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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 185 / 252
Pacific ocean perch Approved DB15543
biotech

Pacific ocean perch allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paclitaxel Approved DB01229
small molecule | CAS: 33069-62-4

Paclitaxel is a chemotherapeutic agent marketed under the brand name Taxol among others. Used as a treatment for various cancers, paclitaxel is a mitotic inhibitor that was first isolated in 1971 from the bark of the Pacific yew tree which contains endophytic…

Kategori:
Agents Causing Muscle ToxicityAlbuminsAmino Acids, Peptides, and Proteins +42
Target Protein:
Tubulin beta-1 chainApoptosis regulator Bcl-2Nuclear receptor subfamily 1 group I member 2
Waktu ParuhWhen a 24 hour infu…
Vol. Distribusi* 227 to 688 L/m^2 …
Klirens* 21.7 L/h/m2 [Dose…
Genetik -
small molecule | CAS: 186040-50-6

Deskripsi belum tersedia.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 199796-52-6

A combination of [docosahexaenoic Acid] (a natural fatty acid) and [paclitaxel] (an anticancer drug) being studied in the treatment of cancer. It is a type of mitotic inhibitor.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Target Protein:
Apoptosis regulator Bcl-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 263351-82-2

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1075214-55-9

Three paclitaxel molecules linked by a cleavable succinyl ester linkage to a brain peptide vector, Angiopep-2, conjugate named ANG1005.

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsCardiotoxic antineoplastic agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pacmilimab DB18873
biotech | CAS: 2145091-51-4

Pacmilimab is under investigation in clinical trial NCT04596150 (Study to Evaluate the Safety and Antitumor Activity of CX-2009 Monotherapy and in Combination With CX-072 in Advanced Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pacritinib Approved DB11697
small molecule | CAS: 937272-79-2

Myelofibrosis (MF) is a rare disorder characterized by hematopoietic abnormalities and fibrosis within the bone marrow.[L40793] The underlying cause of primary MF is unknown, but secondary MF can arise in patients with a history of polycythemia vera or essent…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +29
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK2Receptor-type tyrosine-protein kinase FLT3
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Padeliporfin Approved DB15575
small molecule | CAS: 759457-82-4

Padeliporfin is a water-soluble chlorophyll derivative and cytotoxic photosensitizer used for vascular-targeted photodynamic therapy for malignancies.[A244559] Vascular-targeted photodynamic therapy (VTP), or vascular targeted photochemotherapy, is a focal tr…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +9
Waktu ParuhThe estimated half-…
Vol. DistribusiIn healthy men rece…
KlirensFollowing administr…
Genetik -
Padimate O Approved DB11570
small molecule | CAS: 21245-02-3

Padimate O is an active sunscreen agent in cosmetics and over-the-counter sunscreen drug products in concentrations up to 8%, as regulated by the FDA [L2153]. It is a structurally-related compound to [DB02362] that absorbs UV-B rays to prevent photodamage. It…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +7
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Padnarsertib DB19243
small molecule | CAS: 1643913-93-2

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAcrylatesAmides +2
Target Protein:
Serine/threonine-protein kinase PAK 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Padsevonil DB14977
small molecule | CAS: 1294000-61-5

Padsevonil is under investigation in clinical trial NCT03695094 (A Study in Participants With Epilepsy, to Evaluate the Pharmacokinetics, Safety and Tolerability of Oxcarbazepine on Padsevonil).

Kategori:
AnticonvulsantsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Synaptic vesicle glycoprotein 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paeonol DB16830
small molecule | CAS: 552-41-0

Deskripsi belum tersedia.

Kategori:
Ketones
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pafolacianine Approved DB15413
small molecule | CAS: 1628423-76-6

Pafolacianine, or OTL38, is a folate analogue conjugated with a fluorescent dye that absorbs light in the near-infrared (NIR) spectrum [A242572] within a range of 760 nm to 785 nm, with a peak absorption of 776 nm. It emits fluorescence within a range of 790 …

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic AgentsDiagnostic Uses of Chemicals +10
Target Protein:
Folate receptor alpha
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean plasma cle…
Genetik -
Pafuramidine DB06532
small molecule | CAS: 186953-56-0

Pafuramidine, a prodrug of furamidine, currently has orphan status for _Pneumocystis jiroveci_ pneumonia.

Kategori:
AmidinesAnti-Infective AgentsAntiparasitic Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pagibaximab DB17786
biotech | CAS: 595566-61-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palazestrant DB18971
small molecule | CAS: 2092925-89-6

Palazestrant is under investigation in clinical trial NCT06016738 (OP-1250 (Palazestrant) vs. Standard of Care for the Treatment of ER+/HER2- Advanced Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palbociclib Approved DB09073
small molecule | CAS: 571190-30-2

Palbociclib is a piperazine pyridopyrimidine[A176792] that acts in the cell cycle machinery. It is a second generation cyclin-dependent kinase inhibitor[A176798] selected from a group of pyridopyrimidine compounds due to its favorable physical and pharmaceuti…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +21
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean apparent d…
KlirensThe mean apparent o…
Genetik -
Palifermin Approved DB00039
biotech | CAS: 162394-19-6

Palifermin is a recombinant human keratinocyte growth factor (KGF). It is 140 residues long, and is produced using E. coli. Palifermin was granted FDA approval on 15 December 2004.[L17933]

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsDetoxifying Agents for Antineoplastic Treatment +6
Target Protein:
Fibroblast growth factor receptor 2Fibroblast growth factor receptor 1Basement membrane-specific heparan sulfate proteoglycan core protein
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Palifosfamide DB05668
small molecule | CAS: 31645-39-3

Palifosfamide (ZIO-201) is a proprietary stabilized metabolite of ifosfamide. Ifosfamide has been shown to be effective in high doses in treating testicular cancer, sarcoma and lymphoma.

Kategori:
Alkylating DrugsAmino AcidsAmino Acids, Basic +13
Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Paliperidone Approved DB01267
small molecule | CAS: 144598-75-4

Paliperidone is the primary active metabolite of risperidone. The mechanism of action is unknown but it is likely to act via a similar pathway to risperidone. It has been proposed that the drug's therapeutic activity in schizophrenia is mediated through a com…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +37
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptorD(4) dopamine receptor +12
Waktu ParuhThe terminal elimin…
Vol. Distribusi* 487 L
Klirens-
Genetik -
Paliroden DB05454
small molecule | CAS: 188396-77-2

Paliroden is an orally active neurotrophic, non-peptidic compound that activates synthesis of endogenous neurotrophines. Studies show that use of paliroden increased the rate of formation of both neural progenitors and mature neurons. It is indicated for use …

Target Protein:
Glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palivizumab Approved DB00110
biotech | CAS: 188039-54-5

Humanized monoclonal antibody (IgG1k) produced by recombinant DNA technology, directed to an epitope in the A antigenic site of the F protein of respiratory syncytial virus (RSV). Synagis is a composite of human (95%) and murine (5%) antibody sequences. The h…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +15
Target Protein:
Fusion glycoprotein F0Low affinity immunoglobulin gamma Fc region receptor III-BComplement C1r subcomponent +6
Waktu Paruh18-20 days (in adul…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14967-68-1

Palladium Pd-103 is under investigation in clinical trial NCT00247312 (Pd-103 Dose De-Escalation for Early Stage Prostate Cancer: A Prospective Randomized Trial).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palm oil DB14377
biotech | CAS: 8002-75-3

Palm oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsComplex MixturesDietary Fats +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palmidrol DB14043
small molecule | CAS: 544-31-0

A cannabinoid receptor-inactive eCB-related molecule used as prophylactic in helping to prevent respiratory viral infection. Palmidrol is available for human use as a supplement (400 mg capsules) and as food for medical purposes In Italy and Spain (300 mg and…

Kategori:
Agents producing tachycardiaAlcoholsAmines +15
Target Protein:
Cannabinoid receptor 2Glucose-dependent insulinotropic receptorG-protein coupled receptor 55
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palmitic Acid Approved DB03796
small molecule | CAS: 57-10-3

A common saturated fatty acid found in fats and waxes including olive oil, palm oil, and body lipids.

Kategori:
Enzyme InhibitorsFatty AcidsLipids +1
Target Protein:
Fatty acid-binding protein, adipocyteFatty acid-binding protein 5Alpha-lactalbumin +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 373-49-9

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
Target Protein:
UDP-3-O-[3-hydroxymyristoyl] N-acetylglucosamine deacetylaseFatty-acid peroxygenaseBifunctional cytochrome P450/NADPH--P450 reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 147732-56-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 221227-05-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palomid 529 DB12812
small molecule | CAS: 914913-88-5

Palomid 529 has been used in trials studying the treatment of Age-Related Macular Degeneration.

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Palonosetron Approved DB00377
small molecule | CAS: 135729-56-5

Palonosetron (INN, trade name Aloxi) is an antagonist of 5-HT3 receptors that is indicated for the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV). It is the most effective of the 5-HT3 antagonists in controlling delayed CINV nause…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +22
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu ParuhApproximately 40 ho…
Vol. Distribusi* 8.3 ± 2.5 L/kg
Klirens* 160 +/- 35 mL/h/kg
Genetik -
Palopegteriparatide Approved DB18676
biotech | CAS: 2222514-07-8

Palopegteriparatide is a parathyroid hormone (PTH) analog. Palopegteriparatide is a prodrug consisting of PTH(1-34) conjugated to a methoxy polyethylene glycol carrier (mPEG) via a proprietary TransCon Linker.[L51134] PTH(1-34) contains the N-terminal part of…

Kategori:
Calcium HomeostasisParathyroid Hormones and AnaloguesSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins +1
Target Protein:
Parathyroid hormone/parathyroid hormone-related peptide receptor
Waktu ParuhThe apparent half-l…
Vol. DistribusiThe estimated appar…
KlirensThe estimated clear…
Genetik -
Palovarotene Approved DB05467
small molecule | CAS: 410528-02-8

Fibrodysplasia Ossificans Progressiva (FOP), with an estimated worldwide prevalence of one in 2 million individuals, is an exceptionally rare genetic disorder.[A244920] FOP is caused by a gain-of-function mutation in the ACVR1/ALK2 gene which results in progr…

Kategori:
BCRP/ABCG2 InhibitorsBenzene DerivativesBenzylidene Compounds +17
Target Protein:
Retinoic acid receptor gamma
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent total …
Genetik -
Palucorcel DB17955
biotech

Palucorcel is an investigational stem cell therapy consisting of human umbilical tissue-derived cells. Developed by Janssen Biotech, it is being investigated for the treatment of various conditions such as amyotrophic lateral sclerosis (ALS) and macular degen…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pam2csk4 DB16474
small molecule | CAS: 574741-81-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsDNA-Binding ProteinsExperimental Unapproved Treatments for COVID-19 +5
Target Protein:
Toll-like receptor 6Toll-like receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pamapimod DB19169
small molecule | CAS: 449811-01-2

Pamapimod is under investigation in clinical trial NCT05659459 (The KIN-FAST Trial (KIN001 for Accelerated Symptoms Termination) in Non Hospitalized Patients Infected With Sars-cov-2).

Kategori:
p38 Mitogen-Activated Protein Kinases, antagonists & inhibitorsPyridines
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pamidronic acid Approved DB00282
small molecule | CAS: 40391-99-9

Pamidronic acid is a second generation, nitrogen containing bisphosphonate similar to [neridronic acid] and [alendronic acid].[A203111] Pamidronic acid was first described in the literature in 1977.[A203267] The second generation bisphosphonates are less comm…

Kategori:
Agents Causing Muscle ToxicityAntineoplastic AgentsBisphosphonates +7
Target Protein:
Farnesyl pyrophosphate synthaseHydroxylapatiteGeranylgeranyl pyrophosphate synthase +2
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
KlirensThe mean total clea…
Genetik -
Pamrevlumab DB14952
biotech | CAS: 946415-13-0

Pamrevlumab is under investigation in clinical trial NCT00913393 (Study of FibroGen (FG)-3019 in Subjects With Type 2 Diabetes Mellitus and Kidney Disease on ACEi and/or ARB Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 59763-91-6

Pancreatic Polypeptide has been investigated for the treatment of Diabetes Mellitus, Type 1.

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal AgentsHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pancrelipase Approved DB00085
biotech | CAS: 53608-75-6

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase mixture was developed by Ortho-McNeil-Janssen Pharmace…

Kategori:
Alimentary Tract and MetabolismCarboxylic Ester HydrolasesComplex Mixtures +10
Target Protein:
Dietary fatDietary proteinDietary starch
Waktu ParuhPancrelipase acts l…
Vol. DistribusiPancrelipase acts l…
KlirensPancrelipase acts l…
Genetik -
Pancrelipase amylase Approved DB11065
biotech | CAS: 9000-90-2

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The amylases are enzymes that help in the chemical process of digestion…

Kategori:
AmylasesAmylases, antagonists & inhibitorsEnzymes +3
Target Protein:
Dietary starch
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancrelipase lipase Approved DB13147
biotech | CAS: 9001-62-1

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase lipase is an enzyme secreted by the pancreas that is r…

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +4
Target Protein:
Dietary fat
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancrelipase protease Approved DB11066
biotech | CAS: 9001-94-9

Pancrelipase, in general, is composed of a mixture of pancreatic enzymes which include amylases, lipases, and proteases. These enzymes are extracted from porcine pancreatic glands.[L2509] The pancrelipase protease is a mix of enzymes, formed by trypsin and ch…

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +1
Target Protein:
Dietary protein
Waktu ParuhPlease refer to [DB…
Vol. DistribusiPlease refer to [DB…
KlirensPlease refer to [DB…
Genetik -
Pancuronium Approved DB01337
small molecule | CAS: 16974-53-1

A bis-quaternary steroid that is a competitive nicotinic antagonist. As a neuromuscular blocking agent it is more potent than curare but has less effect on the circulatory system and on histamine release.

Kategori:
Agents producing tachycardiaAndrostanesAndrostanols +19
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu Paruh1.5 to 2.7 hours.
Vol. Distribusi* 241 to 280 mL/kg
Klirens* Plasma cl=1.1–1.9…
Genetik -
Panobacumab DB15342
biotech | CAS: 885053-97-4

Panobacumab is under investigation in clinical trial NCT00851435 (Safety and Pharmacokinetics of KBPA-101 in Hospital Acquired Pneumonia Caused by O11 Pseudomonas Aeruginosa).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Panobinostat Approved DB06603
small molecule | CAS: 404950-80-7

Panobinostat is an oral deacetylace (DAC) inhibitor approved on February 23, 2015 by the FDA for the treatment of multiple myeloma. The approval was accelerated based on progression-free survival, therefore confirmatory trials by the sponsor to demonstrate cl…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Histone deacetylase 1Histone deacetylase
Waktu Paruh30 hours
Vol. Distribusi-
Klirens-
Genetik -
Pantethine Approved DB11190
small molecule | CAS: 16816-67-4

Pantethine is a naturally occurring compound synthesized in the body from pantothenic acid (vitamin B5) via addition of cysteamine. It consists of two molecules of pantetheine that form a dimer via disufide linkages, and acts as an intermediate in the product…

Kategori:
Alimentary Tract and MetabolismSulfhydryl CompoundsSulfur Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Panthenol Approved DB11204
small molecule | CAS: 16485-10-2

Panthenol is an alcohol derivative of pantothenic acid, a component of the B complex vitamins and an essential component of a normally functioning epithelium. Panthenol exists as a racemic mixture containing both the dextrorotatory form (dexpanthenol) and the…

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9201–9250 dari 12560
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