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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

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Hasil Pencarian (14063)

Halaman 184 / 282
small molecule | CAS: 532-40-1

Deskripsi belum tersedia.

Kategori:
MicronutrientsPyrimidinesSulfur Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Monopotassium phosphate Approved DB09413
small molecule | CAS: 7778-77-0

Monopotassium phosphate, MKP, (also potassium dihydrogenphosphate, KDP, or monobasic potassium phosphate), KH2PO4, is a soluble salt of potassium and the dihydrogen phosphate ion. It is a source of phosphorus and potassium as well as a buffering agent. It ca…

Kategori:
AcidsAcids, NoncarboxylicAnions +15
Waktu ParuhIn healthy children…
Vol. DistribusiPotassium first ent…
KlirensPhosphates are rapi…
Genetik -
Monoxerutin DB13764
small molecule | CAS: 23869-24-1

Monoxerutin is a flavonol, a type of flavonoid.

Kategori:
Capillary Stabilizing AgentsFlavonoidsVasoprotectives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Montelukast Approved DB00471
small molecule | CAS: 158966-92-8

Montelukast was first approved for clinical use by the US FDA in 1998 as Merck's brand name Singulair.[L6301] The medication is a member of the leukotriene receptor antagonist (LTRA) category of drugs.[L6301,L6304,L6307,L6310,L6325,L6328,L6331] Although capab…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAgents to Treat Airway Disease +29
Target Protein:
Cysteinyl leukotriene receptor 1Polyunsaturated fatty acid 5-lipoxygenase
Waktu ParuhStudies have demons…
Vol. DistribusiThe steady-state vo…
KlirensThe plasma clearanc…
Genetik -
Monteplase DB12726
biotech | CAS: 156616-23-8

Monteplase has been used in trials studying the treatment of Pulmonary Embolism.

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBlood Proteins +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MOR-22 DB17790
biotech

MOR-22, a Natural human lymphoblastoid interferon-alpha, is currently being investigated to treat papillomavirus warts in the oral cavity of HIV-positive patients.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moricizine Approved DB00680
small molecule | CAS: 31883-05-3

An antiarrhythmia agent used primarily for ventricular rhythm disturbances.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +15
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh2 hours (range 1.5-…
Vol. Distribusi* 300 L
Klirens-
Genetik -
Morin DB16770
small molecule | CAS: 480-16-0

Deskripsi belum tersedia.

Kategori:
AntioxidantsBenzopyransBiological Factors +8
Target Protein:
Estrogen receptor betaSolute carrier family 22 member 12Fatty acid synthase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morinamide DB13417
small molecule | CAS: 952-54-5

Deskripsi belum tersedia.

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsDrugs for Treatment of Tuberculosis
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Moringa oleifera leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morinidazole DB15098
small molecule | CAS: 92478-27-8

Morinidazole is under investigation in clinical trial NCT03380793 (A Trial to Assess the Efficacy and Safety of Morinidazole in Patients With Appendicitis).

Kategori:
ImidazolesNitro Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Morniflumate DB09285
small molecule | CAS: 65847-85-0

Morniflumate is a non-steroidal anti-inflammatory drug with antipyretic properties. It is the morpholinoethyl ester of niflumic acid [L1496]. In one study, post morniflumate ingestion, physical examination and clinical symptoms of those with bronchitis show…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +14
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Polyunsaturated fatty acid 5-lipoxygenase +2
Waktu Paruh2h [L1498]
Vol. Distribusi-
Klirens45 ml/min [L1498]
Genetik -
Moroctocog alfa Approved DB13999
biotech | CAS: 284036-24-4

Moroctocog alfa, also known as BDDrFVIII (B domain deleted recombinant factor VIII), is a recombinant DNA-based drug with functional characteristics comparable to those of endogenous coagulation Factor VIII, the essential human blood clotting protein that is …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor XCoagulation factor IXvon Willebrand factor +8
Waktu ParuhMean terminal elimi…
Vol. DistribusiMean steady-state v…
KlirensMean clearance = 4.…
Genetik -
Morphine Approved DB00295
small molecule | CAS: 57-27-2

Morphine, the main alkaloid of opium, was first obtained from poppy seeds in 1805.[A176035] It is a potent analgesic, though its use is limited due to tolerance, withdrawal, and the risk of abuse.[A176050] Morphine is still routinely used today, though there …

Kategori:
AlkaloidsAnalgesicsAnesthetics +25
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Gen Terkait:
ABCB1 OPRM1
Waktu ParuhMorphine has a half…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik 2 Varian
small molecule | CAS: 20290-10-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingMorphinans +2
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cathepsin S
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 102-77-2

Deskripsi belum tersedia.

Kategori:
Cell-mediated ImmunityHeterocyclic Compounds, Fused-RingIncreased Histamine Release +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Morus alba root bark is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosapride DB11675
small molecule | CAS: 112885-41-3

Mosapride is under investigation for the treatment and prevention of Postoperative Ileus and Gastric Peroral Endoscopic Pyloromyotomy (G-POEM). Mosapride has been investigated for the treatment and diagnostic of Constipation, Type 2 Diabetes, Functional Dyspe…

Kategori:
Acids, CarbocyclicAlimentary Tract and MetabolismAmides +13
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Moschus berezovskii musk sac resin is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosedipimod DB12592
small molecule | CAS: 221139-79-3

Mosedipimod has been used in trials studying the supportive care and treatment of Chemotherapy-induced Neutropenia.

Kategori:
Experimental Unapproved Treatments for COVID-19Lipids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosliciguat DB19425
small molecule | CAS: 2231749-54-3

Mosliciguat is under investigation in clinical trial NCT06635850 (A Phase 2 Study of Mosliciguat in PH-ILD).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mosunetuzumab Approved DB15434
biotech | CAS: 1905409-39-3

Mosunetuzumab is a humanized anti-CD20/CD3 bispecific antibody.[L42230] It can recognize and bind two different targets simultaneously, CD20 on cancer B-cells and CD3 on T-cells, allowing it to redirect T-cell cytotoxic activity to cancer cells.[A249320] The …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +13
Target Protein:
B-lymphocyte antigen CD20T-cell surface glycoprotein CD3 epsilon chain
Waktu ParuhMosunetuzumab has a…
Vol. DistribusiThe estimated centr…
KlirensThe mean steady-sta…
Genetik -
Motesanib DB05575
small molecule | CAS: 453562-69-1

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingNicotinic Acids +3
Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor Kit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 246252-06-2

Motexafin gadolinium is studied in the treatment of cancer by Pharmacyclics. It may make tumor cells more sensitive to radiation therapy, improve tumor images using magnetic resonance imaging (MRI), and kill cancer cells. It belongs to the family of drugs cal…

Kategori:
Antineoplastic AgentsBiological FactorsCompounds used in a research, industrial, or household setting +9
Target Protein:
Peroxiredoxin-5, mitochondrialThioredoxin reductase 1, cytoplasmicThioredoxin reductase 2, mitochondrial +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 246252-04-0

Motexafin lutetium (MLu) is a second-generation photosensitizer for photodynamic therapy (PDT) of cancer. It belongs to the family of drugs called metallotexaphyrins. Also called lutetium texaphyrin. Motexafin lutetium is a pentadentate aromatic metallotexaph…

Kategori:
Biological FactorsCoordination ComplexesDermatologicals +5
Target Protein:
Prostate-specific antigen
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motixafortide Approved DB14939
biotech | CAS: 664334-36-5

Motixafortide is a cyclic peptide hematopoietic stem cell mobilizer used to improve stem cell collection prior to autologous transplantation.[L48116] Hematopoietic stem cell transplantation (HSCT) is commonly employed in the context of hematologic cancers - h…

Kategori:
Amino Acids, Peptides, and ProteinsHematopoietic Stem Cell MobilizerPeptides
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhThe effective half-…
Vol. DistribusiIn a typical patien…
KlirensIn a typical patien…
Genetik -
Motolimod DB12303
small molecule | CAS: 926927-61-9

Motolimod has been used in trials studying the treatment of Lymphoma, Tongue Cancer, Ovarian Cancer, Adult Solid Neoplasm, and Fallopian Tube Cancer, among others.

Kategori:
Heterocyclic Compounds, Fused-RingToll-Like Receptor 8, agonists
Target Protein:
Toll-like receptor 8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motretinide DB13368
small molecule | CAS: 56281-36-8

Deskripsi belum tersedia.

Kategori:
AlkenesAnti-Acne PreparationsAnti-Acne Preparations for Topical Use +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Motuporin DB04738
small molecule | CAS: 141672-08-4

Motuporin is a toxin isolated from the marine sponge Thenonella swinhoie grey.

Kategori:
Amino Acids, Peptides, and ProteinsCytotoxinsPeptides
Target Protein:
Serine/threonine-protein phosphatase PP1-gamma catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moxaverine DB12251
small molecule | CAS: 10539-19-2

Moxaverine has been investigated for the treatment of Retina, Ocular Physiology, and Regional Blood Flow.

Kategori:
Alimentary Tract and MetabolismAlkaloidsAutonomic Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moxestrol DB13418
small molecule | CAS: 34816-55-2

Deskripsi belum tersedia.

Kategori:
Estradiol CongenersEstrogen AntagonistsEstrogenic Steroids, Alkylated +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Moxetumomab pasudotox Approved DB12688
biotech | CAS: 1020748-57-5

CD22 is a lineage-restricted B-cell antigen that is expressed solely in on B-chronic lymphocytic leukemia, hairy cell leukemia, acute lymphocytic leukemiathe and Burkitt's lymphoma. The predecessor of Moxetumab pasudotox (MxP), named BL22, was first created b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
B-cell receptor CD22Elongation factor 2
Waktu ParuhMxP presents a shor…
Vol. DistribusiThe mean volume of …
KlirensThe mean systemic c…
Genetik -
Moxidectin Approved DB11431
small molecule | CAS: 113507-06-5

Moxidectin is a potent, broad-spectrum endectocide (antiparasitic that is active against endo- and ecto-parasites) with activity against nematodes, insects, and acari. It was first used in cattle followed by an approved use in general animals. It is a semi-sy…

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +9
Target Protein:
Glutamate-gated chloride channelGABA-A gated chloride channelABC transporters
Waktu ParuhMoxidectin reporter…
Vol. DistribusiMoxidectin presents…
KlirensThe apparent cleara…
Genetik -
Moxifloxacin Approved DB00218
small molecule | CAS: 151096-09-2

Moxifloxacin is a synthetic fluoroquinolone antibiotic agent. Bayer AG developed the drug (initially called BAY 12-8039) and it is marketed worldwide (as the hydrochloride) under the brand name Avelox (in some countries also Avalox) for oral treatment.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +18
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh11.5-15.6 hours (si…
Vol. Distribusi* 1.7 to 2.7 L/kg
Klirens* 12 +/- 2 L/hr
Genetik -
Moxisylyte Approved DB09205
small molecule | CAS: 54-32-0

Moxisylyte, denominated as thymoxamine in the UK, is a specific and orally active ?1-adrenergic antagonist.[T45] According to the WHO, moxisylyte is approved since 1987[T91] and in the same year, it acquired the denomination of orphan product by the FDA.[L117…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +17
Target Protein:
Alpha-1D adrenergic receptorAlpha adrenergic receptor
Waktu ParuhThe half-life of mo…
Vol. DistribusiIn preclinical tria…
KlirensIn preclinical tria…
Genetik -
Moxonidine Approved DB09242
small molecule | CAS: 75438-57-2

Moxonidine is a new-generation centrally acting antihypertensive drug approved for the treatment of mild to moderate essential hypertension. It is suggested to be effective in cases where other agents such as thiazides, beta-blockers, ACE inhibitors, and calc…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +8
Target Protein:
Alpha-2C adrenergic receptorAlpha-2B adrenergic receptorAlpha-2A adrenergic receptor +1
Waktu ParuhPlasma elimination …
Vol. Distribusi1.8±0.4L/kg. [FDA l…
KlirensAdministered twice …
Genetik -
biotech

RP-L102 is a lentiviral vector carrying the Fanconi Anemia-A (FANCA) gene currently being developed by Rocket Pharmaceuticals for the treatment of Fanconi anemia type A

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mozenavir DB02102
small molecule | CAS: 174391-92-5

Deskripsi belum tersedia.

Kategori:
Amides
Target Protein:
Gag-Pol polyproteinGag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MP-0250 DB17218
biotech | CAS: 1816305-70-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPB-1523 DB18334
small molecule

MPB-1523 is a contrast agent comprising PEGylated iron oxide nanoparticles.[L48161]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPT-0L055 DB17136
small molecule | CAS: 2069950-14-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MPT0B640 DB16512
small molecule

MPT0B640 was under investigation in clinical trials NCT04526717 for COVID-19 infection and NCT04294875 for locally advanced or metastatic solid malignancies.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRK-003 DB17015
small molecule | CAS: 623165-93-5

MRK-003 is a potent and selective ?-secretase inhibitor developed by Merck. It is the preclinical analog of [MK-0752], a drug in clinical development.[A252682]

Kategori:
Amyloid Precursor Protein Secretases, antagonists & inhibitorsEnzyme InhibitorsGamma Secretase Inhibitors and Modulators +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRK-409 DB13993
small molecule | CAS: 233275-76-8

MRK-409 is a GABA-A receptor agonist [A31972].

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3705 DB17668
biotech

mRNA-3705 is an investigational mRNA encoding methylmalonic CoA mutase (MUT) enzyme. Developed by Moderna TX Inc., it is being investigated for the treatment of methylmalonic academia.[A258843]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
mRNA-3927 DB17669
biotech

mRNA-3927 is an investigational mRNA therapy that consists of two mRNAs that encode for the alpha and beta subunits of the mitochondrial enzyme propionyl-CoA carboxylase (PCC) encapsulated within a lipid nanoparticle (LNP). Developed by Moderna Inc., it is be…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRT-2359 DB18015
small molecule | CAS: 2803881-11-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MRT5005 DB18260
biotech

MRT5005 is a human cystic fibrosis transmembrane conductance regulator (hCFTR) messenger RNA (mRNA) complexed with branched polyethyleneimine (bPEI).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 9151–9200 dari 14063
Sebelumnya Halaman 184 / 282 Berikutnya