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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 187 / 252
PCO-371 DB14946
small molecule | CAS: 1613373-33-3

PCO-371 is under investigation in clinical trial NCT02475616 (A Single Ascending Dose Study of PCO371 in Healthy Volunteers).

Kategori:
Imidazoles
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PCS-499 DB15122
small molecule | CAS: 1268605-91-9

PCS-499 is under investigation in clinical trial NCT01487109 (A Phase 2 Study to Evaluate the Safety and Efficacy of CTP-499 in Type 2 Diabetic Nephropathy Patients).

Kategori:
DeuteriumHeterocyclic Compounds, Fused-RingPurines +2
Waktu Paruh-
Vol. Distribusi-
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PD-0299685 DB15264
small molecule | CAS: 313651-33-1

PD-0299685 is under investigation in clinical trial NCT00314964 (Study Evaluating PD-0299685 for the Treatment of Vasomotor Symptoms (Hot Flashes / Flushes) Associated With Menopause).

Waktu Paruh-
Vol. Distribusi-
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PD-166326 DB08339
small molecule | CAS: 185039-91-2

Deskripsi belum tersedia.

Target Protein:
Mast/stem cell growth factor receptor KitMitogen-activated protein kinase 14Tyrosine-protein kinase Lck +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-168393 DB07662
small molecule | CAS: 194423-15-9

PD-168393 is an epidermal growth factor receptor inhibitor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Epidermal growth factor receptorReceptor tyrosine-protein kinase erbB-2Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-169316 DB17040
small molecule | CAS: 152121-53-4

PD-169316 is a p38 MAP kinase inhibitor.[A253062]

Kategori:
Enzyme Inhibitors
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-173952 DB17041
small molecule | CAS: 305820-75-1

PD-173952 is a potent Myt1 kinase inhibitor.[A253067]

Kategori:
Oxazines
Target Protein:
Platelet-derived growth factor receptor alphaProto-oncogene tyrosine-protein kinase SrcTyrosine-protein kinase Lck +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD-98059 DB17042
small molecule | CAS: 167869-21-8

PD-98059 is an inhibitor of MAP-kinase kinase activation.[A253072]

Kategori:
BenzopyransCalcium-Calmodulin-Dependent Protein Kinases, antagonists & inhibitorsChromones +4
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1Dual specificity mitogen-activated protein kinase kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD150606 DB02570
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, Acyclic
Target Protein:
Calpain small subunit 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PD173955 DB02567
small molecule

Deskripsi belum tersedia.

Kategori:
PyridinesTyrosine Kinase Inhibitors
Target Protein:
Platelet-derived growth factor receptor alphaTyrosine-protein kinase LckProto-oncogene tyrosine-protein kinase Src +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
PDPSC18 DB05167
biotech

PDPSC18 is therapeutic DNA vaccine designed to fight chronic infections with the Hepatitis B virus, entering phase I clinical trials.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pea Approved DB10551
biotech

Pea allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peach Approved DB10552
biotech

Peach allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peanut Approved DB10553
biotech

Peanut allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
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Peanut oil Approved DB13964
biotech | CAS: 8002-03-7

Peanut oil is derived from _Arachis hypogaea_ which can be found in South America, Mexico, and Centro America. The kernels are consumed roasted but a large percentage is used for the production of vegetable oil. The peanut oil represents about 45-52% of the k…

Kategori:
Basic Ointments and ProtectantsBiological ProductsDetergents +8
Waktu ParuhThe exact pharmacok…
Vol. DistribusiThe exact pharmacok…
KlirensThe exact pharmacok…
Genetik -
Pear Approved DB10554
biotech

Pear allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
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Pecan Approved DB10555
biotech

Pecan allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
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Pecavaptan DB16279
small molecule | CAS: 1914998-56-3

Pecavaptan is under investigation in clinical trial NCT03901729 (A Trial to Study BAY1753011 in Patients With Congestive Heart Failure).

Target Protein:
Vasopressin V1a receptorVasopressin V2 receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pecilocin DB13459
small molecule | CAS: 19504-77-9

Deskripsi belum tersedia.

Kategori:
Antifungal AgentsAntifungals for Dermatological UseAntifungals for Topical Use +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pectin Approved DB11158
biotech | CAS: 9000-69-5

Pectin is a heteropolysaccharide commercially derived from the cell wall of higher plants.[A32327] It is composed of partially methylated polygalacturonic acid units linked in the positions 1-4.[L1961] The carboxylic group of the constituents of pectin can ex…

Kategori:
Alimentary Tract and MetabolismAntidiarrheals, Intestinal Antiinflammatory/antiinfective AgentsBiological Products +15
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Pefloxacin Approved DB00487
small molecule | CAS: 70458-92-3

A synthetic broad-spectrum fluoroquinolone antibacterial agent active against most gram-negative and gram-positive bacteria.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-betaDNA topoisomerase 4 subunit ADNA gyrase subunit A +2
Waktu Paruh8.6 hours
Vol. Distribusi-
Klirens-
Genetik -
Peg-100 stearate Approved DB11225
small molecule | CAS: 9004-99-3

Deskripsi belum tersedia.

Kategori:
Pegylated agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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PEG-uricase DB05321
biotech

PEG-uricase, a polyethylene glycol ("PEG") conjugate of recombinant porcine uricase (urate oxidase), which breaks down the uric acid deposits is being studied in Phase III clinical trials for the treatment of severe, treatment-refractory gout in the United St…

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEnzymes +8
Target Protein:
Uric acid degradation bifunctional protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegadricase DB15129
biotech | CAS: 1040753-26-1

Pegadricase is under investigation in clinical trial NCT01021241 (Safety and Efficacy Study of Intravenous Uricase-PEG 20).

Waktu Paruh-
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Pegamotecan DB12842
small molecule | CAS: 581079-18-7

Pegamotecan has been used in trials studying the treatment of Cancer of Stomach, Sarcoma, Soft Tissue, and Gastroesophageal Cancer.

Kategori:
AlcoholsAlkaloidsCompounds used in a research, industrial, or household setting +5
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Pegapamodutide DB14817
biotech | CAS: 1492924-65-8

Pegapamodutide is under investigation in clinical trial NCT02188303 (A Study of LY2944876 in Healthy Japanese and Non-Japanese Participants).

Waktu Paruh-
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Pegaptanib Approved DB04895
biotech | CAS: 222716-86-1

Pegaptanib is a polynucleotide aptamer. Pegatinib aids neovascular age-related macular degeneration by binding to VEGF which in order reduces angiogenesis and vessel permeability. Pegaptanib was granted FDA approval on 17 September 2004.[L17903]

Kategori:
Antineovascularisation AgentsCarbohydratesDrugs that are Mainly Renally Excreted +10
Target Protein:
Vascular endothelial growth factor A, long form
Waktu ParuhIn humans, after a …
Vol. DistribusiIt is distributed i…
Klirens-
Genetik -
Pegargiminase DB06592
small molecule | CAS: 1394129-74-8

Pegargiminase is an anticancer agent.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEnzymes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegaspargase Approved DB00059
biotech | CAS: 130167-69-0

Pegaspargase is a conjugate of monomethoxypolyethylene glycol (mPEG) and L-asparaginase (L-asparagine amidohydrolase), an asparagine-specific enzyme that converts L-asparagine into aspartic acid and ammonia.[L44667] Asparagine is an amino acid that is vital f…

Kategori:
AlcoholsAmidohydrolasesAntineoplastic Agents +15
Target Protein:
L-asparagine
Waktu ParuhThe mean eliminatio…
Vol. DistribusiBased on a non-comp…
KlirensFor a single intram…
Genetik -
Pegbelfermin DB15365
biotech | CAS: 2089039-22-3

Pegbelfermin is under investigation in clinical trial NCT03486899 (A Study of Experimental Medication BMS-986036 in Adults With Nonalcoholic Steatohepatitis (NASH) and Stage 3 Liver Fibrosis).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegcetacoplan Approved DB16694
biotech | CAS: 2019171-69-6

Pegcetacoplan is a complement inhibitor indicated in the treatment of paroxysmal nocturnal hemoglobinuria (PNH).[A235000,L34095] Prior to its FDA approval, patients with PNH were typically treated with the C5 inhibiting monoclonal antibody [eculizumab].[A2350…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsComplement Inactivating Agents +6
Target Protein:
Complement C3
Waktu ParuhThe median half lif…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
biotech | CAS: 1448590-54-2

Pegcrisantaspase is under investigation in clinical trial NCT02257684 (A Dose Confirmation and Pharmacokinetic Study of Pegcrisantaspase Administered as Intravenous (IV) Infusion in Children and Young Adults With Acute Lymphoblastic Leukemia (ALL) /Lymphoblas…

Waktu Paruh-
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Pegdinetanib DB05931
small molecule | CAS: 906450-24-6

CT-322 is a proprietary Adnectin(TM) protein therapeutic that, in preclinical studies, specifically binds to vascular endothelial growth factor receptor 2 (VEGFR-2), which regulates the primary tumor angiogenesis pathway. As a result, CT-322 blocks all known …

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsCarbohydrates +11
Target Protein:
Vascular endothelial growth factor receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegenzileukin DB17495
biotech | CAS: 2573074-47-0

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Pegfilgrastim Approved DB00019
biotech | CAS: 208265-92-3

Pegfilgrastim is a PEGylated form of the recombinant human granulocyte colony-stimulating factor (G-CSF) analogue, [filgrastim].[A187601] The drug is approved for use to decrease the incidence of infection, as manifested by febrile neutropenia, in susceptible…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +21
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe serum half-life…
Vol. DistribusiPegfilgrastim appea…
KlirensPegfilgrastim has a…
Genetik -
Pegilodecakin DB15162
biotech | CAS: 1966111-35-2

Pegilodecakin is under investigation in clinical trial NCT03382912 (Study of Pegilodecakin (LY3500518) With Nivolumab Compared to Nivolumab Alone Second-line Tx in Participants With Metastatic Non-Small Cell Lung Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Peginterferon alfa-2a Approved DB00008
biotech | CAS: 198153-51-4

Peginterferon alfa-2a is a form of recombinant interferon used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Adjuvants, ImmunologicAlcoholsAlfa Interferons +29
Target Protein:
Interferon alpha/beta receptor 2Interferon alpha/beta receptor 1
Gen Terkait:
IFNL3
Waktu ParuhThe mean terminal h…
Vol. Distribusi-
KlirensThe mean systemic c…
Genetik 1 Varian
Peginterferon alfa-2b Approved DB00022
biotech | CAS: 215647-85-1

Peginterferon alfa-2b is a form of recombinant interferon used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized in…

Kategori:
Adjuvants, ImmunologicAlcoholsAlfa Interferons +34
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Gen Terkait:
IFNL3
Waktu ParuhThe mean half-life …
Vol. Distribusi-
KlirensThe estimated appar…
Genetik 1 Varian
biotech

PEGylation is a technology for the chemical attachment of polyethylene glycol (PEG) polymer chains to a broad range of drug substances such as peptides and proteins including antibody fragments; small molecules, and other drugs. [Infergen] is a bio-engineered…

Kategori:
Pegylated agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1848968-91-1

Peginterferon Alfacon-2 is under investigation in clinical trial NCT06544551 (Efficacy and Safety Study of Peginterferon Alfacon-2 to Treat Chronic Hepatitis B Virus Infection).

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsInterferons
Waktu Paruh-
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Peginterferon beta-1a Approved DB09122
biotech | CAS: 1211327-92-2

Multiple Sclerosis (MS) is a chronic and inflammatory autoimmune disease of the central nervous system, disrupting communication between the brain and other parts of the body. Most patients diagnosed with this illness experience their initial disease symptoms…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +13
Target Protein:
Interferon alpha/beta receptor 1
Waktu ParuhThe mean half life …
Vol. DistribusiThe volume of distr…
KlirensThe average steady …
Genetik -
biotech | CAS: 914617-98-4

Peginterferon lambda-1a is under investigation in clinical trial NCT01754974 (Safety and Efficacy Study of Peginterferon Lambda-1a vs. Peginterferon Alfa-2a, Plus Ribavirin in Subjects With Genotype 1 Hepatitis C).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegloticase Approved DB09208
biotech | CAS: 885051-90-1

Pegloticase is a porcine recombinant PEGylated uricase indicated for the treatment of chronic gout in adult patients that do not respond to other types of therapies.[L42425] Pegloticase has a similar activity to rasburicase, an enzyme that metabolizes uric ac…

Kategori:
Antigout PreparationsCompounds used in a research, industrial, or household settingEnzymes +6
Target Protein:
Uric acid
Waktu ParuhIn patients with sy…
Vol. DistribusiThe volume of distr…
KlirensIn gout patients gi…
Genetik -
Pegloxenatide DB19230
biotech | CAS: 2420483-82-3

Pegloxenatide is under investigation in clinical trial NCT05172999 (Loxenatide Plus LNG-IUS in Endometrial Atypical Hyperplasia).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsEthylene Glycols +3
Waktu Paruh-
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Klirens-
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Pegnivacogin DB06293
small molecule | CAS: 959716-28-0

Deskripsi belum tersedia.

Kategori:
Factor IXa, antagonists & inhibitorsNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegozafermin DB19062
biotech | CAS: 2489589-60-6

Pegozafermin is under investigation in clinical trial NCT05852431 (To Evaluate the Efficacy and Safety of Pegozafermin in Subjects With Severe Hypertriglyceridemia).

Waktu Paruh-
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Pegpleranib DB06325
small molecule | CAS: 1618657-13-8

Deskripsi belum tersedia.

Kategori:
Pegylated agents
Target Protein:
Platelet-derived growth factor subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pegsitacianine DB19098
small molecule | CAS: 2396651-85-5

Pegsitacianine is under investigation in clinical trial NCT05576974 (A Phase 2a, Single-dose, Open-label Study to Evaluate Diagnostic Performance and Safety of Pegsitacianine, an Intraoperative Fluorescence Imaging Agent for the Detection of Cancer, in Patien…

Waktu Paruh-
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Genetik -
Menampilkan 9301–9350 dari 12560
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