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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Halaman 190 / 236
Ramoplanin DB04952
biotech | CAS: 76168-82-6

Ramoplanin is a novel glycolipodepsipeptide antibiotic under development for the treatment of CDAD.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ramucirumab Approved DB05578
biotech | CAS: 947687-13-0

Ramucirumab is a human monoclonal antibody (IgG1) against vascular endothelial growth factor receptor 2 (VEGFR2), a type II trans-membrane tyrosine kinase receptor expressed on endothelial cells. By binding to VEGFR2, ramucirumab prevents binding of its ligan…

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +20
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh15 days
Vol. Distribusi5.5 L
Klirens0.014 L/hour
Genetik -
Ranibizumab Approved DB01270
biotech | CAS: 347396-82-1

Ranibizumab is a recombinant humanized IgG1 kappa isotype monoclonal antibody fragment directed against human vascular endothelial growth factor A (VEGF-A), which is a glycoprotein implicated in the pathophysiology of age-related macular degeneration.[A2301, …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +19
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhThe estimated avera…
Vol. DistribusiThe apparent volume…
KlirensIn patients with re…
Genetik -
Ranirestat DB05327
small molecule | CAS: 147254-64-6

Ranirestat is a structurally novel and stereospecifically potent aldose reductase (AKR1B; EC 1.1.1.21) inhibitor, which contains a succinimide ring that undergoes ring-opening at physiological pH levels. It has been used in trials studying the treatment of M…

Kategori:
Aldehyde Reductase, antagonists & inhibitorsEnzyme Inhibitors
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ranitidine Approved DB00863
small molecule | CAS: 66357-35-5

Ranitidine is a commonly used drug, classified as a histamine H2-receptor antagonist, and belongs to the same drug class as [cimetidine] and [famotidine]. This drug helps to prevent and treat gastric-acid associated conditions, including ulcers, because of it…

Kategori:
Acid ReducersAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +29
Target Protein:
Histamine H2 receptorAcetylcholinesterase
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensRenal clearance is …
Genetik -
Ranpirnase DB04950
biotech | CAS: 196488-72-9

Ranpirnase is a ribonuclease enzyme found in <i>Rana pipiens</i> oocytes. It is being studied in the treatment of cancer. It is manufactured by Alfacell Corporation. It is the first ribonuclease to enter cancer clinical trials.

Kategori:
Antineoplastic AgentsEgg ProteinsEnzyme Inhibitors +6
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2143578-32-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Rapastinel DB11801
small molecule | CAS: 117928-94-6

Rapastinel has been used in trials studying the treatment of Depressive Disorder, Major and Obsessive-Compulsive Disorder (OCD).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rasagiline Approved DB01367
small molecule | CAS: 136236-51-6

Rasagiline is an irreversible inhibitor of monoamine oxidase and is used as a monotherapy in early Parkinson's disease or as an adjunct therapy in more advanced cases.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Parkinson Drugs +19
Target Protein:
Amine oxidase [flavin-containing] BApoptosis regulator Bcl-2
Waktu ParuhRasagiline has a me…
Vol. Distribusi* 87 L
Klirens-
Genetik -
Rasburicase Approved DB00049
biotech | CAS: 134774-45-1

Rasburicase is a recombinant urate-oxidase enzyme produced by a genetically modified <i>Saccharomyces cerevisiae</i> strain. The cDNA coding for rasburicase was cloned from a strain of _Aspergillus flavus_.

Kategori:
Antigout PreparationsDetoxifying Agents for Antineoplastic TreatmentEnzymes +7
Target Protein:
Uric acid
Waktu Paruh18 hours
Vol. Distribusi* 110 to 127 mL/kg …
Klirens-
Genetik -
biotech | CAS: 1587257-96-2

Rasdegafusp alfa is under investigation in clinical trial NCT03206047 (Atezolizumab, Guadecitabine, and CDX-1401 Vaccine in Treating Patients With Recurrent Ovarian, Fallopian Tube, or Primary Peritoneal Cancer).

Waktu Paruh-
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small molecule | CAS: 8063-17-0

Rauwolfia (Rauwolfia serpentina), also spelled _ravolphia_, is a medicinal plant in the milkweed family. The root of the plant is ground into a powder or sold in tablets or capsules. It is a compound commonly used in Asian medicine, which includes traditional…

Kategori:
AlkaloidsAntiadrenergic Agents, Centrally ActingAntihypertensive Agents +6
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhAfter oral ingestio…
Vol. Distribusi-
KlirensHepatically and ren…
Genetik -
Ravagalimab DB16676
biotech | CAS: 2050816-56-1

Ravagalimab is under investigation in clinical trial NCT03695185 (A Study to Investigate How Well Ravagalimab (ABBV-323) Works and How Safe It Is in Participants With Moderate to Severe Ulcerative Colitis Who Failed Prior Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravidasvir DB15652
small molecule | CAS: 1242087-93-9

Ravidasvir is under investigation in clinical trial NCT02961426 (Sofosbuvir Plus Ravidasvir for the Treatment of HCV Chronic Infection).

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins +6
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Ravoxertinib DB15281
small molecule | CAS: 1453848-26-4

Ravoxertinib is under investigation in clinical trial NCT01875705 (A Dose-Escalation Study of GDC-0994 in Patients With Locally Advanced or Metastatic Solid Tumors).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors +1
Target Protein:
Mitogen-activated protein kinase 3Mitogen-activated protein kinase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravuconazole DB06440
small molecule | CAS: 182760-06-1

Deskripsi belum tersedia.

Kategori:
Antifungal AgentsAzole AntifungalsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ravulizumab Approved DB11580
biotech | CAS: 1803171-55-2

Ravulizumab is a potent and selective complement 5 (C5) inhibitor. It is a humanized monoclonal IgG2/4 kappa antibody produced in Chinese hamster ovary (CHO) cells.[L39690] Ravulizumab was engineered from [eculizumab], another complement inhibitor, to increas…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +15
Target Protein:
Complement C5
Waktu ParuhThe mean (%CV) term…
Vol. DistribusiThe mean (%CV) volu…
KlirensThe mean (%CV) clea…
Genetik -
Razupenem DB12587
small molecule | CAS: 426253-04-5

Razupenem has been used in trials studying the treatment of Skin Infections.

Kategori:
Amidesbeta-LactamsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Razuprotafib DB16353
small molecule | CAS: 1008510-37-9

Razuprotafib, also known as AKB-9778, is a small-molecule inhibitor restoring Tie2 activation by inhibiting VE-PTP.[L27171,L27176] In investigations against diabetes and COVID-19, razuprotafib is self-administered by patients through subcutaneous injection.

Kategori:
AcidsAcids, NoncarboxylicAmines +2
Target Protein:
Receptor-type tyrosine-protein phosphatase betaAngiopoietin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
RC88 DB18697
biotech

RC88 is an antibody-drug conjugate comprising a humanized anti-mesothelin monoclonal antibody conjugated to monomethyl auristatin E (MMAE).

Waktu Paruh-
Vol. Distribusi-
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RCT1100 DB18830
biotech

RCT1100 is an investigational mRNA-based therapeutic that aims to treat primary ciliary dyskinesia caused by pathogenic mutations in DNAI1.[L50788]

Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Rebamipide Approved DB11656
small molecule | CAS: 90098-04-7

Rebamipide has been investigated for the treatment of Stomach Ulcer, Keratoconjunctivitis Sicca, and Gastric Adenoma and Early Gastric Cancer.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Peptides, and Proteins +11
Target Protein:
fMet-Leu-Phe receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebastinib DB13005
small molecule | CAS: 1020172-07-9

Rebastinib has been used in trials studying the treatment of Chronic Myeloid Leukemia. It is an inhibitor of Tie2 tyrosine kinase receptor and an antineoplastic agent.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Tyrosine-protein kinase ABL1Angiopoietin-1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebeccamycin DB14729
small molecule | CAS: 93908-02-2

Rebeccamycin is a weak topoisomerase I inhibitor isolated from _Nocardia sp_.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Rebimastat DB06573
small molecule | CAS: 259188-38-0

Deskripsi belum tersedia.

Kategori:
Matrix Metalloproteinases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1966978-67-5

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Reboxetine Approved DB00234
small molecule | CAS: 71620-89-8

Reboxetine is an antidepressant drug used in the treatment of clinical depression, panic disorder and ADD/ADHD. Its mesylate (i.e. methanesulfonate) salt is sold under tradenames including Edronax, Norebox, Prolift, Solvex, Davedax or Vestra. Reboxetine has t…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAntidepressive Agents +20
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh12.5 hours
Vol. Distribusi-
Klirens-
Genetik -
Recanaclotide DB15417
biotech | CAS: 1667762-62-0

Recanaclotide is under investigation in clinical trial NCT01712412 (Phase 2a Study of IW-9179 to Treat Functional Dyspepsia).

Waktu Paruh-
Vol. Distribusi-
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Recaticimab DB19302
biotech | CAS: 2361290-85-7

Recaticimab is under investigation in clinical trial NCT06467617 (Adebrelimab Plus Chemo and Recaticimab Perioperative Treatment for Resectable NSCLC).

Waktu Paruh-
Vol. Distribusi-
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Recifercept DB17899
biotech | CAS: 2226238-09-9

Deskripsi belum tersedia.

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Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 122320-05-2

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme InhibitorsPeptides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

B38-CAP is structured as a carboxypeptidase and derived from _Paenibacillus sp._ The molecule, an Angiotensin Converting Enzyme 2 (ACE2)-like enzyme, shares structural similarities to the mammalian ACE2. B38-CAP is an ACE2-like enzyme which decreases angioten…

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biotech

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biotech | CAS: 389069-73-2

Recombinant human kallikrein-1 is under investigation in clinical trial NCT01845064 (A Study to Evaluate the Safety and Effectiveness of DM199 in Healthy Subjects and Type 2 Diabetes Patients).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +9
Waktu Paruh-
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biotech

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biotech

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biotech

Plasma gelsolin (pGSN) is a protein found in the blood of healthy individuals which scavenges compounds left over from damaged tissues.

Kategori:
Amino Acids, Peptides, and ProteinsBiopolymersCalcium-Binding Proteins +9
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biotech

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biotech

The Recombinant SARS-CoV-2 Vaccine was created by inserting genes of the SARS-CoV-2 spike protein’s receptor-binding domain into a baculovirus expression system[F4738, A226853]. In pre-clinical trial testing on mice, rabbits, and non-human primates, the candi…

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biotech

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Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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biotech

Recombinant stabilized RSV B prefusion F antigen is one component of a bivalent respiratory syncytial virus (RSV) vaccine called Abrysvo. The vaccine comprises two antigens - the other being [recombinant stabilized RSV A prefusion F antigen] - which have been…

Kategori:
Respiratory syncytial virus (RSV) vaccinesVaccinesViral Vaccines
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