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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 182 / 252
ORG-25435 DB12312
small molecule | CAS: 256456-73-2

Org 25435 has been used in trials studying the treatment of Anaesthesia.

Kategori:
Benzene Derivatives
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
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ORG-25935 DB12220
small molecule | CAS: 1147011-84-4

Org 25935 has been used in trials studying the treatment of Alcoholism, Schizophrenia, and Panic Disorder.

Kategori:
Naphthalenes
Target Protein:
Sodium- and chloride-dependent glycine transporter 1
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ORG-31710 DB15585
small molecule | CAS: 118968-41-5

ORG-31710 is a progestational hormone antagonist.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Progesterone receptor
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ORG-34517 DB05423
small molecule | CAS: 189035-07-2

ORG-34517 is currently under investigation by Organon for the treatment of depression. It has potential to treat a number of diseases such as Cushing’s disease, hypertension, diabetes, glaucoma etc, in which the activity of metabolites corticosterone and cor…

Kategori:
DioxolesFused-Ring CompoundsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Glucocorticoid receptor
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Orgotein DB11444
biotech | CAS: 1569268-91-2

Superoxide is a natural byproduct of oxygen metabolism which, if left unchecked, leads to cell damage. Superoxide dismutase (SOD) is an enzyme that alternately catalyzes the dismutation of the superoxide radical into either the less damaging hydrogen peroxide…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAnalgesics, Non-Narcotic +9
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OriCar-017 DB17280
biotech

Deskripsi belum tersedia.

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Oridonin DB19086
small molecule | CAS: 28957-04-2

Oridonin is under investigation in clinical trial NCT05130892 (Effect of Inflammasome Inhibitor on Hscrp in Patients After PCI).

Kategori:
DiterpenesTerpenes
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Orilanolimab DB15312
biotech | CAS: 2066544-85-0

Orilanolimab is under investigation in clinical trial NCT03075878 (A Safety Study of SYNT001 in Subjects With Chronic, Stable Warm Autoimmune Hemolytic Anemia (WAIHA)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Orismilast DB19042
small molecule | CAS: 1353546-86-7

Orismilast is under investigation in clinical trial NCT05190419 (Study to Assess the Efficacy and Safety of Orismilast in Psoriasis).

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Oritavancin Approved DB04911
small molecule | CAS: 171099-57-3

Oritavancin is a glycopeptide antibiotic used for the treatment of skin infections. It was developed by The Medicines Company (acquired by Novartis).[L12858] Oritavancin was initially approved by the FDA in 2014 and formulated to combat susceptible gram-posit…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +24
Target Protein:
Dihydropteroate synthasePeptidoglycan precursorsBacterial cell wall peptide bridging segments +1
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of or…
Genetik -
Orlistat Approved DB01083
small molecule | CAS: 96829-58-2

The global prevalence of obesity is increasing rapidly. Obesity-related complications lead to significant personal and economic burden by reducing quality of life and increasing the cost of healthcare. In some individuals, diet and exercise are insufficient …

Kategori:
Alimentary Tract and MetabolismAnti-Obesity AgentsAntiobesity Preparations, Excl. Diet Products +11
Target Protein:
Pancreatic triacylglycerol lipaseCannabinoid receptor 1Gastric triacylglycerol lipase +1
Waktu ParuhThe half-life of or…
Vol. DistribusiVolume of distribut…
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ORM-12741 DB12057
small molecule | CAS: 610782-82-6

ORM-12741 has been used in trials studying the basic science and treatment of Alzheimer's Disease.

Kategori:
Adrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +2
Target Protein:
Alpha-2C adrenergic receptor
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ORM-13070 C-11 DB15324
small molecule | CAS: 1227170-74-2

ORM-13070 C-11 is under investigation in clinical trial NCT00735774 (Suitability of 11C-ORM-13070 as a PET Tracer).

Kategori:
Carbon Radioisotopes
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Ormeloxifene DB13310
small molecule | CAS: 31477-60-8

Ormeloxifene is a third-generation selective estrogen receptor (ER) modulator. In India, ormeloxifene has been marketed since the 1990s as a non-hormonal, non-steroidal oral contraceptive taken once a week,[A251450] and it was later introduced for the treatme…

Kategori:
Adrenal Cortex HormonesBenzopyransChromans +13
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu ParuhIn healthy, non-lac…
Vol. DistribusiIn healthy women, t…
KlirensIn healthy, non-lac…
Genetik -
Ornidazole DB13026
small molecule | CAS: 16773-42-5

Ornidazole has been used in trials studying the prevention of Elective Colorectal Surgery.

Kategori:
AmebicidesAnti-Infective AgentsAntibacterials for Systemic Use +13
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Ornithine Approved DB00129
small molecule | CAS: 70-26-8

Produced during the urea cycle, ornithine is an amino acid produced from the splitting off of urea from arginine. L-Ornithine allows for the disposal of excess nitrogen and acts as a precursor of citrulline and arginine.

Kategori:
Alimentary Tract and MetabolismAmino AcidsAmino Acids, Basic +9
Target Protein:
Ornithine aminotransferase, mitochondrialOrnithine transcarbamylase, mitochondrialArginase-1 +7
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Orotic acid DB02262
small molecule | CAS: 65-86-1

Deskripsi belum tersedia.

Kategori:
PyrimidinesPyrimidinones
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialOrotate phosphoribosyltransferaseDihydroorotate dehydrogenase (quinone), mitochondrial +3
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Orotidylic acid DB02957
small molecule | CAS: 2149-82-8

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPyrimidine Nucleotides +3
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ORP-101 DB16072
small molecule | CAS: 1820753-68-1

ORP-101 is under investigation in clinical trial NCT04129619 (A Comparison of the Effects of ORP-101 Versus Placebo in Adult Patients With Irritable Bowel Syndrome With Diarrhea (IBS-D)).

Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
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Orteronel DB12066
small molecule | CAS: 566939-85-3

Orteronel has been investigated for the treatment of Prostate Cancer.

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Orthosiphon aristatus leaf Approved DB15838
biotech

Deskripsi belum tersedia.

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Orticumab DB16653
biotech | CAS: 1314241-10-5

Orticumab is under investigation in clinical trial NCT04776629 (A Proof-of-activity Study With Orticumab in Subjects With Psoriasis and Cardiometabolic Risk Factors).

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biotech

Deskripsi belum tersedia.

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Orvepitant DB12427
small molecule | CAS: 579475-18-6

Orvepitant has been used in trials studying the treatment of Depressive Disorder, Depressive Disorder, Major, Post-Traumatic Stress Disorder, and Posttraumatic Stress Disorder (PTSD).

Kategori:
Antidepressive AgentsCentral Nervous System Depressants
Target Protein:
Substance-P receptor
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OS2966 DB17207
biotech

OS2966 is a humanized integrin ?1 (CD29) blocking antibody currently evaluated for the treatment of acute myeloid leukemia, glioblastoma and ovarian cancer.[A254561, L47351]

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Osalmid DB16273
small molecule | CAS: 526-18-1

Osalmid is under investigation in clinical trial NCT03670173 (Safety and Efficacy Assessments of Osalmid in Multiple Myeloma).

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Osanetant DB04872
small molecule | CAS: 160492-56-8

Developed by Sanofi-Aventis (formerly Sanofi-Synthelabo), osanetant (SR-142801) is an NK3 receptor antagonist which was under development for the treatment of schizophrenia and other Central Nervous System (CNS) disorders. In a review of its R&D portfolio, th…

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +3
Target Protein:
Neuromedin-K receptor
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Osbond acid DB14088
small molecule | CAS: 25182-74-5

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
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OSE-2101 DB17122
biotech

Deskripsi belum tersedia.

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Oseltamivir Approved DB00198
small molecule | CAS: 196618-13-0

Oseltamivir (marketed as the product Tamiflu?), is an antiviral neuraminidase inhibitor used for the treatment and prophylaxis of infection with influenza viruses A (including pandemic H1N1) and B. Oseltamivir exerts its antiviral activity by inhibiting the a…

Kategori:
AcetamidesAcetatesAmides +8
Target Protein:
NeuraminidaseSialidase-1Sialidase-2
Waktu ParuhPlasma concentratio…
Vol. DistribusiThe mean volume of …
KlirensRenal clearance (18…
Genetik -
small molecule | CAS: 187227-45-8

Deskripsi belum tersedia.

Kategori:
AcetamidesAcetatesAcids, Acyclic +8
Target Protein:
Neuraminidase
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Osemitamab DB18219
biotech | CAS: 2460539-61-9

Deskripsi belum tersedia.

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OSI-027 DB12387
small molecule | CAS: 936890-98-1

OSI-027 has been used in trials studying the treatment of Any Solid Tumor or Lymphoma.

Target Protein:
Serine/threonine-protein kinase mTOR
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OSI-461 DB05415
small molecule

OSI-461 is a second-generation molecule belonging to a new class of drugs termed selective apoptotic anti-neoplastic drugs (SAANDs).

Kategori:
IndenesPhosphodiesterase Inhibitors
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
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OSI-7836 DB05837
small molecule

OSI-7836 is a member of the nucleoside class of cytotoxic drugs of which gemcitabine is the market leader. OSI Pharmaceuticals develops OSI-7836 as a next-generation gemcitabine. The anti-tumor activity of OSI-7836 appeares to be less schedule dependent than …

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosides
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OSI-7904L DB05457
small molecule

OSI-7904L is a liposome encapsulated thymidylate synthase inhibitor, which is indicated for use in advanced gastric and/or gastroesophageal adenocarcinoma (A-G/GEJA). Current treatments also inhibit thymidylate synthase but the innovative lipid coating of OSI…

Kategori:
Acids, AcyclicDicarboxylic AcidsHeterocyclic Compounds, Fused-Ring
Target Protein:
Thymidylate synthase
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OSI-930 DB05913
small molecule | CAS: 728033-96-3

OSI-930 is an orally active inhibitor of two clinically validated targets: c-Kit and the vascular endothelial growth factor receptor-2 (VEGFR-2). OSI-930 is designed to target both cancer cell proliferation and blood vessel growth (angiogenesis) in selected t…

Kategori:
Heterocyclic Compounds, Fused-RingSulfur Compounds
Target Protein:
Vascular endothelial growth factor receptor 2Mast/stem cell growth factor receptor KitVascular endothelial growth factor receptor 1
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Osilodrostat Approved DB11837
small molecule | CAS: 928134-65-0

Osilodrostat is an inhibitor of 11?-hydroxylase (also referred to as CYP11B1), the enzyme that catalyzes the final step in the biosynthesis of endogenous cortisol.[L12123] It is used to lower circulating cortisol levels in the treatment of Cushing's disease, …

Kategori:
Antiadrenal PreparationsAnticorticosteroidsCortisol Synthesis Inhibitors +32
Target Protein:
Cytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial
Waktu ParuhThe elimination hal…
Vol. DistribusiThe median apparent…
KlirensData regarding the …
Genetik -
Osimertinib Approved DB09330
small molecule | CAS: 1421373-65-0

Osimertinib is an oral, third-generation epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI) drug developed by AstraZeneca Pharmaceuticals.[A7926,L43453] Its use is indicated for the treatment of metastatic non-small cell lung cancer (NSCL…

Kategori:
Acids, AcyclicAcrylatesAmides +29
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe population esti…
Vol. DistribusiThe mean volume of …
KlirensOral clearance is 1…
Genetik -
Osivelotor DB18071
small molecule | CAS: 2417955-18-9

Deskripsi belum tersedia.

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Osocimab DB14818
biotech | CAS: 2056878-75-0

Osocimab is under investigation in clinical trial NCT03276143 (Factor XIa inhibition for the prevention of venous Thromboembolism in Patients Undergoing Total Knee Arthroplasty).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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OSSM-007 DB18553
biotech

OSSM-007 consists of interferon-gamma primed allogeneic mesenchymal stem cells.

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Ostabolin-C DB05536
small molecule | CAS: 188899-65-2

Ostabolin C was under investigation in clinical trial NCT00787358 (A Proof-of-Concept Study Investigating the Safety and Efficacy of ZT-031 on Hip Fracture Healing in Men and Postmenopausal Women (SHIFT)).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +3
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biotech

Ostrea edulis shell is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

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OSU-6162 DB19178
small molecule | CAS: 146798-66-5

OSU-6162 is under investigation in clinical trial NCT05641623 (OSU6162 as Add-on in Ssri/snri-resistant Depression).

Kategori:
Dopamine AgentsDopamine AntagonistsDopamine D2 Receptor Antagonists +2
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Osugacestat DB12006
small molecule | CAS: 1401066-79-2

Osugacestat (BMS-906024) has been used in trials studying the treatment of Cancer, Lymphoblastic Leukemia, Acute T-cell, and Precursor T-Cell Lymphoblastic Lymphoma.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
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OT-15 DB17950
biotech

Deskripsi belum tersedia.

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OT-551 DB05650
small molecule | CAS: 627085-11-4

OT-551 is a novel small molecule that is topically dosed in an eye drop and has the unique ability to penetrate cell membranes and reach both the front and the back of the eye. It is intended to treat Age-related macular Degeneration (AMD), and preclinical re…

Target Protein:
Nuclear factor erythroid 2-related factor 2
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OT-730 DB16112
small molecule | CAS: 870809-51-1

OT-730 is under investigation in clinical trial NCT00753168 (Phase 1-2 Evaluation of OT-730 Eye Drops in Reducing the Intraocular Pressure in Patients With Ocular Hypertension or Open-angle Glaucoma).

Target Protein:
Beta-3 adrenergic receptor
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Otamixaban DB06635
small molecule | CAS: 193153-04-7

Otamixaban is a novel direct Factor Xa (FXa) inhibitor. It is currently being developed by the French pharmaceutical company Sanofi-Aventis as a treatment for acute coronary syndrome.

Kategori:
AnticoagulantsAntithrombinsEnzyme Inhibitors +4
Target Protein:
Coagulation factor X
Waktu Paruh-
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Genetik -
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