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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 189 / 321
Leridistim DB15095
biotech | CAS: 193700-51-5

Leridistim is under investigation in clinical trial NCT00004215 (Leridistim Compared With Filgrastim in Treating Older Patients With Acute Myeloid Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leriglitazone DB15021
small molecule | CAS: 146062-44-4

Leriglitazone is under investigation in clinical trial NCT03917225 (A Clinical Study to Evaluate the Effect of MIN-102 on the Progression of Friedreich's Ataxia in Male and Female Patients).

Kategori:
Alimentary Tract and MetabolismSulfur CompoundsThiazoles +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerisetron DB12964
small molecule | CAS: 143257-98-1

Lerisetron has been used in trials studying the supportive care of Nausea and Vomiting and Testicular Germ Cell Tumor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerociclib DB16218
small molecule | CAS: 1628256-23-4

Lerociclib is under investigation in clinical trial NCT02983071 (G1T38, a CDK 4/6 Inhibitor, in Combination With Fulvestrant in Hormone Receptor-positive, Her2-negative Locally Advanced or Metastatic Breast Cancer).

Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerodalcibep DB19071
biotech | CAS: 2250073-78-8

Lerodalcibep is under investigation in clinical trial NCT05004675 (Trial to Evaluate Efficacy and Safety of LIB003 and Inclisiran in High-risk CVD Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leronlimab DB05941
biotech | CAS: 674782-26-4

Leronlimab, or PRO-140, is a human monoclonal antibody developed by CytoDyn.[L12684] It was first described in the literature in 2001.[A3922] This antibody binds to CCR5, which may be useful in treating HIV, cancers, and severely ill COVID-19 patients.[A19284…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +17
Target Protein:
C-C chemokine receptor type 5
Waktu ParuhThe half life of a …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Lersivirine DB11649
small molecule | CAS: 473921-12-9

Lersivirine has been used in trials studying the treatment of HIV-1.

Kategori:
RNA-Directed DNA Polymerase
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lesinidase alfa DB15267
biotech | CAS: 1522433-40-4

Lesinidase alfa is under investigation in clinical trial NCT02324049 (Safety, Pharmacokinetics, and Pharmacodynamics/Efficacy of SBC-103 in Mucopolysaccharidosis III, Type B (MPS IIIB)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lesinurad Approved DB11560
small molecule | CAS: 878672-00-5

Lesinurad is an oral uric acid transporter 1 (URAT1) inhibitor indicated for the treatment of hyperuricemia associated with gout. It reduces serum uric acid concentration through the inhibition of URAT1, an enzyme responsible for reuptake of uric acid from th…

Kategori:
AcetatesAcids, AcyclicAntigout Preparations +15
Target Protein:
Solute carrier family 22 member 12Solute carrier family 22 member 11
Waktu Paruh-
Vol. DistribusiThe mean steady sta…
Klirens-
Genetik -
Lesogaberan DB11920
small molecule | CAS: 344413-67-8

Lesogaberan has been used in trials studying the treatment and basic science of GERD, Reflux, Heartburn, Regurgitation, and Reflux Disease, among others.

Kategori:
AcidsAcids, NoncarboxylicAmines +8
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid type B receptor subunit 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lesopitron DB04970
small molecule | CAS: 132449-46-8

Lesopitron is an anxiolytic with pre- and post-synaptic 5-HT1A agonist activity, which is under development by Esteve.

Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh1.1 to 5.6 hours
Vol. Distribusi-
Klirens-
Genetik -
Lestaurtinib DB06469
small molecule | CAS: 111358-88-4

Deskripsi belum tersedia.

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 InhibitorsCytochrome P-450 CYP3A4 Inhibitors (strength unknown) +4
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letaplimab DB16679
biotech | CAS: 2283356-07-8

Letaplimab is under investigation in clinical trial NCT04485052 (Efficacy and Safety Evaluation of IBI188 in Combination With Azacitidine in Treatment of Patients With Acute Myeloid Leukemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letaxaban DB11984
small molecule | CAS: 870262-90-1

Letaxaban has been used in trials studying the treatment and prevention of Venous Thromboembolism and Acute Coronary Syndrome.

Kategori:
AnticoagulantsAntithrombinsEnzyme Inhibitors +6
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letermovir Approved DB12070
small molecule | CAS: 917389-32-3

Letermovir recieved approval from the FDA on November 8th, 2017 for use in prophylaxis of cytomegalovirus (CMV) infection in allogeneic hematopoietic stem cell transplant patients.[L1021] It is the first of a new class of CMV anti-infectives called DNA termin…

Kategori:
Acids, AcyclicAnti-Infective AgentsAntiinfectives for Systemic Use +44
Target Protein:
CMV DNA Terminase Complex
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean steady sta…
KlirensThe mean clearance …
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LetibotulinumtoxinA Approved DB16820
biotech | CAS: 1800016-51-6

The aesthetic utility of botulinum toxin was discovered incidentally following its initial use in the treatment of facial spasmodic disorders in the early 1970s.[A249920] The first aesthetic use of botulinum toxin was reported in 1989, when [onabotulinumtoxin…

Kategori:
Acetylcholine Release InhibitorsBotulinum Toxins, Type ACentral Nervous System Depressants +2
Target Protein:
Synaptosomal-associated protein 25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letolizumab DB19072
biotech | CAS: 1450981-87-9

Letolizumab is under investigation in clinical trial NCT02273960 (Study to Evaluate Safety and Efficacy in Adult Subjects With ITP).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letosteine DB08939
small molecule | CAS: 53943-88-7

Letosteine is a mucolytic used in the treatment of chronic bronchopneumopathies and related conditions.

Kategori:
Cough and Cold PreparationsExpectorantsRespiratory System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letrazuril DB12663
small molecule | CAS: 103337-74-2

Letrazuril has been used in trials studying the treatment of HIV Infections and Cryptosporidiosis.

Kategori:
Nitriles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letrozole Approved DB01006
small molecule | CAS: 112809-51-5

Letrozole, or CGS 20267, is an oral non-steroidal type II aromatase inhibitor first described in the literature in 1990.[A190543,A1559,L11623,L11626] It is a third generation aromatase inhibitor like [exemestane] and [anastrozole], meaning it does not signifi…

Kategori:
Agents Causing Muscle ToxicityAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Aromatase
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Leucanthemum vulgare pollen Approved DB15529
biotech

Leucanthemum vulgare pollen allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leucine DB00149
small molecule | CAS: 61-90-5

An essential branched-chain amino acid important for hemoglobin formation.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +4
Target Protein:
Leucine--tRNA ligase, mitochondrialtRNA wybutosine-synthesizing protein 4Leucine carboxyl methyltransferase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease inhibitor Kazal-type 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leucovorin Approved DB00650
small molecule | CAS: 58-05-9

Folinic Acid (also known as 5-formyl tetrahydrofolic acid or leucovorin) is the 5-formyl derivative of tetrahydrofolic acid, a necessary co-factor in the body. Commercially available leucovorin is composed of a 1:1 racemic mixture of the dextrorotary and levo…

Kategori:
AntidotesCoenzymesCompounds used in a research, industrial, or household setting +15
Target Protein:
Proton-coupled folate transporterDihydrofolate reductase
Waktu Paruh6.2 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leukotriene B4 DB12961
small molecule | CAS: 71160-24-2

Leukotriene B4 has been used in trials studying the treatment of HIV Infections.

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +7
Target Protein:
Leukotriene B4 receptor 1Leukotriene B4 receptor 2Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leukotriene C4 DB08855
small molecule | CAS: 72025-60-6

The conjugation product of LEUKOTRIENE A4 and glutathione. It is the major arachidonic acid metabolite in macrophages and human mast cells as well as in antigen-sensitized lung tissue. It stimulates mucus secretion in the lung, and produces contractions of no…

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +8
Target Protein:
Cysteinyl leukotriene receptor 1Cysteinyl leukotriene receptor 2Multidrug resistance-associated protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leukotriene D4 DB11858
small molecule | CAS: 73836-78-9

Leukotriene D4 has been used in trials studying the diagnostic of Asthma and Allergic Rhinitis.

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +8
Target Protein:
Cysteinyl leukotriene receptor 1Cysteinyl leukotriene receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leupeptin DB16961
small molecule | CAS: 55123-66-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCathepsins, antagonists & inhibitorsCysteine Proteinase Inhibitors +4
Target Protein:
Plasmepsin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leuprolide Approved DB00007
biotech | CAS: 53714-56-0

Leuprolide is a synthetic 9-residue peptide analogue of gonadotropin-releasing hormone (GnRH). Unlike the endogenous decapeptide GnRH, leuprolide contains a single D-amino acid (D-leucyl) residue, which helps to increase its circulating half-life from three t…

Kategori:
Adrenal Cortex HormonesAgents Causing Muscle ToxicityAmino Acids, Peptides, and Proteins +25
Target Protein:
Gonadotropin-releasing hormone receptorProgonadoliberin-1
Waktu ParuhLeuprolide has a te…
Vol. DistribusiLeuprolide has an a…
KlirensLeuprolide administ…
Genetik -
Leuvectin DB17303
biotech

Leuvectin (formerly known as VCL-1102) is a component of gene therapy along with cationic lipid 1,2-dimyristyloxypropyl-3-dimethyl-hydroxyethyl ammonium bromide/dioleyl-phosphatidyl-ethanolamine (DMRIE/DOPE).[A254711]

Kategori:
Biological ProductsComplex MixturesGene Transfer Techniques +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levacetylmethadol Approved DB01227
small molecule | CAS: 1477-40-3

Levacetylmethadol is a narcotic analgesic with a long onset and duration of action. It is used mainly in the treatment of narcotic dependence. Levacetylmethadol was withdrawn from use in the European Union due to its high risk of QT interval prolongation.…

Kategori:
AnalgesicsAnticholinergic AgentsCentral Nervous System Agents +20
Target Protein:
Mu-type opioid receptorNeuronal acetylcholine receptor subunit beta-4Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh2.6 days
Vol. Distribusi-
Klirens-
Genetik -
Levallorphan Approved DB00504
small molecule | CAS: 152-02-3

An opioid antagonist with properties similar to those of naloxone; in addition it also possesses some agonist properties. It should be used cautiously; levallorphan reverses severe opioid-induced respiratory depression but may exacerbate respiratory depressio…

Kategori:
AlkaloidsCentral Nervous System AgentsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Mu-type opioid receptor
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Levamisole Approved DB00848
small molecule | CAS: 14769-73-4

Levamisole is an antihelminthic drug that was commonly used for the treatment of parasitic, viral, and bacterial infections. [A178117] It was manufactured by _Janssen_ and first used in 1969 as an agent to treat worm infestations[A178123] Levamisole was appro…

Kategori:
Adjuvants, ImmunologicAnthelminticsAnti-Infective Agents +10
Target Protein:
Neuronal acetylcholine receptor subunit alpha-3Alkaline phosphatase, tissue-nonspecific isozymeAlkaline phosphatase, germ cell type +4
Waktu Paruh4.4-5.6 hours (biph…
Vol. Distribusi-
Klirens-
Genetik -
Levamlodipine Approved DB09237
small molecule | CAS: 103129-82-4

Levamlodipine, also known as S-amlodipine, is a pharmacologically active enantiomer of [amlodipine], an antihypertensive medication.[L10833] Levamlodipine belongs to the dihydropyridine group of calcium channel blockers.[L10833] This medication was first mark…

Kategori:
Antiarrhythmic agentsAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +11
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent L-type calcium channel subunit alpha-1DNitric oxide synthase 3 +1
Waktu ParuhLevamlodipine has a…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Levetiracetam Approved DB01202
small molecule | CAS: 102767-28-2

Levetiracetam is a drug within the pyrrolidine class that is used to treat various types of seizures stemming from epileptic disorders. It was first approved for use in the United States in 1999 and is structurally and mechanistically unrelated to other anti-…

Kategori:
AcetamidesAmidesAnticonvulsants +8
Target Protein:
5-hydroxytryptamine receptor 3AVoltage-dependent N-type calcium channel subunit alpha-1BSynaptic vesicle glycoprotein 2A
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Levilimab DB16387
biotech | CAS: 2035008-70-7

Levilimab is under investigation in clinical trial NCT04227366 (Study of the Efficacy and Safety of BCD-089 in Combination With Methotrexate in Patients With Active Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levmetamfetamine Approved DB09571
small molecule | CAS: 33817-09-3

Levomethamphetamine, the L-enantiomer of methamphetamine is a sympathomimetic vasoconstrictor used in some over-the-counter (OTC) nasal decongestant inhalers in the United States.

Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Levobetaxolol Approved DB09351
small molecule | CAS: 93221-48-8

Levobetaxolol is a beta-blocker used to lower the pressure in the eye to treat conditions such as glaucoma. It was marketed as a 0.5% ophthalmic solution of levobetaxolol hydrochloride under the trade name Betaxon but has been discontinued.

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +3
Target Protein:
Beta-1 adrenergic receptor
Waktu ParuhThe mean half life …
Vol. Distribusi-
Klirens-
Genetik -
Levobunolol Approved DB01210
small molecule | CAS: 47141-42-4

A nonselective beta-adrenoceptor antagonist used in the treatment of glaucoma.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +22
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
Levobupivacaine Approved DB01002
small molecule | CAS: 27262-47-1

Levobupivacaine is an amino-amide local anaesthetic drug belonging to the family of n-alkylsubstituted pipecoloxylidide. It is the S-enantiomer of bupivacaine. Levobupivacaine hydrochloride is commonly marketed by AstraZeneca under the trade name Chirocaine.…

Kategori:
AmidesAminesAnesthetics +15
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh3.3 hours
Vol. Distribusi66.91 ±18.23 L [aft…
Klirens39.06 ±13.29 L/h [a…
Genetik -
Levocabastine Approved DB01106
small molecule | CAS: 79516-68-0

Levocabastine is a selective second-generation H1-receptor antagonist used for allergic conjunctivitis. Levocabastine was discovered at Janssen Pharmaceutica in 1979.

Kategori:
Anti-Allergic AgentsAntiallergic Agents, Excl. CorticosteroidsCentral Nervous System Depressants +11
Target Protein:
Histamine H1 receptorNeurotensin receptor type 2
Waktu Paruh36 hours (after ora…
Vol. Distribusi-
Klirens-
Genetik -
Levocarnitine Approved DB00583
small molecule | CAS: 541-15-1

Constituent of striated muscle and liver. It is used therapeutically to stimulate gastric and pancreatic secretions and in the treatment of hyperlipoproteinemias.

Kategori:
Alimentary Tract and MetabolismAminesAmino Acids and Derivatives +9
Target Protein:
Carnitine O-palmitoyltransferase 1, muscle isoformXanthine dehydrogenase/oxidaseLiver carboxylesterase 1 +9
Waktu Paruh17.4 hours (elimina…
Vol. DistribusiThe steady state vo…
KlirensTotal body clearanc…
Genetik -
small molecule | CAS: 20064-19-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levocetirizine Approved DB06282
small molecule | CAS: 130018-77-8

Levocetirizine is a selective histamine H<sub>1</sub> antagonist used to treat a variety of allergic symptoms.[A181748,A181790,L7694] It is the R enantiomer of [cetirizine].[L7694] Levocetirizine has greater affinity for the histamine H<sub>1</sub> receptor t…

Kategori:
Antihistamines for Systemic UseCentral Nervous System DepressantsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Histamine H1 receptor
Waktu ParuhThe average half li…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Levodopa Approved DB01235
small molecule | CAS: 59-92-7

Levodopa is a prodrug of dopamine that is administered to patients with Parkinson's due to its ability to cross the blood-brain barrier[Label]. Levodopa can be metabolised to dopamine on either side of the blood-brain barrier and so it is generally administer…

Kategori:
AminesAmino AcidsAmino Acids, Aromatic +21
Target Protein:
D(1A) dopamine receptorD(1B) dopamine receptorD(2) dopamine receptor +2
Waktu Paruh2.3 hours for orall…
Vol. Distribusi168L for orally inh…
KlirensIntravenously admin…
Genetik -
small molecule | CAS: 99291-25-5

Levodropropizine is under investigation in clinical trial NCT01573663 (A Drug-Drug Interaction Study of Ambroxol and Levodropropizine).

Kategori:
AlcoholsAntitussive AgentsCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levofloxacin Approved DB01137
small molecule | CAS: 100986-85-4

Levofloxacin is a fluoroquinolone antibiotic and the optical S-(-) isomer of racemic [ofloxacin].[A190663] It reportedly carries 8 to 128-fold more activity against both gram-negative and gram-positive bacteria compared to R-(+)-ofloxacin[A190663] and remains…

Kategori:
4-QuinolonesAlimentary Tract and MetabolismAnti-Bacterial Agents +35
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu ParuhThe average termina…
Vol. DistribusiLevofloxacin is wid…
KlirensThe average apparen…
Genetik -
Levoglucose DB12970
small molecule | CAS: 921-60-8

Levoglucose has been used in trials studying the diagnostic of Bowel Cleansing Prior to Colonoscopy.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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