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11778

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8554 (72.6%)
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6383 (54.2%)
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11778 (100.0%)

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Halaman 191 / 236
biotech

Recombinant super-compound interferon (rSIFN-co) is a recombinant version of interferon alpha with modified spatial configuration. This interferon has antiviral and antitumor activity.

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biotech

Red blood cell-encapsulated L-asparaginase is [Asparaginase Escherichia coli] encapsulated inside donor-derived red blood cells, which target cancer cells capable of altering asparagine and glutamine metabolism. It is being investigated in cancers.[L44923]

Kategori:
AmidohydrolasesAntineoplastic AgentsEnzymes +2
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Red pepper Approved DB14759
biotech

Red pepper allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Redaporfin DB17219
small molecule | CAS: 1224104-08-8

Deskripsi belum tersedia.

Kategori:
AmidesBiological FactorsHeterocyclic Compounds, Fused-Ring +3
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Refametinib DB06309
small molecule | CAS: 923032-37-5

Deskripsi belum tersedia.

Kategori:
AmidesAminesAniline Compounds +2
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Regadenoson Approved DB06213
small molecule | CAS: 313348-27-5

Regadenoson is an A2A adenosine receptor agonist that causes coronary vasodilation and used for myocardial perfusion imagining. Manufactured by Astellas and FDA approved April 10, 2008.

Kategori:
Adenosine A receptor agonistsAdenosine A2 Receptor AgonistsCardiac Therapy +6
Target Protein:
Adenosine receptor A2a
Waktu ParuhInitial phase: 2-4 …
Vol. DistribusiCentral compartment…
KlirensAverage plasma rena…
Genetik -
Reglitazar DB04971
small molecule | CAS: 170861-63-9

Reglitazar, an isoxazolidine-3,5-dione derivative, is being developed by Pfizer for the treatment of diabetes. It is the first non-thiazolidenedione to enter clinical trials.

Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gamma
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Regorafenib Approved DB08896
small molecule | CAS: 755037-03-7

Regorafenib is an orally-administered inhibitor of multiple kinases. It is used for the treatment of metastatic colorectal cancer, advanced gastrointestinal stromal tumours, and hepatocellular carcinoma. FDA approved on September 27, 2012. Approved use of Reg…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +31
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +15
Waktu ParuhRegorafenib, 160 mg…
Vol. DistribusiRegorafenib undergo…
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Regramostim DB05386
biotech | CAS: 127757-91-9

Regramostim (GM-CSF) is a differentially glycosylated factor produced mainly by activated T cells and macrophages. Endothelial cells and fibroblasts can also produce GM-CSF after exposure to TNF-?, IL-1, IL-2 and IFN-?. GM-CSF is found associated with extrace…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +10
Target Protein:
Granulocyte-macrophage colony-stimulating factor receptor subunit alphaGM-CSF receptor alpha subunit
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Regrelor DB05553
small molecule | CAS: 787548-03-2

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesHeterocyclic Compounds, Fused-RingNeurotransmitter Agents +8
Target Protein:
P2Y purinoceptor 12
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Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
LactonesPolyketides
Target Protein:
Actin, alpha skeletal muscle
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small molecule

Deskripsi belum tersedia.

Target Protein:
Actin, alpha skeletal muscle
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Relacatib DB06367
small molecule | CAS: 362505-84-8

Deskripsi belum tersedia.

Kategori:
Sulfur Compounds
Target Protein:
Cathepsin K
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Relacorilant DB14976
small molecule | CAS: 1496510-51-0

Relacorilant is under investigation in clinical trial NCT02804750 (Study to Evaluate CORT125134 in Patients With Cushing's Syndrome).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Glucocorticoid receptor
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Relamorelin DB12678
small molecule | CAS: 661472-41-9

Relamorelin has been investigated for the treatment and basic science of Gastroparesis, Gastric Motility, Diabetes Mellitus, Parkinson's Disease, and Chronic Constipation, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Relatlimab Approved DB14851
biotech | CAS: 1673516-98-7

Relatlimab is a human IgG4 monoclonal antibody and novel immune checkpoint inhibitor that targets lymphocyte activation gene-3 (LAG-3).[A246165,L41265] It was the first commercially developed anti-LAG-3 antibody, entering clinical trials in 2013,[A246155] and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Lymphocyte activation gene 3 protein
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensAt steady-state, th…
Genetik -
Relcovaptan DB13929
small molecule | CAS: 150375-75-0

Deskripsi belum tersedia.

Kategori:
Antiplatelet agentsHematologic AgentsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Oxytocin receptorVasopressin V1a receptor
Waktu Paruh-
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Reldesemtiv DB15256
small molecule | CAS: 1345410-31-2

Reldesemtiv is under investigation in clinical trial NCT03160898 (A Study to Evaluate Efficacy, Safety and Tolerability of CK-2127107 in Patients With Amyotrophic Lateral Sclerosis (ALS)).

Target Protein:
Troponin C, skeletal muscle
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Relebactam Approved DB12377
small molecule | CAS: 1174018-99-5

Relebactam is a diazabicyclooctane beta-lactamase inhibitor, similar in structure to [avibactam].[A181195,A181207] It includes a piperidine ring which reduces export from bacterial cells by producing a positive charge.[A181207] It is currently available in a …

Kategori:
Antibacterials for Systemic UseAntiinfectives for Systemic UseAza Compounds +6
Target Protein:
Beta-lactamaseBeta-lactamase TEMBeta-lactamase SHV-1 +3
Waktu ParuhRelebactam has a ha…
Vol. DistribusiRelebactam has a vo…
KlirensRelebactam has a re…
Genetik -
Relenopride DB12798
small molecule | CAS: 1221416-43-8

Relenopride has been used in trials studying the treatment of Chronic Idiopathic Constipation.

Kategori:
Acids, AcyclicAcids, CarbocyclicAmides +2
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
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biotech

Deskripsi belum tersedia.

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Relmapirazin DB19130
small molecule | CAS: 1313706-17-0

Relmapirazin is under investigation in clinical trial NCT05425719 (Pharmacokinetics and Safety of MB-102 (Relmapirazin) and the Medibeacon Transdermal GFR Measurement System in Evaluation of Kidney Function in Normal and Renal Compromised Subjects).

Target Protein:
Interleukin-3 receptor subunit alpha
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Reloxaliase DB15560
biotech | CAS: 202011-67-4

Reloxaliase is a crystalline formulation of oxalate decarboxylase derived from _Bacillus Subtilis_. Reloxaliase is under investigation in clinical trial NCT03456830 (Evaluate ALLN-177 in Patients With Enteric Hyperoxaluria).

Kategori:
Carbon-Carbon LyasesEnzymesEnzymes and Coenzymes +1
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Reloxiliase DB17653
biotech

Reloxiliase is a first-in-class, oral crystalline formulation of the oxalate-specific, microbial enzyme oxalate decarboxylase. It is being investigated for the treatment of hyperoxaluria.[A258823]

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Reltecimod DB16687
small molecule | CAS: 1447799-33-8

Reltecimod is under investigation in clinical trial NCT02469857 (Phase III Efficacy and Safety Study of AB103 in the Treatment of Patients With Necrotizing Soft Tissue Infections).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Differentiation +7
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Relugolix Approved DB11853
small molecule | CAS: 737789-87-6

Relugolix is a gonadotropin-releasing hormone (GnRH) receptor antagonist used in the treatment of several hormone-responsive conditions. It was first approved in Japan in 2019, under the brand name Relumina, for the symptomatic treatment of uterine fibroids,[…

Kategori:
AmidesAnti-Gonadotropin-Releasing HormonesAntiandrogens +30
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe average effecti…
Vol. Distribusi-
KlirensThe average renal c…
Genetik -
Remdesivir Approved DB14761
small molecule | CAS: 1809249-37-3

Severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) is the causative agent of coronavirus disease 2019 (COVID-19), which is a respiratory disease that is capable of progressing to viral pneumonia and acute respiratory distress syndrome (ARDS); COVID-…

Kategori:
Adenine NucleotidesAmino AcidsAmino Acids, Peptides, and Proteins +37
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1abReplicase polyprotein 1ab +1
Waktu ParuhRemdesivir has an e…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Remestemcel-L Approved DB13973
biotech

Remestemcel-L is a third-party, off-the-shelf suspension of ex-vivo cultured adult human mesenchymal stem cells intended for intravenous infusion. The mesenchymal stem cells are derived from the bone marrow of unrelated and human leukocyte antigen (HLA)–unmat…

Kategori:
Anti-Infective AgentsAnti-Inflammatory AgentsAntiviral Agents +6
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Remetinostat DB14869
small molecule | CAS: 946150-57-8

Remetinostat is under investigation in clinical trial NCT02213861 (Efficacy, Safety and Tolerability Study of SHAPE in IA, IB or IIA Cutaneous T-cell Lymphoma).

Kategori:
Acids, CarbocyclicBenzene Derivatives
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Remibrutinib DB16852
small molecule | CAS: 1787294-07-8

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
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Remifentanil Approved DB00899
small molecule | CAS: 132875-61-7

Remifentanil (marketed by Abbott as Ultiva) is a potent ultra short-acting synthetic opioid given to patients during surgery for pain relief and adjunctive to an anaesthetic. Remifentanil is a specific mu-type-opioid receptor agonist which means it reduces sy…

Kategori:
Acids, AcyclicAgents producing tachycardiaAgents that produce hypertension +24
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh1-20 minutes
Vol. Distribusi* 350 mL/kg * 452 …
Klirens* 40 mL/min/kg [you…
Genetik -
Remimazolam Approved DB12404
small molecule | CAS: 308242-62-8

Remimazolam is an ultra short-acting benzodiazepine used in the induction and maintenance of sedation during short (<30 minute) procedures.[L14647] Recent trends in anesthesia-related drug development have touted the benefits of so-called "soft drugs" - these…

Kategori:
BenzazepinesBenzodiazepine hypnotics and sedativesBenzodiazepines and benzodiazepine derivatives +8
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of re…
Genetik -
Remlarsen DB19131
biotech | CAS: 1848266-71-6

Remlarsen is under investigation in clinical trial NCT03601052 (Efficacy, Safety, and Tolerability of Remlarsen (MRG-201) Following Intradermal Injection in Subjects With a History of Keloids).

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Remternetug DB18994
biotech | CAS: 2571940-41-3

Remternetug is under investigation in clinical trial NCT05463731 (A Study of Remternetug (LY3372993) in Participants With Alzheimer's Disease (TRAILRUNNER-ALZ 1)).

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Remtolumab DB15128
biotech | CAS: 1791410-27-9

Remtolumab is under investigation in clinical trial NCT02433340 (Phase 2, Multicenter, Open-Label Extension (OLE) Study With ABT-122 in Rheumatoid Arthritis Subjects Who Have Completed the Preceding M12-963 Study).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +3
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Remune DB17772
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesHIV +2
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Renadirsen DB19132
small molecule | CAS: 1782108-31-9

Renadirsen is under investigation in clinical trial NCT04433234 (Long-term, Extension Study of Ds-5141b in Patients With Duchenne Muscular Dystrophy).

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Renvistobart DB19065
biotech | CAS: 2725062-35-9

Renvistobart is under investigation in clinical trial NCT02913313 (A Study of BMS-986207 Given Alone and in Combination With Nivolumab or With Nivolumab and Ipilimumab in Advanced Solid Tumors).

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Renzapride DB04917
small molecule | CAS: 112727-80-7

Renzapride is currently in Phase III clinical development in the United States for the treatment of constipation-predominant irritable bowel syndrome (IBS-C). It has been suggested that renzapride is effective in the treatment of irritable bowel syndrome with…

Kategori:
Acids, CarbocyclicAmidesAntidepressive Agents +8
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3A
Waktu Paruh-
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Repifermin DB06434
small molecule | CAS: 219527-63-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsFibroblast Growth Factors +3
Waktu Paruh-
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Repotrectinib Approved DB16826
small molecule | CAS: 1802220-02-5

Repotrectinib is a next-generation tyrosine kinase inhibitor (TKI) specifically designed to address resistance in the treatment of non-small cell lung cancer (NSCLC), specifically due to mutations in the ROS1 gene.[A262056] ROS1 mutations are one of the defin…

Kategori:
BCRP/ABCG2 InhibitorsCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +28
Target Protein:
Proto-oncogene tyrosine-protein kinase ROSHigh affinity nerve growth factor receptorBDNF/NT-3 growth factors receptor +1
Waktu ParuhThe repotrectinib m…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Reproterol DB12846
small molecule | CAS: 54063-54-6

Reproterol has been used in trials studying the treatment of Asthma, Exercise-Induced.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-Agonists +25
Waktu Paruh-
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Reproxalap DB16688
small molecule | CAS: 916056-79-6

Reproxalap (previously ADX 102 or NS-2) is a small molecule inhibitor being developed by Aldeyra Therapeutics investigated against dry eye disease, allergic conjunctivitis, noninfectious anterior uveitis, and Sjögren-Larsson syndrome.[L32990] NS-2 has orphan …

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
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biotech | CAS: 2085240-27-1

AT132 is under investigation in clinical trial NCT03199469 (Gene Transfer Clinical Study in X-linked Myotubular Myopathy).

Kategori:
Adeno-associated Viral Vector Therapies
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Reserpine Approved DB00206
small molecule | CAS: 50-55-5

An alkaloid found in the roots of Rauwolfia serpentina and R. vomitoria. Reserpine inhibits the uptake of norepinephrine into storage vesicles resulting in depletion of catecholamines and serotonin from central and peripheral axon terminals. It has been used …

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAlkaloids +37
Target Protein:
Synaptic vesicular amine transporterChromaffin granule amine transporterBaculoviral IAP repeat-containing protein 5
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Resiniferatoxin DB06515
small molecule | CAS: 57444-62-9

Resiniferatoxin (RTX) is a naturally occurring, ultrapotent capsaicin analog that activates the vanilloid receptor in a subpopulation of primary afferent sensory neurons involved in nociception (the transmission of physiological pain).

Kategori:
NeurotoxinsTerpenes
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
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Resiquimod DB06530
small molecule | CAS: 144875-48-9

A substance being studied in the treatment of some types of skin cancer. When put on the skin, resiquimod causes some immune cells to make certain chemicals that may help them kill tumor cells. It is also being studied to find out if adding it to a tumor vacc…

Kategori:
Immunologic FactorsImmunomodulatory AgentsToll-Like Receptor Agonists
Target Protein:
Toll-like receptor 7Toll-like receptor 8
Waktu Paruh-
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Reslizumab Approved DB06602
biotech | CAS: 241473-69-8

Reslizumab is a humanized interleukin-5 (IL-5) antagonist monoclonal antibody (IgG4 kappa) that is produced by recombinant DNA technology in murine myeloma non-secreting 0 (NS0) cells. IL-5 is a pro-inflammatory cytokine that is responsible for the growth and…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAntibodies +12
Target Protein:
Interleukin-5
Waktu ParuhThe half-life is ap…
Vol. DistribusiThe approximate vol…
KlirensReslizumab clearanc…
Genetik -
RESP301 DB16497
small molecule

RESP301 was under investigation in clinical trials for various conditions. It was studied in community patients at risk of viral infections, including SARS-CoV-2, in a terminated trial (NCT04858451) and adults with rifampicin-susceptible pulmonary tuberculosi…

Kategori:
Experimental Unapproved Treatments for COVID-19
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Respigam DB17765
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +8
Waktu Paruh-
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