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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 189 / 252
Pentazocine Approved DB00652
small molecule | CAS: 359-83-1

The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97)

Kategori:
Adjuvants, AnesthesiaAgents that reduce seizure thresholdAlkaloids +20
Target Protein:
Sigma non-opioid intracellular receptor 1Mu-type opioid receptorKappa-type opioid receptor
Waktu Paruh2 to 3 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentetic acid Approved DB14007
small molecule | CAS: 67-43-6

Pentetic acid, also known as diethylenetriaminepentaacetic acid (DTPA), is a synthetic polyamino carboxylic acid with eight coordinate bond forming sites that can sequester metal ions and form highly stable DTPA-metal ion complexes. DTPA, along with its calci…

Kategori:
AcetatesAcids, AcyclicAmines +10
Target Protein:
Transuranium elements
Waktu ParuhIn preclinical stud…
Vol. DistribusiThe volume of distr…
KlirensPentetic acid prese…
Genetik -
Pentetrazol DB13415
small molecule | CAS: 54-95-5

Pentetrazol, also known as pentylenetetrazole, is a gamma-aminobutyric acid type A (GABA<sub>A</sub>) receptor antagonist that was approved by the FDA until 1982.[A254437]

Kategori:
AzepinesCentral Nervous System AgentsCentral Nervous System Stimulants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penthienate DB13695
small molecule | CAS: 22064-27-3

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentobarbital Approved DB00312
small molecule | CAS: 76-74-4

A short-acting barbiturate that is effective as a sedative and hypnotic (but not as an anti-anxiety) agent and is usually given orally. It is prescribed more frequently for sleep induction than for sedation but, like similar agents, may lose its effectiveness…

Kategori:
Adjuvants, AnesthesiaAnticholinergic AgentsAnticonvulsants +23
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3 +10
Waktu Paruh5 to 50 hours (dose…
Vol. Distribusi-
Klirens-
Genetik -
Pentolinium Approved DB01090
small molecule | CAS: 144-44-5

Pentolinium is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.

Kategori:
Anticholinergic AgentsAntihypertensive AgentsAutonomic Agents +7
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit alpha-3Neuronal acetylcholine receptor subunit beta-4 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentostatin Approved DB00552
small molecule | CAS: 53910-25-1

A potent inhibitor of adenosine deaminase. The drug is effective in the treatment of many lymphoproliferative malignancies, particularly hairy-cell leukemia. It is also synergistic with some other antineoplastic agents and has immunosuppressive activity.

Kategori:
Adenosine Deaminase InhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
Adenosine deaminase
Waktu Paruh5.7 hours (with a r…
Vol. Distribusi-
Klirens* 68 mL/min/m2
Genetik -
Pentoxifylline Approved DB00806
small molecule | CAS: 6493-05-6

Pentoxifylline (PTX) is a synthetic dimethylxanthine derivative that modulates the rheological properties of blood and also has both anti-oxidant and anti-inflammatory properties.[A226415, L30300] Although originally developed to treat intermittent claudicati…

Kategori:
AlkaloidsAntioxidantsAntiplatelet agents +23
Target Protein:
Adenosine receptor A2aTumor necrosis factorPhosphodiesterase enzymes +2
Waktu ParuhOverall, pentoxifyl…
Vol. DistribusiPentoxifylline has …
KlirensPentoxifylline give…
Genetik -
Peoniflorin DB16288
small molecule | CAS: 23180-57-6

Peoniflorin is under investigation in clinical trial NCT02878863 (Paeoniflorin Combination of Hepatoprotective Drugs Versus Hepatoprotective Drugs Only for Auto-immune Hepatitis).

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +8
Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PEP0101 DB18572
biotech

PEP0101 is a nanocomplex consisting of elastin-like polypeptides and a small interfering RNA (siRNA) designed to down-regulate the expression of EVI1 oncogene in cancer cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pepinemab DB15155
biotech | CAS: 2097151-87-4

Pepinemab is under investigation in clinical trial NCT03769155 (VX15/2503 With or Without Ipilimumab and/or Nivolumab in Patients With Resectable Stage IIIB-D Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peppermint oil Approved DB11198
biotech | CAS: 8006-90-4

Extracted from the stem, leaves, and flowers of _Mentha piperita_ L. plant, peppermint oil (Mentha piperita) is a popular essential oil used in aromatherapy for both external and internal use. Mentha piperita is a hybrid of spearmint (Mentha spicata) and wate…

Kategori:
Alimentary Tract and MetabolismAngiospermsAntiemetics +31
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Pepsin Approved DB13198
biotech | CAS: 9001-75-6

Pepsin is a potent enzyme in gastric juice that digests proteins such as those in meat, eggs, seeds, and dairy products [L2358]. Studies on gastric digestion from 1820-1840 led to the discovery of pepsin as the substance which, in the presence of stomach a…

Kategori:
Alimentary Tract and MetabolismAspartic Acid EndopeptidasesAspartic Acid Proteases +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 123583-37-9

Peptide YY (3-36), a synthetic human PYY 3-36, is a compound being evaluated for the treatment of obesity. It reduces appetite and increases satiety in obese patients.

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesHormones +3
Target Protein:
Neuropeptide Y receptor type 2Neuropeptide Y receptor type 1Neuropeptide Y receptor type 5 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peracetic acid DB14556
small molecule | CAS: 79-21-0

A liquid that functions as a strong oxidizing agent. It has an acrid odor and is used as a disinfectant.

Kategori:
AcetatesAcids, AcyclicAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peramivir Approved DB06614
small molecule | CAS: 330600-85-6

Peramivir is an antiviral agent developed by Biocryst Pharmaceuticals to treat influenza A/B. The development of peramivir has been supported by the US Department of Health and Human Services as part of the government's effort to prepare for a flu pandemic. B…

Kategori:
AmidinesAnti-Infective AgentsAntiinfectives for Systemic Use +6
Target Protein:
NeuraminidaseNeuraminidaseNeuraminidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perampanel Approved DB08883
small molecule | CAS: 380917-97-5

Perampanel is a noncompetitive AMPA glutamate receptor antagonist. It is marketed under the name Fycompa™ and is indicated as an adjunct in patients over 12 years old for the treatment of partial-onset seizures that may or may not occur with generalized seizu…

Kategori:
AMPA Receptor AntagonistsAnticonvulsantsCentral Nervous System Depressants +23
Target Protein:
Glutamate receptor 2Glutamate receptor 3Glutamate receptor 4 +1
Waktu ParuhPerampanel has a lo…
Vol. DistribusiThe volume of distr…
KlirensIn healthy patients…
Genetik -
Perboric acid Approved DB13235
small molecule | CAS: 14034-78-7

Perboric acid is mainly found in its salt form of sodium perborate and it can be found as a monohydrate or tetrahydrate.[A33037] It is one of the peroxy acid salts with very wide functionalities in industrial settings.[F66] Perboric acid in the form of sodium…

Kategori:
AcidsAlimentary Tract and MetabolismAnions +7
Waktu ParuhAs perboric acid an…
Vol. DistribusiAs perboric acid an…
KlirensAs perboric acid an…
Genetik -
Peresolimab DB18874
biotech | CAS: 2411580-63-5

Peresolimab is under investigation in clinical trial NCT04634253 (A Study of LY3462817 in Participants With Rheumatoid Arthritis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peretinoin DB16291
small molecule | CAS: 81485-25-8

Deskripsi belum tersedia.

Kategori:
AlkenesAnticarcinogenic AgentsBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perflenapent DB11625
small molecule | CAS: 678-26-2

Dodecafluoropentane is also known as perfluoropentane or perflenapent.

Kategori:
AlkanesCompounds used in a research, industrial, or household settingContrast Media +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perflexane Approved DB09531
small molecule | CAS: 355-42-0

Deskripsi belum tersedia.

Kategori:
Diagnostic AgentsHydrocarbons, FluorinatedHydrocarbons, Halogenated +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perflubron DB05791
small molecule | CAS: 423-55-2

Perflubron (Oxygent) is being developed as an intravascular oxygen carrier designed to augment oxygen delivery in surgical patients.

Kategori:
Anti-Obesity AgentsCompounds used in a research, industrial, or household settingContrast Media +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perflubutane Approved DB12821
small molecule | CAS: 355-25-9

Perflubutane has been used in trials studying the diagnostic of Liver Mass, Liver Diseases, Liver Metastasis, Portal Hypertension, and Peripheral Artery Disease. It is a cardiovascular drug designed to enable ultrasound to compete more effectively with nuclea…

Kategori:
AnionsCompounds used in a research, industrial, or household settingContrast Media +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 306-94-5

Perfluorodecalin is under investigation in clinical trial NCT03668665 (Influencing Wound Healing Through the Application of Hyaluronic Acid With Perfluorodecalin and Physalis Angulata Extract After Split Skin Removal From the Thigh - a Study in "Split Wound D…

Kategori:
Blood SubstitutesHydrocarbons, FluorinatedHydrocarbons, Halogenated +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perfluorohexyloctane Approved DB17823
small molecule | CAS: 133331-77-8

Perfluorohexyloctane is a semifluorinated alkane that contains six perfluorinated carbon atoms and eight hydrogenated carbon atoms.[L46491] It is an inert, slightly amphiphilic compound.[A259746] Because it is a completely non-aqueous liquid, microbial growth…

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, HalogenatedOphthalmic Solutions +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perfluorooctane DB15997
small molecule | CAS: 307-34-6

Deskripsi belum tersedia.

Kategori:
Hydrocarbons, FluorinatedHydrocarbons, Halogenated
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perflutren Approved DB00556
small molecule | CAS: 76-19-7

Perflutren, a diagnostic drug that is intended to be used for contrast enhancement during the indicated echocardiographic procedures, is comprised of lipid-coated microspheres filled with octafluoropropane(OFP) gas. When exposed to ultrasound waves, the micro…

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingContrast Media +10
Waktu ParuhThe mean half-life …
Vol. Distribusi-
Klirens-
Genetik -
Perfosfamide DB12727
small molecule | CAS: 62435-42-1

Perfosfamide has been used in trials studying the treatment of Lymphoma, Neuroblastoma, and Multiple Myeloma and Plasma Cell Neoplasm.

Kategori:
Hydrocarbons, HalogenatedMustard CompoundsNitrogen Mustard Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pergolide Approved DB01186
small molecule | CAS: 66104-22-1

Pergolide is a long-acting dopamine agonist approved in 1982 for the treatment of Parkinson’s Disease. It is an ergot derivative that acts on the dopamine D2 and D3, alpha2- and alpha1-adrenergic, and 5-hydroxytryptamine (5-HT) receptors. It was indicated as …

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +24
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +12
Waktu Paruh27 hours
Vol. Distribusi-
Klirens-
Genetik -
Perifosine DB06641
small molecule | CAS: 157716-52-4

Perifosine is a novel alkylphospholipid with antiproliferative properties attributed to protein kinase B inhibition.

Kategori:
AminesOnium CompoundsQuaternary Ammonium Compounds +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformRAC-alpha serine/threonine-protein kinaseMitogen-activated protein kinase 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18457-55-1

Perillyl alcohol is under investigation in clinical trial NCT02704858 (Safety and Efficacy Study in Recurrent Grade IV Glioma).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsPerilla +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perindoprilat DB14213
small molecule | CAS: 95153-31-4

The active metabolite of the prodrug [Perindopril].

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Permethrin Approved DB04930
small molecule | CAS: 52645-53-1

A pyrethroid insecticide commonly used in the treatment of lice infestations and scabies. It is a yellow to light orange-brown, low melt-ing solid or viscous liquid.

Kategori:
AgrochemicalsAntiparasitic Products, Insecticides and RepellentsBenzene Derivatives +22
Target Protein:
Sodium channel protein type 1 subunit alphaEstrogen receptorNuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perospirone DB08922
small molecule | CAS: 150915-41-6

Perospirone is an atypical or second-generation antipsychotic of the azapirone family that antagonizes serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist. Dainippon Sumitomo Pharma devel…

Kategori:
Antipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical])Central Nervous System Agents +13
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +3
Gen Terkait:
HTR1A
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean volume of …
KlirensApparent clearance …
Genetik 1 Varian
Perphenazine Approved DB00850
small molecule | CAS: 58-39-9

An antipsychotic phenothiazine derivative with actions and uses similar to those of chlorpromazine.

Kategori:
Antipsychotic AgentsAntipsychotic Agents (First Generation [Typical])Central Nervous System Agents +28
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorCalmodulin
Waktu Paruh8-12 hours, but ran…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 17528-28-8

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pertussis vaccine Approved DB15274
biotech

Pertussis vaccine is under investigation in clinical trial NCT01698346 (Pertussis (Tdap) Vaccination in Pregnancy).

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pertuzumab Approved DB06366
biotech | CAS: 380610-27-5

Pertuzumab is a recombinant humanized monoclonal antibody that targets the extracellular dimerization domain (subdomain II) of the human epidermal growth factor receptor 2 protein (HER2). It consists of two heavy chains and two lights chains that have 448 and…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhThe median half-lif…
Vol. DistribusiThe average steady-…
KlirensThe median clearanc…
Genetik -
Peruvoside DB13756
small molecule | CAS: 1182-87-2

Deskripsi belum tersedia.

Kategori:
CardanolidesCardiac GlycosidesCardiac Therapy +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Perzinfotel DB12365
small molecule | CAS: 144912-63-0

Perzinfotel has been used in trials studying the treatment of Diabetes Mellitus and Diabetic Neuropathy, Painful.

Kategori:
Aza CompoundsOrganophosphorus Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Petesicatib DB15297
small molecule | CAS: 1252637-35-6

Petesicatib is under investigation in clinical trial NCT02295332 (A Study of RG7625 in Healthy Volunteers).

Kategori:
Enzyme Inhibitors
Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Petosemtamab DB18948
biotech | CAS: 2213450-26-9

Petosemtamab is under investigation in clinical trial NCT03526835 (A Study of Bispecific Antibody MCLA-158 in Patients With Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Petrelintide DB19442
biotech | CAS: 2766385-23-1

Petrelintide is under investigation in clinical trial NCT06662539 (Once-weekly Petrelintide Versus Placebo for Obesity or Overweight With Co-morbidities).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Petrolatum Approved DB11058
small molecule | CAS: 8009-03-8

A colloidal system of semisolid hydrocarbons obtained from petroleum. It is used as an ointment base, topical protectant, and lubricant.

Kategori:
Basic Ointments and ProtectantsCompounds used in a research, industrial, or household settingDermatologicals +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PEV3A DB05144
biotech

PEV3A is a prophylactic malaria vaccine that acts against various stages of the disease. It is a two-component vaccine that contains the virosome formulated peptide mimetics PEV301 and PEV302. The two synthetic peptide vaccine components mimic the native stru…

Kategori:
Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pevonedistat DB11759
small molecule | CAS: 905579-51-3

Pevonedistat has been used in trials studying the treatment of Lymphoma, Solid Tumors, Multiple Myeloma, Hodgkin Lymphoma, and Metastatic Melanoma, among others.

Kategori:
CycloparaffinsEnzyme Inhibitors
Target Protein:
NEDD8-activating enzyme E1 catalytic subunitUbiquitin-like protein NEDD8NEDD8-activating enzyme E1 regulatory subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pexacerfont DB12572
small molecule | CAS: 459856-18-9

Pexacerfont has been investigated for the treatment of Alcoholism, Anxiety Disorder, Alcohol Dependence, and Alcohol-Related Disorders.

Target Protein:
Corticotropin-releasing factor receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1058624-46-6

Pexastimogene devacirepvec is under investigation in clinical trial NCT00429312 (A Study of Recombinant Vaccinia Virus to Treat Malignant Melanoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pexelizumab DB04949
biotech | CAS: 219685-93-5

Pexelizumab is a humanized monoclonal antibody used as an immunosuppressive drug. It is being investigated by Alexion Pharmaceuticals.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Waktu Paruh7.0 hours to 14.5 h…
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9401–9450 dari 12560
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