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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (11778)

Halaman 186 / 236
small molecule | CAS: 139-85-5

Also known as protocatechuic aldehyde, protocatechualdehyde is a naturally-occuring phenolic aldehyde that is found in barley, green cavendish bananas, grapevine leaves and root of the herb S. miltiorrhiza [A27224]. Protocatechualdehyde possesses antiprolifer…

Kategori:
AldehydesAnticoagulantsBenzene Derivatives +2
Target Protein:
Amine oxidase [flavin-containing] B
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Protokylol Approved DB06814
small molecule | CAS: 136-70-9

Protokylol is a ?-adrenergic receptor agonist used as a bronchodilator in Europe and the United States.

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +15
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptor
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Protriptyline Approved DB00344
small molecule | CAS: 438-60-8

Protriptyline hydrochloride is a dibenzocycloheptene-derivative tricyclic antidepressant (TCA). TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents that produce hypertension +24
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter
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Proxalutamide DB16065
small molecule | CAS: 1398046-21-3

Proxalutamide is under investigation in clinical trial NCT03899467 (The Safety and Tolerability of Proxalutamide (GT0918) in Subjects With Metastatic Castrate Resistant Prostate Cancer).

Kategori:
HydantoinsImidazolesImidazolidines
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Proxibarbal Approved DB13253
small molecule | CAS: 2537-29-3

Proxibarbal is a derivative of barbiturates, which has been used to treat migraines. Proxibarbal was approved in France but was withdrawn from the market due to the risk of inducing immunoallergic thrombocytopenia [L5476].

Kategori:
Barbiturates, PlainCentral Nervous System AgentsCentral Nervous System Depressants +5
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PRTX-100 DB05947
small molecule

PRTX-100 is a highly-purified form of Staphylococcal Protein A that binds directly to monocytes and a subset of B-cells that are involved in the development and progression of various autoimmune diseases. These binding interactions enable the compound to modu…

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Prucalopride Approved DB06480
small molecule | CAS: 179474-81-8

Prucalopride is a dihydrobenzofurancarboxamide derivative from the benzofurane family that selectively stimulates 5-HT4 receptors and thus, it presents enterokinetic properties.[A37348] The high selectivity of prucalopride allowed further development as it pr…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsCentral Nervous System Depressants +17
Target Protein:
5-hydroxytryptamine receptor 4
Waktu ParuhThe reported half-l…
Vol. DistribusiThe mean volume of …
KlirensPrucalopride renal …
Genetik -
Prulifloxacin DB11892
small molecule | CAS: 123447-62-1

Prulifloxacin has been investigated for the treatment of Urinary Tract Infection.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA topoisomerase 4 subunit ADNA gyrase subunit ADNA gyrase subunit B
Waktu Paruh-
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Prussian blue Approved DB06783
small molecule | CAS: 14038-43-8

Prussian blue is described as a deep blue pigment that is produced when the oxidation of ferrous ferrocyanide salts occurs. It contains ferric hexacyanoferrate(II) in a cubic lattice crystal structure. It is insoluble in water but also tends to form a colloid…

Kategori:
AnionsAntidotesChelating Activity +11
Waktu Paruh-
Vol. DistribusiHistopathological e…
KlirensThe clearance from …
Genetik -
PRX-07034 DB05993
small molecule | CAS: 903580-39-2

Deskripsi belum tersedia.

Target Protein:
5-hydroxytryptamine receptor 6
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PRX-08066 DB05607
small molecule

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT2 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 2B
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PRX-ASL DB17679
biotech

PRX-ASL is an intracellular enzyme replacement therapy designed to replace the missing or defective enzyme in patients with argininosuccinate lyase deficiency.

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PRX-OTC DB17680
biotech

PRX-OTC is an intracellular enzyme replacement therapy designed to replace missing or defective enzyme in patients with ornithine transcarbamylase deficiency.

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Pseudoephedrine Approved DB00852
small molecule | CAS: 90-82-4

Pseudoephedrine is structurally related to [ephedrine] but exerts a weaker effect on the sympathetic nervous system.[A188820,A188823] Both drugs naturally occur in in ephedra plant which have a history of use in traditional Eastern medicine and were first res…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +30
Target Protein:
Sodium-dependent noradrenaline transporterD(2) dopamine receptorSodium-dependent dopamine transporter +10
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe apparent volume…
KlirensA 60mg oral dose of…
Genetik -
biotech

Deskripsi belum tersedia.

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small molecule | CAS: 567-19-1

Deskripsi belum tersedia.

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Pseudotropine DB04026
small molecule | CAS: 135-97-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsAza CompoundsAzabicyclo Compounds
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PSI-697 DB12211
small molecule | CAS: 851546-61-7

PSI-697 has been used in trials studying the treatment of Scleritis.

Kategori:
Heterocyclic Compounds, Fused-RingP-SelectinQuinolines
Target Protein:
P-selectin
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Psicose DB15087
small molecule | CAS: 23140-52-5

Psicose is under investigation in clinical trial NCT02459834 (The Fructose and Allulose Catalytic Effects (FACE) Trial).

Kategori:
CarbohydratesHexosesKetoses +1
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PSN357 DB05044
small molecule

PSN357 is a glycogen phosphorylase inhibitor (GPI), which is designed to rapidly lower blood glucose levels by preventing glycogen breakdown to glucose in the liver.

Target Protein:
Glycogen phosphorylase, liver form
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Psoralen DB18665
small molecule | CAS: 66-97-7

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +13
Target Protein:
Amine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
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PT-2385 DB16055
small molecule | CAS: 1672665-49-4

PT-2385 is under investigation in clinical trial NCT03108066 (PT2385 for the Treatment of Von Hippel-lindau Disease-associated Clear Cell Renal Cell Carcinoma).

Target Protein:
Endothelial PAS domain-containing protein 1Hypoxia-inducible factor 1-alpha
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PT217 DB18472
biotech

PT217 is a bispecific Antibody against DLL3 and CD47

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PT886 DB18471
biotech

PT886 is a bispecific antibody against Claudin 18.2 and cluster of differentiation 47 (CD47)

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PTC299 DB05173
small molecule

PTC299 is a novel, orally administered small-molecule designed to inhibit the production of vascular endothelial growth factor (VEGF) in tumors. Overexpression of VEGF plays a key role in multiple diseases including cancer and macular degeneration. PTC299 was…

Kategori:
Acids, AcyclicHeterocyclic Compounds, Fused-RingIndoles
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Pteric acid DB04357
small molecule

Deskripsi belum tersedia.

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Pterostilbene DB17939
small molecule | CAS: 18259-15-9

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene Compounds
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PTI-110 DB18298
small molecule | CAS: 633700-15-9

Deskripsi belum tersedia.

Target Protein:
Amyloid-beta precursor protein
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PTI-801 DB05300
small molecule | CAS: 615580-67-1

PTI-801 represents a new class of drugs to treat pain. PTI-801 can minimize the opioid tolerance, dependence or addiction that is often associated with repeat use of oxycodone. It is a combination of oxycodone with ultralow-dose naltrexone, an opioid antagoni…

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PTR-01 DB17900
biotech

Deskripsi belum tersedia.

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Puccinia graminis Approved DB10706
biotech

Puccinia graminis is a fungus which can provoke allergic reactions. Puccinia graminis extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Genetik -
biotech

Puccinia striiformis var. striiformis is a fungus which can provoke allergic reactions. Puccinia striiformis var. striiformis extract is used in allergenic testing.

Kategori:
Non-Standardized Fungal Allergenic Extract
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Pucotenlimab Approved DB17552
biotech | CAS: 2403647-03-8

Pucotenlimab is a recombinant humanized anti-PD-1 monoclonal antibody. It received its first global approval in China in July 2022 for the treatment of solid tumours.[A257296] It is being investigated in other cancers.

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Pudexacianinium DB19161
small molecule | CAS: 2243793-21-5

Pudexacianinium is under investigation in clinical trial NCT05754333 (A Study to Find Out if ASP5354 Can Clearly Help Show the Ureter During Surgery).

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Pumice DB14374
biotech | CAS: 1332-09-8

Pumice is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
MineralsSilicon Compounds
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Ribonuclease pancreatic
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Puromycin DB08437
small molecule | CAS: 53-79-2

Puromycin is an antibiotic that prevents bacterial protein translation. It is utilized as a selective agent in laboratory cell cultures. Puromycin is toxic to both prokaryotic and eukaryotic cells, resulting in significant cell death at appropriate doses.

Kategori:
Acids, CarbocyclicAgents that produce neuromuscular block (indirect)Aminoglycoside Antibacterials +20
Target Protein:
Ribosomal protein uL16-likeLarge ribosomal subunit protein uL13Large ribosomal subunit protein uL14 +10
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Purslane Approved DB14327
biotech

Purslane is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Purvalanol DB02733
small molecule

Deskripsi belum tersedia.

Target Protein:
Cyclin-dependent kinase 1Beta-3 adrenergic receptorCyclin-dependent kinase 5 +6
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Purvalanol A DB04751
small molecule | CAS: 212844-53-6

Deskripsi belum tersedia.

Kategori:
CDC2 Protein Kinase, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 1Casein kinase I isoform gamma-3 +2
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Putrescine DB01917
small molecule | CAS: 110-60-1

Putrescine is a toxic diamine formed by putrefaction from the decarboxylation of arginine and ornithine. Putrescine is a solid. This compound belongs to the polyamines. These are compounds containing more than one amine group. Known drug targets of putrescine…

Kategori:
AminesBiogenic AminesBiogenic Polyamines +3
Target Protein:
S-adenosylmethionine decarboxylase proenzymeOrnithine decarboxylaseBeta-1 adrenergic receptor +2
Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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biotech | CAS: 1200123-84-7

Deskripsi belum tersedia.

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biotech | CAS: 1200123-78-9

Deskripsi belum tersedia.

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biotech | CAS: 1200123-74-5

Deskripsi belum tersedia.

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PX-102 DB15416
small molecule | CAS: 1268244-88-7

PX-102 is under investigation in clinical trial NCT01998672 (Multiple Ascending Oral Dose Phase I Study With Px-102).

Target Protein:
Bile acid receptor
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PX-478 DB06082
small molecule | CAS: 685898-44-6

PX-478 is a small molecule inhibitor of hypoxia inducible factor (HIF)-1 alpha currently in a clinical trial in patients with advanced metastatic cancer and lymphoma. PX-478 was effective in models of both non-small cell lung cancer and small cell lung cance…

Kategori:
Acids, CarbocyclicHydrocarbons, Halogenated
Target Protein:
Hypoxia-inducible factor 1-alpha
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small molecule

Deskripsi belum tersedia.

Kategori:
NaphthalenesPyridines
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small molecule | CAS: 1478364-40-7

PXS-4728A free base is under investigation in clinical trial NCT05904717 (Effect of PXS-4728A on Microglia Activation in Participants With Isolated Rapid Eye Movement Sleep Behaviour Disorder).

Kategori:
Acids, CarbocyclicAlkenesAllyl Compounds +5
Target Protein:
Amine oxidase [copper-containing] 3
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PXS-5505 DB17510
small molecule | CAS: 2409963-83-1

Deskripsi belum tersedia.

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