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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 183 / 252
Otelixizumab DB05496
biotech | CAS: 881191-44-2

Otelixizumab is a monoclonal antibody that binds to a receptor found on all T cells called CD3, which is involved in normal T cell signaling. Otelixizumab is believed to inhibit the function of autoreactive T cells, which are important in propagating autoimmu…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otenabant DB11745
small molecule | CAS: 686344-29-6

Otenabant has been investigated for the treatment of Obesity.

Kategori:
Cannabinoid Receptor AntagonistsCannabinoids and similarsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Cannabinoid receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oteracil Approved DB03209
small molecule | CAS: 937-13-3

Oteracil is an adjunct to antineoplastic therapy, used to reduce the toxic side effects associated with chemotherapy. Approved by the European Medicines Agency (EMA) in March 2011, Oteracil is available in combination with [DB09257] and [DB09256] within the c…

Kategori:
Triazines
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Oteseconazole Approved DB13055
small molecule | CAS: 1340593-59-0

Oteseconazole is an azole metalloenzyme inhibitor that targets fungal CYP51.[L41635] CYP51, also known as 14? demethylase, participates in the formation of ergosterol, a compound that plays a vital role in the integrity of cell membranes.[L41635,A247020] By b…

Kategori:
14-alpha Demethylase InhibitorsAntifungal AgentsAntiinfectives for Systemic Use +5
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe median terminal…
Vol. DistribusiOn average, the vol…
KlirensClinical phase I st…
Genetik -
OTI-030 DB05648
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otilimab DB06303
biotech | CAS: 1638332-55-4

Investigated for the treatment of osteoarthritis and rheumatoid arthritis (RA).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otilonium DB13500
small molecule | CAS: 105360-89-2

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents producing tachycardiaAlimentary Tract and Metabolism +26
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OTL-103 DB17593
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OTL-201 DB17652
biotech

OTL-201 is an investigational hematopoietic stem cell (HSC) gene therapy being developed by Orchard Therapeutics for the treatment of mucopolysaccharidosis type IIIA (MPS-IIIA). It consists of a lentiviral vector to insert a functional copy of the human N-Sul…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Otlertuzumab DB16275
biotech | CAS: 1372645-37-8

Otlertuzumab is under investigation in clinical trial NCT01188681 (Safety and Efficacy Study of TRU-016 Plus Bendamustine vs. Bendamustine in Relapsed Chronic Lymphocytic Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Leukocyte antigen CD37
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ouabain Approved DB01092
small molecule | CAS: 630-60-4

A cardioactive glycoside consisting of rhamnose and ouabagenin, obtained from the seeds of Strophanthus gratus and other plants of the Apocynaceae; used like digitalis. It is commonly used in cell biological studies as an inhibitor of the NA(+)-K(+)-exchangin…

Kategori:
CarbohydratesCardanolidesCardenolides +16
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1Sodium/potassium-transporting ATPase subunit alpha-2Sodium/potassium-transporting ATPase subunit alpha-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ovatodiolide DB19264
small molecule | CAS: 3484-37-5

Ovatodiolide is under investigation in clinical trial NCT04220411 (A Study for AR100DP1 in Mild to Moderate Atopic Dermatitis (AD)).

Kategori:
Terpenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ovemotide DB19156
biotech | CAS: 181477-91-8

Ovemotide is under investigation in clinical trial NCT00357461 (Ipilimumab With or Without Vaccine Therapy in Treating Patients With Previously Treated Stage IV Melanoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxabolone DB01500
small molecule | CAS: 4721-69-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1254-35-9

Oxabolone cipionate is the C17? cypionate ester and a prodrug of [DB01500]. A synthetic anabolic-androgenic (AAS) steroid, it is a derivative of 19-nortestosterone (nandrolone). It is considered as a performance enhancing drug thus is prohibited from use in s…

Kategori:
Alimentary Tract and MetabolismAnabolic Agents for Systemic UseAnabolic Steroids +11
Waktu Paruh-
Vol. Distribusi-
KlirensThe elimination on …
Genetik -
Oxacillin Approved DB00713
small molecule | CAS: 66-79-5

An antibiotic similar to [flucloxacillin] used in resistant staphylococci infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2aPenicillin-binding protein 1A +7
Waktu Paruh20 to 30 minutes
Vol. Distribusi-
Klirens-
Genetik -
Oxaflozane DB13457
small molecule | CAS: 26629-87-8

Deskripsi belum tersedia.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsNervous System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxaliplatin Approved DB00526
small molecule | CAS: 61825-94-3

Oxaliplatin is a platinum-based chemotherapy drug in the same family as cisplatin and carboplatin. Compared to cisplatin the two amine groups are replaced by diamino cyclohexane (DACH) group to provide a greater antitumor effect.[A797] However, this leads to …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +9
Target Protein:
DNA
Waktu ParuhThe decline of ultr…
Vol. DistribusiAfter a single 2-ho…
KlirensPlatinum was cleare…
Genetik -
Oxametacin DB13308
small molecule | CAS: 27035-30-9

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAntiinflammatory and Antirheumatic ProductsAntiinflammatory and Antirheumatic Products, Non-Steroids +1
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxandrolone Approved DB00621
small molecule | CAS: 53-39-4

A synthetic hormone with anabolic and androgenic properties.

Kategori:
Alimentary Tract and MetabolismAnabolic AgentsAnabolic Agents for Systemic Use +13
Target Protein:
Androgen receptor
Waktu Paruh0.55 hours (1st pha…
Vol. Distribusi-
Klirens-
Genetik -
Oxantel DB13670
small molecule | CAS: 36531-26-7

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxaprotiline DB09307
small molecule | CAS: 56433-44-4

Oxaprotiline is a norepinephrine reuptake inhibitor of the tetracyclic antidepressant family that is related to maprotiline. This drug was never marketed. Oxaprotiline is a racemic mixture of the isomers levoprotiline and dextroprotiline. Levoprotiline is the…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnthracenes +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxaprozin Approved DB00991
small molecule | CAS: 21256-18-8

Oxaprozin is a non-narcotic, non-steroidal anti-inflammatory drug (NSAID), used to relieve the inflammation, swelling, stiffness, and joint pain associated with osteoarthritis and rheumatoid arthritis.

Kategori:
Acids, AcyclicAgents causing hyperkalemiaAgents that produce hypertension +22
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh54.9 hours
Vol. Distribusi* 11 to 17 L/70 kg
Klirens-
Genetik -
Oxazepam Approved DB00842
small molecule | CAS: 604-75-1

Oxazepam is an intermediate-acting, 3-hydroxybenzodiazepine used in the treatment of alcohol withdrawal and anxiety disorders. Oxazepam, like related 3-hydroxybenzodiazepine [lorazepam], is considered less susceptible to pharmacokinetic variability based on p…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +16
Target Protein:
GABA(A) ReceptorTranslocator proteinGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe mean eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
Oxazolam DB15491
small molecule | CAS: 24143-17-7

Deskripsi belum tersedia.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OXB-301 DB19269
biotech

OXB-301 is under investigation in clinical trial NCT00397345 (Trovax Renal Immunotherapy Survival Trial).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxcarbazepine Approved DB00776
small molecule | CAS: 28721-07-5

Oxcarbazepine is an anti-epileptic medication used in the treatment of partial onset seizures that was first approved for use in the United States in 2000.[L8627,L8630,L8633] It is a structural derivative of [carbamazepine][A186101] and exerts a majority of i…

Kategori:
Anti-epileptic AgentAnticonvulsantsCarboxamide Derivatives +29
Target Protein:
Sodium channel protein type 11 subunit alphaSodium channel protein
Gen Terkait:
HLA-B
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensPlasma clearance of…
Genetik 1 Varian
Oxelumab DB16663
biotech | CAS: 1186098-83-8

Oxelumab is under investigation in clinical trial NCT00983658 (A Study of HuMAb OX40L in the Prevention of Allergen-induced Airway Obstruction in Adults With Mild Allergic Asthma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxerutins DB15826
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxetacaine Approved DB12532
small molecule | CAS: 126-27-2

Oxetacaine, also called oxethazaince, is a potent surface analgesic with the molecular formula N, N-bis-(N-methyl-N-phenyl-t-butyl-acetamide)-beta-hydroxyethylamine that conserves its unionized form at low pH levels. Its actions have shown to relieve dysphagi…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAnestheticsAnesthetics, Local +5
Target Protein:
Gastrin
Waktu ParuhOxetacaine presents…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Oxetorone DB13463
small molecule | CAS: 26020-55-3

Deskripsi belum tersedia.

Kategori:
AnalgesicsAntimigraine PreparationsHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxfendazole DB11446
small molecule | CAS: 53716-50-0

Oxfendazole is a sulfoxide metabolite of fenbendazole. This benzimidazole antihelminthic protects livestock from roundworm. strongyles, and pinworn.

Kategori:
AnthelminticsAnti-Infective AgentsAntinematodal Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
OXI-4503 DB05143
small molecule | CAS: 288847-35-8

OXI-4503 is investigated in clinical trials for treating cancer/tumors. OXI-4503 is a solid. OXI-4503 blocks and destroys tumor vasculature, resulting in extensive tumor cell death and necrosis. OXI-4503 (combretastatin A1 di-phosphate / CA1P) is a unique and…

Kategori:
AcidsAcids, NoncarboxylicAnions +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxibendazole DB04910
small molecule | CAS: 20559-55-1

Oxibendazole is a polymerase inhibitor in phase III trials for the treatment of helminth intestinal infections.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +1
Target Protein:
Tubulin beta-4B chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxiconazole Approved DB00239
small molecule | CAS: 64211-45-6

Oxiconazole is an antifungal agent that is commonly found in topical formulations. It is marketed under the brand names Oxistat and Oxistat, and is used in the treatment of various skin infections such as athlete's foot, jock itch and ringworm.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +13
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol synthaseNuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 9032-53-5

Deskripsi belum tersedia.

Kategori:
BiopolymersBlood and Blood Forming OrgansCarbohydrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxidronic acid Approved DB14159
small molecule | CAS: 15468-10-7

Deskripsi belum tersedia.

Kategori:
OrganophosphonatesOrganophosphorus Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxilofrine Approved DB11610
small molecule | CAS: 365-26-4

Oxilofrine is used in combination with [DB11609] as an antitussive. It is currently marketed in Canada by Valeant under the tradename Cophylac.

Kategori:
AlcoholsAminesAmino Alcohols +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxiracetam DB13601
small molecule | CAS: 62613-82-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsNervous System +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxitriptan Approved DB02959
small molecule | CAS: 4350-09-8

5-Hydroxytryptophan (5-HTP), also known as oxitriptan (INN), is a naturally occurring amino acid and metabolic intermediate in the synthesis of serotonin and melatonin. 5-HTP is sold over-the-counter in the United Kingdom, United States and Canada as a dietar…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +8
Target Protein:
Tryptophan--tRNA ligase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxitropium DB12086
small molecule | CAS: 99571-64-9

Oxitropium has been investigated for the treatment of Pulmonary Disease, Chronic Obstructive.

Kategori:
Agents producing tachycardiaAlkaloidsAnticholinergic Agents +9
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxogluric acid DB08845
small molecule | CAS: 328-50-7

Oxogluric acid (?-Ketoglutarate) is not approved for any indication in the world but is an investigational drug in the United States. In the United States a phase I clinical trial is investigating whether oxogluric acid precursors found in nutritional supplem…

Kategori:
Acids, AcyclicDicarboxylic AcidsGlutarates +2
Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxolamine Approved DB13216
small molecule | CAS: 959-14-8

Oxolamine is not approved in the USA, it may be marketed elsewhere internationally as a cough suppressant [L5416]. It is listed as a prescription drug in New Zealand legislation [L5419]. Oxolamine is also approved in Taiwan for the treatment of respiratory tr…

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxomemazine DB13820
small molecule | CAS: 3689-50-7

Deskripsi belum tersedia.

Kategori:
Antihistamines for Systemic UseHeterocyclic Compounds, Fused-RingPhenothiazine Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxprenolol Approved DB01580
small molecule | CAS: 6452-71-7

A beta-adrenergic antagonist used in the treatment of hypertension, angina pectoris, arrhythmias, and anxiety.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +32
Target Protein:
Beta-1 adrenergic receptorBeta-3 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Oxtriphylline Approved DB01303
small molecule | CAS: 4499-40-5

Oxtriphylline is the choline salt form of [theophylline]. Once in the body, theophylline is released and acts as a phosphodiesterase inhibitor, adenosine receptor blocker, and histone deacetylase activator. Its main physiological reponse is to dilate the bron…

Kategori:
AlcoholsAlkaloidsAmines +19
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A3',5'-cyclic-AMP phosphodiesterase 4AAdenosine receptor A2a +2
Waktu ParuhThe serum half life…
Vol. DistribusiTheophylline has an…
KlirensTheophylline has an…
Genetik -
Oxybenzone Approved DB01428
small molecule | CAS: 131-57-7

Oxybenzone is an organic compound used in sunscreens. It is a derivative of benzophenone. It forms colorless crystals that are readily soluble in most organic solvents. It is used as an ingredient in sunscreen and other cosmetics because it absorbs UV-A ultra…

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingCosmetics +6
Target Protein:
Hormone-sensitive lipaseProgesterone receptorAndrogen receptor +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxybutynin Approved DB01062
small molecule | CAS: 5633-20-5

Overactive bladder (OAB) is a common condition negatively impacting the lives of millions of patients worldwide. Due to its urinary symptoms that include nocturia, urgency, and frequency, this condition causes social embarrassment and a poor quality of life.…

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAnticholinergic Agents +23
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M1
Waktu ParuhThe plasma eliminat…
Vol. DistribusiOxybutynin has a wi…
Klirens-
Genetik -
Oxycinchophen DB13596
small molecule | CAS: 485-89-2

Deskripsi belum tersedia.

Kategori:
Antiinflammatory and Antirheumatic ProductsMusculo-Skeletal SystemQuinolines +1
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Oxycodone Approved DB00497
small molecule | CAS: 76-42-6

Oxycodone is a semisynthetic opioid analgesic derived from thebaine in Germany in 1917.[A178696] It is currently indicated as an immediate release product for moderate to severe pain and as an extended release product for chronic moderate to severe pain requi…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +21
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu ParuhThe apparent elimin…
Vol. Distribusi2.6L/kg.[Label]
KlirensTotal plasma cleara…
Genetik -
Menampilkan 9101–9150 dari 12560
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