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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Halaman 192 / 236
biotech

Arexvy (respiratory syncytial virus vaccine, adjuvanted) is an adjuvanted vaccine developed by GlaxoSmithKline Biologicals. It comprises lyophilized recombinant respiratory syncytial virus glycoprotein F (RSVPreF3) stabilized in pre-fusion conformation as the…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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Resveratrol DB02709
small molecule | CAS: 501-36-0

Resveratrol (3,5,4'-trihydroxystilbene) is a polyphenolic phytoalexin. It is a stilbenoid, a derivate of stilbene, and is produced in plants with the help of the enzyme stilbene synthase. It exists as cis-(Z) and trans-(E) isomers. The trans- form can undergo…

Kategori:
Angiogenesis InhibitorsAnticarcinogenic AgentsAntioxidants +33
Target Protein:
NAD-dependent protein deacetylase sirtuin-1Ribosyldihydronicotinamide dehydrogenase [quinone]Casein kinase II subunit alpha +23
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Retagliptin DB14898
small molecule | CAS: 1174122-54-3

Retagliptin is under investigation in clinical trial NCT02822534 (The Pharmacokinetics and Pharmacodynamics Study of Single and Multiple Dose of SP2086 in Type 2 Diabetes Patients).

Target Protein:
Dipeptidyl peptidase 4
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Retapamulin Approved DB01256
small molecule | CAS: 224452-66-8

Retapamulin, marketed by GlaxoSmithKline as the ointment Altabax, is an antibiotic for skin infections like impetigo. It was approved by the FDA in April 2007.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibiotics for Topical Use +6
Target Protein:
50S ribosomal protein L3
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Retaspimycin DB05626
small molecule | CAS: 857402-23-4

Deskripsi belum tersedia.

Kategori:
AmidesHSP90 Heat-Shock Proteins, antagonists & inhibitorsLactams +2
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Reteplase Approved DB00015
biotech | CAS: 133652-38-7

Human tissue plasminogen activator, purified, glycosylated, 355 residues purified from CHO cells. Retavase is considered a "third-generation" thrombolytic agent, genetically engineered to retain and delete certain portions of human tPA. Retavase is a deletion…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnticoagulants +17
Target Protein:
PlasminogenFibrinogen alpha chainPlasminogen activator inhibitor 1
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Retifanlimab Approved DB15766
biotech | CAS: 2079108-44-2

Retifanlimab is a humanized IgG4 kappa monoclonal antibody that binds to the programmed death receptor-1 (PD-1), blocking PD-1 interaction with its ligands, programmed death-ligand 1 (PD-L1) and programmed death-ligand 2 (PD-L2). By blocking the PD-1/PD-L1/2 …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +11
Target Protein:
Programmed cell death protein 1
Waktu ParuhAt steady-state, re…
Vol. DistribusiAt steady-state, re…
KlirensFollowing the first…
Genetik -
small molecule | CAS: 74193-17-2

Deskripsi belum tersedia.

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Genetik -
biotech | CAS: 2395839-91-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
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Retosiban DB11818
small molecule | CAS: 820957-38-8

Retosiban has been used in trials studying the treatment of Premature Labor and Obstetric Labour, Premature.

Target Protein:
Oxytocin receptor
Waktu Paruh-
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Revaprazan DB16308
small molecule | CAS: 199463-33-7

Revaprazan is under investigation in clinical trial NCT01750437 (Phase 2 Clinical Trial to Investigate the Safety, Tolerability and Efficacy of YH1885L in Patients With Non-erosive Reflux Disease(nerd)).

Kategori:
Heterocyclic Compounds, Fused-RingIsoquinolinesPyrimidines
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Revefenacin Approved DB11855
small molecule | CAS: 864750-70-9

Revefenacin is a novel biphenyl carbamate tertiary amine agent that belongs to the family of the long-acting muscarinic antagonists (LAMA). The labile primary amide in the structure produces a "soft-drug" site that allows rapid systemic clearance and minimizi…

Kategori:
AmidesAnticholinergic AgentsBCRP/ABCG2 Substrates +9
Target Protein:
Muscarinic acetylcholine receptor
Waktu ParuhThe apparent termin…
Vol. DistribusiAfter intravenous a…
KlirensThe renal clearance…
Genetik -
biotech | CAS: 1446198-96-4

Deskripsi belum tersedia.

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Reversin 121 DB14072
small molecule | CAS: 174630-04-7

Reversin 121 is a hydrophobic peptide chemosensitizer that can reverse P-glycoprotein-mediated multidrug resistance.

Kategori:
Amino Acids, Peptides, and ProteinsDrug Resistance, MultipleP-glycoprotein inhibitors +1
Target Protein:
ATP-dependent translocase ABCB1
Waktu Paruh-
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Reversine DB07340
small molecule | CAS: 656820-32-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingOxazinesProtein Kinase Inhibitors
Target Protein:
Adenosine receptor A3Dual specificity mitogen-activated protein kinase kinase 1Aurora kinase B +1
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Revumenib Approved DB18515
small molecule | CAS: 2169919-21-3

Abnormal gene rearrangements at chromosome locus 11q23, called KMT2A rearrangements or translocations, are present in 5%-10% of patients with acute leukemias and are the sole genetic aberration found in the majority of infant acute lymphoblastic leukemia case…

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +17
Target Protein:
Menin
Waktu ParuhFollowing oral admi…
Vol. DistribusiThe the geometric m…
KlirensFollowing oral admi…
Genetik -
Revusiran DB16309
biotech | CAS: 1438322-82-7

Revusiran is under investigation in clinical trial NCT02319005 (ENDEAVOUR: Phase 3 Multicenter Study of Revusiran (ALN-TTRSC) in Patients With Transthyretin (TTR) Mediated Familial Amyloidotic Cardiomyopathy (FAC)).

Kategori:
Antisense Elements (Genetics)Molecular ProbesNucleic Acid Probes +5
Target Protein:
Transthyretin
Waktu Paruh-
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biotech | CAS: 2172954-10-6

Rexlemestrocel-L is an investigational human bone marrow-derived allogeneic mesenchymal precursor cell (MPC) product. It is being investigated in various cardiac conditions, such as chronic heart failure and acute myocardial infarction.

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Rezafungin Approved DB16310
small molecule | CAS: 1396640-59-7

Rezafungin is an echinocandin antifungal drug.[A258393,L45633] Unlike other echinocandins such as [caspofungin] and [micafungin], rezafungin has long?acting pharmacokinetics and a high stability that allows for it to have long dosing intervals maintaining hig…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +8
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu ParuhRezafungin has a te…
Vol. DistribusiRezafungin has a vo…
KlirensRezafungin has an e…
Genetik -
Rezatapopt DB18980
small molecule | CAS: 2636846-41-6

Rezatapopt is under investigation in clinical trial NCT04585750 (The Evaluation of PC14586 in Patients With Advanced Solid Tumors Harboring a TP53 Y220C Mutation (PYNNACLE)).

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Rezatomidine DB12143
small molecule | CAS: 847829-38-3

Rezatomidine has been used in trials studying the treatment of Fibromyalgia, Cystitis, Interstitial, Irritable Bowel Syndrome, and Diabetic Neuropathy, Painful.

Target Protein:
Alpha-2C adrenergic receptor
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biotech | CAS: 2641686-76-0

Rezpegaldesleukin is under investigation in clinical trial NCT04433585 (A Study of LY3471851 in Adults With Systemic Lupus Erythematosus (SLE)).

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Rezvilutamide DB19133
small molecule | CAS: 1572045-62-5

Rezvilutamide is under investigation in clinical trial NCT05956639 (Comparing a 6-month vs Long-term Course of Rezvilutamide With ADT Plus Chemotherapy in Mhspc).

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RG-4733 DB11870
small molecule | CAS: 847925-91-1

Ro4929097 has been used in trials studying the treatment of Sarcoma, LYMPHOMA, Neoplasms, Wilm's Tumor, and OSTEOSARCOMA, among others.

Kategori:
Amyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme InhibitorsGamma Secretase Inhibitors and Modulators +3
Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
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RG-7795 DB06329
small molecule | CAS: 892498-64-5

Deskripsi belum tersedia.

Target Protein:
Toll-like receptor 7
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RG2417 DB05055
small molecule

RG2417 is a proprietary formulation of uridine, a biological compound essential for the synthesis of DNA and RNA, the basic hereditary material found in all cells, and numerous other factors essential for cell metabolism. Uridine is synthesized by the mitocho…

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RGLS-8429 DB18127
biotech

RGLS-8429 is an investigational anti-miR-17 oligonucleotide.

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RGX-111 DB17632
biotech

RGX-111 is an adeno-associated virus vector AAV9 designed to deliver the ?-L-iduronidase (IDUA) gene. Developed by REGENXBIO Inc., it was investigated for the treatment of mucopolysaccharidosis Type I (MPS I).[L46666]

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RGX-121 DB17681
biotech

RGX-121 is designed to use the NAV AAV9 vector to deliver the human iduronate-2-sulfatase gene to the central nervous system.

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RGX-181 DB17942
biotech

RGX-181 consists of an adeno-associated virus serotype 9 (AAV9) vector designed to deliver the soluble lysosomal enzyme tripeptidyl peptidase I (TPP1) gene. Developed by REGENXBIO, it is being investigated for the treatment of late-infantile neuronal ceroid l…

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RGX-202 DB18397
biotech

RGX-202 is a recombinant AAV8 that contains a vector genome encoding a miniaturized dystrophin protein (microdystrophin).

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RGX-501 DB17639
biotech

RGX-501 is an adeno-associated virus vector 8 (AAV8)-mediated gene therapy that delivers a functional copy of the human low-density lipoprotein receptor (LDLR) gene to liver cells. It is being investigated for the treatment of homozygous familial hypercholest…

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Rhamnetin DB16772
small molecule | CAS: 90-19-7

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +3
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Rhein DB13174
small molecule | CAS: 478-43-3

Rhein is an anthraquinone metabolite of rheinanthrone and senna glycoside is present in many medicinal plants including Rheum palmatum, Cassia tora, Polygonum multiflorum, and Aloe barbadensis [A19247]. It is known to have hepatoprotective, nephroprotective, …

Kategori:
AnthracenesCytochrome P-450 CYP1A2 InhibitorsCytochrome P-450 CYP1A2 Inhibitors (strength unknown) +10
Target Protein:
Heat shock protein HSP 90-alphaOxysterols receptor LXR-alphaOxysterols receptor LXR-beta +2
Waktu Paruh4-10h [A19300].
Vol. Distribusi15-60L [A19300].
KlirensTotal CL is 1.5 L/h…
Genetik -
Rheinanthrone DB13175
small molecule | CAS: 480-09-1

Rheinanthrone is the active metabolite of senna glycoside [DB11365] known for its laxative effect [A19235]. It is commonly produced by plants of the Rheum species [L772].

Kategori:
Anthracenes
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small molecule

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsTherapeutic Radiopharmaceuticals
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Rhenium re-188 DB19267
small molecule | CAS: 14378-26-8

Rhenium re-188 is under investigation in clinical trial NCT03458559 (Rhenium-188-hedp vs. Radium-223-chloride in Patients With Advanced Prostate Cancer Refractory to Hormonal Therapy).

Kategori:
ElementsIsotopesMetals +2
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rhIGFBP-3 DB05897
biotech

rhIGFBP-3 (recombinant human insulin-like growth factor binding protein-3) is Insmed’s proprietary anti-cancer compound that has demonstrated significant decreases in cancerous growth in several models of human. It is developed by Insmed and is currently unde…

Target Protein:
Insulin-like growth factor 1 receptor
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rhMBL DB05237
biotech

rhMBL is a protein therapeutic being developed by Enzon for the prevention and treatment of severe infections in individuals with low levels of Mannose-Binding Lectin (MBL). Over 10 percent of the general population is estimated to be MBL-deficient. Natural M…

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small molecule | CAS: 104114-27-4

Deskripsi belum tersedia.

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Rhodotorula mucilaginosa Approved DB10701
biotech

Rhodotorula mucilaginosa is a fungus which can provoke allergic reactions. Rhodotorula mucilaginosa is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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rhThrombin Approved DB04923
biotech | CAS: 1270043-60-1

rhThrombin (recombinant human thrombin) is being developed by ZymoGenetics, Inc. as a general aid to achieving hemostasis during surgery. ZymoGenetics is developing rhThrombin, a recombinant form of human thrombin that is not derived from animal or human bloo…

Waktu ParuhApproximately 15 ho…
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Ribavirin Approved DB00811
small molecule | CAS: 36791-04-5

Producing a broad-spectrum activity against several RNA and DNA viruses, Ribavirin is a synthetic guanosine nucleoside and antiviral agent that interferes with the synthesis of viral mRNA. It is primarily indicated for use in treating hepatitis C and viral he…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +13
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1RNA-directed RNA polymerase LGenome polyprotein +2
Gen Terkait:
IFNL3
Waktu ParuhThe terminal half-l…
Vol. DistribusiRibavirin displays …
KlirensThe total apparent …
Genetik 1 Varian
small molecule | CAS: 1352921-29-9

Deskripsi belum tersedia.

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Ribaxamase DB16311
biotech | CAS: 1792207-66-9

Ribaxamase is under investigation in clinical trial NCT02563106 (A Study of SYN-004 for the Prevention of c.diff in Patients With a LRTI).

Kategori:
AmidohydrolasesAmino Acids, Peptides, and ProteinsEnzymes +3
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Ribitol DB14704
small molecule | CAS: 488-81-3

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydratesSugar Alcohols
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Ribociclib Approved DB11730
small molecule | CAS: 1211441-98-3

Ribociclib is a selective cyclin-dependent kinase inhibitor, a class of drugs that help slow the progression of cancer by inhibiting two proteins called cyclin-dependent kinase 4 and 6 (CDK4/6). These proteins, when over-activated, can enable cancer cells to …

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +17
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhAt steady-state in …
Vol. DistribusiAt steady-state, th…
KlirensAt steady-state in …
Genetik -
Riboflavin Approved DB00140
small molecule | CAS: 83-88-5

Nutritional factor found in milk, eggs, malted barley, liver, kidney, heart, and leafy vegetables. The richest natural source is yeast. It occurs in the free form only in the retina of the eye, in whey, and in urine; its principal forms in tissues and cells a…

Kategori:
Alimentary Tract and MetabolismBiological FactorsCoenzymes +14
Target Protein:
Riboflavin kinaseRiboflavin synthaseFlavin reductase (NADPH)
Waktu Paruh66-84 minutes
Vol. Distribusi-
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small molecule | CAS: 752-56-7

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +4
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Riboprine DB11933
small molecule | CAS: 7724-76-7

Ipa has been used in trials studying the treatment of Nausea and Surgical Site Infection.

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