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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 194 / 252
Piperine DB12582
small molecule | CAS: 94-62-2

Bioperine has been used in trials studying the treatment of Multiple Myeloma and Deglutition Disorders.

Kategori:
AlkenesAlkynesAmides +11
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] BNuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperonyl butoxide Approved DB09350
small molecule | CAS: 51-03-6

Piperonyl butoxide (PBO) is an organic compound used as a component of pesticide formulations. It is used for the treatment of head, pubic (crab), and body lice. Piperonyl butoxide is a synergist. It has no pesticidal activity of its own, but acts to increase…

Kategori:
AgrochemicalsBenzodioxolesCompounds used in a research, industrial, or household setting +6
Waktu Paruh32 hours.
Vol. DistribusiPiperonyl butoxide …
KlirensClearance of pipero…
Genetik -
Pipethanate DB15888
small molecule | CAS: 4546-39-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pipobroman Approved DB00236
small molecule | CAS: 54-91-1

An antineoplastic agent that acts by alkylation.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +4
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipradrol Approved DB11584
small molecule | CAS: 467-60-7

Pipradrol (Meratran) [L2523] was initially developed in the 1950s as an antidepressant, however, the adverse effects associated with its use and its abuse potential led to its withdrawal and international regulation [L2524]. Pipradrol was made illegal in man…

Kategori:
Central Nervous System StimulantsNervous SystemPsychoanaleptics +1
Target Protein:
D(1) dopamine receptor
Waktu Paruh-
Vol. DistribusiDistributed in the …
KlirensRapidly cleared [T1…
Genetik -
Piprinhydrinate DB15987
small molecule | CAS: 606-90-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Piracetam Approved DB09210
small molecule | CAS: 7491-74-9

Piracetam is a nootropic drug in the racetams group, with chemical name 2-oxo-1-pyrrolidine acetamide. It shares the same 2-oxo-pyrrolidone base structure with pyroglutamic acid and is a cyclic derivative of the neurotransmitter ?-aminobutyric acid (GABA). Ho…

Kategori:
AcetamidesAcetatesAcids, Acyclic +12
Waktu ParuhThe plasma half lif…
Vol. DistribusiVd is approximately…
KlirensThe apparent total …
Genetik -
Pirbuterol Approved DB01291
small molecule | CAS: 38677-81-5

Pirbuterol is a beta-2 adrenergic bronchodilator. In vitro studies and in vivo pharmacologic studies have demonstrated that pirbuterol has a preferential effect on beta-2 Adrenergic receptors compared with isoproterenol. While it is recognized that beta-2 adr…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +21
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh2 hours.
Vol. Distribusi-
Klirens-
Genetik -
Pirenoxine DB15945
small molecule | CAS: 1043-21-6

Deskripsi belum tersedia.

Kategori:
Cataract, drug therapy
Waktu Paruh-
Vol. Distribusi-
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Pirenzepine Approved DB00670
small molecule | CAS: 28797-61-7

An antimuscarinic agent that inhibits gastric secretion at lower doses than are required to affect gastrointestinal motility, salivary, central nervous system, cardiovascular, ocular, and urinary function. It promotes the healing of duodenal ulcers and due to…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Ulcer Agents +10
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirepemat DB19165
small molecule | CAS: 1227638-29-0

Pirepemat is under investigation in clinical trial NCT05258071 (A Clinical Study Evaluating Efficacy of Pirepemat on Falls Frequency in Patients With Parkinson's Disease (PD)).

Waktu Paruh-
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Piretanide Approved DB02925
small molecule | CAS: 55837-27-9

Piretanide (INN, trade names Arelix, Eurelix, Tauliz) has been synthesized in 1973 at Hoechst AG (Germany) as a loop diuretic compound by using a then-new method for introducing cyclic amine residues in an aromatic nucleus in the presence of other aromaticall…

Kategori:
AmidesCardiovascular AgentsDiuretics +9
Target Protein:
Solute carrier family 12 member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirfenidone Approved DB04951
small molecule | CAS: 53179-13-8

Pirfenidone is a synthetic pyridone drug.[A251370] It is an antifibrotic agent with anti-inflammatory and antioxidant properties [A251370] that is used to treat idiopathic pulmonary fibrosis (IPF),[L26801] which is a chronic, progressive form of interstitial …

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +29
Target Protein:
Transforming growth factor beta-1 proprotein
Waktu ParuhThe mean terminal h…
Vol. DistribusiMean apparent oral …
KlirensFollowing administr…
Genetik -
Piribedil DB12478
small molecule | CAS: 3605-01-4

Piribedil has been investigated in Parkinson's Disease.

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +7
Target Protein:
D(3) dopamine receptorAlpha-2C adrenergic receptor5-hydroxytryptamine receptor 1A +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirisudanol DB13412
small molecule | CAS: 33605-94-6

Deskripsi belum tersedia.

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Piritrexim DB03695
small molecule | CAS: 72732-56-0

Piritrexim has been used in trials studying the treatment of Bladder Cancer, Urethral Cancer, and Transitional Cell Cancer of the Renal Pelvis and Ureter.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsFolic Acid Antagonists
Target Protein:
Dihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirlimycin DB11537
small molecule | CAS: 79548-73-5

Pirlimycin hydrochloride is an antibiotic belonging to the _lincosamide_ class. Often marketed as _Pirsue_, this drug is used to treat mastitis in cattle.

Kategori:
Anti-Bacterial AgentsCarbohydratesGlycosides +3
Waktu Paruh-
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Pirlindole DB09244
small molecule | CAS: 60762-57-4

This drug is classified as a reversible inhibitor of monoamine oxidase A enzyme (also known as a RIMA drug). It was developed and is currently used as an antidepressant in Russia. Its chemical structure is similar to metralindole, and it also shares pharmacol…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +14
Target Protein:
Amine oxidase [flavin-containing] A5-hydroxytryptamine receptor 1AAlpha-2A adrenergic receptor
Waktu Paruh0.7±0.3 in one stud…
Vol. Distribusi-
KlirensHigh plasma clearan…
Genetik -
Pirmitegravir DB18974
small molecule | CAS: 2245231-10-9

Pirmitegravir is under investigation in clinical trial NCT05869643 (A Clinical Trial of STP0404 in Treatment-naïve Adults With HIV-1 Infection).

Waktu Paruh-
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Pirnabine DB12840
small molecule | CAS: 19825-63-9

Pirnabine has been used in trials studying the treatment of Chronic Idiopathic Constipation.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme ActivatorsGastrointestinal Agents +6
Waktu Paruh-
Vol. Distribusi-
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Piroctone DB15946
small molecule | CAS: 50650-76-5

Piroctone olamine is used in combination with other substances as a part of shampoo effectively reduced the amount of dandruff and, at the same time, provided hair conditioning advantages. Recently was shown, that piroctone olamine could induce apoptosis and …

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
Vol. Distribusi-
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Pirodavir DB08012
small molecule | CAS: 124436-59-5

Pirodavir is an antipicornavirus agent.

Kategori:
Antiviral Agents
Target Protein:
Genome polyproteinGenome polyproteinGenome polyprotein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Piromidic acid DB13744
small molecule | CAS: 19562-30-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piroxicam Approved DB00554
small molecule | CAS: 36322-90-4

A cyclooxygenase inhibiting, non-steroidal anti-inflammatory agent (NSAID) that is well established in treating rheumatoid arthritis and osteoarthritis and used for musculoskeletal disorders, dysmenorrhea, and postoperative pain. Its long half-life enables it…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +33
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh30 to 86 hours
Vol. Distribusi* 0.14 L/kg
Klirens-
Genetik -
small molecule | CAS: 87234-24-0

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsSulfur CompoundsThiazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirtobrutinib Approved DB17472
small molecule | CAS: 2101700-15-4

Pirtobrutinib is a small molecule and a highly selective non-covalent inhibitor of Bruton’s tyrosine kinase (BTK). Its high selectivity has been associated with lower discontinuation rates due to adverse events and a lower incidence of atrial fibrillation.[A2…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +42
Target Protein:
Tyrosine-protein kinase BTK
Waktu ParuhPirtobrutinib has a…
Vol. DistribusiPirtobrutinib has a…
KlirensPirtobrutinib has a…
Genetik -
Pistachio Approved DB10559
biotech

Pistachio allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
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Pisum sativum whole Approved DB15545
biotech

Pisum sativum whole allergenic extract is used in allergenic testing.

Waktu Paruh-
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Pitavastatin Approved DB08860
small molecule | CAS: 147511-69-1

Pitavastatin, also known as the brand name product Livalo, is a lipid-lowering drug belonging to the statin class of medications. By inhibiting the endogenous production of cholesterol within the liver, statins lower abnormal cholesterol and lipid levels and …

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +20
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-L
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean volume of …
KlirensFollowing a single …
Genetik -
Pitofenone DB15947
small molecule | CAS: 54063-52-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesDrugs for Functional Gastrointestinal Disorders +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pitolisant Approved DB11642
small molecule | CAS: 362665-56-3

Pitolisant is a selective antagonist or inverse agonist of the histamine H3 receptor used to treat type 1 or 2 narcolepsy.[L8063] Narcolepsy is a chronic neurological disorder that affects 1 in 2,000 individuals and is characterized by excessive daytime sleep…

Kategori:
Cytochrome P-450 CYP1A2 InducersCytochrome P-450 CYP1A2 Inducers (strength unknown)Cytochrome P-450 CYP2B6 Inducers +25
Target Protein:
Histamine H3 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhPitolisant has a pl…
Vol. DistribusiFollowing single an…
KlirensThe apparent oral c…
Genetik -
small molecule | CAS: 566170-04-5

Pittsburgh Compound B is under investigation in clinical trial NCT01723553 (Amyloid-related Imaging Abnormalities (Microbleeds) in Atypical AD).

Kategori:
AminesCarbon RadioisotopesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivagabine DB12951
small molecule | CAS: 69542-93-4

Pivagabine has been used in trials studying the treatment of Stress and Anxiety.

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivhydrazine DB09252
small molecule | CAS: 306-19-4

Pivhydrazine, also known as pivazide, is a member of the hydrazine family with irreversible and non-selective inhibitory activity against monoamine oxidases. In 1960, it was widely used as an antidepressant agent but it is now discontinued.

Kategori:
Acids, AcyclicAgents that produce hypertensionAgents that reduce seizure threshold +7
Waktu Paruh-
Vol. Distribusi-
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Pivmecillinam Approved DB01605
small molecule | CAS: 32886-97-8

Pivmecillinam is a mecillinam prodrug, a pivaloyloxymethyl ester of amdinocillin that is well absorbed orally, but broken down to amdinocillin in the intestinal mucosa. It is active against gram-negative organisms and used as for amdinocillin. [PubChem]

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pixantrone Approved DB06193
small molecule | CAS: 144510-96-3

Pixantrone is an aza-anthracenedione and DNA intercalator which inhibits topoisomerase II. It is similar in structure to anthracyclines such as mitoxantrone, but exerts fewer toxic effects on cardiac tissue. [2] The lower cardio-toxic effects of pixantrone ma…

Kategori:
Anthracyclines and Related SubstancesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +6
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu ParuhHalf life ranges fr…
Vol. Distribusi9.7-29.7 L/kg. [2]
KlirensPlasma clearance is…
Genetik -
Pixatimod DB19166
small molecule | CAS: 1144617-49-1

Pixatimod is under investigation in clinical trial NCT05061017 (Pixatimod (PG545) Plus Nivolumab in PD-1 Relapsed/refractory Metastatic Melanoma and NSCLC and With Nivolumab and Low-dose Cyclophosphamide in MSS Metastatic Colorectal Carcinoma (Mcrc)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pixofisiran DB17294
biotech | CAS: 1152798-48-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Pizotifen Approved DB06153
small molecule | CAS: 15574-96-6

Pizotifen belongs to the class of antamines and is related to [cyproheptadine].[A32532] It is a potent serotonin and tryptamine antagonist that has been used for migraine prevention for many years. It exhibits weak anticholinergic, antihistamine, and antikini…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +27
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +12
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
PL-3994 DB15355
small molecule | CAS: 952295-80-6

PL-3994 is under investigation in clinical trial NCT01304628 (Cross-Over Study of Subcutaneous Study Drug for the Treatment of Patients With Mild to Moderate Asthma).

Kategori:
Amino Acids, Peptides, and ProteinsBronchodilator AgentsPeptides +1
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The placenta serves many purposes, with one of the many being a bank of mesenchymal stem cells (MSCs). It can be obtained relatively easily as medical waste from which MSCs can be non-invasively extracted and without the ethical issues that come with embryoni…

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Placulumab DB11983
biotech | CAS: 945781-29-3

Placulumab has been used in trials studying the treatment of Rheumatoid Arthritis.

Waktu Paruh-
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Plamotamab DB18944
biotech | CAS: 2138442-31-4

Plamotamab is under investigation in clinical trial NCT05328102 (Phase 2 Study of Plamotamab Combined With Tafasitamab Plus Lenalidomide Versus Tafasitamab Plus Lenalidomide in Relapsed or Refractory (R/R) Diffuse Large-cell B-cell Lymphoma (DLBCL)).

Waktu Paruh-
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Genetik -
biotech

The Covifenz COVID-19 vaccine (plant-based virus-like particles (VLP), recombinant, adjuvanted) is a plant-based vaccine developed in partnership by Medicago and GlaxoSmithKline which is approved in Canada for the prevention of COVID-19.[L40694] It is compose…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
Waktu Paruh-
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Plantago ovata seed Approved DB14585
biotech

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAngiospermsBiological Products +15
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Plantago seed Approved DB11097
biotech | CAS: 8063-16-9

Platango seeds refer to the seeds collected from various species of plantago trees. It is found in some laxatives for treating occasional constipation and restoring regularity in bowel movements. Its potential benefit in maintaining remission in ulcerative co…

Kategori:
Biological ProductsBulk-Forming LaxativesComplex Mixtures +5
Waktu ParuhThe half-life of ps…
Vol. DistribusiPsyllium husk when …
KlirensPsyllium husk when …
Genetik -
biotech

The plasma protein fraction human (PPFh) is defined as a sterile solution of proteins composed mainly of albumin and globulin derived from human plasma.[A32512] It is already reviewed under the category of biologics by the FDA where the processing, required t…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood Derivatives +9
Waktu ParuhThe registered clea…
Vol. DistribusiThe registered volu…
KlirensThe registered clea…
Genetik -
PlasmaCord DB16363
biotech

PlasmaCord is platelet-poor plasma that is derived by fractionation from sterile umbilical cord and placental blood.[L27581] It is developed by Cellpraxis and is currently being investigated against severe acute respiratory syndrome (SARS).

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Plasminogen Approved DB16701
biotech | CAS: 9001-91-6

Plasminogen is a pro-enzyme (i.e. a zymogen) which is cleaved to form plasmin - also known as [fibrinolysin] - as part of the fibrinolytic pathway that breaks down fibrin blood clots.[A236035] This pathway is activated when a clot is no longer needed or to pr…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBeta-Globulins +11
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean steady-sta…
KlirensThe clearance of Ry…
Genetik -
Platelet Lysate DB15869
biotech

Platelet lysate is an acellular compound composed of platelet proteins while also being void of cellular debris, thus making the lysate rich with growth factors.[A220188] It is extracted through lysis of the plasma membrane of platelets. Because white cell an…

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Menampilkan 9651–9700 dari 12560
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