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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 195 / 272
small molecule | CAS: 373-44-4

Deskripsi belum tersedia.

Kategori:
AminesPolyamines
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxypeptidase A1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Octasulfur Approved DB09353
small molecule | CAS: 10544-50-0

Sulfur is a chemical element that is present in all living tissues. The most commonly used form of pharmaceutical sulfur is Octasulfur (S8). After calcium and phosphorus, it is the third most abundant mineral in the human body. Sulfur is also found in garlic,…

Kategori:
ChalcogensElementsKeratolytic Agents
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Octinoxate Approved DB09496
small molecule | CAS: 5466-77-3

Octinoxate is a cinnamate ester and common ingredient in sunscreen and other skin care products to minimize DNA photodamage. It was originally developed in 1950's as an organic UV-B filter that absorbs UV-B rays from sun. It is often combined with nanoparticl…

Kategori:
Acids, CarbocyclicCompounds used in a research, industrial, or household settingCosmetics +8
Waktu Paruh-
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Genetik -
Octisalate Approved DB11062
small molecule | CAS: 118-60-5

Also known as Ethylhexyl Salicylate. Octyl salicylate is an oil soluble chemical sunscreen agent that absorbs UVB radiation. It does not protect against UVA. Octyl salicylate is used to augment the UVB protection in a sunscreen. Salicylates are weak UVB absor…

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Octocrylene Approved DB09535
small molecule | CAS: 6197-30-4

Octocrylene is a compound often used as an additive in sun screen, and is thought to have skin moisturizing effects because of its emollient properties. What makes this chemical such a popular additive to sun block, is its ability to neutralize UV radiation d…

Kategori:
Acids, AcyclicSunscreen Agents
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
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Genetik -
OCTODRINE DB19374
small molecule | CAS: 543-82-8

Deskripsi belum tersedia.

Kategori:
AlkanesHydrocarbons, Acyclic
Waktu Paruh-
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Octopamine DB13251
small molecule | CAS: 104-14-3

Octopamine is structurally similar to norepinephrine. It has been used as a nootropic, and therefore it and all of its enantiomer are prohibited by the World Anti-doping Agency (WADA) as of 2014.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-Agonists +16
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Octreotide Approved DB00104
biotech | CAS: 83150-76-9

Acromegaly is a disorder caused by excess growth hormone (GH), increasing the growth of body tissues and causing metabolic dysfunction.[L14501] In most cases, it results from an anterior pituitary growth hormone-releasing tumor. Typically, the feet, hands, an…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Hormonal +19
Target Protein:
Somatostatin receptor type 2Somatostatin receptor
Waktu ParuhAfter a subcutaneou…
Vol. DistribusiIn a pharmacokineti…
KlirensThe total body clea…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Histo-blood group ABO system transferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Histo-blood group ABO system transferase
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aquaporin Z
Waktu Paruh-
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Genetik -
Octyldodecanol DB14134
small molecule | CAS: 5333-42-6

Deskripsi belum tersedia.

Kategori:
AlcoholsLipids
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 9036-19-5

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAlcoholsAntifoaming Agents +21
Target Protein:
Troponin C, skeletal muscle
Waktu Paruh-
Vol. Distribusi-
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Genetik -
OCU-100 DB17853
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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OCU400 DB18277
biotech

OCU400 is a novel gene therapy comprising an adeno-associated viral vector expressing human nuclear hormone receptor subfamily 2 group E member 3 (hNR2E3).

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OCU410ST DB18326
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Odalasvir DB13041
small molecule | CAS: 1415119-52-6

Odalasvir has been used in trials studying the treatment of Hepatitis C, Chronic and Chronic Hepatitis C Infection.

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiviral Agents +1
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Odanacatib DB06670
small molecule | CAS: 603139-19-1

Odanacatib is an inhibiter of cathepsin K which was originally developed be Merck & Co as a new treatment for osteoporosis [A19388]. The drug made it to phase III trials before abandoned due to increased stroke.

Kategori:
Benzene DerivativesCytochrome P-450 CYP2C8 SubstratesCytochrome P-450 CYP3A Substrates +3
Target Protein:
Cathepsin K
Waktu ParuhApparent half life …
Vol. Distribusi100L [A19391]
KlirensTotal clearance of …
Genetik -
Odesivimab Approved DB15900
biotech | CAS: 2135632-30-1

Ebola virus (EBOV) remains an important human pathogen within the _Ebolavirus_ genus, having been responsible for at least 17 known outbreaks with an average case fatality rate of 43.92%.[A221825] Immune therapy using monoclonal antibodies (mAbs) is becoming …

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +10
Target Protein:
Envelope glycoprotein
Waktu ParuhOdesivimab administ…
Vol. DistribusiOdesivimab administ…
KlirensOdesivimab administ…
Genetik -
Odetiglucan DB17468
biotech | CAS: 53238-80-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Odevixibat Approved DB16261
small molecule | CAS: 501692-44-0

Odevixibat, or A4250, is an ileal sodium/bile acid cotransporter inhibitor indicated for the treatment of pruritus in patients older than 3 months, with progressive familial intrahepatic cholestasis (PFIC).[A236808,L34793] Odevixibat is the first approved non…

Kategori:
Acids, AcyclicAlimentary Tract and MetabolismBenzazepines +9
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu ParuhA 7.2 mg oral dose …
Vol. DistribusiThe majority of adu…
KlirensThe majority of adu…
Genetik -
Odiparcil DB06609
small molecule | CAS: 137215-12-4

Deskripsi belum tersedia.

Kategori:
Carbohydrates
Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ODM-203 DB16843
small molecule | CAS: 1430723-35-5

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
ODM-207 DB18820
small molecule | CAS: 1801503-93-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Genetik -
ODN M362 DB16485
biotech

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19Nucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Target Protein:
Toll-like receptor 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Odronextamab DB16684
biotech | CAS: 1801338-64-6

Odronextamab is a hinge-stabilized, fully human immunoglobulin G4 (IgG4)-based CD20×CD3 bispecific antibody currently evaluated for the treatment of relapsed/refractory (R/R) B-Cell non-Hodgkin lymphoma (NHL).[A254187,A254197] Preliminary studies have shown t…

Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ofatumumab Approved DB06650
biotech | CAS: 679818-59-8

Ofatumumab is a novel anti-CD20 monoclonal antibody that targets B-cells. It is an IgG1? human monoclonal antibody produced from a recombinant murine cell line (NS0) via transgenic mouse and hybridoma technology.[L12612] Ofatumumab works by recognizing antige…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +17
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhIn patients with CL…
Vol. DistribusiIn patients with CL…
KlirensIn patients with CL…
Genetik -
Ofloxacin Approved DB01165
small molecule | CAS: 82419-36-1

A synthetic fluoroquinolone (fluoroquinolones) antibacterial agent that inhibits the supercoiling activity of bacterial DNA gyrase, halting DNA replication.

Kategori:
4-QuinolonesAgents Causing Muscle ToxicityAnti-Bacterial Agents +22
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu Paruh9 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1476737-24-2

Ofranergene obadenovec is under investigation in clinical trial NCT01229865 (Safety and Efficacy of VB-111 in Subjects With Advanced Differentiated Thyroid Cancer).

Waktu Paruh-
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Oglemilast DB12375
small molecule | CAS: 778576-62-8

Oglemilast has been investigated for the treatment of Pulmonary Disease, Chronic Obstructive.

Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4B3',5'-cyclic-AMP phosphodiesterase 4D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oglufanide DB05779
small molecule | CAS: 38101-59-6

Oglufanide is a synthetic dipeptide immunomodulator in development for the treatment of chronic hepatitis C viral infection. Oglufanide was originally developed to treat severe infectious disease in Russia (where it is a registered pharmaceutical), and was ex…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAngiogenesis Modulating Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ohmefentanyl DB01570
small molecule | CAS: 78995-14-9

Ohmefentanyl is an extremely potent opioid analgesic drug which selectively binds to the µ-opioid receptor. The Chinese have recorded ohmefentanyl as having a potency that is 6,300 times morphine. Ohmefentanyl is one of the most potent ? -receptor agonists kn…

Kategori:
AnalgesicsCentral Nervous System AgentsPeripheral Nervous System Agents +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
OKI-179 DB17583
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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Olacaftor DB16262
small molecule | CAS: 1897384-89-2

Olacaftor is under investigation in clinical trial NCT02951182 (A Study Evaluating the Safety and Efficacy of VX-440 Combination Therapy in Subjects With Cystic Fibrosis).

Waktu Paruh-
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Olafertinib DB17179
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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Olaflur DB13290
small molecule | CAS: 6818-37-7

Olaflur which is also referred to as elmex gel is an ingredient used in toothpaste which helps in the prevention of dental caries.

Kategori:
Alimentary Tract and MetabolismAminesAnions +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olanexidine DB16889
small molecule | CAS: 146510-36-3

Deskripsi belum tersedia.

Kategori:
AmidinesGuanidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olanzapine Approved DB00334
small molecule | CAS: 132539-06-1

Olanzapine is a thienobenzodiazepine classified as an atypical or second-generation antipsychotic agent.[A176996] The second-generation antipsychotics were introduced in the 90s and quickly gained traction due to their impressive efficacy, reduced risk for ex…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +50
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorD(1A) dopamine receptor +17
Gen Terkait:
HTR1A
Waktu ParuhOlanzapine presents…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik 1 Varian
Olaparib Approved DB09074
small molecule | CAS: 763113-22-0

Olaparib is a selective and potent inhibitor of poly (ADP-ribose) polymerase (PARP) enzymes, PARP1 and PARP2.[L41100, L40908, L43792] PARP inhibitors represent a novel class of anti-cancer therapy and they work by taking advantage of a defect in DNA repair in…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +38
Target Protein:
Poly [ADP-ribose] polymerase 1Poly [ADP-ribose] polymerase 2Protein mono-ADP-ribosyltransferase PARP3 +1
Waktu ParuhFollowing a single …
Vol. DistribusiThe mean (± standar…
KlirensFollowing a single …
Genetik -
small molecule | CAS: 1380359-84-1

Olaparib-bodipy FL is under investigation in clinical trial NCT03085147 (A Dye for the Detection of Cancer of the Tongue and Mouth).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Olaptesed Pegol DB11707
small molecule | CAS: 1390628-22-4

Olaptesed Pegol has been investigated for the treatment of Hematopoietic Stem Cell Transplantation.

Kategori:
Pegylated agents
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Olaratumab Approved DB06043
biotech | CAS: 1024603-93-7

Olaratumab (IMC-3G3) is a fully human IgG1 monoclonal antibody with antitumor activity that selectively binds the external domain of human platelet-derived growth factor receptor (PDGFR)-? with high affinity and blocks ligand binding. It is composed of two he…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Platelet-derived growth factor receptor alpha
Waktu ParuhEstimated value of …
Vol. Distribusi7.7 L at steady sta…
KlirensMean value of 0.56L…
Genetik -
Olea europaea pollen Approved DB10378
biotech

Olea europaea pollen is the pollen of the Olea europaea plant. Olea europaea pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oleandomycin DB11442
small molecule | CAS: 3922-90-5

Oleandomycin is a macrolide antibiotic, though it is less effective than erythromycin. It is synthesized from strains of _Streptomyces antibioticus_.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oleandrin DB12843
small molecule | CAS: 465-16-7

Oleandrin has been used in trials studying the treatment of Lung Cancer and Chemotherapeutic Agent Toxicity.

Kategori:
CardanolidesCardiac GlycosidesFused-Ring Compounds +2
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1Sodium/potassium-transporting ATPase subunit alpha-2Sodium/potassium-transporting ATPase subunit alpha-3 +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oleclumab DB15088
biotech | CAS: 1803176-05-7

Oleclumab is under investigation in clinical trial NCT03819465 (A Study of Novel Anti-cancer Agents in Patients With Previously Untreated NSCLC).

Waktu Paruh-
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Genetik -
biotech | CAS: 2096510-84-6

Olenasufligene relduparvovec is under investigation in clinical trial NCT03612869 (Study of aavrh10-h.sgsh Gene Therapy in Patients With Mucopolysaccharidosis Type IIIA (MPS IIIA)). It is an adeno-associated virus (AAV) vector that delivers a functional copy …

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Olendalizumab DB14834
biotech | CAS: 1337966-73-0

Olendalizumab is under investigation in clinical trial NCT01883544 (Study to Evaluate the Safety, Tolerability, Pharmacokinetics, and Pharmacodynamics of ALXN1007 in Healthy Male and Female Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oleoyl-estrone DB04870
small molecule | CAS: 180003-17-2

Oleoyl-estrone (OE) is a fatty acid ester of estrone. This hormone occurs naturally and is found circulating in various animal species and humans. It has been shown in animal studies to promote the loss of body fat while maintaining body protein storage, main…

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAnti-Obesity Agents +15
Target Protein:
Metabotropic glutamate receptor 3Metabotropic glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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