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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 185 / 236
Progabide DB00837
small molecule | CAS: 62666-20-0

Progabide is an analog and prodrug of gamma-aminobutyric acid. It is commonly used in the treatment of epilepsy. It has agonistic activity for both the GABAA and GABAB receptors. In clinical trials, progabide has been investigated for Parkinson's disease, sch…

Kategori:
Acids, AcyclicAmino AcidsAmino Acids, Peptides, and Proteins +14
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 2Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid type B receptor subunit 1
Waktu Paruh4 hours
Vol. Distribusi-
Klirens-
Genetik -
Progerinin DB17634
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Progesterone Approved DB00396
small molecule | CAS: 57-83-0

Progesterone is a hormone that occurs naturally in females, and is essential for endometrial receptivity, embryo implantation, and the successful establishment of pregnancy. A low progesterone concentration or an insufficient response to progesterone can caus…

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InducersBCRP/ABCG2 Inhibitors +47
Target Protein:
Progesterone receptorMineralocorticoid receptorEstrogen receptor +7
Waktu ParuhAbsorption half-lif…
Vol. DistribusiWhen administered v…
Klirens**Apparent clearanc…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Immunoglobulin heavy constant gamma 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proglumetacin DB13527
small molecule | CAS: 57132-53-3

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 67422-14-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolectin-M DB16521
small molecule

Prolectin-M is a (1-6)-alpha-D-mannopyranose[L31338] and acts as an antagonist of galectin.[L31343] It is being investigated in the clinical trial NCT04512027 (Prolectin-M in COVID-19 Patients Having Mild to Moderate Symptoms Not Requiring Oxygen Support. (Pr…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prolgolimab DB16740
biotech | CAS: 2093956-19-3

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsMonoclonal antibodies and antibody drug conjugates +2
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proline DB00172
small molecule | CAS: 147-85-3

Proline is one of the twenty amino acids used in living organisms as the building blocks of proteins. Proline is sometimes called an imino acid, although the IUPAC definition of an imine requires a carbon-nitrogen double bond. Proline is a non-essential amino…

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +4
Target Protein:
Peptidyl-prolyl cis-trans isomerase BPeptidyl-prolyl cis-trans isomerase APyrroline-5-carboxylate reductase 1, mitochondrial +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promegestone DB13602
small molecule | CAS: 34184-77-5

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promestriene DB12487
small molecule | CAS: 39219-28-8

Promestriene (3-propyl ethyl, 17B-methyl estradiol) has been used in trials studying the prevention of Hypospadias. It is a synthetic estrogen analog, which is used in topical estrogen therapy. Promestriene’s potential for treating vaginal atrophy symptoms as…

Kategori:
Estradiol CongenersEstranesEstrenes +10
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Promethazine Approved DB01069
small molecule | CAS: 60-87-7

Promethazine, originally known as 3,277 R.P., is an N-dimethylaminopropyl derivative of [phenothiazine] that was developed in France in 1946.[A189901] Promethazine antagonizes a variety of receptors, allowing it to be used for a number of indications includin…

Kategori:
Acid ReducersAgents producing tachycardiaAgents that reduce seizure threshold +44
Target Protein:
Histamine H1 receptorD(2) dopamine receptorMuscarinic acetylcholine receptor M1 +10
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe intravenous cle…
Genetik -
Propacetamol DB09288
small molecule | CAS: 66532-85-2

Propacetamol is a non-opioid analgesic devoid of the major contraindications.[A32051] It is a derivative of [acetaminophen], or paracetamol, with the molecular formula glycine, N, N-diethyl-,4-(acetylamino)phenyl ester. Propacetamol is a parenteral formulatio…

Kategori:
Acetaminophen and ProdrugsAcetanilidesAgents causing hyperkalemia +37
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Transient receptor potential cation channel subfamily V member 1 +1
Waktu ParuhThe half-life of pr…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Propagermanium DB17608
small molecule | CAS: 12758-40-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntineoplastic AgentsElements +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propanoic acid Approved DB03766
small molecule | CAS: 79-09-4

Sodium propionate is the sodium salt of propionic acid that exists as colorless, transparent crystals or a granular crystalline powder. It is considered generally recognized as safe (GRAS) food ingredient by FDA, where it acts as an antimicrobial agent for fo…

Kategori:
Acids, AcyclicAnti-Infective AgentsFatty Acids +4
Target Protein:
Alanine racemaseGephyrin2-hydroxy-6-oxo-7-methylocta-2,4-dienoate hydrolase
Waktu ParuhThe half-life of iv…
Vol. DistribusiThree days after a …
KlirensReadily accessible …
Genetik -
Propanoyl-CoA DB02912
small molecule | CAS: 317-66-8

Deskripsi belum tersedia.

Kategori:
Adenine NucleotidesCoenzymesEnzymes and Coenzymes +7
Target Protein:
Propionyl-CoA carboxylase complex B subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propantheline Approved DB00782
small molecule | CAS: 298-50-0

A muscarinic antagonist used as an antispasmodic, in rhinitis, in urinary incontinence, and in the treatment of ulcers. At high doses it has nicotinic effects resulting in neuromuscular blocking.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAmines +13
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proparacaine Approved DB00807
small molecule | CAS: 499-67-2

Proparacaine is a topical anesthetic drug of the amino ester group. It is found in ophthalmic solutions at a concentration of 0.5% as the hydrochloride salt.

Kategori:
Acids, CarbocyclicAminobenzoatesAnesthetics +18
Target Protein:
Sodium channel protein type 10 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propenidazole DB13319
small molecule | CAS: 76448-31-2

Deskripsi belum tersedia.

Kategori:
Antiparasitic Products, Insecticides and RepellentsAntiprotozoalsGenito Urinary System and Sex Hormones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propentofylline DB06479
small molecule | CAS: 55242-55-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnti-Ulcer AgentsCentral Nervous System Agents +12
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propicillin DB13660
small molecule | CAS: 551-27-9

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiolactone Approved DB09348
small molecule | CAS: 57-57-8

Propiolactone is a lactone compound with a four-membered ring. It is a colorless liquid with a pungent slightly sweet odor. Propiolactone is a disinfectant used for the sterilization of blood plasma, vaccines, tissue grafts, surgical instruments, and enzymes.…

Kategori:
Anti-Infective AgentsCompounds used in a research, industrial, or household settingDisinfectants +1
Target Protein:
DNA
Waktu ParuhThe half-life of pr…
Vol. Distribusi-
Klirens-
Genetik -
Propiomazine Approved DB00777
small molecule | CAS: 362-29-8

Propiomazine, an atypical antipsychotic agent, is used to treat both negative and positive symptoms of schizophrenia, acute mania with bipolar disorder, agitation, and psychotic symptoms in dementia. Future uses may include the treatment of obsessive-compulsi…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +20
Target Protein:
Histamine H1 receptorMuscarinic acetylcholine receptorAlpha-1A adrenergic receptor +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propionamide DB04161
small molecule | CAS: 79-05-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propionate ion DB19384
small molecule | CAS: 72-03-7

Propionate ion is under investigation in clinical trial NCT00846326 (Preventing Tolerance to Oxymetazoline in Allergic Rhinitis).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propiverine Approved DB12278
small molecule | CAS: 60569-19-9

Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB) [A32576]. Overactive bladder (OAB) is a chronic condition of the lower urinary tract characterized by urinary…

Kategori:
Acids, CarbocyclicAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +22
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +4
Waktu ParuhIn three studies in…
Vol. DistribusiIn one study, the v…
KlirensMean total clearanc…
Genetik -
Propofol Approved DB00818
small molecule | CAS: 2078-54-8

Propofol is an intravenous anaesthetic agent used for induction and maintenance of general anaesthesia. IV administration of propfol is used to induce unconsciousness after which anaesthesia may be maintained using a combination of medications. Recovery from …

Kategori:
Agents Causing Muscle ToxicityAgents that produce hypertensionAgents that reduce seizure threshold +32
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit beta-3GABA(A) Receptor +2
Waktu ParuhInitial distributio…
Vol. Distribusi* 60 L/kg [healthy …
Klirens* 23 - 50 mL/kg/min…
Genetik -
small molecule | CAS: 184869-48-5

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, General
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propranolol Approved DB00571
small molecule | CAS: 525-66-6

Propranolol is a racemic mixture of 2 enantiomers where the S(-)-enantiomer has approximately 100 times the binding affinity for beta adrenergic receptors.[L6904] Propranolol is used to treat a number of conditions but most commonly is used for hypertension.[…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +37
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta-3 adrenergic receptor +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of pr…
Genetik -
Propyl acetate DB01670
small molecule | CAS: 109-60-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Carboxylesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propyl alcohol Approved DB03175
small molecule | CAS: 71-23-8

A colorless liquid made by oxidation of aliphatic hydrocarbons that is used as a solvent and chemical intermediate.

Kategori:
AlcoholsAntiseptics and DisinfectantsDermatologicals +1
Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propyl Gallate DB12450
small molecule | CAS: 121-79-9

Propyl Gallate is under investigation in clinical trial NCT01450098 (A Study of LY2484595 in Healthy Subjects).

Kategori:
Acids, CarbocyclicAntioxidantsBenzene Derivatives +7
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propylene glycol Approved DB01839
small molecule | CAS: 57-55-6

A clear, colorless, viscous organic solvent and diluent used in pharmaceutical preparations.

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingDrug Delivery Systems +7
Target Protein:
B12-independent glycerol dehydratase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propylhexedrine Approved DB06714
small molecule | CAS: 101-40-6

Propylhexedrine is an alpha-adrenergic agonist often used in nasal decongestant inhalers. It is used to give temporary relief for nasal congestion from colds, allergic rhinitis, or allergies.

Kategori:
Adrenergic AgonistsAdrenergic alpha-AgonistsAmines
Target Protein:
Synaptic vesicular amine transporterAlpha-2C adrenergic receptorTrace amine-associated receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propyliodone Approved DB09366
small molecule | CAS: 587-61-1

Radiopaque medium usually in oil; used in bronchography.

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propylparaben Approved DB14177
small molecule | CAS: 94-13-3

Propylparaben is used in allergenic testing.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Propyphenazone DB13524
small molecule | CAS: 479-92-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proquazone DB13649
small molecule | CAS: 22760-18-5

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Proscillaridin DB13307
small molecule | CAS: 466-06-8

Proscillaridin is a cardiac glycoside that is derived from plants of the genus Scilla and in Drimia maritima (Scilla maritima). Studies suggest the potential cytotoxic and anticancer property of proscillaridin, based on evidence of the drug potently disruptin…

Kategori:
BufanolidesCarbohydratesCardanolides +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prosopis juliflora pollen Approved DB10371
biotech

Prosopis juliflora pollen is the pollen of the Prosopis juliflora plant. Prosopis juliflora pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 13367-85-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 41598-07-6

The principal cyclooxygenase metabolite of arachidonic acid. It is released upon activation of mast cells and is also synthesized by alveolar macrophages. Among its many biological actions, the most important are its bronchoconstrictor, platelet-activating-fa…

Kategori:
AutacoidsBiological FactorsEicosanoids +7
Target Protein:
Prostaglandin D2 receptorProstaglandin F2-alpha receptorProstaglandin E2 receptor EP1 subtype +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protamine DB13700
small molecule | CAS: 9012-00-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntidotesCoagulants +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protamine sulfate Approved DB09141
biotech | CAS: 9009-65-8

Since it's earliest discovery in salmon rine sperm heads in the late 1800's to its formal introduction via US FDA approval in 1939, protamine sulfate has occupied an important therapeutic niche as perhaps the only viable option for reversing the anticoagulant…

Kategori:
Amino Acids, Peptides, and ProteinsAntiheparin AgentsHematologic Agents +5
Waktu ParuhThe half-life of pr…
Vol. DistribusiIn a study group of…
KlirensIn a study group of…
Genetik -
Protego-PD DB18279
biotech

Protego-PD is a post-delivery placental extract.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Prothrombin Approved DB11311
biotech | CAS: 9001-26-7

Prothrombin Complex Concentrate (Human), is indicated for the urgent reversal of acquired coagulation factor deficiency induced by Vitamin K antagonist (VKA, e.g., warfarin) therapy in adult patients with acute major bleeding.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +7
Target Protein:
Fibrinogen alpha chainFibrinogen beta chainCoagulation factor XIII A chain +1
Waktu ParuhApproximately 60h […
Vol. Distribusi-
Klirens-
Genetik -
Protionamide Approved DB12667
small molecule | CAS: 14222-60-7

Prothionamide has been used in trials studying the treatment of MDR-TB and HIV Infections.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiinfectives for Systemic Use +5
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Protirelin Approved DB09421
small molecule | CAS: 24305-27-9

Protirelin is the pharmaceutically available synthetic analogue of the endogenous peptide thyrotropin-releasing hormone (TRH). It is a tri-peptide tropic hormone, released by the hypothalamus, that stimulates the release of Thyroid Stimulating Hormone (TSH) a…

Kategori:
Amino Acids, Peptides, and ProteinsDiagnostic AgentsHormones +12
Target Protein:
Thyrotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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