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12560

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9109 (72.5%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 195 / 252
biotech

Deskripsi belum tersedia.

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Platensimycin DB08407
small molecule | CAS: 835876-32-9

Deskripsi belum tersedia.

Kategori:
3-Oxoacyl-(Acyl-Carrier-Protein) SynthaseAcids, CarbocyclicAmides +10
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 2
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Platinum DB12257
small molecule | CAS: 7440-06-4

Platinum is under investigation for the treatment of Metastatic Breast Cancer, Non-small Cell Lung Cancer, Gastric Large Cell Neuroendocrine Carcinoma, Colorectal Large Cell Neuroendocrine Carcinoma, and Pancreatic Large Cell Neuroendocrine Carcinoma, among o…

Kategori:
Antineoplastic AgentsChlorine CompoundsCompounds used in a research, industrial, or household setting +9
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biotech

Platycodon grandiflorus leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Plazomicin Approved DB12615
small molecule | CAS: 1154757-24-0

Developed by Achaogen biopharmaceuticals, plazomicin is a next-generation aminoglycoside synthetically derived from [DB12604]. The structure of plazomicin was established via appending hydroxylaminobutyric acid to [DB12604] at position 1 and 2-hydroxyethyl gr…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +12
Target Protein:
rRNA methyltransferase 2, mitochondrial30S ribosomal protein S1130S ribosomal protein S14
Waktu ParuhThe mean (±SD) half…
Vol. DistribusiThe mean (±SD) volu…
KlirensFollowing administr…
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Plecanatide Approved DB13170
small molecule | CAS: 467426-54-6

Plecanatide is a drug approved in January 2017 by the FDA for the treatment of chronic idiopathic constipation (CIC). It should not be used in children less than six years of age, and should be avoided in patients six years to 18 years of age

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +12
Target Protein:
Guanylyl cyclase CGuanylate cyclase soluble subunit alpha-2
Waktu Paruhhalf-life (t½) cann…
Vol. DistribusiConcentrations of p…
KlirensNo excretion studie…
Genetik -
Pleconaril DB05105
small molecule | CAS: 153168-05-9

Pleconaril is an antiviral drug from _viral capsid inhibitor_ class, manufactured by _Schering-Plough_ and intended for the prevention of acute asthma exacerbations and common cold symptoms in asthmatic patients who have had exposure to _picornavirus_. It act…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +4
Target Protein:
Genome polyprotein
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Pleospora herbarum Approved DB10825
biotech

Pleospora herbarum is a fungus which can provoke allergic reactions. Pleospora herbarum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Plerixafor Approved DB06809
small molecule | CAS: 110078-46-1

Plerixafor is a small-molecule inhibitor of C-X-C chemokine receptor type 4 (CXCR4) that acts as a hematopoietic stem cell mobilizer.[A7117,L45678] It is used to stimulate the release of stem cells from the bone marrow into the blood in patients with non-Hodg…

Kategori:
Adjuvants, ImmunologicAminesAnti-HIV Agents +9
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhPlerixafor has a di…
Vol. DistribusiPlerixafor has an a…
KlirensPlerixafor has a to…
Genetik -
Plevitrexed DB06163
small molecule | CAS: 153537-73-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Thymidylate synthase
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Plinabulin DB05992
small molecule | CAS: 714272-27-2

Deskripsi belum tersedia.

Kategori:
DeuteriumPiperazines
Target Protein:
Translation initiation factor eIF2B subunit alphaTranslation initiation factor eIF2B subunit betaTumor necrosis factor
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Plitidepsin DB04977
small molecule | CAS: 137219-37-5

Aplidine is a peptide found in tunicates which shows promise in shrinking tumors in pancreatic, stomach, bladder, and prostate cancers. The specific marine organism is _Aplidium albicans_. Aplidine is also of interest as a potential treatment for some leukemi…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Palmitoyl-protein thioesterase 1Elongation factor 1-alpha 2
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PLN-74809 DB16515
small molecule

PLN-74809 is a small-molecule that dually inhibits both ?<sub>v</sub>?<sub>6</sub> and ?<sub>v</sub>?<sub>1</sub> to treat both idiopathic pulmonary fibrosis (IPF) and primary sclerosing cholangitis (PSC)[L31693]. The compound was granted orphan drug designat…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Integrin alpha-VIntegrin beta-1Integrin beta-6
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Plozalizumab DB12520
biotech | CAS: 1610761-46-0

Plozalizumab has been investigated for the treatment of Atherosclerosis. Plozalizumab, a novel humanized monoclonal antibody, specifically targets CCR2 chemokine receptors found on the surface of certain white blood cells including macrophages and monocytes. …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
C-C chemokine receptor type 2
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Plozasiran DB18997
biotech | CAS: 2379776-40-4

Plozasiran is under investigation in clinical trial NCT05089084 (Study of ARO-APOC3 (Plozasiran) in Adults With Familial Chylomicronemia Syndrome (FCS)).

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Plum Approved DB10560
biotech

Plum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Plumbagin DB17048
small molecule | CAS: 481-42-5

Plumbagin is a compound investigated for its anticancer activity. It has been found that it inactivates the Akt/NF-kB, MMP-9 and VEGF pathways.[A253102]

Kategori:
Adjuvants, ImmunologicAdrenal Cortex HormonesAnthelmintics +17
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
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Plutavimab DB18856
biotech | CAS: 2529854-88-2

Plutavimab is under investigation in clinical trial NCT04900428 (Study to Evaluate a Single Intranasal Dose of STI-2099 (COVI-DROPS™) in Outpatient Adults With COVID-19 (UK)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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PLX-4720 DB06999
small molecule | CAS: 918505-84-7

Deskripsi belum tersedia.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Vascular endothelial growth factor receptor 2Serine/threonine-protein kinase B-raf
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PLX51107 DB17543
small molecule | CAS: 1627929-55-8

PLX51107 is a potent and selective inhibitor of the bromodomain and extraterminal (BET) protein family.[A257246,A257251] PLX51107 is under investigation in clinical trial NCT04022785 (PLX51107 and Azacitidine in Treating Patients With Acute Myeloid Leukemia o…

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PM-060184 DB13137
small molecule | CAS: 960210-99-5

PM060184 has been used in trials studying Solid Tumors.

Kategori:
LactonesPyrans
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pM-81 DB17432
biotech

Deskripsi belum tersedia.

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PM02734 DB05158
small molecule

PM02734 is a marine derived compound. PM02734 as a new antiproliferative drug demonstrating activity against a broad spectrum of tumor types: breast, colon, pancreas, lung and prostate, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic
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PMI-001 DB05730
small molecule

PMI-001 is a stand-alone, disease-modifying, anti-rheumatic drug (DMARD) being developed by Phytomedics Inc. It is an extract of the roots of an undisclosed perennial shrub which interferes with the production of IL-2 and COX-2 proteins, for the potential tre…

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small molecule

Deskripsi belum tersedia.

Target Protein:
Alanine racemase
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PMX-205 DB17938
small molecule | CAS: 514814-49-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesReceptor, Anaphylatoxin C5a, antagonists & inhibitors
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PN0621 DB05218
biotech

PN0621 is an anti-TNF, domain antibody (dAb) based therapeutic. It targets tumour necrosis factor (TNF) to treat auto-immune inflammatory diseases such as rheumatoid arthritis. It is being developed by Peptech.

Target Protein:
Tumor necrosis factor
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PNT001 DB18375
biotech

PNT001 is a humanized IgG4 S228P monoclonal antibody targeting the cis conformation of the phosphorylated Thr231-Pro232 motif in tau.

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PNU-142721 DB08414
small molecule | CAS: 185220-03-5

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
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Poa annua pollen Approved DB10353
biotech

Poa annua pollen is the pollen of the Poa annua plant. Poa annua pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
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Pocapavir DB17736
small molecule | CAS: 146949-21-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsBenzene Derivatives +2
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Pociredir DB18070
small molecule | CAS: 2490676-18-9

Deskripsi belum tersedia.

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Podofilox Approved DB01179
small molecule | CAS: 518-28-5

A lignan found in podophyllin resin from the roots of podophyllum plants. It is a potent spindle poison, toxic if taken internally, and has been used as a cathartic. It is very irritating to skin and mucous membranes, has keratolytic actions, has been used to…

Kategori:
Antimitotic AgentsAntineoplastic Agents, PhytogenicAntiviral Agents +11
Target Protein:
DNA topoisomerase 2-betaTubulin alpha-4A chainTubulin beta chain +1
Waktu Paruh1.0 to 4.5 hours.
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Podophyllin Approved DB09094
small molecule | CAS: 9000-55-9

Podophyllin is a resin extracted from the roots of _Podophyllum peltatum_ (American mandrake) and _Podophyllum emodi_, which contains numerous compounds, amongst which is podophyllin (as well as the drug [podophyllotoxin]). Podophyllin is the principal active…

Kategori:
Antineoplastic AgentsAntineoplastic Agents, PhytogenicBiological Products +11
Waktu ParuhNo data available.
Vol. DistribusiNo data available.
KlirensNo data available.
Genetik -
Polaprezinc DB09221
small molecule | CAS: 107667-60-7

Polaprezinc is a chelated form of zinc and L-carnosine. It is a zinc-related medicine approved for the first time in Japan, which has been clinically used to treat gastric ulcers [L1307, L1308]. It was determined that polaprezinc may be effective in pressure…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Ulcer AgentsDipeptides +10
Target Protein:
Tumor necrosis factorInterleukin-6Interleukin-3 +5
Waktu ParuhThe half-life of po…
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Polatuzumab vedotin Approved DB12240
biotech | CAS: 1313206-42-6

Polatuzumab vedotin is a CD79b-directed antibody-drug conjugate that delivers monomethyl auristatin E (MMAE), an anti-mitotic agent, to cancer cells.[L6658] The drug consists of three components - a humanized immunoglobulin G1 (IgG1) monoclonal antibody speci…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +22
Target Protein:
B-cell antigen receptor complex-associated protein beta chain
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe estimated centr…
KlirensThe predicted clear…
Genetik -
Poldine DB13507
small molecule | CAS: 596-50-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +7
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Polidocanol Approved DB06811
small molecule | CAS: 9002-92-0

Polidocanol is a sclerosing agent indicated to treat uncomplicated spider veins (varicose veins ?1 mm in diameter) and uncomplicated reticular veins (varicose veins 1 to 3 mm in diameter) in the lower extremity. It is marketed under the brand names Asclera an…

Kategori:
AlcoholsAntivaricose TherapyCardiovascular Agents +18
Waktu ParuhThe half-life is ap…
Vol. DistribusiWhen given intraven…
KlirensSytemic clearance w…
Genetik -
Polihexanide Approved DB12277
small molecule | CAS: 28757-47-3

Polihexanide has been used in trials studying the treatment, prevention, and supportive care of Caries, Neoplasm, Skin Diseases, Nail Diseases, and Dental Plaque, among others.

Kategori:
AmidinesAnti-Infective AgentsAntiseptics and Disinfectants +7
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biotech

Deskripsi belum tersedia.

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biotech

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biotech

Poliovirus type 1 antigen is a suspension of poliovirus Type 1 (Mahoney) used in the active immunization of infants (as young as 6 weeks of age), children, and adults for the prevention of poliomyelitis caused by poliovirus Type 1. The vaccine contains purifi…

Kategori:
Actively Acquired ImmunityInactivated Poliovirus Vaccine
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biotech

Polistes fuscatus venom protein is an extract of Polistes fuscatus venom. Polistes fuscatus venom protein is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +3
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Poloxalene DB11451
small molecule | CAS: 691397-13-4

Ethylene oxide/propylene oxide copolymer is used as a food additive. It belongs to the family of Epoxides. These are compounds containing a cyclic ether with three ring atoms (one oxygen and two carbon atoms).

Kategori:
AlcoholsAnti-Infective AgentsCompounds used in a research, industrial, or household setting +8
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Poloxamer 237 DB16553
small molecule

Deskripsi belum tersedia.

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Poloxamer 407 DB11252
small molecule | CAS: 691397-13-4

Poloxamer 407 is a polyoxyethylene polymer and hydrophilic non-ionic surfactant. It consists of a central hydrophobic block of polypropylene glycol that is flanked on each side by polyethylene glycol blocks, both hydrophilic in nature. Poloxamer 407 is used a…

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +9
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Poloxamine 1304 DB19167
small molecule | CAS: 11111-34-5

Poloxamine 1304 is under investigation in clinical trial NCT00483795 (Pilot Evaluation of Two Multipurpose Solutions in Regards to Corneal Staining).

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small molecule | CAS: 26811-96-1

Poly(lactic acid) is under investigation in clinical trial NCT00126308 (Facial Lipoatrophy Trial: Immediate Versus Deferred Injections of Poly-L-Lactic Acid for HIV Facial Lipoatrophy).

Kategori:
Dental ImplantsMacromolecular SubstancesPolymers
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small molecule | CAS: 9003-05-8

Polyacrylamide (crosslinked; 2 mole percent bisacrylamide) is under investigation in clinical trial NCT00629083 (Bulking Agents for the Treatment of Stress Urinary Incontinence in Females).

Kategori:
Biocompatible MaterialsColloidsComplex Mixtures +6
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small molecule | CAS: 133029-32-0

Deskripsi belum tersedia.

Kategori:
AmidinesGuanidinesPreservatives, Pharmaceutical
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