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state vo…
KlirensBased on a populati…
Genetik -
Ixekizumab Approved DB11569
biotech | CAS: 1143503-69-8

Ixekizumab is a humanized immunoglobulin G subclass 4 (IgG4) monoclonal antibody (mAb) against interleukin-17A (IL-17A) and prevents it from interacting with the IL-17A receptor. As IL-17A is a pro-inflammatory cytokine involved in inflammation and immune res…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +14
Target Protein:
Interleukin-17A
Waktu Paruh13 days
Vol. DistribusiThe mean (geometric…
Klirens0.39 L/day
Genetik -
Ixmyelocel-T DB17601
biotech

Ixmyelocel-T is an expanded, autologous multicellular therapy cultured from bone-marrow mononuclear cells. Developed by Vericel Corporation, it is being investigated for cardiomyopathy.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2538429-16-0

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Izaflortaucipir DB18282
small molecule | CAS: 2173361-80-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Izencitinib DB16660
small molecule | CAS: 2051918-33-1

Izencitinib is under investigation in clinical trial NCT03920254 (TD-1473 Long-term Safety (LTS) Ulcerative Colitis (UC) Study).

Kategori:
Colitis, Ulcerative, drug therapyHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Izokibep DB19081
biotech | CAS: 2226130-02-3

Izokibep is under investigation in clinical trial NCT05623345 (Psoriatic Arthritis Study of Izokibep).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Izuralimab DB18933
biotech | CAS: 2329669-80-7

Izuralimab is under investigation in clinical trial NCT05879185 (A Study of Xmab23104 in People With Sarcoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
J147 DB13957
small molecule | CAS: 1146963-51-0

J147 is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging. [A31606,A31607,A31608] It is a curcumin derivative and a potent neurogenic and neuroprotective drug candidate initially develo…

Kategori:
AlkanesBenzene DerivativesCatechols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JAB-21822 DB17478
small molecule

JAB-21822 is an oral small-molecule KRAS G12C inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JAB-3068 DB17131
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein phosphatase non-receptor type 11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JAG101 DB18321
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JAK4D DB18527
small molecule | CAS: 882400-49-9

JAK4D is a first-in-class thyrotropin-releasing hormone (TRH)-based compound.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Jaktinib DB17545
small molecule

Jaktinib is a JAK 1, JAK 2 and JAK 3 inhibitor, being developed by Suzhou Zelgen Biopharmaceuticals. Jaktinib is under investigation in clinical trial NCT04866056 (Jaktinib and Azacitidine in Treating Patients With MDS With MF or MDS/MPN With MF.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Janagliflozin DB16209
small molecule | CAS: 1800115-22-3

Janagliflozin is under investigation in clinical trial NCT03851432 (Janagliflozin Treat Type 2 Diabetes Mellitus (T2DM) Inadequately Controlled With Metformin).

Kategori:
AlcoholsCarbohydratesCyclohexanes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Janssen COVID-19 Vaccine Approved DB15857
biotech

The Janssen COVID-19 vaccine (Ad26.COV2.S) is a recombinant vaccine that contains an adenovirus serotype 26 (Ad26) vector expressing a stabilized SARS-CoV-2 spike protein. The vaccine was created in collaboration with Johnson and Johnson (J&J), Janssen Pharma…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Actively Acquired ImmunityBiological ProductsComplex Mixtures +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Inactivated Japanese Encephalitis Virus Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Jaspisamide A DB03850
small molecule

Deskripsi belum tersedia.

Target Protein:
Actin, alpha skeletal muscle
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JB991 DB05081
small molecule

JB991 is a cyclopentenone prostaglandin analogue intended for treatment of psoriasis. The drug exerts marked antiproliferative and pro-apoptotic effect in human keratinocytes and fibroblasts in vitro. In addition a closely related cyclopentenone prostaglandin…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JBI-778 DB18074
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JBI-802 DB17399
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JBPOS0101 DB16034
small molecule | CAS: 1353949-71-9

JBPOS0101 is under investigation in clinical trial NCT03976076 (A Study of Orally Administered JBPOS0101 in Refractory Infantile Spasms Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JCAR014 DB17232
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
jCell DB17906
biotech

jCell is an human retinal progenitor cell therapy for retinitis pigmentosa.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JE-2147 DB02668
small molecule | CAS: 186538-00-1

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmino Acids, Peptides, and ProteinsAntiviral Agents +4
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JHU-75528 C-11 DB14902
small molecule | CAS: 942063-86-7

JHU-75528 C-11 is under investigation in clinical trial NCT03204305 (Brain Imaging of Cannabinoid Receptors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JLK-247 DB17637
biotech

JLK-247 is an adeno-associated viral vector serotype 9 (AAV9)-mediated gene replacement therapy for the treatment of Sanfilippo Syndrome Type C or MPS IIIC.[L46686]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-17216498 DB17087
small molecule | CAS: 1035626-05-1

JNJ-17216498 is a histamine receptor H3 antagonist developed by Johnson and Johnson for the treatment of narcolepsy.[A253997]

Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-1802 DB17734
small molecule | CAS: 2043343-94-6

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-26489112 DB15203
small molecule | CAS: 871824-55-4

JNJ-26489112 is under investigation in clinical trial NCT00579384 (A Study of the Effects of JNJ-26489112 on the Photic Induced Paroxysmal Electroencephalogram (EEG) Response in Patients With Photosensitive Epilepsy).

Kategori:
AmidesAnticonvulsantsCentral Nervous System Depressants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-27390467 DB06962
small molecule | CAS: 1025795-11-2

JNJ-27390467 is a potent, nonpeptide inhibitor of human mast cell tryptase.

Target Protein:
Tryptase beta-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-27548547 DB15372
small molecule | CAS: 303983-00-8

JNJ-27548547 is under investigation in clinical trial NCT01705002 (Intravenously Administered Pegylated Liposomal Mitomycin-C Lipid-based Prodrug (PROMITIL) in Cancer Patients With Solid Tumors.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-28312141 DB17140
small molecule | CAS: 885692-52-4

Deskripsi belum tersedia.

Kategori:
Receptors, Colony-Stimulating Factor, antagonists & inhibitors
Target Protein:
NT-3 growth factor receptorMast/stem cell growth factor receptor KitTyrosine-protein kinase Lck +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-28330835 DB13936
small molecule | CAS: 888072-47-7

A selective androgen receptor modulator with minimal prostate hypertrophic activity, enhances lean body mass in male rats and stimulates sexual behavior in female rats.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-37822681 DB12579
small molecule | CAS: 935776-74-2

JNJ-37822681 has been used in trials studying the treatment of Schizophrenia.

Kategori:
Dopamine AgentsDopamine AntagonistsDopamine D2 Receptor Antagonists +1
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-38877605 DB13113
small molecule | CAS: 943540-75-8

JNJ-38877605 has been used in trials studying the treatment of Neoplasms.

Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-38877618 DB16883
small molecule | CAS: 943540-74-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-39220675 DB12929
small molecule | CAS: 959740-39-7

JNJ-39220675 has been used in trials studying the treatment of Allergic Rhinitis.

Kategori:
Histamine H3 Antagonists
Target Protein:
Histamine H3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-39393406 DB11867
small molecule | CAS: 953428-73-4

JNJ-39393406 has been used in trials studying the treatment and basic science of DEPRESSION, Schizophrenia, Smoking Cessation, Cognition Disorders, and Alzheimer's Disease.

Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-39758979 DB18899
small molecule | CAS: 1046447-90-8

JNJ-39758979 is under investigation in clinical trial NCT01480388 (A Dose Range Finding Study of JNJ-39758979 in Patients With Active Rheumatoid Arthritis Currently Treated With Methotrexate).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-40346527 DB12504
small molecule | CAS: 1142363-52-7

JNJ-40346527 has been used in trials studying the treatment of Health and Arthritis, Rheumatoid.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
JNJ-40411813 DB12059
small molecule | CAS: 1127498-03-6

JNJ-40411813 has been used in trials studying the treatment and basic science of Confusion, Schizophrenia, Perceptual Disorders, and Major Depressive Disorder.

Kategori:
Pyridines
Target Protein:
Metabotropic glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9701–9750 dari 17430
Sebelumnya Halaman 195 / 349 Berikutnya