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14063

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Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
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14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 195 / 282
NAV 1800 DB05437
biotech

RIGScan CR49, a 125I-labelled CR monoclonal antibody directed against the tumour-associated antigen TAG-72, is undergoing development with Neoprobe for the intraoperative detection of metastatic colorectal cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Navafenterol DB19195
small molecule | CAS: 1435519-06-4

Navafenterol is under investigation in clinical trial NCT02971293 (Efficacy, Pharmacokinetics (PK), Safety and Tolerability Study of Inhaled AZD8871).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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Navarixin DB11711
small molecule | CAS: 473727-83-2

Navarixin has been investigated for the treatment of Asthma.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +4
Waktu Paruh-
Vol. Distribusi-
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Naveglitazar DB12662
small molecule | CAS: 476436-68-7

Naveglitazar has been used in trials studying the treatment of Diabetes Mellitus, Non-Insulin-Dependent.

Kategori:
Acids, CarbocyclicPPAR alpha, agonistsPPAR gamma, agonists
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Navicixizumab DB12634
biotech | CAS: 1638338-43-8

Navicixizumab is under investigation in clinical trial NCT02298387 (A Phase 1 Study of Navicixizumab in Subjects With Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
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Navitoclax DB12340
small molecule | CAS: 923564-51-6

Navitoclax has been used in trials studying the treatment and basic science of Solid Tumors, Non-Hodgkin's Lymphoma, EGFR Activating Mutation, Chronic Lymphoid Leukemia, and Hematological Malignancies, among others. Navitoclax is an orally bioavailable sma…

Kategori:
AmidesAminesAntineoplastic Agents +3
Target Protein:
Bcl-2-like protein 1G1/S-specific cyclin-D1Apoptosis regulator Bcl-2 +2
Waktu Paruh-
Vol. Distribusi-
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Navocaftor DB19039
small molecule | CAS: 2159103-66-7

Navocaftor is under investigation in clinical trial NCT04853368 (Study to Evaluate Adverse Events and Change in Disease Activity With Oral Capsules of Galicaftor/navocaftor/abbv-119 or Galicaftor/navocaftor/abbv-576 Combination Therapies in Adult Participants…

Waktu Paruh-
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Navoximod DB15439
small molecule | CAS: 1402837-78-8

Navoximod is under investigation in clinical trial NCT02048709 (Indoleamine 2,3-Dioxygenase (IDO) Inhibitor in Advanced Solid Tumors).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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Navtemadlin DB15299
small molecule | CAS: 1352066-68-2

Navtemadlin (AMG-232) is under investigation in clinical trial NCT03041688 (MDM2 Inhibitor AMG-232 and Decitabine in Treating Patients With Relapsed, Refractory, or Newly-Diagnosed Acute Myeloid Leukemia).

Kategori:
Acids, AcyclicAntineoplastic AgentsFatty Acids +3
Target Protein:
E3 ubiquitin-protein ligase Mdm2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Navuridine DB17759
small molecule | CAS: 84472-85-5

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesDideoxynucleosidesNucleic Acids, Nucleotides, and Nucleosides +3
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
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Naxifylline DB06471
small molecule | CAS: 166374-49-8

Deskripsi belum tersedia.

Kategori:
Adenosine A1 Receptor AntagonistsAlkaloidsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Naxitamab Approved DB15965
biotech | CAS: 1879925-92-4

Naxitamab (humanized 3F8, hu3F8) is an IgG1 monoclonal antibody directed against the oncofetal differentiation antigen GD2 disialoganglioside.[L24454,A224604] Normally expressed during fetal development and in mature neurons, pain fibers, and skin cells, GD2 …

Kategori:
Agents that produce hypertensionAmino Acids, Peptides, and ProteinsAntibodies +18
Target Protein:
GD2 disialoganglioside
Waktu ParuhThe mean terminal h…
Vol. Distribusi-
KlirensThe clearance of na…
Genetik -
Nazartinib DB16250
small molecule | CAS: 1508250-71-2

Nazartinib is under investigation in clinical trial NCT03529084 (Phase III Study of Nazartinib (EGF816) Versus Erlotinib/gefitinib in First-line Locally Advanced / Metastatic NSCLC With EGFR Activating Mutations).

Kategori:
AlkaloidsAntineoplastic AgentsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NB-001 DB12716
small molecule | CAS: 686301-48-4

NB-001 has been investigated for the treatment of Recurrent Herpes Labialis.

Kategori:
Adenine NucleotidesAdenylyl Cyclase InhibitorsEnzyme Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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NB-124 sulfate DB16951
small molecule | CAS: 1375073-96-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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NBI-6024 DB05819
biotech

NBI-6024 is an altered peptide ligand that is designed to cause an immune response which result in preservation of beta-cell function and endogenous insulin production.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +3
Waktu Paruh-
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NBI-98782 Approved DB16905
small molecule | CAS: 85081-18-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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NBL-015 DB18183
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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NC-6300 DB17341
small molecule

NC-6300, also known as K-912, is a novel [epirubicin] drug-conjugated polymeric micelle.

Kategori:
Amino Acids, Peptides, and ProteinsAminoglycoside AntibacterialsAnthracyclines +5
Waktu Paruh-
Vol. Distribusi-
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NCATS-BL0746 DB18322
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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NCX 1015 DB05825
small molecule

NCX 1015 is nitric oxide-releasing derivative of prednisolone developed for the treatment of inflammatory bowel disease (IBD) by NicOx SA.

Kategori:
Fused-Ring CompoundsPregnadienesPregnadienetriols +2
Waktu Paruh-
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NCX 1022 DB05410
small molecule | CAS: 571186-50-0

NCX is an NO-releasing derivative of hydrocortisone.

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +8
Waktu Paruh-
Vol. Distribusi-
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NCX 950 DB05849
small molecule

NCX 950, beta2-adrenoceptor agonists is widely used in the treatment of pulmonary diseases.

Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
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NCX-1000 DB16026
small molecule | CAS: 401519-96-8

NCX-1000 is under investigation in clinical trial NCT00414869 (Preliminary Efficacy and Tolerability of NCX-1000 After Repeated Oral Doses in Patients With Elevated Portal Pressure).

Kategori:
AnionsBile Acids and SaltsCholanes +6
Waktu Paruh-
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ND1251 DB05132
small molecule

ND1251 is an orally active phosphodiesterase-4 (PDE4) inhibitor, a mechanism clinically proven to play a role in alleviating symptoms of depression. ND1251 is a very potent compound with a large safety margin. ND1251 may also have applications in other disord…

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ND7001 DB05142
small molecule

ND7001, a selective PDE2 inhibitor is in clinical trials for the treatment of depression. ND7001 is a solid. Known drug targets of ND7001 including phosphodiesterase 2A, cGMP-stimulated and cGMP-dependent 3',5'-cyclic phosphodiesterase. It is a new type of an…

Target Protein:
cGMP-dependent 3',5'-cyclic phosphodiesterase
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Ornithine carbamoyltransferase chain I
Waktu Paruh-
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NDI-5001 DB17609
small molecule | CAS: 1365571-66-9

Deskripsi belum tersedia.

Waktu Paruh-
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NE-180 DB05619
small molecule

NE-180 was under investigation in a clinical trial conducted in the European Union.

Waktu Paruh-
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Neamine DB04808
small molecule | CAS: 3947-65-7

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +3
Waktu Paruh-
Vol. Distribusi-
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Nebicapone DB14849
small molecule | CAS: 274925-86-9

Nebicapone is under investigation in clinical trial NCT03097211 (Effect of BIA 6-512 at Steady-state on the Levodopa Pharmacokinetics With a Single-dose of Levodopa/Benserazide 200/50 mg or With a Single-dose of Levodopa/Benserazide 200/50 mg Plus a Single-do…

Kategori:
COMT InhibitorsKetones
Target Protein:
Catechol O-methyltransferase
Waktu Paruh-
Vol. Distribusi-
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Nebivolol Approved DB04861
small molecule | CAS: 118457-14-0

Nebivolol is a racemic mixture of 2 enantiomers where one is a beta adrenergic antagonist and the other acts as a cardiac stimulant without beta adrenergic activity.[A182579] Treatment with nebivolol leads to a greater decrease in systolic and diastolic blood…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor
Waktu Paruhd-nebivolol has a h…
Vol. DistribusiFor a 20mg dose, d-…
KlirensFor a 20mg dose, th…
Genetik -
Necuparanib DB16251
small molecule | CAS: 1415139-34-2

Necuparanib is under investigation in clinical trial NCT01621243 (M402 in Combination With Nab-paclitaxel and Gemcitabine in Pancreatic Cancer).

Waktu Paruh-
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Nedaplatin Approved DB13145
small molecule | CAS: 95734-82-0

Nedaplatin is a second generation platinum analog [A20300]. It is less nephrotoxic than [DB00515] but has proven equally effective. It was approved for use in Japan in 1995.

Kategori:
Antineoplastic AgentsDrugs that are Mainly Renally ExcretedDrugs that are Mainly Renally Excreted with a Narrow Therapeutic Index +3
Target Protein:
DNAGlutathione
Waktu Paruh-
Vol. DistribusiThe volume of distr…
KlirensClearance of the fr…
Genetik -
Nedisertib DB16252
small molecule | CAS: 1637542-33-6

Nedisertib is under investigation in clinical trial NCT03770689 (Study of M3814 in Combination With Capecitabine and Radiotherapy in Rectal Cancer).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
DNA-dependent protein kinase catalytic subunit
Waktu Paruh-
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Nedocromil Approved DB00716
small molecule | CAS: 69049-73-6

A pyranoquinolone derivative that inhibits activation of inflammatory cells which are associated with asthma, including eosinophils, neutrophils, macrophages, mast cells, monocytes, and platelets.

Kategori:
4-QuinolonesAnti-Allergic AgentsAnti-Asthmatic Agents +16
Target Protein:
Cysteinyl leukotriene receptor 1Cysteinyl leukotriene receptor 2fMet-Leu-Phe receptor +2
Waktu Paruh~3.3 hours
Vol. Distribusi-
Klirens-
Genetik -
Nedometinib DB18102
small molecule | CAS: 2252314-46-6

Deskripsi belum tersedia.

Waktu Paruh-
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Nedosiran Approved DB17635
biotech | CAS: 2266591-83-5

Nedosiran is an RNA interference targeting hepatic lactate dehydrogenase, the enzyme responsible for the conversion of glyoxylate to oxalate.[A261690] Oxalate, particularly calcium oxalate, precipitation is the main cause of kidney stones formation; therefore…

Target Protein:
L-lactate dehydrogenase A chain
Waktu ParuhThe half-life of ne…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ne…
Genetik -
Nefazodone Approved DB01149
small molecule | CAS: 83366-66-9

Nefazodone hydrochloride (trade name Serzone) is an antidepressant drug marketed by Bristol-Myers Squibb. Its sale was discontinued in 2003 in some countries, due to the small possibility of hepatic (liver) injury. Drug-induced hepatic injuries were associate…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +44
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2CSodium-dependent serotonin transporter +7
Waktu Paruh2-4 hours
Vol. Distribusi* 0.22 to 0.87 L/kg
Klirens-
Genetik -
Nefiracetam DB13082
small molecule | CAS: 77191-36-7

Nefiracetam has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCompounds used in a research, industrial, or household setting +5
Waktu Paruh-
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Neflamapimod DB07138
small molecule | CAS: 209410-46-8

Neflamapimod has been used in trials studying the treatment of Alzheimer's Disease and Mild Cognitive Impairment.

Target Protein:
Mitogen-activated protein kinase 11Mitogen-activated protein kinase 12Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
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Nefopam Approved DB12293
small molecule | CAS: 13669-70-0

Nefopam is under investigation for the prevention of Cholecystitis and Post Anaesthetic Shivering. Nefopam has been investigated for the prevention of Kidney Transplantation.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAzocines +5
Waktu Paruh-
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Neihulizumab DB16698
biotech

Neihulizumab is a novel immune checkpoint agonistic antibody that binds to human CD162 (PSGL-1), thereby preferentially inducing apoptosis in late stage activated T cells.[L34450]

Target Protein:
P-selectin glycoprotein ligand 1
Waktu Paruh-
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Genetik -
biotech

Neisseria meningitidis group a capsular oligosaccharide diphtheria crm197 protein conjugate antigen is a vaccine.

Kategori:
Actively Acquired ImmunityInactivated Meningococcal Vaccine
Waktu Paruh-
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biotech

Neisseria meningitidis group c capsular oligosaccharide diphtheria crm197 protein conjugate antigen is a vaccine.

Kategori:
Actively Acquired ImmunityInactivated Meningococcal Vaccine
Waktu Paruh-
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biotech

Neisseria meningitidis group w-135 capsular oligosaccharide diphtheria crm197 protein conjugate antigen is a vaccine.

Kategori:
Actively Acquired ImmunityInactivated Meningococcal Vaccine
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biotech

Neisseria meningitidis serogroup B recombinant lp2086 a05 protein variant antigen is a sterile vaccine for intramuscular injection indicated for the active immunization to prevent invasive disease caused by *Neisseria meningitidis* serogroup B. It is containe…

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biotech

Neisseria meningitidis serogroup b recombinant lp2086 b01 protein variant antigen is a sterile vaccine for intramuscular injection indicated for the active immunization to prevent invasive disease caused by *Neisseria meningitidis* serogroup B. It is containe…

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Genetik -
biotech

Deskripsi belum tersedia.

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