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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 195 / 321
biotech | CAS: 1703749-62-5

Lutetium Lu-177 vipivotide tetraxetan is a radioligand therapeutic agent. It consists of a radionuclide, [lutetium Lu-177], linked to a moiety that binds to PSMA, a transmembrane protein that is expressed in prostate cancer.[L41280] Lutetium Lu-177 vipivot…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic Uses of ChemicalsRadioactive Therapeutic Agent +6
Target Protein:
Prostate-specific antigen
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 321835-55-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lutikizumab DB16224
biotech | CAS: 1791411-57-8

Lutikizumab is under investigation in clinical trial NCT02087904 (A Study Evaluating the Safety, Efficacy, and Pharmacodynamic Effects of ABT-981 in Patients With Knee Osteoarthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lutropin alfa Approved DB00044
biotech | CAS: 152923-57-4

Lutropin alfa is a recombinant human luteinizing hormone produced in yeast with 2 subunits, alpha = 92 residues, beta = 121 residues. It is a heterodimeric glycoprotein made up of monomeric units. Lutropin alfa was the first and only recombinant human form of…

Kategori:
Genito Urinary System and Sex HormonesGonadotropinsGonadotropins and Antigonadotropins +1
Target Protein:
Lutropin-choriogonadotropic hormone receptor
Waktu ParuhBiphasic; terminal …
Vol. DistribusiThe steady state vo…
Klirens* 2 – 3 L/h [health…
Genetik -
Luvadaxistat DB16067
small molecule | CAS: 1425511-32-5

Luvadaxistat is under investigation in clinical trial NCT03214588 (Efficacy, Tolerability, and Pharmacokinetics of Multiple Doses of Oral TAK-831 in Adults With Friedreich Ataxia).

Kategori:
D-Amino Acid Oxidase Inhibitor
Target Protein:
D-amino-acid oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Luveltamab tazevibulin, formerly known as STRO-002, is novel homogeneous folate receptor alpha (FolR?) targeting antibody-drug conjugate.[A257414] It is under investigation in clinical trial NCT05200364 (A Study of STRO-002, an Anti-folate Receptor Alpha Anti…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luvixasertib DB19200
small molecule | CAS: 1610759-22-2

Luvixasertib is under investigation in clinical trial NCT05251714 (CFI-402257, a Potent and Selective TTK Inhibitor, in Solid Tumors and With Fulvestrant in Breast Cancer).

Waktu Paruh-
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Luxeptinib DB19179
small molecule | CAS: 1616428-23-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LV-FAH DB17686
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

LV-SMENP-DC is a vaccine candidate being developed by Shenzhen Geno-Immune Medical Institute that comprises dendritic cells that are modified with lentiviral vector-expressing synthetic minigene which are based on domains of selected viral proteins. This vacc…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LV305 DB17288
biotech

LV305 is a lentiviral vector encoding NY-ESO-1 gene. LV305 is an active component of CMB305 along with [G305].[L47346]

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LX-1004 DB18272
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LX-2931 DB06297
small molecule | CAS: 948840-25-3

Deskripsi belum tersedia.

Kategori:
AminesHydroxylamines
Target Protein:
Sphingosine-1-phosphate lyase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LX-7101 DB16009
small molecule | CAS: 1192189-69-7

LX-7101 is under investigation in clinical trial NCT01528111 (Study to Evaluate the Safety, Tolerability, and Efficacy of LX7101 in Subjects With Primary Open-angle Glaucoma or Ocular Hypertension).

Waktu Paruh-
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LX1031 DB05199
small molecule

LX1031 is an orally-dosed drug candidate for irritable bowel syndrome and other gastrointestinal disorders. LX1031 was generated by Lexicon medicinal chemists, and its target was internally identified as a key control point for the regulation of peripheral se…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +3
Target Protein:
Tryptophan 5-hydroxylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2090314 DB11913
small molecule | CAS: 603288-22-8

Ly2090314 has been used in trials studying the treatment of Leukemia, Advanced Cancer, and Pancreatic Cancer.

Kategori:
Acids, AcyclicDicarboxylic AcidsGlycogen Synthase Kinase 3, antagonists & inhibitors +3
Target Protein:
Glycogen synthase kinase-3 alphaGlycogen synthase kinase-3 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2183240 DB17035
small molecule | CAS: 874902-19-9

LY-2183240 is an inhibitor of endocannabinoid reuptake/breakdown.[A253037]

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LY-2300559 DB13016
small molecule | CAS: 889116-06-7

Ly2300559 has been used in trials studying the prevention of Migraine Headache.

Kategori:
Acids, CarbocyclicBenzene DerivativesKetones
Target Protein:
Metabotropic glutamate receptor 2Cysteinyl leukotriene receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2334737 DB12906
small molecule | CAS: 892128-60-8

LY2334737 has been used in trials studying the treatment of Solid Tumor, Metastatic Tumor, and Malignant Solid Tumor.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2452473 DB12573
small molecule | CAS: 1029692-15-6

Ly2452473 is under investigation for the supportive care of Prostate Cancer. Ly2452473 has been investigated for the treatment of Erectile Dysfunction.

Kategori:
Acids, Acyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2584702 DB12690
small molecule | CAS: 1082949-67-4

LY2584702 has been used in trials studying the treatment of Cancer, Advanced Cancer, Renal Cell Carcinoma, Metastases, Neoplasm, and Neuroendocrine Tumors, among others.

Kategori:
Ribosomal Protein S6 Kinases, 70-kDa, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2599506 DB05970
small molecule | CAS: 745051-65-4

LY2599506 was under investigation in clinical trials NCT01024244 and NCT01029795 for the treatment of patients with type 2 diabetes.

Target Protein:
Hexokinase-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2608204 DB12284
small molecule | CAS: 1234703-40-2

LY2608204 has been used in trials studying the treatment of Diabetes Mellitus, Type 2.

Kategori:
Enzyme ActivatorsSulfur Compounds
Target Protein:
Hexokinase-4Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2623091 DB15367
small molecule | CAS: 1162264-07-4

LY-2623091 is under investigation in clinical trial NCT02194465 (A Study of LY2623091 in Participants With High Blood Pressure).

Target Protein:
Mineralocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2624803 DB15092
small molecule | CAS: 879409-35-5

LY-2624803 is under investigation in clinical trial NCT01236105 (Effect of Activated Charcoal and Time of Dose on the Pharmacokinetics of LY2624803 in Healthy Subject).

Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2811376 DB13065
small molecule | CAS: 1194044-20-6

LY2811376 has been used in trials studying the basic science of Alzheimer's Disease.

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2874455 DB13022
small molecule | CAS: 1254473-64-7

LY2874455 has been used in trials studying the treatment of Advanced Cancer.

Kategori:
Heterocyclic Compounds, Fused-RingPyrazolesReceptors, Fibroblast Growth Factor, antagonists & inhibitors
Target Protein:
Fibroblast growth factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2881835 DB15046
small molecule | CAS: 1292290-38-0

LY-2881835 is under investigation in clinical trial NCT01358981 (A Study of LY2881835 in Healthy People and People With Diabetes).

Target Protein:
Free fatty acid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2886721 DB12547
small molecule | CAS: 1262036-50-9

LY2886721 has been used in trials studying the basic science of Alzheimer's Disease.

Kategori:
Heterocyclic Compounds, Fused-RingPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-294002 DB02656
small molecule | CAS: 154447-36-6

Specific inhibitor of phosphatidylinositol 3-kinase.

Kategori:
BenzopyransEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase pim-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-295501 DB12574
small molecule | CAS: 150869-74-2

ILX-295501 has been used in trials studying the treatment of Ovarian Cancer, Metastatic Cancer, Fallopian Tube Cancer, and Primary Peritoneal Cavity Cancer.

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-3023414 DB12167
small molecule | CAS: 1386874-06-1

LY3023414 has been used in trials studying the treatment of Neoplasm, Solid Tumor, COLON CANCER, BREAST CANCER, and Advanced Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-3039478 DB12050
small molecule | CAS: 1421438-81-4

LY3039478 has been used in trials studying the treatment and basic science of LYMPHOMA, Neoplasms, Solid Tumor, COLON CANCER, and BREAST CANCER, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Neurogenic locus notch homolog protein 4Neurogenic locus notch homolog protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-3200882 DB16064
small molecule | CAS: 1898283-02-7

LY-3200882 is under investigation in clinical trial NCT04158700 (A Study of LY3200882 and Pembrolizumab in Participants With Advanced Cancer).

Target Protein:
TGF-beta receptor type-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-3499446 DB17486
small molecule | CAS: 2409131-50-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-377604 DB12858
small molecule | CAS: 204592-94-9

Ly377604 has been used in trials studying the treatment of Obesity.

Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-517717 DB05713
small molecule | CAS: 313489-71-3

LY517717 is an investigational oral direct inhibitor of activated Factor Xa. It is believed to be Lilly's PMD-3112 (licensed from Amgen).

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-518674 DB12988
small molecule | CAS: 425671-29-0

LY518674 has been used in trials studying the treatment of Metabolic Syndrome X.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY2181308 DB05141
small molecule

LY2181308 is investigated in clinical trials for treating solid tumors. LY2181308 is a solid. LY2181308 is directed against a molecular target called survivin. LY2181308 is known to target baculoviral IAP repeat-containing protein 5. LY2181308 is an anti-sens…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Baculoviral IAP repeat-containing protein 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY2275796 DB05165
small molecule

LY2275796 is a second-generation antisense anti-cancer drug candidate for clinical development. LY2275796 targets eukaryotic initiation factor- 4E (eIF-4E), a protein involved in the translation of key growth and survival factors that drive tumor progression,…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
Eukaryotic translation initiation factor 4E
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY2828360 DB16074
small molecule | CAS: 1231220-79-3

LY2828360 is under investigation in clinical trial NCT01319929 (A Study of LY2828360 in Patients With Osteoarthritic Knee Pain).

Kategori:
Cannabinoid Receptor AgonistsCannabinoids and similarsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY3884961 DB17070
biotech

LY3884961 (previously PR001) is being developed by Prevail Therapeutics as a single-dose gene therapy for patients with Parkinson's disease and Gaucher disease.[L43468]

Waktu Paruh-
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Genetik -
Lycopene Approved DB11231
small molecule | CAS: 502-65-8

Lycopene is a naturally occurring red carotenoid pigment that is responsible for red to pink colors seen in tomatoes, pink grapefruit, and other foods [A27242]. Having a chemical formula of C40H56, lycopene is a tetraterpene assembled from eight isoprene unit…

Kategori:
AlkenesAnti-Inflammatory AgentsAnticarcinogenic Agents +13
Waktu Paruh-
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Genetik -
Lym-1-I-131 DB17445
biotech

Lym-1-I-131 is a monoclonal antibody labeled with iodine-131 (131I) that preferentially targets malignant lymphocytes.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lymecycline Approved DB00256
small molecule | CAS: 992-21-2

Lymecycline is a broad-spectrum second-generation tetracycline antibiotic used for the treatment of acne and other susceptible bacterial infections.[L13880,L13883] It has been proven a cost-effective alternative to treatment with [minocycline] with comparable…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
30S ribosomal protein S4
Waktu ParuhThe half-life of ly…
Vol. DistribusiLymecycline is lipo…
KlirensLymecycline is part…
Genetik -
Lynestrenol Approved DB12474
small molecule | CAS: 52-76-6

Lynestrenol is a progestin and prodrug of [norethisterone].

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lypressin Approved DB14642
small molecule | CAS: 50-57-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntidiuretic AgentsCardiovascular Agents +20
Target Protein:
Vasopressin V1a receptorVasopressin V2 receptorVasopressin V1b receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Lysergic acid 2,4-dimethylazetidide is under investigation in clinical trial NCT02765802 (A Study to Evaluate Pegylated Interferon Lambda Monotherapy in Patients With Chronic Hepatitis Delta Virus Infection).

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Genetik -
small molecule | CAS: 50-37-3

Debate continues over the nature and causes of chronic flashbacks. Explanations in terms of LSD physically remaining in the body for months or years after consumption have been discounted by experimental evidence. Some say HPPD is a manifestation of post-trau…

Kategori:
Agents that produce hypertensionAlkaloidsAntidepressive Agents +18
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2B +1
Waktu Paruh3 hours
Vol. Distribusi-
Klirens-
Genetik -
Lysine Approved DB00123
small molecule | CAS: 56-87-1

Lysine (abbreviated as Lys or K) is an ?-amino acid with the chemical formula HO2CCH(NH2)(CH2)4NH2. This amino acid is an essential amino acid, which means that humans cannot synthesize it. Its codons are AAA and AAG. Lysine is a base, as are arginine and his…

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +10
Target Protein:
High affinity cationic amino acid transporter 1Cationic amino acid transporter 4Cationic amino acid transporter 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9701–9750 dari 16004
Sebelumnya Halaman 195 / 321 Berikutnya