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11778

Total database: 17430
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8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 181 / 236
Platensimycin DB08407
small molecule | CAS: 835876-32-9

Deskripsi belum tersedia.

Kategori:
3-Oxoacyl-(Acyl-Carrier-Protein) SynthaseAcids, CarbocyclicAmides +10
Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 2
Waktu Paruh-
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Platinum DB12257
small molecule | CAS: 7440-06-4

Platinum is under investigation for the treatment of Metastatic Breast Cancer, Non-small Cell Lung Cancer, Gastric Large Cell Neuroendocrine Carcinoma, Colorectal Large Cell Neuroendocrine Carcinoma, and Pancreatic Large Cell Neuroendocrine Carcinoma, among o…

Kategori:
Antineoplastic AgentsChlorine CompoundsCompounds used in a research, industrial, or household setting +9
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Genetik -
biotech

Platycodon grandiflorus root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsBiological ProductsCampanulaceae +8
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Plazomicin Approved DB12615
small molecule | CAS: 1154757-24-0

Developed by Achaogen biopharmaceuticals, plazomicin is a next-generation aminoglycoside synthetically derived from [DB12604]. The structure of plazomicin was established via appending hydroxylaminobutyric acid to [DB12604] at position 1 and 2-hydroxyethyl gr…

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +12
Target Protein:
rRNA methyltransferase 2, mitochondrial30S ribosomal protein S1130S ribosomal protein S14
Waktu ParuhThe mean (±SD) half…
Vol. DistribusiThe mean (±SD) volu…
KlirensFollowing administr…
Genetik -
Plecanatide Approved DB13170
small molecule | CAS: 467426-54-6

Plecanatide is a drug approved in January 2017 by the FDA for the treatment of chronic idiopathic constipation (CIC). It should not be used in children less than six years of age, and should be avoided in patients six years to 18 years of age

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +12
Target Protein:
Guanylyl cyclase CGuanylate cyclase soluble subunit alpha-2
Waktu Paruhhalf-life (t½) cann…
Vol. DistribusiConcentrations of p…
KlirensNo excretion studie…
Genetik -
Plerixafor Approved DB06809
small molecule | CAS: 110078-46-1

Plerixafor is a small-molecule inhibitor of C-X-C chemokine receptor type 4 (CXCR4) that acts as a hematopoietic stem cell mobilizer.[A7117,L45678] It is used to stimulate the release of stem cells from the bone marrow into the blood in patients with non-Hodg…

Kategori:
Adjuvants, ImmunologicAminesAnti-HIV Agents +9
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhPlerixafor has a di…
Vol. DistribusiPlerixafor has an a…
KlirensPlerixafor has a to…
Genetik -
Plevitrexed DB06163
small molecule | CAS: 153537-73-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Thymidylate synthase
Waktu Paruh-
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PLG-0206 DB18116
biotech | CAS: 847061-43-2

PLG-0206 is a peptide antibiotic under investigation for the treatment of periprosthetic joint infections.[L48106]

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Plicamycin Approved DB06810
small molecule | CAS: 18378-89-7

Plicamycin is an antineoplastic antibiotic produced by Streptomyces plicatus. It has been used in the treatment of testicular cancer, Paget's disease of bone, and, rarely, the management of hypercalcemia. The manufacturer discontinued plicamycin in 2000.

Kategori:
AnthracyclinesAntibiotics, AntineoplasticAntineoplastic Agents +15
Target Protein:
DNA
Waktu Paruh-
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Plinabulin DB05992
small molecule | CAS: 714272-27-2

Deskripsi belum tersedia.

Kategori:
DeuteriumPiperazines
Target Protein:
Translation initiation factor eIF2B subunit alphaTranslation initiation factor eIF2B subunit betaTumor necrosis factor
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Plitidepsin DB04977
small molecule | CAS: 137219-37-5

Aplidine is a peptide found in tunicates which shows promise in shrinking tumors in pancreatic, stomach, bladder, and prostate cancers. The specific marine organism is _Aplidium albicans_. Aplidine is also of interest as a potential treatment for some leukemi…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Palmitoyl-protein thioesterase 1Elongation factor 1-alpha 2
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PLN-74809 DB16515
small molecule

PLN-74809 is a small-molecule that dually inhibits both ?<sub>v</sub>?<sub>6</sub> and ?<sub>v</sub>?<sub>1</sub> to treat both idiopathic pulmonary fibrosis (IPF) and primary sclerosing cholangitis (PSC)[L31693]. The compound was granted orphan drug designat…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Integrin alpha-VIntegrin beta-1Integrin beta-6
Waktu Paruh-
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Plozalizumab DB12520
biotech | CAS: 1610761-46-0

Plozalizumab has been investigated for the treatment of Atherosclerosis. Plozalizumab, a novel humanized monoclonal antibody, specifically targets CCR2 chemokine receptors found on the surface of certain white blood cells including macrophages and monocytes. …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
C-C chemokine receptor type 2
Waktu Paruh-
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Plozasiran DB18997
biotech | CAS: 2379776-40-4

Plozasiran is under investigation in clinical trial NCT05089084 (Study of ARO-APOC3 (Plozasiran) in Adults With Familial Chylomicronemia Syndrome (FCS)).

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Plumbagin DB17048
small molecule | CAS: 481-42-5

Plumbagin is a compound investigated for its anticancer activity. It has been found that it inactivates the Akt/NF-kB, MMP-9 and VEGF pathways.[A253102]

Kategori:
Adjuvants, ImmunologicAdrenal Cortex HormonesAnthelmintics +17
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
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PLX-4720 DB06999
small molecule | CAS: 918505-84-7

Deskripsi belum tersedia.

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Vascular endothelial growth factor receptor 2Serine/threonine-protein kinase B-raf
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PLX-PAD DB17990
biotech

Deskripsi belum tersedia.

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PLX-R18 DB17989
biotech

Deskripsi belum tersedia.

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PLX51107 DB17543
small molecule | CAS: 1627929-55-8

PLX51107 is a potent and selective inhibitor of the bromodomain and extraterminal (BET) protein family.[A257246,A257251] PLX51107 is under investigation in clinical trial NCT04022785 (PLX51107 and Azacitidine in Treating Patients With Acute Myeloid Leukemia o…

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PLX8394 DB16038
small molecule | CAS: 1393466-87-9

PLX8394 is under investigation in clinical trial NCT02428712 (A Study of PLX8394 as a Single Agent in Patients With Advanced Unresectable Solid Tumors).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +1
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu Paruh-
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PM-060184 DB13137
small molecule | CAS: 960210-99-5

PM060184 has been used in trials studying Solid Tumors.

Kategori:
LactonesPyrans
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pM-81 DB17432
biotech

Deskripsi belum tersedia.

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PM02734 DB05158
small molecule

PM02734 is a marine derived compound. PM02734 as a new antiproliferative drug demonstrating activity against a broad spectrum of tumor types: breast, colon, pancreas, lung and prostate, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic
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PMI-001 DB05730
small molecule

PMI-001 is a stand-alone, disease-modifying, anti-rheumatic drug (DMARD) being developed by Phytomedics Inc. It is an extract of the roots of an undisclosed perennial shrub which interferes with the production of IL-2 and COX-2 proteins, for the potential tre…

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small molecule

Deskripsi belum tersedia.

Target Protein:
Alanine racemase
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PMX-205 DB17938
small molecule | CAS: 514814-49-4

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesReceptor, Anaphylatoxin C5a, antagonists & inhibitors
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PNT001 DB18375
biotech

PNT001 is a humanized IgG4 S228P monoclonal antibody targeting the cis conformation of the phosphorylated Thr231-Pro232 motif in tau.

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PNU-142721 DB08414
small molecule | CAS: 185220-03-5

Deskripsi belum tersedia.

Target Protein:
Gag-Pol polyprotein
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PNU177836 DB02977
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
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Poa compressa pollen Approved DB10713
biotech

Poa compressa pollen is the pollen of the Poa compressa plant. Poa compressa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityGrass Pollen Allergen ExtractsIncreased Histamine Release +2
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Pocapavir DB17736
small molecule | CAS: 146949-21-5

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntiviral AgentsBenzene Derivatives +2
Waktu Paruh-
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Pociredir DB18070
small molecule | CAS: 2490676-18-9

Deskripsi belum tersedia.

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Podofilox Approved DB01179
small molecule | CAS: 518-28-5

A lignan found in podophyllin resin from the roots of podophyllum plants. It is a potent spindle poison, toxic if taken internally, and has been used as a cathartic. It is very irritating to skin and mucous membranes, has keratolytic actions, has been used to…

Kategori:
Antimitotic AgentsAntineoplastic Agents, PhytogenicAntiviral Agents +11
Target Protein:
DNA topoisomerase 2-betaTubulin alpha-4A chainTubulin beta chain +1
Waktu Paruh1.0 to 4.5 hours.
Vol. Distribusi-
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Genetik -
Polaprezinc DB09221
small molecule | CAS: 107667-60-7

Polaprezinc is a chelated form of zinc and L-carnosine. It is a zinc-related medicine approved for the first time in Japan, which has been clinically used to treat gastric ulcers [L1307, L1308]. It was determined that polaprezinc may be effective in pressure…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Ulcer AgentsDipeptides +10
Target Protein:
Tumor necrosis factorInterleukin-6Interleukin-3 +5
Waktu ParuhThe half-life of po…
Vol. Distribusi-
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Polatuzumab vedotin Approved DB12240
biotech | CAS: 1313206-42-6

Polatuzumab vedotin is a CD79b-directed antibody-drug conjugate that delivers monomethyl auristatin E (MMAE), an anti-mitotic agent, to cancer cells.[L6658] The drug consists of three components - a humanized immunoglobulin G1 (IgG1) monoclonal antibody speci…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +22
Target Protein:
B-cell antigen receptor complex-associated protein beta chain
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe estimated centr…
KlirensThe predicted clear…
Genetik -
Poldine DB13507
small molecule | CAS: 596-50-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents producing tachycardiaAlimentary Tract and Metabolism +7
Waktu Paruh-
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Polifeprosan 20 DB16298
small molecule | CAS: 90409-78-2

Polifeprosan 20 is under investigation in clinical trial NCT00003878 (Carmustine Implants in Treating Patients With Brain Metastases).

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Poliglusam DB11234
small molecule | CAS: 9012-76-4

Poliglusam, or chitosan, is a linear polysaccharide consisting of D-glucosamine and N-acetyl-D-glucosamine. Naturally-occuring poliglusam is found in the cell walls of fungi, soil and sediments where it is produced from degradation of chitin induced by certai…

Kategori:
Anticholesteremic AgentsBiocompatible MaterialsBiopolymers +14
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Polihexanide Approved DB12277
small molecule | CAS: 28757-47-3

Polihexanide has been used in trials studying the treatment, prevention, and supportive care of Caries, Neoplasm, Skin Diseases, Nail Diseases, and Dental Plaque, among others.

Kategori:
AmidinesAnti-Infective AgentsAntiseptics and Disinfectants +7
Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
biotech

Deskripsi belum tersedia.

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biotech

Poliovirus type 1 antigen is a suspension of poliovirus Type 1 (Mahoney) used in the active immunization of infants (as young as 6 weeks of age), children, and adults for the prevention of poliomyelitis caused by poliovirus Type 1. The vaccine contains purifi…

Kategori:
Actively Acquired ImmunityInactivated Poliovirus Vaccine
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biotech

Poliovirus type 2 antigen is a suspension of poliovirus Type 2 (MEF-1) used in the active immunization of infants (as young as 6 weeks of age), children, and adults for the prevention of poliomyelitis caused by poliovirus Type 2. The vaccine contains purified…

Kategori:
Actively Acquired ImmunityInactivated Poliovirus Vaccine
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biotech

Poliovirus type 3 antigen is a suspension of poliovirus Type 3 (Saukett) used in the active immunization of infants (as young as 6 weeks of age), children, and adults for the prevention of poliomyelitis caused by poliovirus Type 3. The vaccine contains purifi…

Kategori:
Actively Acquired ImmunityInactivated Poliovirus Vaccine
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biotech

Polistes annularis venom protein is an extract of Polistes annularis venom. Polistes annularis venom protein is used in allergenic testing.

Kategori:
Bee and Wasp Venom
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Polmacoxib DB12399
small molecule | CAS: 301692-76-2

Polmacoxib has been used in trials studying the treatment of Osteoarthritis, Osteoarthritis, Hip, Osteoarthritis, Knee, Localized Primary Osteoarthritis of Hip, and Localized Primary Osteoarthritis of Knee.

Kategori:
AmidesAnti-Inflammatory AgentsAnti-Inflammatory Agents, Non-Steroidal +8
Target Protein:
Prostaglandin G/H synthase 2Carbonic anhydrase 1Carbonic anhydrase 2
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Poloxalene DB11451
small molecule | CAS: 691397-13-4

Ethylene oxide/propylene oxide copolymer is used as a food additive. It belongs to the family of Epoxides. These are compounds containing a cyclic ether with three ring atoms (one oxygen and two carbon atoms).

Kategori:
AlcoholsAnti-Infective AgentsCompounds used in a research, industrial, or household setting +8
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Poloxamer 188 Approved DB11333
small molecule | CAS: 691397-13-4

Poloxamer 188 (P188) is a nonionic block linear copolymer that exhibits rheologic, anti-thrombotic, anti-inflammatory, and cytoprotective activities in various tissue injury models [A33121]. Composed of two hydrophilic side-chains attached to a hydrophobic ce…

Kategori:
AlcoholsCompounds used in a research, industrial, or household settingEthylene Glycols +9
Waktu ParuhIn humans, P188 has…
Vol. DistribusiThe volume of distr…
KlirensFollowing a 48-hour…
Genetik -
Poloxamer 237 DB16553
small molecule

Deskripsi belum tersedia.

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Poloxamer 331 DB17761
small molecule

Deskripsi belum tersedia.

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