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12560

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9109 (72.5%)
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6912 (55.0%)
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12560 (100.0%)

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Halaman 188 / 252
Pegsunercept DB06611
biotech | CAS: 330988-75-5

Pegsunercept is used for treating rheumatoid arthritis. Phase II clinical trials were completed in January 2010.

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household setting +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegtarazimod DB19318
biotech | CAS: 2056232-82-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegtarviliase DB18999
biotech | CAS: 2649372-23-4

Pegtarviliase is under investigation in clinical trial NCT05154890 (A Multiple Ascending Dose Study of ACN00177 (Pegtarviliase) in Subjects With CBS Deficiency).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pegteograstim DB15290
biotech | CAS: 1329602-23-4

Pegteograstim is under investigation in clinical trial NCT02787876 (Pegteograstim in Children With Solid Tumors).

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsColony-Stimulating Factors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegtibatinase DB17677
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pegulicianine Approved DB18731
small molecule | CAS: 2230217-17-9

Pegulicianine is an optical imaging agent indicated for fluorescence imaging in patients with breast cancer. It is used following surgical resection of the primary tumor to detect areas of remaining cancer. Pegulicianine itself is a prodrug comprising three m…

Kategori:
Contrast MediaFluorescent Dyes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegunigalsidase alfa Approved DB14992
biotech | CAS: 1644392-61-9

Pegunigalsidase alfa (PRX-102) is a recombinant form of human ?-galactosidase-A indicated for long-term enzyme replacement therapy in patients with Fabry disease, a rare genetic disorder characterized by the deficiency of alpha-galactosidase A.[A259352,L46342…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Alpha-galactosidase AGlobotriaosylceramide
Waktu ParuhPegunigalsidase alf…
Vol. DistribusiIn enzyme replaceme…
KlirensPatients treated wi…
Genetik -
Pegvaliase Approved DB12839
biotech | CAS: 1585984-95-7

Pegvaliase is a recombinant phenylalanine ammonia lyase (PAL) enzyme derived from _Anabaena variabilis_ that converts phenylalanine to ammonia and _trans_-cinnamic acid [A33284]. Both the U.S. Food and Drug Administration and European Medicines Agency approve…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAmmonia-Lyases +7
Target Protein:
Phenylalanine-4-hydroxylase
Waktu ParuhFollowing once-dail…
Vol. DistribusiThe mean ± SD (rang…
KlirensAt steady state fol…
Genetik -
Pegvisomant Approved DB00082
biotech | CAS: 218620-50-9

Pegvisomant is a highly selective growth hormone (GH) receptor antagonist. It is used to treat acromegaly. Unlike dopamine or somatostatin analogs (which inhibit growth hormone secretion), this drug actually blocks the hepatic (GH-mediated) production of ins…

Kategori:
AcromegalyAmino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and Analogues +17
Target Protein:
Growth hormone receptor
Waktu Paruh~6 days
Vol. Distribusi* 7 L
Klirens* 36 - 28 mL/h [SC …
Genetik -
biotech | CAS: 1620390-06-8

Pegvorhyaluronidase alfa is under investigation in clinical trial NCT02241187 (Two Stage Study Of Single Dose PEGPH20 And Cetuximab In Patients With Pancreatic Adenocarcinoma Prior To Surgical Resection).

Kategori:
Carbon-Oxygen LyasesEnzymesEnzymes and Coenzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1417412-83-9

PEGylated Recombinant Factor VIII is under investigation in clinical trial NCT02585960 (BAX 855 Pk-guided Dosing).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 1433787-75-7

Pegylated Recombinant Human Arginase I is under investigation in clinical trial NCT03455140 (A Study Evaluating the Safety and Activity of Pegylated Recombinant Human Arginase (BCT-100)).

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsEnzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1350661-05-0

Deskripsi belum tersedia.

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegzilarginase Approved DB14780
biotech | CAS: 1659310-95-8

Pegzilarginase is under investigation in clinical trial NCT02488044 (A Phase 1/2 Study of AEB1102 in Patients With Arginase I Deficiency).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1380087-89-7

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Bromodomain-containing protein 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelacarsen DB16284
biotech | CAS: 1637637-70-7

Pelacarsen is under investigation in clinical trial NCT03070782 (Phase 2 Study of ISIS 681257 (Akcea-apo(a)-lrx) in Participants With Hyperlipoproteinemia(a) and Cardiovascular Disease).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Pelcitoclax DB16285
small molecule | CAS: 1619923-36-2

Pelcitoclax is under investigation in clinical trial NCT04210037 (Study of Combination APG-1252 Plus Paclitaxel in Patients With Relapsed/refractory Small Cell Lung Cancer).

Kategori:
Amines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peldesine DB02568
small molecule | CAS: 133432-71-0

Peldesine is a potent inhibitor of human CCRF-CEM T-cell proliferation. It has undergone phase I trials for the treatment of Human Immunodeficiency Virus (HIV) infections.

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 SubstratesHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelitinib DB05524
small molecule | CAS: 257933-82-7

Pelitinib (EKB-569) is a potent, low molecular weight, selective, and irreversible inhibitor of epidermal growth factor receptor (EGFR) that is being developed as an anticancer agent.

Kategori:
AminesAntineoplastic AgentsEnzyme Inhibitors +4
Target Protein:
Epidermal growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelitrexol DB12757
small molecule | CAS: 446022-33-9

Pelitrexol has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Sulfur Compounds
Target Protein:
Trifunctional purine biosynthetic protein adenosine-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pelubiprofen DB12150
small molecule | CAS: 69956-77-0

Pelubiprofen has been investigated for the treatment of Chronic Back Pain.

Kategori:
Acids, Carbocyclic
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemafibrate DB15212
small molecule | CAS: 848259-27-8

Pemafibrate is under investigation in clinical trial NCT03350165 (A Study of Pemafibrate in Patients With Nonalcoholic Fatty Liver Disease (NAFLD)).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +6
Target Protein:
Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pembrolizumab Approved DB09037
biotech | CAS: 1374853-91-4

Pembrolizumab is a highly selective IgG4-kappa humanized monoclonal antibody against PD-1 receptors. It was generated by grafting the variable sequences of a very high-affinity mouse antihuman PD-1 antibody onto a human IgG4-kappa isotype containing a stabili…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Programmed cell death protein 1Programmed cell death 1 ligand 1
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state vo…
KlirensClearance is modera…
Genetik -
Pemetrexed Approved DB00642
small molecule | CAS: 137281-23-3

Pemetrexed is a chemotherapy drug that is manufactured and marketed by Eli Lilly and Company under the brand name Alimta. It is indicated for use in combination with cisplatin for the treatment of patients with malignant pleural mesothelioma whose disease is …

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +19
Target Protein:
Thymidylate synthaseThymidylate synthaseBifunctional purine biosynthesis protein ATIC +2
Waktu ParuhThe elimination hal…
Vol. DistribusiPemetrexed has a st…
KlirensThe total systemic …
Genetik -
Pemigatinib Approved DB15102
small molecule | CAS: 1513857-77-6

Pemigatinib is a small molecule kinase inhibitor with antitumour activity. It works by inhibiting fibroblast growth factor receptors (FGFRs), which are receptor tyrosine kinases that activate signalling pathways in tumour cells.[A193719] FGFRs gained attentio…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +16
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +1
Waktu ParuhFollowing administr…
Vol. DistribusiThe apparent volume…
KlirensFollowing administr…
Genetik -
Pemirolast Approved DB00885
small molecule | CAS: 69372-19-6

Pemirolast potassium is a slightly yellow powder that is soluble in water. It is a mast cell stabilizer that acts as an antiallergic agent. As an ophthalmic aqueous sterile solution, pemirolast is used for the prevention of itching of the eyes caused by aller…

Kategori:
Decreased Histamine ReleaseHistamine AgentsMast Cell Stabilizers +3
Target Protein:
Histamine H1 receptor
Waktu Paruh4.5 hours (Ophthalm…
Vol. Distribusi-
Klirens-
Genetik -
Pemivibart DB18720
biotech | CAS: 2858673-18-2

Pemivibart (Pemgarda) is a human IgG1 monoclonal antibody targeting the SARS-CoV-2 spike protein receptor binding domain.[L50326] It received emergency use authorization (EUA) from the FDA in March 2024 for pre-exposure prophylaxis (PrEP) of COVID-19 in certa…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalApproved Treatments for COVID-19 +4
Target Protein:
Spike glycoprotein
Waktu ParuhPemivibart has an e…
Vol. DistribusiFollowing the admin…
KlirensFollowing the admin…
Genetik -
biotech

Pemlimogene merolisbac is under investigation in clinical trial NCT03371381 (An Efficacy and Safety Study of JNJ-64041757, a Live Attenuated Listeria Monocytogenes Immunotherapy, in Combination With Nivolumab Versus Nivolumab Monotherapy in Participants With …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemoline Approved DB01230
small molecule | CAS: 2152-34-3

In 2005, the Food and Drug Administration (FDA) withdrew approval for pemoline. In March 2005, Abbott Laboratories (Cylert marketer) had discontinued the production of Cylert arguing economic reasons.

Kategori:
Central Nervous System AgentsCentral Nervous System StimulantsCentrally Acting Sympathomimetics +4
Waktu ParuhThe serum half-life…
Vol. Distribusi-
Klirens-
Genetik -
Pemrametostat DB19170
small molecule | CAS: 1616392-22-3

Pemrametostat is under investigation in clinical trial NCT03614728 (Study to Investigate the Safety and Clinical Activity of GSK3326595 and Other Agents to Treat Myelodysplastic Syndrome (MDS) and Acute Myeloid Leukemia (AML)).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Protein arginine N-methyltransferase 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemtumomab DB18563
biotech

Pemtumomab is a murine monoclonal antibody radiolabeled with Yttrium-90. It targets the mucin 1 (MUC1) protein.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pemvidutide DB18998
biotech | CAS: 2538014-94-5

Pemvidutide is under investigation in clinical trial NCT05989711 (Efficacy and Safety of Pemvidutide in Subjects With Nonalcoholic Steatohepatitis (NASH) (IMPACT Trial)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penamecillin DB13739
small molecule | CAS: 983-85-7

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penbutolol Approved DB01359
small molecule | CAS: 38363-40-5

Penbutolol is a drug in the beta-blocker class used to treat hypertension. Penbutolol binds both beta-1 and beta-2 adrenergic receptors, rendering it a non-selective beta-blocker. Penbutolol can act as a partial agonist at beta adrenergic receptors, since it …

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor5-hydroxytryptamine receptor 1A +1
Waktu ParuhPlasma= approximate…
Vol. Distribusi-
KlirensApproximately 90% o…
Genetik -
Penciclovir Approved DB00299
small molecule | CAS: 39809-25-1

Penciclovir is a synthetic acyclic guanine derivative with antiviral activity used for the treatment of various herpes simplex virus (HSV) infections. Displaying low toxicity and good selectivity, penciclovir is a nucleoside analogue.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
Thymidine kinase, cytosolicDNA polymerase catalytic subunitThymidine kinase
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Penfluridol DB13791
small molecule | CAS: 26864-56-2

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntipsychotic Agents +20
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1G
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penicillamine Approved DB00859
small molecule | CAS: 52-67-5

Penicillamine is a pharmaceutical of the chelator class. The pharmaceutical form is D-penicillamine, as L-penicillamine is toxic (it inhibits the action of pyridoxine). It is an ?-amino acid metabolite of penicillin, although it has no antibiotic properties.

Kategori:
Agents Causing Muscle ToxicityAmino AcidsAmino Acids, Peptides, and Proteins +16
Target Protein:
Copper
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Penimepicycline DB13264
small molecule | CAS: 4599-60-4

Penimepicycline is a tetracycline-class antibiotic. It is mentioned on List A produced by the Government of Canada, which is a list of antimicrobial active pharmaceutical ingredients [L2791]. In the classification of the active ingredients included on this li…

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Penpulimab DB16747
biotech | CAS: 2350298-92-7

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaerithrityl DB13526
small molecule | CAS: 115-77-5

Deskripsi belum tersedia.

Kategori:
AlcoholsAlimentary Tract and MetabolismDrugs for Constipation +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaerythritol tetranitrate Approved DB06154
small molecule | CAS: 78-11-5

Pentaerythritol tetranitrate is the nitrate ester of pentaerythritol that possesses explosive properties. When mixed with a plasticizer, this chemical forms a plastic explosive. It is recognized by the FDA to be a coronary vasodilator in the treatment of hear…

Kategori:
AlcoholsAntianginal AgentsCarbohydrates +11
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit betaFree radicals
Waktu ParuhThe elimination hal…
Vol. DistribusiThe steady-state vo…
KlirensIn a pharmacokineti…
Genetik -
Pentagastrin Approved DB00183
small molecule | CAS: 5534-95-2

A synthetic pentapeptide that mimics the actions of endogenous gastrin when given parenterally. It works by stimulating the secretion of gastric acid, pepsin, and intrinsic factor. It has also been used as a diagnostic aid.

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsGastrins +8
Target Protein:
Gastrin/cholecystokinin type B receptor
Waktu Paruh10 minutes or less
Vol. Distribusi-
Klirens-
Genetik -
Pentaglobin DB15865
biotech | CAS: 97794-27-9

Pentaglobin, also known as IgM-enriched immunoglobulin, falls under a group of polyclonal immunoglobulin preparations.[A220173] It is comprised of [immunoglobulin G (IgG)](https://www.drugbank.ca/drugs/DB00028) and immunoglobulin A (IgA) while also being enri…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentaglyme DB02580
small molecule | CAS: 1191-87-3

Deskripsi belum tersedia.

Target Protein:
Profilin-2Restriction endonuclease R.BpuJICytochrome c-552 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentamidine Approved DB00738
small molecule | CAS: 100-33-4

Antiprotozoal agent effective in trypanosomiasis, leishmaniasis, and some fungal infections; used in treatment of pneumocystis pneumonia in HIV-infected patients. It may cause diabetes mellitus, central nervous system damage, and other toxic effects.

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAgents causing hyperkalemiaAmidines +20
Target Protein:
Tryptase alpha/beta-1tRNA (cytosine(38)-C(5))-methyltransferaseDNA
Waktu Paruh9.1-13.2 hours
Vol. Distribusi-
Klirens-
Genetik -
Pentamycin DB13571
small molecule | CAS: 6834-98-6

Deskripsi belum tersedia.

Kategori:
AlkenesAntifungal AgentsGenito Urinary System and Sex Hormones +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pentastarch Approved DB09111
small molecule | CAS: 9005-27-0

Pentastarch is an artificial colloid (hydroxyethyl starch derivative). Pentastarch is characterized by presenting five hydroxyethyl groups, which signifies an approximate 50% hydroxyethylation. It is sold under the name Pentaspan by Bristol-Myers Squibb and i…

Kategori:
Blood SubstitutesCarbohydratesCompounds used in a research, industrial, or household setting +9
Waktu Paruh~2.5 hours.
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Sulfide dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22537-51-5

Pentavalent Antimony has been investigated for the treatment of Cutaneous Leishmaniasis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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