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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 194 / 236
Rivaroxaban Approved DB06228
small molecule | CAS: 366789-02-8

Rivaroxaban is an anticoagulant and the first orally active direct factor Xa inhibitor. Unlike warfarin, routine lab monitoring of INR is not necessary. However there is no antidote available in the event of a major bleed. Only the 10 mg tablet can be taken w…

Kategori:
AnticoagulantsAntithrombinsBCRP/ABCG2 Substrates +17
Target Protein:
Coagulation factor X
Waktu ParuhThe terminal half l…
Vol. DistribusiThe steady state Vd…
KlirensSystemic clearance …
Genetik -
Rivipansel DB12778
small molecule | CAS: 927881-99-0

Rivipansel has been used in trials studying the other, basic science, and treatment of Pain Crisis, Renal impairment, Anemia, Sickle Cell, Sickle Cell Disease, and Sickle Cell Disorders, among others.

Kategori:
CarbohydratesGlycoconjugatesLipids
Target Protein:
E-selectinL-selectinP-selectin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rivoceranib DB14765
small molecule | CAS: 811803-05-1

Rivoceranib is under investigation in clinical trial NCT02726854 (Apatinib as Second-line Treatment of Advanced Pancreatic Cancer).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
RLY-2608 DB16751
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
RLYB212 DB17727
biotech

RLYB212 is a human monoclonal antibody against Antigen-1A Immunoglobulin (HPA-1A). It is currently being developed by Rallybio for the prevention of fetal and neonatal alloimmune thrombocytopenia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ro 12-7310 DB08455
small molecule | CAS: 65316-65-6

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ro 24-7429 DB16062
small molecule | CAS: 139339-45-0

Ro 24-7429 is under investigation in clinical trial NCT00002314 (A Study of Ro 24-7429 in Patients With Hiv-related Kaposi's Sarcoma).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-4584820 DB08094
small molecule | CAS: 741713-40-6

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 1Cyclin-dependent kinase 7 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-4987655 DB12933
small molecule | CAS: 874101-00-5

RO4987655 has been used in trials studying the treatment of Neoplasms.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-5028442 DB12721
small molecule | CAS: 920022-47-5

RO5028442 has been used in trials studying Autistic Disorder.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-5045337 DB14793
small molecule | CAS: 939981-39-2

RO-5045337 is under investigation in clinical trial NCT01164033 (A Study of RO5045337 in Patients With Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-6870810 DB15151
small molecule | CAS: 1349719-98-7

RO-6870810 is under investigation in clinical trial NCT02308761 (A Study of RO6870810/TEN-010 in Participants With Acute Myeloid Leukemia and Myelodysplastic Syndrome).

Kategori:
Sulfur CompoundsThiazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RO-7293583 DB17455
biotech

RO-7293583 is a TYRP1-Targeting CD3 T-Cell Engager.

Waktu Paruh-
Vol. Distribusi-
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RO6953958 DB17081
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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RO7200220 DB18437
biotech

RO7200220 is a recombinant fully humanized anti-IL 6 monoclonal antibody.

Waktu Paruh-
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RO7284755 DB17527
biotech

RO7284755 is an investigational cancer drug: it is a PD-1-targeted IL-2 variant antibody fusion protein. RO7284755 is under investigation in clinical trial NCT04303858 (A Study to Evaluate Safety and Anti-tumor Activity of RO7284755 Alone or in Combination Wi…

Waktu Paruh-
Vol. Distribusi-
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RO7296682 DB17531
biotech

RO7296682 is a monoclonal antibody against CD25 (IL-2R alpha) expressed on tumour-infiltrating regulatory T (T<sub>reg</sub>) cells. RO7296682 is under investigation in clinical trial NCT04642365 (A Study to Evaluate the Safety and Tolerability of RO7296682 i…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
RO7300490 DB17535
biotech

RO7300490 is an investigational Fibroblast Activation Protein-? (FAP) targeted CD40 agonist. RO7300490 is under investigation in clinical trial NCT04857138 (A Study to Evaluate Safety, Pharmacokinetics and Anti-tumor Activity of RO7300490, as Single Agent or …

Waktu Paruh-
Vol. Distribusi-
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Genetik -
RO7502175 DB17502
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Robalzotan DB06538
small molecule | CAS: 169758-66-1

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Robatumumab DB12976
biotech | CAS: 934235-44-6

Robatumumab has been used in trials studying the treatment of Osteosarcoma, Sarcoma, Ewing's, and Peripheral Neuroectodermal Tumor.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Robenidine DB11542
small molecule | CAS: 25875-51-8

Robenidine is identified as a coccidiostat drug, which slows both the growth and reproductive cycles of coccidian parasites. Robenidine is used to control coccidiosis, a lethal infection in poultry which has shown a significant economic burden. Despite the av…

Kategori:
AmidinesAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Robinia pseudoacacia pollen Approved DB10474
biotech

Robinia pseudoacacia pollen is the pollen of the Robinia pseudoacacia plant. Robinia pseudoacacia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roblitinib DB16845
small molecule | CAS: 1708971-55-4

Deskripsi belum tersedia.

Target Protein:
Fibroblast growth factor receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocacetrapib DB15437
small molecule | CAS: 1402796-27-3

Rocacetrapib is under investigation in clinical trial NCT02156544 (Study to Investigate the Safety/Tolerability and Pharmacokinetics/Pharmacodynamics of CKD-519).

Kategori:
Hydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocaglamide DB15495
small molecule | CAS: 84573-16-0

Rocaglamide, also referred to as rocaglamide-A, is the eponymous member of a class of anti-cancer phytochemicals known as rocaglamides.[A186760] Rocaglamides are secondary metabolites of the plant genus _Aglaia_, and extracts of the plant have traditionally b…

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prohibitin 1Transcription factor RelBNuclear factor NF-kappa-B p100 subunit +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2253753-17-0

Rocakinogene sifuplasmid is under investigation in clinical trial NCT03491683 (INO-5401 and INO-9012 Delivered by Electroporation (EP) in Combination With Cemiplimab (REGN2810) in Newly-diagnosed Glioblastoma (GBM)).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocapuldencel-T DB17588
biotech

Rocapuldencel-T is an autologous dendritic cell immunotherapy that was investigated in NCT02662634 (A Safety and Feasibility Study of AGS-003-LNG for the Treatment of Stage 3 Non Small Cell Lung Cancer).

Kategori:
Autologous Cellular Immunotherapy
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocatinlimab DB18809
biotech | CAS: 2431972-52-8

Rocatinlimab is a subcutaneously administered anti-OX40 antibody developed for the treatment of moderate-to-severe atopic dermatitis. In clinical trials, it has shown significant efficacy and safety compared to a placebo. The drug works by targeting the OX40 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Tumor necrosis factor receptor superfamily member 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocbrutinib DB19445
small molecule | CAS: 2485861-07-0

Rocbrutinib is under investigation in clinical trial NCT05716087 (A Study of Rocbrutinib in Participants With Relapse or Refractory Mantle Cell Lymphoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Rociletinib DB11907
small molecule | CAS: 1374640-70-6

Rociletinib has been used in trials studying the treatment and prevention of Nonsmall Cell Lung Cancer, Non-small Cell Lung Cancer, and Locally Advanced or Metastatic Non-small Cell Lung Cancer.

Kategori:
Acids, AcyclicAcrylatesAmides +4
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rociverine DB13581
small molecule | CAS: 53716-44-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +9
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rocuronium Approved DB00728
small molecule | CAS: 143558-00-3

Rocuronium (rapid onset-curonium) is a desacetoxy analogue of vecuronium with a more rapid onset of action. It is an aminosteroid non-depolarizing neuromuscular blocker or muscle relaxant used in modern anaesthesia, to facilitate endotracheal intubation and t…

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +16
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M25-hydroxytryptamine receptor 3A
Waktu ParuhThe rapid distribut…
Vol. Distribusi* 0.3 L/kg [3 to <1…
Klirens* 0.25 L/kg/hr [Adu…
Genetik -
Rodatristat DB18478
small molecule | CAS: 1673568-73-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1673571-51-1

Deskripsi belum tersedia.

Target Protein:
Tryptophan 5-hydroxylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rofecoxib Approved DB00533
small molecule | CAS: 162011-90-7

Rofecoxib is used for the treatment of osteoarthritis, rheumatoid arthritis, acute pain in adults, and primary dysmenorrhea, as well as acute treatment of migraine attacks with or without auras. Rofecoxib is a solid. This compound belongs to the stilbenes. Th…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +29
Target Protein:
Prostaglandin G/H synthase 2Elastin
Waktu Paruh17 hours
Vol. Distribusi-
Klirens-
Genetik -
Roflumilast Approved DB01656
small molecule | CAS: 162401-32-3

Roflumilast is a highly selective phosphodiesterase-4 (PDE4) inhibitor.[A251385] PDE4 is a major cyclic-3',5?-adenosinemonophosphate (cyclic AMP, cAMP)-metabolizing enzyme [L37564] expressed on nearly all immune and pro-inflammatory cells, in addition to stru…

Kategori:
Acids, CarbocyclicAgents to Treat Airway DiseaseAmides +17
Target Protein:
cAMP-specific 3',5'-cyclic phosphodiesterase 4 (PDE4)
Waktu ParuhFollowing oral admi…
Vol. DistribusiFollowing a single …
KlirensPlasma clearance of…
Genetik -
Rogaratinib DB15078
small molecule | CAS: 1443530-05-9

Rogaratinib is under investigation in clinical trial NCT03762122 (Rogaratinib in Patients With Advanced Pretreated Squamous-cell Non-small Cell Lung Cancer (SQCLC)).

Kategori:
Sulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roginolisib DB18088
small molecule | CAS: 1305267-37-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rokitamycin DB13409
small molecule | CAS: 74014-51-0

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolapitant Approved DB09291
small molecule | CAS: 552292-08-7

Rolapitant is a potent, highly selective, long-acting Neurokinin-1 (NK-1) receptor antagonist approved for the prevention of delayed chemotherapy-induced nausea and vomiting (CINV) in adults. Delayed-phase CINV typically occurs >24 hours after chemotherapy tr…

Kategori:
Alimentary Tract and MetabolismAntiemetics and AntinauseantsBCRP/ABCG2 Inhibitors +11
Target Protein:
Substance-P receptor
Waktu ParuhMean terminal half …
Vol. Distribusi460 L
Klirens0.96 L/hour
Genetik -
Roledumab DB16317
biotech | CAS: 1174008-79-7

Roledumab is under investigation in clinical trial NCT02287896 (Pharmacokinetics and Safety of Roledumab in Rhd-negative Pregnant Women Carrying an Rhd-positive Foetus).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolicyclidine DB01549
small molecule | CAS: 2201-39-0

Rolicyclidine (PCPy) is classified as a dissociative anesthetic agent. It also has hallucinogenic and sedative properties. Because of its pharmacodynamic similarity to the drug phencyclidine (PCP), rolicyclidine was added to the Schedule I list of illegal dr…

Kategori:
Piperidines
Target Protein:
Glutamate receptor ionotropic, NMDA 3AD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolitetracycline Approved DB01301
small molecule | CAS: 751-97-3

A pyrrolidinylmethyl tetracycline.

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
30S ribosomal protein S916S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rolofylline DB12670
small molecule | CAS: 136199-02-5

Rolofylline is under clinical development by pharmaceutical company NovaCardia for the treatment of congestive heart failure.

Kategori:
AlkaloidsDiureticsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Roluperidone DB13080
small molecule | CAS: 359625-79-9

Roluperidone has been used in trials studying the treatment of Schizophrenia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Sigma intracellular receptor 25-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romidepsin Approved DB06176
small molecule | CAS: 128517-07-7

Romidepsin is a selective inhibitor of histone deacetylase, approved in the US in 2009 for the treatment of cutaneous T-cell lymphoma (CTCL) in patients who have received at least one prior systemic therapy.

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntineoplastic Agents +30
Target Protein:
Histone deacetylase 1Histone deacetylase 2Histone deacetylase 4 +3
Waktu ParuhApproximately 3 hou…
Vol. Distribusi44.5L
Klirens8.4L/h
Genetik -
Romilkimab DB16318
biotech | CAS: 1399584-78-1

Romilkimab is under investigation in clinical trial NCT02345070 (Efficacy and Safety of SAR156597 in the Treatment of Idiopathic Pulmonary Fibrosis).

Target Protein:
Interleukin-13Interleukin-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Romiplostim Approved DB05332
biotech | CAS: 267639-76-9

Romiplostim is a thrombopoiesis stimulating dimer Fc-peptide fusion protein (peptibody) to increase platelet production through activation of the thrombopoietin receptor. The peptibody molecule has two identical single-chain subunits, each one is made up of 2…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +17
Target Protein:
Thrombopoietin receptor
Waktu ParuhImmune thrombocytop…
Vol. DistribusiIn healthy voluntee…
Klirens-
Genetik -
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