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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 193 / 272
Normethadone Approved DB11609
small molecule | CAS: 467-85-6

Normethadone is used as an opioid antitussive in combination with [DB11610]. It is marketed in Canada by Valeant under the tradename Cophylac.

Kategori:
AnalgesicsAntitussive AgentsCentral Nervous System Agents +10
Waktu Paruh-
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Genetik -
small molecule | CAS: 156126-12-4

Deskripsi belum tersedia.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
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Northern brown shrimp Approved DB15539
biotech

Northern brown shrimp allergenic extract is used in allergenic testing.

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Nortriptyline Approved DB00540
small molecule | CAS: 72-69-5

Nortriptyline hydrochloride, the active metabolite of [amitriptyline], is a tricyclic antidepressant (TCA).[L11878] It is used in the treatment of major depression and is also used off-label for chronic pain and other conditions.[L11881]

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +59
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +12
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +4
Waktu ParuhThe average plasma …
Vol. DistribusiThe apparent volume…
KlirensThe average plasma …
Genetik 7 Varian
small molecule | CAS: 99697-24-2

norUrsodeoxycholic acid is under investigation in clinical trial NCT03872921 (Norursodeoxycholic Acid vs Placebo in PSC).

Kategori:
Bile Acids and SaltsCholanesCholic Acids +2
Waktu Paruh-
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Noscapine Approved DB06174
small molecule | CAS: 128-62-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntitussive AgentsCentral Nervous System Agents +12
Target Protein:
Sigma non-opioid intracellular receptor 1
Waktu Paruh-
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Genetik -
NOV-002 DB05393
small molecule

NOV-002, the lead compound acts as a chemoprotectant and an immunomodulator, in combination with chemotherapy. NOV-002 is approved and marketed in the Russian Fereration by Pharma BAM under the trade name Glutoxim. It has been administered to over 10,000 pati…

Kategori:
Amino Acids, Peptides, and ProteinsChlorine CompoundsNitrogen Compounds +3
Waktu Paruh-
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Novaferon DB16483
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +4
Waktu Paruh-
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Novobiocin Approved DB01051
small molecule | CAS: 303-81-1

Novobiocin is an antibiotic compound derived from _Streptomyces niveus_. It has a chemical structure similar to coumarin. Novobiocin binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. (From Reynolds, Martindale The Extra Pharmacopoeia,…

Kategori:
AminocoumarinsAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA gyrase subunit B +1
Waktu Paruh6 hours
Vol. Distribusi-
Klirens-
Genetik -
Novolimus DB19085
small molecule | CAS: 151519-50-5

Novolimus is under investigation in clinical trial NCT04483791 (Dynamx Bioadaptor Hong Kong Registry).

Kategori:
LactonesPolyketides
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
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Noxytiolin Approved DB13838
small molecule | CAS: 15599-39-0

Local antibacterial that probably acts by releasing formaldehyde in aqueous solutions. It is used for THERAPEUTIC IRRIGATION of infected body cavities - bladder, peritoneum, etc. and as a spray for burns.

Kategori:
AmidesAnti-Infective AgentsAnti-Infective Agents, Local +5
Waktu Paruh-
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Genetik -
NP-10679 DB18040
small molecule | CAS: 2914889-88-4

Deskripsi belum tersedia.

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NP-50301 DB05662
small molecule

NP-50301 is an ophthalmic therapeutic eye drop treating post-menopausal Dry Eye Syndrome (DES). It is being developed by Nascent Pharmaceuticals. It is estimated that about 30% of postmenopausal women suffer symptoms of DES, which accounts for over 12 million…

Target Protein:
Estrogen receptor
Waktu Paruh-
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NP-51 DB16995
small molecule | CAS: 66611-38-9

Deskripsi belum tersedia.

Kategori:
AminesEnzyme InhibitorsHydroxylamines
Target Protein:
Mitogen-activated protein kinase 8Mitogen-activated protein kinase 9Mitogen-activated protein kinase 10
Waktu Paruh-
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Genetik -
NP-6A4 DB17599
biotech

NP-6A4 is a peptide designed to specifically bind and activate angiotensin II receptor type 2 (AT2R). It has an Orphan Drug designation from the FDA for pediatric cardiomyopathy.[A258523]

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NP-G2-044 DB14995
small molecule | CAS: 1807454-59-6

NP-G2-044 is under investigation in clinical trial NCT03199586 (Phase 1 Clinical Trial of Metastasis Inhibitor NP-G2-044 in Patients With Advanced or Metastatic Solid Tumors (Including Lymphoma)).

Kategori:
Heterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Fascin
Waktu Paruh-
Vol. Distribusi-
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NP2 DB06308
small molecule

NP2 is a replication defective HSV-1 based gene transfer vector engineered to express human preproenkephalin. It was under investigation in clinical trial NCT01291901 (NP2 Enkephalin For Treatment of Intractable Cancer Pain).

Waktu Paruh-
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NPI 32101 DB05264
small molecule

NPI 32101 possesses both anti-inflammatory and broad spectrum antimicrobial activities. This combination of pharmacological properties may have additional therapeutic uses beyond dermatology.

Target Protein:
Cytokine receptor common subunit beta
Waktu Paruh-
Vol. Distribusi-
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NPS-2143 DB05695
small molecule | CAS: 284035-33-2

Deskripsi belum tersedia.

Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NPT520-34 DB17920
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
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NRC-AN-019 DB17110
small molecule | CAS: 879507-25-2

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +2
Waktu Paruh-
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NRP290 DB06383
small molecule

NRP290 is a hydrocodone derivative under investigation for the treatment of pain (moderate to moderately severe).

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NRP369 DB06384
small molecule

NRP369 is an oxycodone derivative under investigation for the treatment of pain (moderate to moderately severe). NRP369 was developed by New River Pharmaceuticals as a backup therapeutic to [NRP290].

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NRP409 DB05235
small molecule

NRP409 is a triiodothyronine (T3) hormone, being investigated by New River Pharmaceuticals as a treatment for patients with primary hypothyroidism.

Target Protein:
Ketimine reductase mu-crystallinThyroid hormone receptor alpha
Waktu Paruh-
Vol. Distribusi-
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NS-2359 DB05805
small molecule | CAS: 195875-68-4

NS2359 is a triple monoamine re-uptake inhibitor with a new, unique drug profile expected to yield important benefits compared to existing treatments of depression. Enhancing the function of the three neurotransmitters serotonin, noradrenalin and dopamine, NS…

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds +1
Target Protein:
Sodium-dependent dopamine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
Waktu Paruh-
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NS-3728 DB05835
small molecule | CAS: 265646-85-3

NS3728 is an orally active chloride channel blocker for the treatment of cancer.

Kategori:
AmidesAminesAnilides +3
Waktu Paruh-
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NS-398 DB14060
small molecule | CAS: 123653-11-2

NS-398 is a COX-2 inhibitor. It was developed as part of the mechanistic study of the cyclooxygenases.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +14
Target Protein:
Prostaglandin G/H synthase 2Cyclooxygenase 2
Waktu Paruh-
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NS-8593 DB16897
small molecule | CAS: 875755-39-8

Deskripsi belum tersedia.

Kategori:
AminesNaphthalenes
Waktu Paruh-
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NS13001 DB16898
small molecule | CAS: 1063331-94-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Waktu Paruh-
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NSC-663284 DB17038
small molecule | CAS: 383907-43-5

NSC-663284 is a potent quinolinedione Cdc25 phosphatase inhibitor.[A253052]

Kategori:
cdc25 Phosphatases, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
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NSI-189 DB16230
small molecule | CAS: 1270138-40-3

NSI-189 is under investigation in clinical trial NCT02695472 (Study of NSI-189 for Major Depressive Disorder).

Kategori:
AminesPyridines
Waktu Paruh-
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NT 13 DB16953
small molecule | CAS: 117928-93-5

Deskripsi belum tersedia.

Waktu Paruh-
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NT-102 DB18112
small molecule | CAS: 1607447-79-9

Deskripsi belum tersedia.

Waktu Paruh-
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NT-219 DB17490
small molecule | CAS: 1198078-60-2

Deskripsi belum tersedia.

Target Protein:
Insulin receptor substrate 2Insulin receptor substrate 1Signal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
NTLA-2002 DB17597
biotech

NTLA-2002 is a lipid nanoparticle encapsulating single guide RNA (G012267) targeting the human KLKB1 gene and messenger RNA (mRNA000042) encoding Cas9. It is an investigational therapy designed to knock out the target gene kallikrein B1 (KLKB1) to reduce plas…

Waktu Paruh-
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NTP-42 DB18302
small molecule | CAS: 2055599-51-2

Deskripsi belum tersedia.

Waktu Paruh-
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NU1025 DB02690
small molecule | CAS: 90417-38-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Poly [ADP-ribose] polymerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
NUC B1000 DB05242
biotech

NUC B1000 is an expressed interfering RNA (eiRNA)- based product consisting of a plasmid DNA construct designed to produce four short interfering RNA (siRNA) molecules, formulated with a proprietary cationic-lipid delivery system. [F3910] eiRNA is an approach…

Waktu Paruh-
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NUC-7738 DB19148
small molecule | CAS: 2348493-39-8

NUC-7738 is under investigation in clinical trial NCT03829254 (A Safety, Pharmacokinetic and Clinical Activity Study of NUC-7738 in Patients With Advanced Solid Tumours and Lymphoma).

Kategori:
Benzene DerivativesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Nurulimab DB18946
biotech | CAS: 2168561-20-2

Nurulimab is under investigation in clinical trial NCT05732805 (A Clinical Study of BCD-217 (Nurulimab + Prolgolimab) Followed by Anti-pd-1 Compared to Anti-pd-1 Monotherapy as First-line Treatment in Subjects With Unresectable/metastatic Melanoma).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Nusinersen Approved DB13161
small molecule | CAS: 1258984-36-9

An antisense oligonucleotide that induces survival motor neuron (SMN) protein expression, it was approved by the U.S. FDA in December, 2016 as Spinraza for the treatment of children and adults with spinal muscular atrophy (SMA). It is adminstrated as direct i…

Kategori:
Antisense OligonucleotidesIncreased Protein SynthesisMusculo-Skeletal System +4
Target Protein:
Survival motor neuron protein
Waktu ParuhThe mean terminal e…
Vol. DistribusiCSF: 0.4 L Plasma…
KlirensSlow clearance is o…
Genetik -
Nutlin-3 DB17039
small molecule | CAS: 548472-68-0

Nutlin-3 is a small molecule inhibitor that targets p53-Mdm2 interaction.[A253057]

Kategori:
Stereoisomerism
Target Protein:
Cellular tumor antigen p53
Waktu Paruh-
Vol. Distribusi-
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Nuvaxovid Approved DB15810
biotech

SARS-CoV-2, the causative agent of COVID-19, relies on the interaction between its trimeric spike (S) glycoprotein and angiotensin-converting enzyme 2 (hACE2) expressed on host cells in order to establish a productive infection in humans.[A243789] Antibodies …

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
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NV-354 DB18392
small molecule | CAS: 866465-21-6

Deskripsi belum tersedia.

Waktu Paruh-
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NV-5138 DB19180
small molecule | CAS: 2095886-80-7

NV-5138 is under investigation in clinical trial NCT06235905 (Open-label of SPN-820 in Adults With Major Depressive Disorder).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +1
Waktu Paruh-
Vol. Distribusi-
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NV-52 DB05673
small molecule

NV-52 is an investigational synthetic flavonoid thromboxane synthase (TXS) inhibitor developed for the maintenance of remission in inflammatory bowel disease.

Target Protein:
Thromboxane-A synthase
Waktu Paruh-
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NVS antibody DB05312
small molecule

This drug has been developed using Medarex's UltiMAb Human Antibody Development System to treat autoimmune diseases.

Waktu Paruh-
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NX-1207 DB05493
small molecule

NX-1207 is an investigational new drug for BPH, whose chemical entity and mechanism of action remain undisclosed. Nymox Pharmaceutical Corporation recently completed studies of NX-1207 for treatment of benign prostatic hyperplasia (BPH).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
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NXC680 DB18366
small molecule

NXC680 is a small molecule under investigation for the treatment of idiopathic pulmonary fibrosis (IPF).

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Nylidrin Approved DB06152
small molecule | CAS: 447-41-6

Nylidrin, also known as _buphenine_ belongs to the category of drugs called _vasodilators_, which relax blood vessels and increase blood flow. Nylidrin is a peripheral vasodilator. Some studies show the evidence of improving cognitive impairment in selected i…

Kategori:
2-Amino-1-Phenylethanol DerivativesAdrenergic AgentsAdrenergic Agonists +29
Target Protein:
Interferon alpha/beta receptor 2Voltage-dependent T-type calcium channel subunit alpha-1I
Waktu ParuhDuration of action …
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9601–9650 dari 13591
Sebelumnya Halaman 193 / 272 Berikutnya