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2279

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Halaman 19 / 46
Galcanezumab Approved DB14042
biotech | CAS: 1578199-75-3

Galcanezumab is a humanized monoclonal antibody developed by Eli Lilly and Company against human calcitonin gene-related peptide (CGRP).[A33105] Although several small-molecule CGRP receptor antagonists have been developed, humanized monoclonal antibodies lik…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +15
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhBetween 1 and 600 m…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Galegenimab DB18860
biotech | CAS: 2403683-24-7

Galegenimab is under investigation in clinical trial NCT03972709 (A Study Assessing the Safety, Tolerability, and Efficacy of Galegenimab (FHTR2163) in Participants With Geographic Atrophy Secondary to Age-related Macular Degeneration (AMD)).

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Galidesivir DB11676
small molecule | CAS: 249503-25-1

Galidesivir is an adenosine analogue that has been investigated for use against Zaire Ebolavirus.[A191451] In animal studies, galidesivir was effective in increasing the survival rates from infections caused by various pathogens, including Ebola, Marburg, Yel…

Kategori:
Anti-Infective AgentsAntiviral AgentsCarbohydrates +9
Target Protein:
RNA-directed RNA polymerase L
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gallium Ga-68 gozetotide Approved DB16019
small molecule | CAS: 1906894-20-9

Gallium (Ga) 68 prostate-specific membrane antigen (PSMA)-11, or Ga-68 gozetotide, is a radiopharmaceutical agent used to identify and assess prostate-specific membrane antigen (PSMA)-positive lesions in adult men with prostate cancer during positron emission…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic RadiopharmaceuticalsDiagnostic Uses of Chemicals +14
Target Protein:
Prostate-specific antigenGlutamate carboxypeptidase 2
Waktu ParuhGallium-68 (Ga-68) …
Vol. DistribusiGa-68 PSMA-11 accum…
KlirensThere is limited in…
Genetik -
Galsulfase Approved DB01279
biotech | CAS: 552858-79-4

Galsufase is a variant form of the polymorphic human enzyme N-acetylgalactosamine 4-sulfatase of recombinant DNA origin. Galsulfase is a glycoprotein with a molecular weight of approximately 56 kD. The recombinant protein is comprised of 495 amino acids and c…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsArylsulfatases +9
Target Protein:
Dermatan sulfate
Waktu Paruh9 (6 to 21) minutes…
Vol. DistribusiWeek 1: 56-323 mL/k…
Klirens-
Genetik -
Gam-COVID-Vac DB15848
biotech

Gam-COVID-Vac was created by Gamaleya Research Institute of Epidemiology and MIcrobiology in Russia. The vaccine candidate is a heterologous COVID-19 vaccine containing two components, recombinant adenovirus type 26 (rAd26) vector and recombinant adenovirus t…

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Genetik -
Gamolenic acid Approved DB13854
small molecule | CAS: 506-26-3

Gamolenic acid, or gamma-linolenic acid (?-Linolenic acid) or GLA, is an essential fatty acid (EFA) comprised of 18 carbon atoms with three double bonds [F27] that is most commonly found in human milk and other botanical sources [A32848]. It is an omega-6 pol…

Kategori:
Agents that reduce seizure thresholdDermatologicalsFatty Acids +5
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Gantenerumab DB12034
biotech | CAS: 1043556-46-2

Alzheimer's disease (AD) is the most common cause of dementia in elderly patients, with classical histopathological hallmarks including extracellular amyloid-beta (A?) plaques and intraneuronal neurofibrillary tangles (NFTs). As the classical view of AD patho…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhGantenerumab admini…
Vol. Distribusi-
Klirens-
Genetik -
Garadacimab DB15629
biotech | CAS: 2162134-62-3

Garadacimab is under investigation in clinical trial NCT04281524 (A Clinical Study to Test the Efficacy and Safety of CSL312 on Catheter-associated Blood Clot Formation in Subjects With Cancer Who Receive Chemotherapy Through a PICC Line).

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Gatipotuzumab DB18861
biotech | CAS: 1264737-26-9

Gatipotuzumab is under investigation in clinical trial NCT01899599 (Pankomab-gex™ Versus Placebo as Maintenance Therapy in Advanced Ovarian Cancer).

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Genetik -
biotech

Gavocabtagene autoleucel is a novel cell therapy consisting of autologous genetically engineered T cells expressing a single-domain antibody that recognizes human Mesothelin, fused to the CD3-epsilon subunit which, upon expression, is incorporated into the en…

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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
GDP-mannose 6-dehydrogenase
Waktu Paruh-
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Genetik -
Gebasaxturev DB17296
biotech | CAS: 2122169-83-7

Deskripsi belum tersedia.

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Gefitinib Approved DB00317
small molecule | CAS: 184475-35-2

Gefitinib (originally coded ZD1839) is a drug used in the treatment of certain types of cancer. Acting in a similar manner to erlotinib (marketed as Tarceva), gefitinib selectively targets the mutant proteins in malignant cells. It is marketed by AstraZeneca …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +25
Target Protein:
Epidermal growth factor receptor
Gen Terkait:
EGFR EGFR EGFR +1
Waktu Paruh48 hours [IV admini…
Vol. Distribusi* 1400 L [IV admini…
Klirens* 595 mL/min [IV ad…
Genetik 4 Varian
Gefurulimab DB18928
biotech | CAS: 2456407-94-4

Gefurulimab is under investigation in clinical trial NCT05556096 (Safety and Efficacy of ALXN1720 in Adults With Generalized Myasthenia Gravis).

Waktu Paruh-
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Gemtuzumab ozogamicin Approved DB00056
biotech | CAS: 220578-59-6

Gemtuzumab ozogamicin is a recombinant humanized IgG4 kappa antibody which is conjugated with calicheamicin derivative, a cytotoxic antitumor antibiotic isolated from fermentation of Micromonospora echinospora ssp. calichensis. Gemtuzumab ozogamicin has appro…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +28
Target Protein:
Myeloid cell surface antigen CD33Low affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +1
Waktu ParuhIn pediatric patien…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Genistein DB01645
small molecule | CAS: 446-72-0

An isoflavonoid derived from soy products. It inhibits protein-tyrosine kinase and topoisomerase-II (DNA topoisomerases, type II) activity and is used as an antineoplastic and antitumor agent. Experimentally, it has been shown to induce G2 phase arrest in hum…

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsBCRP/ABCG2 Inhibitors +31
Target Protein:
Estrogen receptor betaNuclear receptor coactivator 1Estrogen receptor +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gentulizumab DB18148
biotech

Deskripsi belum tersedia.

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Genetik -
Geraniol Approved DB14183
small molecule | CAS: 106-24-1

Geraniol is a monoterpene that is found within many essential oils of fruits, vegetables, and herbs including rose oil, citronella, lemongrass, lavender, and other aromatic plants. It is emitted from the flowers of many species of plant and is commonly used b…

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseMonoterpenes +2
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu ParuhIn vitro measuremen…
Vol. Distribusi-
Klirens-
Genetik -
GI-101 DB17243
biotech

GI-101 is a bi-specific fragment crystallizable region (Fc) fusion protein containing a cluster of differentiation 80 ectodomain as an N-terminal moiety and interleukin-2 variant as a C-terminal moiety conjugated with human immunoglobulin G4 Fc.

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Genetik -
GI-181771X DB12309
small molecule | CAS: 305366-98-7

Gski181771 X is under investigation in clinical trial NCT00600743 (Effect of a CCK-1R Agonist on Food Intake in Humans).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-RingReceptor, Cholecystokinin A, agonists
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Giloralimab DB18862
biotech | CAS: 2226292-20-0

Giloralimab is under investigation in clinical trial NCT04807972 (Study to Evaluate Adverse Events and Change in Disease Activity When Intravenous (IV) Infusion of ABBV-927 Is Administered in Combination With IV Modified FOLFIRINOX (Mffx) With or Without IV B…

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Genetik -
Gingerol DB19255
small molecule | CAS: 23513-14-6

Gingerol is under investigation in clinical trial NCT05882864 (Efficacy of Ginger Muco-bioadhesive Gel in Management of Oral Lichen Planus With Immunohistochemical Analysis).

Kategori:
AlcoholsBenzene DerivativesLipids +2
Target Protein:
Transient receptor potential cation channel subfamily A member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginisortamab DB18863
biotech | CAS: 2390147-17-6

Ginisortamab is under investigation in clinical trial NCT04393298 (A Study to Assess the Safety, Pharmacokinetics and Anti Tumor Activity of UCB6114 Administered Intravenously to Participants With Advanced Solid Tumors).

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Ginkgo biloba Approved DB01381
biotech | CAS: 90045-36-6

_Ginkgo biloba_ extract contains a group of terpene lactones (notably, ginkgolides and diterpenes) and ginkgo flavone glycosides (notably, ginkgetin, bilobetin, and sciadopitysin) that have antioxidant and vasoactive properties.[A232389] Most of the studies t…

Kategori:
Anti-Dementia DrugsBiological ProductsBlood Circulation +27
Target Protein:
Sodium-dependent noradrenaline transporterPhospholipase A2, membrane associatedGlycine receptor subunit alpha-1 +5
Waktu ParuhUnpublished human d…
Vol. DistribusiNo data available.
KlirensNo data available.
Genetik -
Girentuximab DB05304
biotech | CAS: 916138-87-9

Girentuximab is a monoclonal chimeric (mouse/human) antibody directed against carbonic anhydrase IX, an antigen expressed in 95% of clear cell renal cell carcinomas (RCC).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Carbonic anhydrase 9Interleukin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2166101-71-7

Giroctocogene fitelparvovec is under investigation in clinical trial NCT04370054 (Study to Evaluate the Efficacy and Safety of PF-07055480 in Moderately Severe to Severe Hemophilia a Adults).

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GIVI-MPC DB17905
biotech

GIVI-MPC is a therapy that uses human-induced pluripotent stem cell-derived myogenic progenitor cells.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Givosiran Approved DB15066
biotech | CAS: 1639325-43-1

Givosiran is a small interfering RNA (siRNA) directed towards 5-aminolevulinic acid synthase, a critical enzyme in the heme biosynthesis pathway.[L10202] It is manufactured by Alnylam Pharmaceuticals and was first approved for use in the United States in Nove…

Kategori:
Alimentary Tract and MetabolismAmino SugarsAminolevulinate Synthase 1-directed RNA Interaction +13
Target Protein:
ALAS1 mRNA5-aminolevulinate synthase, non-specific, mitochondrial
Waktu ParuhBoth givosiran and …
Vol. DistribusiThe apparent centra…
KlirensThe apparent cleara…
Genetik -
GL-2045 DB16971
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Glatiramer Approved DB05259
biotech | CAS: 28704-27-0

Glatiramer acetate is a mix of synthetic polypeptides that includes L-glutamic acid, L-alanine, L-tyrosine, and L-lysine at an average molar fraction of 0.141, 0.427, 0.095, and 0.338, respectively.[L41940] Since glatiramer acetate is a heterogeneous drug, th…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +5
Target Protein:
MHC class II protein complex
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Glenzocimab DB16175
biotech | CAS: 2101829-58-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glimepiride Approved DB00222
small molecule | CAS: 93479-97-1

First introduced in 1995, glimepiride is a member of the second-generation sulfonylurea (SU) drug class used for the management of type 2 diabetes mellitus (T2DM) to improve glycemic control. Type 2 diabetes is a metabolic disorder with increasing prevalences…

Kategori:
Alimentary Tract and MetabolismAmidesBlood Glucose Lowering Agents +12
Target Protein:
ATP-binding cassette sub-family C member 9ATP-sensitive inward rectifier potassium channel 11ATP-sensitive inward rectifier potassium channel 1 +1
Waktu ParuhThe elimination hal…
Vol. DistribusiFollowing intraveno…
KlirensA single-dose, cros…
Genetik -
Glofitamab Approved DB16371
biotech | CAS: 2229047-91-8

Glofitamab is a full-length bispecific monoclonal antibody with affinity for both CD20 and CD3 surface antigens found on B- and T-cells, respectively. It has a 2:1 configuration, with bivalency towards CD20 and monovalency towards CD3, and works by recruiting…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3
Waktu ParuhThe transition from…
Vol. DistribusiFollowing intraveno…
KlirensGlofitamab's serum …
Genetik -
biotech | CAS: 107444-51-9

GLP-1 (7-36) amide is under investigation in clinical trial NCT01185119 (Effect of GLP-1 on Glucose Metabolism in CNS Assessed by PET).

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesGlucagon-Like Peptides +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GLPG-0492 DB12461
small molecule | CAS: 1215085-92-9

Glpg0492 is under investigation in clinical trial NCT01130818 (First-in-Human Single Ascending Dose of GLPG0492).

Kategori:
AndrogensImidazolesImidazolidines
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glucagon Approved DB00040
biotech | CAS: 16941-32-5

Glucagon is a 29 amino acid hormone used as a diagnostic aid in radiologic exams to temporarily inhibit the movement of the gastrointestinal tract and to treat severe hypoglycemia.[L7634,L7637,L7640,L7643,L8519] Glucagon raises blood sugar through activation …

Kategori:
Amino Acids, Peptides, and ProteinsAntihypoglycemic AgentDecreased GI Motility +19
Target Protein:
Glucagon receptorGlucagon-like peptide 2 receptorGlucagon-like peptide 1 receptor
Waktu ParuhThe half life of gl…
Vol. DistribusiThe volume of distr…
KlirensA 1mg intravenous d…
Genetik -
Glucarpidase Approved DB08898
biotech | CAS: 9074-87-7

Glucarpidase is a recombinant carboxypeptidase G2 produced by genetically modified _Escherichia coli_ bacteria. It is a 390-amino acid homodimer protein.[L39855] High-dose [methotrexate], an antifolate agent, has been widely and safely used for many decades i…

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesCarboxypeptidases +8
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn healthy adults w…
KlirensThe mean systemic c…
Genetik -
small molecule | CAS: 56-73-5

An ester of glucose with phosphoric acid, made in the course of glucose metabolism by mammalian and other cells. It is a normal constituent of resting muscle and probably is in constant equilibrium with fructose-6-phosphate. (Stedman, 26th ed)

Kategori:
CarbohydratesGlucosephosphatesHexosephosphates +1
Target Protein:
Glutamine--fructose-6-phosphate aminotransferase [isomerizing]Glucose-6-phosphate isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 80143-57-3

Glutamine 2-n-15 is under investigation in clinical trial NCT01912235 (Arginine Synthesis in Healthy Adult Humans).

Waktu Paruh-
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Genetik -
Glutathione Approved DB00143
small molecule | CAS: 70-18-8

A tripeptide with many roles in cells. It conjugates to drugs to make them more soluble for excretion, is a cofactor for some enzymes, is involved in protein disulfide bond rearrangement and reduces peroxides.

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesDietary Supplements +4
Target Protein:
Aldo-keto reductase family 1 member B1Matrix metalloproteinase-9Cytochrome P450 3A4 +38
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Glyburide Approved DB01016
small molecule | CAS: 10238-21-8

Glyburide is a second generation sulfonylurea used to treat patients with diabetes mellitus type II.[L8123] It is typically given to patients who cannot be managed with the standard first line therapy, [metformin].[L8123] Glyburide stimulates insulin secretio…

Kategori:
Alimentary Tract and MetabolismAmidesBCRP/ABCG2 Substrates +28
Target Protein:
ATP-binding cassette sub-family C member 8Sulfonylurea receptor 1, Kir6.2ATP-binding cassette sub-family C member 9 +6
Waktu ParuhElderly patients ha…
Vol. DistribusiElderly patients ha…
KlirensElderly patients ha…
Genetik -
Glycol salicylate Approved DB11323
small molecule | CAS: 87-28-5

Glycol salicylate, also known as _2-hydroxyethyl salicylate_, is a benzoate ester formed from the condensation of the carboxy group of salicylic acid with one of the hydroxy groups of ethylene glycol. It is found as an active ingredient and topical analgesic …

Kategori:
Acids, CarbocyclicAnti-Inflammatory AgentsAnti-Inflammatory Agents, Non-Steroidal +5
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhThe serum half-life…
Vol. Distribusi-
Klirens-
Genetik -
Goflikicept DB16396
biotech | CAS: 2416984-26-2

Goflikicept is under investigation in clinical trial NCT04380519 (Study of the Efficacy and Safety of a Single Administration of Olokizumab and RPH-104 With Standard Therapy in Patients With Severe Severe Acute Respiratory Syndrome Coronavirus 2 (Sars-cov-2) …

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gold DB14154
small molecule | CAS: 7440-57-5

A yellow metallic element with the atomic symbol Au, atomic number 79, and atomic weight 197. It is used in jewelry, goldplating of other metals, as currency, and in dental restoration. Many of its clinical applications, such as ANTIRHEUMATIC AGENTS, are in t…

Kategori:
Cell-mediated ImmunityElementsGold Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Golimumab Approved DB06674
biotech | CAS: 476181-74-5

Golimumab is a human IgG1? monoclonal antibody derived from immunizing genetically engineered mice with human TNF?. Golimumab binds and inhibits soluble and transmembrane human TNF?. Increased TNF? is associated with chronic inflammation. Thus golimumab is in…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +17
Target Protein:
Tumor necrosis factor
Waktu ParuhGolimumab has a lon…
Vol. DistribusiAfter IV administra…
KlirensAfter one IV dose o…
Genetik -
Golodirsen Approved DB15593
biotech | CAS: 1422959-91-8

Golodirsen is a morpholino antisense oligomer designed to treat about 8% of patients with Duchenne Muscular Dystrophy (DMD). This is an X-linked condition leading to progressive muscle degeneration that begins in early childhood, rendering many patients wheel…

Kategori:
Antisense Elements (Genetics)Antisense OligonucleotidesCompounds used in a research, industrial, or household setting +10
Target Protein:
Dystrophin
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe volume of distr…
KlirensThis drug is rapidl…
Genetik -
GPI-0100 DB05929
small molecule

GPI-0100 is Avantogen’s lead adjuvanat-immunopotentiator, a key component of vaccines for boosting the immune response. The GPI-0100 adjuvant, which has been shown to significantly enhance the immune response with a variety of vaccines, has been shown to hav…

Kategori:
CarbohydratesGlycosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Grazoprevir Approved DB11575
small molecule | CAS: 1350514-68-9

Grazoprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nin…

Kategori:
Acids, AcyclicAmidesAnti-Infective Agents +24
Target Protein:
Genome polyprotein
Waktu ParuhThe geometric mean …
Vol. DistribusiGrazoprevir has an …
KlirensThe clearance of Gr…
Genetik -
Gresonitamab DB18210
biotech | CAS: 2413817-97-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Menampilkan 901–950 dari 2279
Sebelumnya Halaman 19 / 46 Berikutnya