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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
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16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 194 / 321
LS11 DB05918
small molecule

LS11(talaporfin sodium) is an agent consisting of chlorin e6, derived from chlorophyll, and L-aspartic acid with photosensitizing activity. After intratumoral activation by light emitting diodes, taporfin sodium forms an extended high energy conformational st…

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LSALT Peptide DB16472
biotech

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
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LSP-GR3 DB16934
biotech

Deskripsi belum tersedia.

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LSTA1 DB17346
biotech | CAS: 1392278-76-0

Deskripsi belum tersedia.

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LSZ-102 DB15362
small molecule | CAS: 2135600-76-7

LSZ-102 is under investigation in clinical trial NCT02734615 (Phase I/Ib Trial of LSZ102 Single Agent or LSZ102 + LEE011 or LSZ102 + BYL719 in ER+ Breast Cancers).

Kategori:
Sulfur Compounds
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LTI-03 DB18491
biotech | CAS: 1504575-10-3

LTI-03 is a caveolin-1 Scaffolding Domain 7-Mer

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LTX-109 DB12711
small molecule | CAS: 1166254-80-3

LTX-109 has been investigated for the treatment of Atopic Dermatitis, Mild Eczema/Dermatoses, and Gram-positive, Skin Infections.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptidomimetics
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LTX-315 DB12748
small molecule | CAS: 1345407-05-7

LTX-315 has been used in trials studying the treatment of Cancer, Lymphoma, Melanoma, Carcinoma, and Breast Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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LU-31130 DB05828
small molecule

LU-31130 is a rapid acting therapy developed by H. Lundbeck A/S to treat Psychosis, Schizophrenia and Schizoaffective Disorders. It acts at the Dopamine D4 receptors in the cortex and has low affinity for D2 receptors, adrenoceptors, muscarinic and histaminer…

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Lubazodone DB09196
small molecule | CAS: 161178-07-0

Lubazodone (YM-992, YM-35,995) is an arylpiperazine antidepressant which was being developed as a treatment for depression and obsessive compulsive disorder, and reached phase II clinical trials, but was discontinued. It acts as a serotonin reuptake inhibitor…

Kategori:
Oxazines
Target Protein:
5-hydroxytryptamine receptor 2ASodium-dependent serotonin transporter
Waktu Paruh-
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Lubiprostone Approved DB01046
small molecule | CAS: 136790-76-6

Lubiprostone is a medication used in the management of idiopathic chronic constipation. A prostaglandin E1 derivative, lubiprostone is a bicyclic fatty acid that activates ClC-2 chloride channels located on the apical side of the gastrointestinal epithelial c…

Kategori:
Alimentary Tract and MetabolismChloride Channel AgonistsDrugs for Constipation +9
Target Protein:
Chloride channel protein 2
Waktu Paruh0.9 to 1.4 hours
Vol. Distribusi-
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Lucanthone DB04967
small molecule | CAS: 479-50-5

One of the schistosomicides, it has been replaced largely by hycanthone and more recently praziquantel. (From Martindale The Extrapharmacopoeia, 30th ed., p46). It is currently being tested as a radiation sensitizer.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +7
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA repair nuclease/redox regulator APEX1 +2
Waktu Paruh-
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Lucatumumab DB06360
biotech | CAS: 903512-50-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Tumor necrosis factor receptor superfamily member 5
Waktu Paruh-
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Lucerastat DB14872
small molecule | CAS: 141206-42-0

Lucerastat is under investigation in clinical trial NCT03425539 (Efficacy and Safety of Lucerastat Oral Monotherapy in Adult Subjects With Fabry Disease).

Kategori:
AlkaloidsCarbohydratesImines +3
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Lucinactant Approved DB04897
biotech | CAS: 825600-90-6

Lucinactant is a new synthetic peptide-containing surfactant for intratracheal use. It contains sinapultide, a novel, hydrophobic, 21-amino acid peptide (leucine and lysine repeating units, KL4 peptide) designed to mimic human surfactant protein-B (SB-P). Mor…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +11
Waktu Paruh-
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Lucitanib DB11845
small molecule | CAS: 1058137-23-7

Lucitanib has been used in trials studying the treatment of ER+, MBC, SCLC, HER2+, and NSCLC, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Vascular endothelial growth factor receptor 2 +5
Waktu Paruh-
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Lufenuron DB11424
small molecule | CAS: 103055-07-8

Lufenuron is used in veterinary for the control of flea.

Kategori:
Acids, CarbocyclicAgrochemicalsAmides +9
Waktu Paruh-
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Luliconazole Approved DB08933
small molecule | CAS: 187164-19-8

Luliconazole is a topical antifungal agent that acts by unknown mechanisms but is postulated to involve altering the synthesis of fungi cell membranes. It was approved by the FDA (USA) in November 2013 and is marketed under the brand name Luzu. Luliconazole i…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +10
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe half life of lu…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of lu…
Genetik -
Lulizumab pegol DB15441
biotech | CAS: 1421830-13-8

Lulizumab pegol is under investigation in clinical trial NCT02843659 (Proof of Concept Study to Evaluate the Efficacy and Safety of BMS-931699 (Lulizumab) or BMS-986142 in Primary Sjögren's Syndrome).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntibodies, Monoclonal +11
Waktu Paruh-
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LuLym-T DB17405
biotech

LuLym-T is an investigational autologous immune cell therapy consisting of activated T Lymphocytes. Developed by Lukas Biomedical, Inc., it is currently being investigated in hepatocellular carcinoma.

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Lumacaftor Approved DB09280
small molecule | CAS: 936727-05-8

Lumacaftor is a drug used in combination with [DB08820] as the fixed dose combination product Orkambi for the management of Cystic Fibrosis (CF) in patients aged 6 years and older. Cystic Fibrosis is an autosomal recessive disorder caused by one of several di…

Kategori:
AminesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +21
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe half-life of lu…
Vol. DistribusiFollowing oral admi…
KlirensThe typical apparen…
Genetik -
Lumasiran Approved DB15935
biotech | CAS: 1834610-13-7

Lumasiran is a small interfering RNA used in the treatment of primary hyperoxaluria type 1 (PH1).[L23554] This condition, caused by a deficiency in the enzyme alanine-glyoxylate aminotransferase, leads to an accumulation of oxalate, causing calcium crystal fo…

Kategori:
Alimentary Tract and MetabolismAntisense Elements (Genetics)Cytochrome P-450 CYP2C8 Inhibitors +12
Target Protein:
2-Hydroxyacid oxidase 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent centra…
KlirensThe apparent plasma…
Genetik -
Lumateperone Approved DB06077
small molecule | CAS: 313368-91-1

Schizophrenia is a complex mental illness and impacts approximately 1% of the population.[L10902] Although there are several antipsychotics including [aripiprazole], [paliperidone] and [clozapine] available for clinical use, they are generally accompanied by …

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +21
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 2AD(2) dopamine receptor +1
Waktu ParuhLumateperone's half…
Vol. DistribusiThe volume of distr…
KlirensLumateperone's clea…
Genetik -
Lumefantrine Approved DB06708
small molecule | CAS: 82186-77-4

Lumefantrine is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with artemether for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +11
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh~ 4.5 days
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Lumefantrine co-artemether Approved DB13085
small molecule | CAS: 141204-94-6

Lumefantrine Co-Artemether (Riamet) has been investigated for the treatment of Malaria, Malaria, Falciparum, Malaria in Pregnancy, Uncomplicated Malaria, and Uncomplicated Knowlesi Malaria. Lumefantrine Co-Artemether is a tablet formulation of artemether and …

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Lumichrome DB04345
small molecule | CAS: 1086-80-2

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +3
Target Protein:
Flavin reductase (NADPH)Riboflavin biosynthesis protein
Waktu Paruh-
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Lumicitabine DB14808
small molecule | CAS: 1445385-02-3

Lumicitabine is under investigation in clinical trial NCT03010059 (A Study to Assess the Relative Bioavailability of JNJ64041575 Administered as 2 Different New Concept Formulations (Oral Suspension and Tablet) Compared to Their Respective Current Formulation…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
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Lumiflavin DB04726
small molecule | CAS: 1088-56-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +3
Waktu Paruh-
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Lumiliximab DB06162
biotech | CAS: 357613-86-6

Lumiliximab is a chimeric monoclonal antibody which is used as an immunosuppressive drug. It is a primatized anti-CD23 macaque/human chimeric antibody that inhibits the production of the IgE antibody, for the potential treatment of allergic conditions. Lumili…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Low affinity immunoglobulin epsilon Fc receptor
Waktu Paruh-
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Luminol DB18536
small molecule | CAS: 521-31-3

Deskripsi belum tersedia.

Kategori:
Compounds used in a research, industrial, or household settingIndicators and ReagentsLaboratory Chemicals +2
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Lumiracoxib Approved DB01283
small molecule | CAS: 220991-20-8

Lumiracoxib is a COX-2 selective non-steroidal anti-inflammatory drug (NSAID). On August 11, 2007, Australia's Therapeutic Goods Administration (TGA, the Australian equivalent of the FDA) cancelled the registration of lumiracoxib in Australia due to concerns …

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +21
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhTerminal half-life …
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Lumretuzumab DB12683
biotech | CAS: 1448327-63-6

Lumretuzumab has been used in trials studying the treatment of Neoplasms, Breast Cancer, Squamous Non-Small Cell Lung Cancer, and Non-Squamous Non-Small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
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Lunasine DB16223
small molecule | CAS: 6901-22-0

Lunasine is under investigation in clinical trial NCT02709330 (ALS Reversals - Lunasin Regimen).

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Lunresertib DB19241
small molecule | CAS: 2719793-90-3

Deskripsi belum tersedia.

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Lunsekimig DB19009
biotech | CAS: 2770858-49-4

Lunsekimig is under investigation in clinical trial NCT06102005 (Dose Ranging Study of Lunsekimig Compared With Placebo-control in Adult Participants With Moderate-to-severe Asthma).

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Lupeol DB12622
small molecule | CAS: 545-47-1

Lupeol has been investigated for the treatment of Acne.

Kategori:
Anti-Inflammatory AgentsPentacyclic TriterpenesTerpenes +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaNeutrophil elastase
Waktu Paruh-
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Luprostiol DB11425
small molecule | CAS: 67110-79-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lurasidone Approved DB08815
small molecule | CAS: 367514-87-2

Lurasidone is an atypical antipsychotic developed by Dainippon Sumitomo Pharma. It was approved by the U.S. Food and Drug Administration (FDA) for treatment of schizophrenia on October 29, 2010 and is currently pending approval for the treatment of bipolar di…

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +34
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 7 +3
Waktu Paruh40 mg dose= 18 hour…
Vol. Distribusi6173 L
Klirens3902 mL/min
Genetik -
Lurbinectedin Approved DB12674
small molecule | CAS: 497871-47-3

Lurbinectedin is a DNA alkylating agent that has been investigated in the treatment of a variety of cancers, including mesothelioma,[A214325] chronic lymphocytic leukemia (CLL),[A214328] breast cancer,[A214322] and small-cell lung cancer (SCLC).[A214310] It i…

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +12
Target Protein:
DNA
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state vo…
KlirensThe total plasma cl…
Genetik -
Lurtotecan DB12222
small molecule | CAS: 149882-10-0

Lurtotecan is under investigation in clinical trial NCT00022594 (Liposomal Lurtotecan in Treating Patients With Metastatic or Locally Recurrent Head and Neck Cancer).

Kategori:
AlkaloidsAntineoplastic Agents
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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Klirens-
Genetik -
Lusacomfar Alfa DB18526
biotech | CAS: 2640087-71-2

Lusacomfar Alfa is a recombinant complement factor H

Waktu Paruh-
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Luseogliflozin DB12214
small molecule | CAS: 898537-18-3

Luseogliflozin has been used in trials studying the treatment of Diabetes Melltius, Type 2.

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood Glucose Lowering Agents +5
Waktu Paruh-
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Luspatercept Approved DB12281
biotech | CAS: 1373715-00-4

Luspatercept is a recombinant fusion protein comprised of a modified extracellular domain of activin receptor type IIB fused to the FC domain of human IgG1.[A187829,L42455] It was first approved for use in the United States in November 2019 under the brand na…

Kategori:
Activin ReceptorsAmino Acids, Peptides, and ProteinsAntianemia Drugs +25
Waktu ParuhThe average half-li…
Vol. DistribusiThe average apparen…
KlirensThe total apparent …
Genetik -
Lusutrombopag Approved DB13125
small molecule | CAS: 1110766-97-6

Lusutrombopag is an orally bioavailable thrombopoietin receptor (TPOR) agonist developed by Shionogi & Company (Osaka, Japan). TPOR is a regulatory target site for endogenous thrombopoietin, which acts as a primary cytokine to promote megakaryocyte proliferat…

Kategori:
Acids, CarbocyclicBCRP/ABCG2 SubstratesBlood and Blood Forming Organs +4
Target Protein:
Thrombopoietin receptor
Waktu ParuhIn healthy adult su…
Vol. DistribusiThe mean (%CV) lusu…
KlirensThe approximate mea…
Genetik -
Lusvertikimab DB18778
biotech | CAS: 2375835-91-7

Deskripsi belum tersedia.

Waktu Paruh-
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Lutein Approved DB00137
small molecule | CAS: 127-40-2

Lutein is an xanthophyll and one of 600 known naturally occurring carotenoids. Lutein is synthesized only by plants and like other xanthophylls is found in high quantities in green leafy vegetables such as spinach, kale and yellow carrots. In green plants, xa…

Kategori:
AlkenesBiological FactorsCarotenoids +10
Waktu Paruh-
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Luteinizing hormone Approved DB14741
biotech | CAS: 9002-67-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsGonadotropinsGonadotropins, Pituitary +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luteolin DB15584
small molecule | CAS: 491-70-3

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
Signal transducer and activator of transcription 3Lysophosphatidylcholine acyltransferase 2Lysophosphatidylcholine acyltransferase 1 +1
Waktu Paruh-
Vol. Distribusi-
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Lutetium Lu 177 dotatate Approved DB13985
small molecule | CAS: 437608-50-9

A 177Lu-labeled somatostatin analog peptide, Lutetium Lu 177 dotatate belongs to an emerging form of treatments called Peptide Receptor Radionuclide Therapy (PRRT), which involves targeting tumours with molecules carrying radioactive particles that bind to sp…

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +8
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 1Somatostatin receptor type 3 +2
Waktu ParuhThe mean (± standar…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Lutetium Lu-177 Approved DB13982
small molecule | CAS: 14265-75-9

Deskripsi belum tersedia.

Kategori:
ElementsIsotopesLanthanoid Series Elements +3
Waktu Paruh-
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Genetik -
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