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11778

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Halaman 180 / 236
Pinus palustris pollen Approved DB10745
biotech

Pinus palustris pollen is the pollen of the Pinus palustris plant. Pinus palustris pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinus ponderosa pollen Approved DB10746
biotech

Pinus ponderosa pollen is the pollen of the Pinus ponderosa plant. Pinus ponderosa pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinus taeda pollen Approved DB10744
biotech

Pinus taeda pollen is the pollen of the Pinus taeda plant. Pinus taeda pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pinus virginiana pollen Approved DB10748
biotech

Pinus virginiana pollen is the pollen of the Pinus virginiana plant. Pinus virginiana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pioglitazone Approved DB01132
small molecule | CAS: 111025-46-8

Pioglitazone is an antihyperglycemic used as an adjunct to diet, exercise, and other antidiabetic medications to manage type 2 diabetes mellitus.[L11416,L11419,L11422,L11425] It is administered as a racemic mixture, though there is no pharmacologic difference…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCytochrome P-450 CYP2C8 Inhibitors +21
Target Protein:
Peroxisome proliferator-activated receptor gammaAmine oxidase [flavin-containing] B
Waktu ParuhThe mean serum half…
Vol. DistribusiThe average apparen…
KlirensThe apparent cleara…
Genetik -
Pipazethate DB08796
small molecule | CAS: 2167-85-3

A non-narcotic oral antitussive agent.

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipenzolate DB13844
small molecule | CAS: 13473-38-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipequaline DB13991
small molecule | CAS: 77472-98-1

Pipequaline is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It presents a unique chemical structure that does not follow the structural properties of other drugs of its class. Pipequaline has a simil…

Kategori:
Central Nervous System AgentsHeterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piperacillin Approved DB00319
small molecule | CAS: 66258-76-2

Semisynthetic, broad-spectrum, ampicillin derived ureidopenicillin antibiotic proposed for pseudomonas infections. It is also used in combination with other antibiotics.

Kategori:
Agents that produce neuromuscular block (indirect)AmidesAnti-Bacterial Agents +15
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 2BPenicillin-binding protein 2a +1
Waktu Paruh36-72 minutes
Vol. Distribusi* 101 mL/kg [intrav…
Klirens* 32 - 41 mL/min/1.…
Genetik -
Piperaquine Approved DB13941
small molecule | CAS: 4085-31-8

Piperaquine is an antimalarial agent first synthesized in the 1960's and used throughout China [A31550]. Its use declined in the 1980's as piperaquine resistant strains of *Plasmodium falciparum* appeared and artemisinin derivatives became available. It has c…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +19
Waktu ParuhThe terminal elimin…
Vol. DistribusiPiperaquine is thou…
KlirensThe mean apparent t…
Genetik -
Piperidione DB13224
small molecule | CAS: 77-03-2

Piperidione was cough medicine marketed by Roche under the trade name Sedulon.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pipradrol Approved DB11584
small molecule | CAS: 467-60-7

Pipradrol (Meratran) [L2523] was initially developed in the 1950s as an antidepressant, however, the adverse effects associated with its use and its abuse potential led to its withdrawal and international regulation [L2524]. Pipradrol was made illegal in man…

Kategori:
Central Nervous System StimulantsNervous SystemPsychoanaleptics +1
Target Protein:
D(1) dopamine receptor
Waktu Paruh-
Vol. DistribusiDistributed in the …
KlirensRapidly cleared [T1…
Genetik -
Piprinhydrinate DB15987
small molecule | CAS: 606-90-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piprozolin DB13202
small molecule | CAS: 17243-64-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBile and Liver TherapyBile Therapy +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piracetam Approved DB09210
small molecule | CAS: 7491-74-9

Piracetam is a nootropic drug in the racetams group, with chemical name 2-oxo-1-pyrrolidine acetamide. It shares the same 2-oxo-pyrrolidone base structure with pyroglutamic acid and is a cyclic derivative of the neurotransmitter ?-aminobutyric acid (GABA). Ho…

Kategori:
AcetamidesAcetatesAcids, Acyclic +12
Waktu ParuhThe plasma half lif…
Vol. DistribusiVd is approximately…
KlirensThe apparent total …
Genetik -
Pirarubicin DB11616
small molecule | CAS: 72496-41-4

Deskripsi belum tersedia.

Kategori:
AnthracyclinesAnthracyclines and Related SubstancesAntineoplastic Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirbuterol Approved DB01291
small molecule | CAS: 38677-81-5

Pirbuterol is a beta-2 adrenergic bronchodilator. In vitro studies and in vivo pharmacologic studies have demonstrated that pirbuterol has a preferential effect on beta-2 Adrenergic receptors compared with isoproterenol. While it is recognized that beta-2 adr…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +21
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptor
Waktu Paruh2 hours.
Vol. Distribusi-
Klirens-
Genetik -
Pirenzepine Approved DB00670
small molecule | CAS: 28797-61-7

An antimuscarinic agent that inhibits gastric secretion at lower doses than are required to affect gastrointestinal motility, salivary, central nervous system, cardiovascular, ocular, and urinary function. It promotes the healing of duodenal ulcers and due to…

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnti-Ulcer Agents +10
Target Protein:
Muscarinic acetylcholine receptor M1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirepemat DB19165
small molecule | CAS: 1227638-29-0

Pirepemat is under investigation in clinical trial NCT05258071 (A Clinical Study Evaluating Efficacy of Pirepemat on Falls Frequency in Patients With Parkinson's Disease (PD)).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Piretanide Approved DB02925
small molecule | CAS: 55837-27-9

Piretanide (INN, trade names Arelix, Eurelix, Tauliz) has been synthesized in 1973 at Hoechst AG (Germany) as a loop diuretic compound by using a then-new method for introducing cyclic amine residues in an aromatic nucleus in the presence of other aromaticall…

Kategori:
AmidesCardiovascular AgentsDiuretics +9
Target Protein:
Solute carrier family 12 member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirfenidone Approved DB04951
small molecule | CAS: 53179-13-8

Pirfenidone is a synthetic pyridone drug.[A251370] It is an antifibrotic agent with anti-inflammatory and antioxidant properties [A251370] that is used to treat idiopathic pulmonary fibrosis (IPF),[L26801] which is a chronic, progressive form of interstitial …

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +29
Target Protein:
Transforming growth factor beta-1 proprotein
Waktu ParuhThe mean terminal h…
Vol. DistribusiMean apparent oral …
KlirensFollowing administr…
Genetik -
Piribedil DB12478
small molecule | CAS: 3605-01-4

Piribedil has been investigated in Parkinson's Disease.

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson Agents (Dopamine Agonist)Anti-Parkinson Drugs +7
Target Protein:
D(3) dopamine receptorAlpha-2C adrenergic receptor5-hydroxytryptamine receptor 1A +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piritrexim DB03695
small molecule | CAS: 72732-56-0

Piritrexim has been used in trials studying the treatment of Bladder Cancer, Urethral Cancer, and Transitional Cell Cancer of the Renal Pelvis and Ureter.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsFolic Acid Antagonists
Target Protein:
Dihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirlimycin DB11537
small molecule | CAS: 79548-73-5

Pirlimycin hydrochloride is an antibiotic belonging to the _lincosamide_ class. Often marketed as _Pirsue_, this drug is used to treat mastitis in cattle.

Kategori:
Anti-Bacterial AgentsCarbohydratesGlycosides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirlindole DB09244
small molecule | CAS: 60762-57-4

This drug is classified as a reversible inhibitor of monoamine oxidase A enzyme (also known as a RIMA drug). It was developed and is currently used as an antidepressant in Russia. Its chemical structure is similar to metralindole, and it also shares pharmacol…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +14
Target Protein:
Amine oxidase [flavin-containing] A5-hydroxytryptamine receptor 1AAlpha-2A adrenergic receptor
Waktu Paruh0.7±0.3 in one stud…
Vol. Distribusi-
KlirensHigh plasma clearan…
Genetik -
Pirmitegravir DB18974
small molecule | CAS: 2245231-10-9

Pirmitegravir is under investigation in clinical trial NCT05869643 (A Clinical Trial of STP0404 in Treatment-naïve Adults With HIV-1 Infection).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piroctone DB15946
small molecule | CAS: 50650-76-5

Piroctone olamine is used in combination with other substances as a part of shampoo effectively reduced the amount of dandruff and, at the same time, provided hair conditioning advantages. Recently was shown, that piroctone olamine could induce apoptosis and …

Kategori:
AlcoholsAminesAmino Alcohols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Piromidic acid DB13744
small molecule | CAS: 19562-30-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 87234-24-0

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsSulfur CompoundsThiazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirprofen DB13722
small molecule | CAS: 31793-07-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pirtobrutinib Approved DB17472
small molecule | CAS: 2101700-15-4

Pirtobrutinib is a small molecule and a highly selective non-covalent inhibitor of Bruton’s tyrosine kinase (BTK). Its high selectivity has been associated with lower discontinuation rates due to adverse events and a lower incidence of atrial fibrillation.[A2…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +42
Target Protein:
Tyrosine-protein kinase BTK
Waktu ParuhPirtobrutinib has a…
Vol. DistribusiPirtobrutinib has a…
KlirensPirtobrutinib has a…
Genetik -
Pitavastatin Approved DB08860
small molecule | CAS: 147511-69-1

Pitavastatin, also known as the brand name product Livalo, is a lipid-lowering drug belonging to the statin class of medications. By inhibiting the endogenous production of cholesterol within the liver, statins lower abnormal cholesterol and lipid levels and …

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBCRP/ABCG2 Substrates +20
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-L
Waktu ParuhThe mean plasma eli…
Vol. DistribusiThe mean volume of …
KlirensFollowing a single …
Genetik -
Pitofenone DB15947
small molecule | CAS: 54063-52-4

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesDrugs for Functional Gastrointestinal Disorders +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pitolisant Approved DB11642
small molecule | CAS: 362665-56-3

Pitolisant is a selective antagonist or inverse agonist of the histamine H3 receptor used to treat type 1 or 2 narcolepsy.[L8063] Narcolepsy is a chronic neurological disorder that affects 1 in 2,000 individuals and is characterized by excessive daytime sleep…

Kategori:
Cytochrome P-450 CYP1A2 InducersCytochrome P-450 CYP1A2 Inducers (strength unknown)Cytochrome P-450 CYP2B6 Inducers +25
Target Protein:
Histamine H3 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhPitolisant has a pl…
Vol. DistribusiFollowing single an…
KlirensThe apparent oral c…
Genetik -
small molecule | CAS: 566170-04-5

Pittsburgh Compound B is under investigation in clinical trial NCT01723553 (Amyloid-related Imaging Abnormalities (Microbleeds) in Atypical AD).

Kategori:
AminesCarbon RadioisotopesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pivampicillin Approved DB01604
small molecule | CAS: 33817-20-8

Pivalate ester analog of ampicillin.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Pivmecillinam Approved DB01605
small molecule | CAS: 32886-97-8

Pivmecillinam is a mecillinam prodrug, a pivaloyloxymethyl ester of amdinocillin that is well absorbed orally, but broken down to amdinocillin in the intestinal mucosa. It is active against gram-negative organisms and used as for amdinocillin. [PubChem]

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pixatimod DB19166
small molecule | CAS: 1144617-49-1

Pixatimod is under investigation in clinical trial NCT05061017 (Pixatimod (PG545) Plus Nivolumab in PD-1 Relapsed/refractory Metastatic Melanoma and NSCLC and With Nivolumab and Low-dose Cyclophosphamide in MSS Metastatic Colorectal Carcinoma (Mcrc)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pixofisiran DB17294
biotech | CAS: 1152798-48-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Pizotifen Approved DB06153
small molecule | CAS: 15574-96-6

Pizotifen belongs to the class of antamines and is related to [cyproheptadine].[A32532] It is a potent serotonin and tryptamine antagonist that has been used for migraine prevention for many years. It exhibits weak anticholinergic, antihistamine, and antikini…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +27
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3 +12
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
PKI-179 DB13109
small molecule | CAS: 1197160-28-3

PKI-179 has been used in trials studying the treatment of Advanced Malignant Solid Tumors.

Kategori:
AmidesOxazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The placenta serves many purposes, with one of the many being a bank of mesenchymal stem cells (MSCs). It can be obtained relatively easily as medical waste from which MSCs can be non-invasively extracted and without the ethical issues that come with embryoni…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Placulumab DB11983
biotech | CAS: 945781-29-3

Placulumab has been used in trials studying the treatment of Rheumatoid Arthritis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plamotamab DB18944
biotech | CAS: 2138442-31-4

Plamotamab is under investigation in clinical trial NCT05328102 (Phase 2 Study of Plamotamab Combined With Tafasitamab Plus Lenalidomide Versus Tafasitamab Plus Lenalidomide in Relapsed or Refractory (R/R) Diffuse Large-cell B-cell Lymphoma (DLBCL)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The Covifenz COVID-19 vaccine (plant-based virus-like particles (VLP), recombinant, adjuvanted) is a plant-based vaccine developed in partnership by Medicago and GlaxoSmithKline which is approved in Canada for the prevention of COVID-19.[L40694] It is compose…

Kategori:
COVID-19 VaccinesVaccinesViral Vaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plantago seed Approved DB11097
biotech | CAS: 8063-16-9

Platango seeds refer to the seeds collected from various species of plantago trees. It is found in some laxatives for treating occasional constipation and restoring regularity in bowel movements. Its potential benefit in maintaining remission in ulcerative co…

Kategori:
Biological ProductsBulk-Forming LaxativesComplex Mixtures +5
Waktu ParuhThe half-life of ps…
Vol. DistribusiPsyllium husk when …
KlirensPsyllium husk when …
Genetik -
biotech

The plasma protein fraction human (PPFh) is defined as a sterile solution of proteins composed mainly of albumin and globulin derived from human plasma.[A32512] It is already reviewed under the category of biologics by the FDA where the processing, required t…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood Derivatives +9
Waktu ParuhThe registered clea…
Vol. DistribusiThe registered volu…
KlirensThe registered clea…
Genetik -
PlasmaCord DB16363
biotech

PlasmaCord is platelet-poor plasma that is derived by fractionation from sterile umbilical cord and placental blood.[L27581] It is developed by Cellpraxis and is currently being investigated against severe acute respiratory syndrome (SARS).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Plasminogen Approved DB16701
biotech | CAS: 9001-91-6

Plasminogen is a pro-enzyme (i.e. a zymogen) which is cleaved to form plasmin - also known as [fibrinolysin] - as part of the fibrinolytic pathway that breaks down fibrin blood clots.[A236035] This pathway is activated when a clot is no longer needed or to pr…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsBeta-Globulins +11
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean steady-sta…
KlirensThe clearance of Ry…
Genetik -
small molecule | CAS: 74389-68-7

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAlcoholsAmines +21
Target Protein:
Platelet-activating factor receptorGanglioside GM2 activator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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