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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 190 / 315
Manitimus DB06481
small molecule | CAS: 202057-76-9

FK778, a novel compound with multiple mechanisms of action, is efficacious, well tolerated and safe in kidney transplant patients, potentially offering a breakthrough in immunosuppressive therapy.

Kategori:
Hydrocarbons, Acyclic
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mannitol Approved DB00742
small molecule | CAS: 69-65-8

Mannitol is an osmotic diuretic that is metabolically inert in humans and occurs naturally, as a sugar or sugar alcohol, in fruits and vegetables. Mannitol elevates blood plasma osmolality, resulting in enhanced flow of water from tissues, including the brain…

Kategori:
Agents causing hyperkalemiaAlcoholsAlimentary Tract and Metabolism +31
Waktu ParuhMannitol has an eli…
Vol. DistribusiMannitol administer…
KlirensIntravenous adminis…
Genetik -
Mannitol busulfan Approved DB12097
small molecule | CAS: 1187-00-4

Mm has been used in trials studying the treatment of Cocaine Dependence and Diabetes Mellitus, Type 2.

Kategori:
Agents causing hyperkalemia
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mannose DB12907
small molecule | CAS: 3458-28-4

Mannose is under investigation for the basic science of IUGR and Pregnancy.

Kategori:
CarbohydratesHexosesMonosaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 3672-15-9

Mannose 6-phosphate has been used in trials studying the treatment of Wound, Cicatrix, Wound-healing, and Re-epithelialisation.

Target Protein:
Cation-independent mannose-6-phosphate receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mannosulfan DB13334
small molecule | CAS: 7518-35-6

Deskripsi belum tersedia.

Kategori:
AlkanesAlkanesulfonatesAlkanesulfonic Acids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mant-Adp DB03126
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAdenine NucleotidesAminobenzoates +8
Target Protein:
Myosin-14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mapatumumab DB18945
biotech | CAS: 658052-09-6

Mapatumumab is under investigation in clinical trial NCT00094848 (Study of TRM-1 (TRAIL-R1 Monoclonal Antibody) in Subjects With Relapsed or Refractory Non-hodgkin's Lymphoma (NHL)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Maplirpacept DB18441
biotech

Maplirpacept is a recombinant fusion protein consisting of the CD47-binding domain of human signal regulatory protein alpha (SIRPa) linked to the IgG4 Fc region of human IgG.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mapracorat DB12041
small molecule | CAS: 887375-26-0

Mapracorat has been investigated for the treatment of Eczema and Atopic Dermatitis.

Kategori:
AlcoholsFatty AlcoholsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Maprotiline Approved DB00934
small molecule | CAS: 10262-69-8

Maprotiline is a tetracyclic antidepressant with similar pharmacological properties to tricyclic antidepressants (TCAs). Similar to TCAs, maprotiline inhibits neuronal norepinephrine reuptake, possesses some anticholinergic activity, and does not affect monoa…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +29
Target Protein:
Sodium-dependent noradrenaline transporterHistamine H1 receptorMuscarinic acetylcholine receptor M1 +10
Waktu ParuhAverage ~ 51 hours …
Vol. DistribusiMaprotiline and its…
Klirens-
Genetik -
Maralixibat Approved DB16226
small molecule | CAS: 716313-53-0

Maralixibat (also known as SHP625, LUM001, and lopixibat) is an ileal bile acid transporter inhibitor, like [odevixibat].[A236823,A239249,L38834] Maralixibat is indicated for the treatment of cholestatic pruritus in patients with Alagille syndrome.[L38834] …

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyBile Therapy +9
Target Protein:
Ileal sodium/bile acid cotransporterHepatic sodium/bile acid cotransporter
Waktu ParuhThe mean half life …
Vol. Distribusi-
Klirens-
Genetik -
Maraviroc Approved DB04835
small molecule | CAS: 376348-65-1

Maraviroc (brand-named Selzentry, or Celsentri outside the U.S.) is a chemokine receptor antagonist drug developed by the drug company Pfizer that is designed to act against HIV by interfering with the interaction between HIV and CCR5. It was originally label…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +15
Target Protein:
C-C chemokine receptor type 5
Waktu Paruh14-18 hours
Vol. Distribusi* 194 L
Klirens-
Genetik -
Marbofloxacin DB11426
small molecule | CAS: 115550-35-1

Marbofloxacin is a carboxylic acid, part of the third generation of antibiotic fluoroquinolones. It is used in veterinary medicine. A formulation of marbofloxacin combined with clotrimazole and dexamethasone is available under the name Aurizon.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mardepodect DB08387
small molecule | CAS: 898562-94-2

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Margetuximab Approved DB14967
biotech | CAS: 1350624-75-7

The HER2 oncoprotein, the product of the human _ERBB2_/mouse _neu_ genes, is a member of the HER family of receptor tyrosine kinases that includes the epidermal growth factor receptor (EGFR). Of the various subtypes of breast cancer, HER2-positive breast canc…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhMargetuximab has a …
Vol. DistribusiMargetuximab has a …
KlirensMargetuximab has a …
Genetik -
Maribavir Approved DB06234
small molecule | CAS: 176161-24-3

Maribavir is an inhibitor of the cytomegalovirus (CMV; HHV5) pUL97 kinase which is used to treat CMV infections in patients post-transplantation.[L39322] Most standard CMV therapies, such as [ganciclovir] or [foscarnet], target CMV DNA polymerase - while gene…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +14
Target Protein:
Serine/threonine protein kinase UL97
Waktu ParuhIn post-transplant …
Vol. DistribusiThe mean apparent s…
KlirensIn post-transplant …
Genetik -
biotech | CAS: 2760218-55-9

Maridebart Cafraglutide is under investigation in clinical trial NCT05669599 (Dose-ranging Study to Evaluate the Efficacy, Safety, and Tolerability of AMG 133 in Adult Subjects With Overweight or Obesity, With or Without Type 2 Diabetes Mellitus).

Waktu Paruh-
Vol. Distribusi-
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Marimastat DB00786
small molecule | CAS: 154039-60-8

Used in the treatment of cancer, Marmiastat is an angiogenesis and metastasis inhibitor. As an angiogenesis inhibitor it limits the growth and production of blood vessels. As an antimetatstatic agent it prevents malignant cells from breaching the basement mem…

Kategori:
AminesEnzyme InhibitorsHydroxy Acids +2
Target Protein:
Interstitial collagenase72 kDa type IV collagenaseStromelysin-1 +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 9007-34-5

Marine collagen, soluble is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAntioxidantsAntiplatelet agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Marizomib DB11762
small molecule | CAS: 437742-34-2

Marizomib has been used in trials studying the treatment of Cancer, Melanoma, Lymphoma, Glioblastoma, and Malignant Glioma, among others.

Waktu Paruh-
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Genetik -
Maropitant DB11427
small molecule | CAS: 147116-67-4

Maropitant, used as maropitant citrate, is a neurokinin receptor antagonist, which was developed by Zoetis specifically for the treatment of motion sickness and vomiting in dogs. It was approved by the FDA in 2007 for use in dogs, and more recently has also b…

Kategori:
AntiemeticsAutonomic AgentsBenzene Derivatives +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Marstacimab Approved DB17725
biotech | CAS: 1985638-39-8

Marstacimab is a human monoclonal immunoglobulin G Type 1 (IgG1) antibody produced by Chinese hamster ovary (CHO) cells by recombinant DNA technology.[L51803] It is a tissue factor pathway inhibitor (TFPI) antagonist, which is an endogenous anticoagulant.[A26…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Tissue factor pathway inhibitor
Waktu ParuhIn a study consisti…
Vol. DistribusiIn patients with he…
KlirensIn a study consisti…
Genetik -
Martinostat DB14979
small molecule | CAS: 1629052-58-9

Martinostat is under investigation in clinical trial NCT03721211 (Imaging With [11C]Martinostat in Breast Cancer).

Kategori:
AminesBridged-Ring CompoundsCarbon Radioisotopes +3
Target Protein:
Histone deacetylase 7Histone deacetylase 9Histone deacetylase 8 +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1600492-21-4

Marzeptacog alfa (activated) is under investigation in clinical trial NCT01439971 (Phase 1 Safety, Pharmacokinetics And Pharmacodynamics Study Of Recombinant Factor VIIa Variant (813d) In Adult Subjects With Hemophilia).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +10
Waktu Paruh-
Vol. Distribusi-
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Genetik -
MAS825 DB16452
small molecule

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Masilukast DB16227
small molecule | CAS: 136564-68-6

Masilukast is under investigation in clinical trial NCT01740986 (Safety and Efficacy of SA09012 in Asthma).

Target Protein:
Cysteinyl leukotriene receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Masitinib DB11526
small molecule | CAS: 790299-79-5

Masitinib is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in dogs. It has been available in Europe since 2009, under the brand name Masivet. In the USA it is distributed under the name Kinavet and has been available for veterinaries s…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +5
Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Masoprocol Approved DB00179
small molecule | CAS: 27686-84-6

A potent lipoxygenase inhibitor that interferes with arachidonic acid metabolism. The compound also inhibits formyltetrahydrofolate synthetase, carboxylesterase, and cyclooxygenase to a lesser extent. It also serves as an antioxidant in fats and oils. [PubChe…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +16
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenaseReceptor tyrosine-protein kinase erbB-2Transient receptor potential cation channel subfamily M member 7 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Matairesinol DB04200
small molecule | CAS: 580-72-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzyl CompoundsPlants
Target Protein:
Dehydrogenase/reductase SDR family member 4-like 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Matrix-M DB16369
biotech

Matrix-M is a saponin-based adjuvant made of nanometer particles, cholesterol, and phospholipid that is developed by Novavax.[L27981] This compound is administered alongside vaccines to enhance biological functions: creating robust and long-lasting immune res…

Kategori:
CarbohydratesGlycosidesNanostructures
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Matuzumab DB05101
biotech | CAS: 339186-68-4

Matuzumab (formerly known as the experimental drug, EMD 72000) is a humanized monoclonal antibody used in cancer treatment. It has a high affinity for EGFR (epithelial growth factor receptor), frequently associated with the growth of blood vessels in malignan…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Epidermal growth factor receptor
Waktu Paruh196 hours
Vol. Distribusi-
Klirens-
Genetik -
Mavacamten Approved DB14921
small molecule | CAS: 1642288-47-8

Mavacamten is a myosin inhibitor indicated for the treatment of adults with symptomatic New York Heart Association (NYHA) class II-III obstructive hypertrophic cardiomyopathy (HCM). It received initial US FDA approval in 2022, and it is one of the first myosi…

Kategori:
AminesBenzene DerivativesBenzyl Compounds +21
Target Protein:
Myosin-7
Waktu ParuhMavacamten has a va…
Vol. DistribusiThrough the use of …
KlirensMavacamten demonstr…
Genetik -
Mavatrep DB12875
small molecule | CAS: 956274-94-5

Mavatrep has been used in trials studying the treatment of Osteoarthritis, Knee.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mavelertinib DB16228
small molecule | CAS: 1776112-90-3

Mavelertinib is under investigation in clinical trial NCT02349633 (Study for Patients With NSCLC EGFR Mutations (Del 19 or L858R +/- T790M)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Maveropepimut-S DB17339
biotech

Maveropepimut-S is a T cell activating immunotherapy.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mavodelpar DB17662
small molecule | CAS: 942594-93-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mavoglurant DB13004
small molecule | CAS: 543906-09-8

Mavoglurant has been used in trials studying the treatment of Patient Diagnosed With OCD and and Resistant to SSRI Treatment (Failed SSRI Over 12 Weeks at Appropriate Doses).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mavorixafor Approved DB05501
small molecule | CAS: 558447-26-0

Mavorixafor is a CXC chemokine receptor 4 (CXCR4) antagonist.[L50642] It was first approved by the FDA on April 30, 2024, for the treatment of warts, hypogammaglobulinemia, infections, and myelokathexis (WHIM) syndrome, a genetic immunodeficiency disorder cha…

Kategori:
AlkanesAminesButanes +38
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiMavorixafor volume …
KlirensThe mean (CV%) appa…
Genetik -
Mavrilimumab DB12534
biotech | CAS: 1085337-57-0

Mavrilimumab has been investigated for the treatment of Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MAX-40279 DB15191
small molecule | CAS: 2070931-57-4

MAX-40279 is under investigation in clinical trial NCT03412292 (MAX-40279 in Subjects With Acute Myelogenous Leukemia (AML)).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Maxacalcitol DB06272
small molecule | CAS: 103909-75-7

Deskripsi belum tersedia.

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsCholestanes +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MaxAdFVIII DB17713
biotech

MaxAdFVIII is an adenoviral vector that expresses the full-length human Factor VIII (hFVIII) cDNA. First developed by GenStar, it is being investigated for the treatment of hemophilia.

Waktu Paruh-
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Maxy-G34 DB05718
biotech

MAXY-G34 is a pegylated variant of human granulocyte-colony stimulating factor (G-CSF). This variant contains multiple non-naturally occurring lysines that have been introduced into alpha helixes of wild type human G-CSF as PEGylation sites, and from which mu…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mazaticol DB13448
small molecule | CAS: 42024-98-6

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAgents producing tachycardia +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mazdutide DB19099
biotech | CAS: 2259884-03-0

Mazdutide is under investigation in clinical trial NCT06143956 (A Chronic Weight Management Master Protocol Study (LY900038) of Multiple Intervention-specific-appendices (Isas) in Adult Participants With Obesity or Overweight).

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mazindol Approved DB00579
small molecule | CAS: 22232-71-9

Mazindol is a tricyclic anorexigenic agent that is unrelated to and less toxic than [amphetamine], but with some similar side effects. It inhibits uptake of catecholamines and blocks the binding of cocaine to the dopamine uptake transporter. Mazindol is only …

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAlimentary Tract and Metabolism +19
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent dopamine transporterSodium-dependent serotonin transporter +1
Waktu Paruh10-13 hours
Vol. Distribusi-
Klirens-
Genetik -
Mazorelvimab DB17767
biotech | CAS: 2419087-89-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

MB-102 are autologous T cells genetically modified to express CD123-specific, hinge-optimized CD28-costimulatory chimeric receptor and a truncated human epidermal growth factor receptor.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Menampilkan 9451–9500 dari 15718
Sebelumnya Halaman 190 / 315 Berikutnya