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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 181 / 252
Onatasertib DB12570
small molecule | CAS: 1228013-30-6

Onatasertib (CC-223) has been used in trials studying the treatment and basic science of Multiple Myeloma, Glioblastoma Multiforme, HepatoCellular Carcinoma, Non-small Cell Lung Cancer, and Diffuse Large B-Cell Lymphoma, among others.

Target Protein:
Serine/threonine-protein kinase mTOR
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ONCOS-102 DB17274
biotech | CAS: 1802359-98-3

Deskripsi belum tersedia.

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ONCOS?102 DB17173
biotech

Deskripsi belum tersedia.

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Ondansetron Approved DB00904
small molecule | CAS: 99614-02-5

A competitive serotonin type 3 receptor antagonist. It is effective in the treatment of nausea and vomiting caused by cytotoxic chemotherapy drugs, including cisplatin, and has reported anxiolytic and neuroleptic properties. Having been developed in the 19…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +29
Target Protein:
5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 4Mu-type opioid receptor +2
Gen Terkait:
CYP2D6 CYP2D6
Waktu ParuhThe half-life of on…
Vol. DistribusiThe volume of distr…
KlirensThe clearance value…
Genetik 2 Varian
Ondelopran DB12585
small molecule | CAS: 676501-25-0

Ondelopran has been used in trials studying the treatment of Alcohol Dependence.

Kategori:
AminesBenzene DerivativesBenzyl Compounds +3
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Onercept DB06495
biotech | CAS: 199685-57-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsMembrane ProteinsPolyethylene Glycols +3
Target Protein:
Tumor necrosis factor
Waktu Paruh-
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Onfekafusp alfa DB16269
biotech | CAS: 1957239-88-1

Onfekafusp alfa is under investigation in clinical trial NCT02938299 (Neoadjuvant L19IL2/L19TNF- Pivotal Study).

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Ongericimab DB18949
biotech | CAS: 2145096-91-7

Ongericimab is under investigation in clinical trial NCT05325203 (A Study to Evaluate the Efficacy and Safety of JS002 in Patients With Heterozygous Familial Hypercholesterolemia (Hefh).).

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Onion Approved DB10548
biotech

Onion allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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ONL-1204 DB18239
biotech | CAS: 2040964-58-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and Proteins
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ONO-2952 DB14802
small molecule | CAS: 895169-20-7

ONO-2952 is under investigation in clinical trial NCT01887002 (Study to Evaluate the Effects of ONO-2952 on Pain Perception Produced by Rectal Distention in Female Subjects With Diarrhea-Predominant Irritable Bowel Syndrome (IBS-D)).

Kategori:
CycloparaffinsHeterocyclic Compounds, Fused-Ring
Target Protein:
Translocator protein
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ONO-5334 DB19206
small molecule | CAS: 620614-15-5

ONO-5334 is under investigation in clinical trial NCT00532337 (Controlled Study of ONO-5334 in Postmenopausal Women With Osteopenia or Osteoporosis).

Kategori:
Osteoporosis, Postmenopausal, drug therapySulfur CompoundsThiazoles
Target Protein:
Cathepsin K
Waktu Paruh-
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ONO-7579 DB17236
small molecule | CAS: 1622212-25-2

Deskripsi belum tersedia.

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
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ONO-8539 DB15325
small molecule | CAS: 459842-29-6

ONO-8539 is under investigation in clinical trial NCT01707901 (A Study of the Effect of ONO-8539 on Oesophageal Pain Hypersensitivity in Patients With Non-erosive Reflux Disease).

Kategori:
Acids, CarbocyclicBenzene DerivativesReceptors, Prostaglandin E, EP1 Subtype, antagonists & inhibitors +1
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ONT-093 DB14069
small molecule | CAS: 216227-54-2

ONT-093 is an orally bioavailable inhibitor of P-glycoprotein (P-gp). In pre-clinical studies, ONT-093 could inhibit P-gp and reverse multidrug resistance at nM concentrations with no effect on paclitaxel pharmacokinetics.

Kategori:
Drug Resistance, MultipleP-glycoprotein inhibitors
Target Protein:
ATP-dependent translocase ABCB1
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Ontamalimab DB15298
biotech | CAS: 2098790-40-8

Ontamalimab is under investigation in clinical trial NCT03627091 (Efficacy and Safety Study of SHP647 as Maintenance Treatment in Participants With Moderate to Severe Crohn's Disease (CARMEN CD 307)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Onternabez DB18076
small molecule | CAS: 256934-39-1

Deskripsi belum tersedia.

Kategori:
Cannabinoid Receptor AgonistsCannabinoids and similarsHormones +3
Waktu Paruh-
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Ontuxizumab DB16270
biotech | CAS: 946415-62-9

Ontuxizumab is a humanized monoclonal antibody that targets endosialin or tumour endothelial marker 1 (TEM-1). It is under investigation in clinical trial NCT01574716 (Sarcoma Study of Morab-004 Utilization: Research and Clinical Evaluation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Onvansertib DB15110
small molecule | CAS: 1034616-18-6

Onvansertib is under investigation in clinical trial NCT03303339 (Onvansertib in Combination With Either Low-dose Cytarabine or Decitabine in Adult Patients With Acute Myeloid Leukemia (AML).).

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingProtein Kinase Inhibitors
Target Protein:
Serine/threonine-protein kinase PLK1
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biotech | CAS: 1620643-19-7

Onvitrelin ucalontide is under investigation in clinical trial NCT01485848 (EP-100 Plus Paclitaxel Versus Paclitaxel Alone in Patients With Ovarian Cancer).

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OP-145 DB05672
biotech | CAS: 732984-79-1

OP-145 is a synthetic antimicrobial peptide developed from human cathelicidin LL-37.

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Opaganib DB12764
small molecule | CAS: 915385-81-8

Opaganib, also known as ABC294640, is a selective [sphingosine kinase-2 (SK2)](https://go.drugbank.com/polypeptides/Q9NRA0) inhibitor that is orally administered.[L27436] This drug has potential anticancer, anti-inflammatory, and antiviral activities, with po…

Kategori:
Bridged-Ring CompoundsCycloparaffins
Target Protein:
Sphingosine kinase 2
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OPC-14523 DB05422
small molecule | CAS: 145969-30-8

OPC-14523 is an antidepressant drug developed by Otsuka America Pharmaceutical.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Sigma non-opioid intracellular receptor 15-hydroxytryptamine receptor 1ASodium-dependent serotonin transporter
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OPC-28326 DB05461
small molecule

At low doses, OPC 28326 selectively vasodilates the femoral arterial bed due to its inhibitory action at alpha-2-adrenoceptors while having minimal action on systemic blood pressure, heart rate and coronary, carotid, vertebral, renal, and mesenteric blood flo…

Kategori:
Amines
Target Protein:
5-hydroxytryptamine receptor 2BAlpha-2C adrenergic receptorAlpha-2B adrenergic receptor
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OPC-51803 DB05838
small molecule

OPC-51803 is the first nonpeptide vasopressin (AVP) V(2)-receptor-selective agonist. It is a V(2)-selective agonist that produces a significant antidiuretic action after single and multiple oral dosing in AVP-deficient and normal AVP states. It is useful ther…

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Vasopressin, agonists
Target Protein:
Vasopressin V2 receptor
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Opebacan DB06161
biotech | CAS: 206254-79-7

Deskripsi belum tersedia.

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Opelconazole DB18251
small molecule | CAS: 1931946-73-4

Deskripsi belum tersedia.

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small molecule

Deskripsi belum tersedia.

Target Protein:
Deoxyribose-phosphate aldolaseDeoxyribose-phosphate aldolase
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Opicapone Approved DB11632
small molecule | CAS: 923287-50-7

Opicapone is a potent, reversible, and peripherally-acting third-generation inhibitor of catechol-o-methyltransferase (COMT), an enzyme involved in the breakdown of various catecholamines including dopamine.[A36938, A203048] Many patients with Parkinson’s dis…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBCRP/ABCG2 Substrates +25
Target Protein:
Catechol O-methyltransferase
Waktu ParuhThe mean eliminatio…
Vol. DistribusiFollowing oral admi…
KlirensFollowing oral admi…
Genetik -
Opicinumab DB14959
biotech | CAS: 1422268-07-2

Opicinumab is under investigation in clinical trial NCT02641041 (Safety, Tolerability, and Pharmacokinetics of Single and Multiple Doses of BIIB033 in Healthy Japanese Participants).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Opilio crab Approved DB10855
biotech

Opilio crab allergenic extract is used in allergenic testing.

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Opipramol DB12930
small molecule | CAS: 315-72-0

Opipramol has been used in trials studying the treatment of Dementia, Depression, Schizophrenia, Anxiety Disorders, and Psychosomatic Disorders.

Kategori:
Adrenergic AgentsAgents that produce hypertensionAgents that reduce seizure threshold +16
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Opiranserin DB16271
small molecule | CAS: 1441000-45-8

Opiranserin is under investigation in clinical trial NCT03997838 (Evaluate the Efficacy and Safety of VVZ-149 Injections for the Treatment of Post-operative Pain Following Abdominoplasty).

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Opium Approved DB11130
small molecule | CAS: 8008-60-4

Opium is the first substance of the diverse group of the opiates. It has been known for a long time, and the first evidence of a poppy culture dates from 5 thousand years by the Sumerians. During the years, opium was used as a sedative and hypnotic, but it wa…

Kategori:
Alimentary Tract and MetabolismAnalgesicsAntidiarrheals +25
Target Protein:
Delta-type opioid receptorKappa-type opioid receptorMu-type opioid receptor
Waktu ParuhThe half-life of op…
Vol. DistribusiOpium presents a la…
Klirens-
Genetik -
biotech | CAS: 945228-48-8

VB4-845 is studied in the treatment of certain types of head and neck cancer. VB4-845 is made by linking a monoclonal antibody fragment to a toxic protein that may kill cancer cells. VB4-845 is a fusion protein containing humanized scFv specific for the epith…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +8
Target Protein:
Epithelial cell adhesion molecule
Waktu Paruh-
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Oprelvekin Approved DB00038
biotech | CAS: 145941-26-0

Oprelvekin, the active ingredient in Neumega®, is recombinant Interleukin-11 (IL-11), which is produced in Escherichia coli (E. coli) by recombinant DNA technology. With a molecular mass of approximately 19,000 daltons, the non-glycosylated protein is 177 ami…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +7
Target Protein:
Interleukin-11 receptor subunit alpha
Waktu Paruh6.9 +/- 1.7 hrs
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Oprozomib DB11991
small molecule | CAS: 935888-69-0

Oprozomib has been used in trials studying the treatment of Solid Tumors, Multiple Myeloma, Waldenstrom Macroglobulinemia, Advanced Hepatocellular Carcinoma, and Advanced Non-Central Nervous System (CNS) Malignancies.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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OptPA DB18325
biotech

Optimized tPA (OptPA; W253R/R275S-tPA) is an engineered variant of tPA designed to exhibit reduced neurotoxicity.[A261486]

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biotech

The oral polio vaccine (OPV) is a live attenuated vaccine containing a mixture of one or more strains of poliovirus serotypes. Strains of the virus are selected based on their reduced incidence of spreading to the central nervous system but still having the a…

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Orange Approved DB10549
biotech

Orange allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Orantinib DB12072
small molecule | CAS: 252916-29-3

Orantinib has been used in trials studying the treatment of Lung Cancer, Breast Cancer, Kidney Cancer, Gastric Cancer, and Prostate Cancer, among others.

Kategori:
Acids, AcyclicAlkaloidsEnzyme Inhibitors +9
Target Protein:
Vascular endothelial growth factor receptor 2Aurora kinase AFibroblast growth factor receptor 1 +2
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ORC-13661 DB18903
small molecule | CAS: 1979935-33-5

ORC-13661 is under investigation in clinical trial NCT05730283 (Prevention of Ototoxicity in NTM Patients Treated With IV Amikacin).

Kategori:
AmidesSulfur Compounds
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Orciprenaline Approved DB00816
small molecule | CAS: 586-06-1

A beta-adrenergic agonist used in the treatment of asthma and bronchospasms. [PubChem]

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +26
Target Protein:
Beta-2 adrenergic receptor
Waktu Paruh6 hours
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Ordesekimab DB16649
biotech | CAS: 2394931-19-0

Ordesekimab is under investigation in clinical trial NCT02633020 (Study to Evaluate the Efficacy and Safety of AMG 714 in Adult Patients With Type II Refractory Celiac Disease).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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ORE-1001 DB12271
small molecule | CAS: 305335-31-3

ORE1001 has been used in trials studying the treatment of Mild to Moderate Ulcerative Colitis. It is an ACE2 inhibitor.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Peptides, and Proteins
Target Protein:
Angiotensin-converting enzyme 2Carboxypeptidase N catalytic chainCarboxypeptidase N subunit 2
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

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Oregovomab DB04964
biotech | CAS: 213327-37-8

Oregovomab is a murine monoclonal antibody that attaches to the tumor-associated antigen CA125.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Target Protein:
Mucin-16
Waktu Paruh-
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Orelabrutinib DB16272
small molecule | CAS: 1655504-04-3

Orelabrutinib is under investigation in clinical trial NCT04305197 (A Study of ICP-022 in Patients With Systemic Lupus Erythematosus (SLE)).

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBruton's tyrosine kinase (BTK) inhibitors +1
Target Protein:
Tyrosine-protein kinase BTK
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Orellanine DB19263
small molecule | CAS: 37338-80-0

Orellanine is under investigation in clinical trial NCT05287945 (Study of Orellanine in Metastatic Clear-cell or Papillary Renal Cell Carcinoma).

Kategori:
AgaricalesPyridines
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Orforglipron DB18964
small molecule | CAS: 2212020-52-3

Orforglipron is under investigation in clinical trial NCT06010004 (A Long-term Safety Study of Orforglipron (LY3502970) in Participants With Type 2 Diabetes).

Kategori:
Oxazoles
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh-
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