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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 180 / 282
Metyrosine Approved DB00765
small molecule | CAS: 672-87-7

An inhibitor of the enzyme tyrosine 3-monooxygenase, and consequently of the synthesis of catecholamines. It is used to control the symptoms of excessive sympathetic stimulation in patients with pheochromocytoma. (Martindale, The Extra Pharmacopoeia, 30th ed)

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +6
Target Protein:
Tyrosine 3-monooxygenase
Waktu Paruh3.4 to 3.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Mevidalen DB19034
small molecule | CAS: 1638667-79-4

Mevidalen is under investigation in clinical trial NCT03305809 (A Study of LY3154207 in Participants With Dementia Due to Lewy Body Dementia (LBD) Associated With Idiopathic Parkinson's Disease (PD) or Dementia With Lewy Bodies (DLB)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75225-51-3

Deskripsi belum tersedia.

Kategori:
Naphthalenes
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevonlerbart DB19416
biotech | CAS: 2453195-99-6

Mevonlerbart is under investigation in clinical trial NCT06602726 (A Study to Demonstrate How Well REGN1908-1909 Works in Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Cat Allergy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mexiletine Approved DB00379
small molecule | CAS: 31828-71-4

Antiarrhythmic agent pharmacologically similar to lidocaine. It may have some anticonvulsant properties.

Kategori:
AminesAntiarrhythmic agentsAntiarrhythmics, Class I +20
Target Protein:
Sodium channel protein type 5 subunit alphaAryl hydrocarbon receptor
Waktu Paruh10-12 hours
Vol. Distribusi* 5 to 7 L/lg
Klirens-
Genetik -
Mezagitamab DB16370
biotech | CAS: 2227490-52-8

Mezagitamab is under investigation in clinical trial NCT04278924 (Study to Evaluate Safety, Tolerability, and Efficacy of TAK-079 in Participants With Persistent/chronic Primary Immune Thrombocytopenia).

Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezigdomide DB17584
small molecule | CAS: 2259648-80-9

Mezigdomide is under investigation in clinical trial NCT05372354 (A Study to Evaluate Safety, Drug Levels and Effectiveness of CC-92480 (BMS-986348) in Combination With Other Treatments in Participants With Relapsed or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezlocillin Approved DB00948
small molecule | CAS: 51481-65-3

Semisynthetic ampicillin-derived acylureido penicillin. It has been proposed for infections with certain anaerobes and may be useful in inner ear, bile, and CNS infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1APeptidoglycan synthase FtsIPenicillin-binding protein 3 +1
Waktu Paruh1.3 to 4.4 hours
Vol. Distribusi-
Klirens-
Genetik -
MF101 DB05052
small molecule

MF101 is a novel estrogen receptor beta (ER?) selective agonist and unlike currently available hormone therapies, does not activate the estrogen receptor alpha (ER?), known to be implicated in tumor formation. MF101 is an oral drug designed for the treatment …

Target Protein:
Estrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MF268 DB04021
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MG-S-2525 DB18063
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGB-BP-3 DB12892
small molecule | CAS: 1000277-08-6

Mgb Bp 3 is under investigation in clinical trial NCT02518607 (Safety, Blood Levels and Effects of MGB-BP-3).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGD-024 DB17265
biotech

MGD-024 is an anti-CD123/anti-CD3 bispecific DART molecule.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGN-4893 DB17338
biotech

MGN-4893 is an inhibitor of microRNA-451. In February 2011, it was granted FDA orphan designation for the treatment of polycythemia vera.[L47356]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mianserin Approved DB06148
small molecule | CAS: 24219-97-4

A tetracyclic compound with antidepressant effects. Mianserin was previously available internationally, however in most markets it has been phased out in favour of [mirtazapine].

Kategori:
Adrenergic AgentsAgents that produce hypertensionAntidepressive Agents +29
Target Protein:
Alpha-2A adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C +17
Waktu Paruh10-17 hours
Vol. Distribusi-
Klirens-
Genetik -
Mibampator DB12717
small molecule | CAS: 375345-95-2

Mibampator has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
AmidesBenzene DerivativesSulfones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibavademab DB16673
biotech | CAS: 2305770-44-7

Mibavademab is under investigation in clinical trial NCT04159415 (Study of REGN4461, a Leptin Receptor Agonist Antibody, in Patients With Generalized Lipodystrophy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibefradil DB01388
small molecule | CAS: 116644-53-2

Mibefradil was withdrawn from the market in 1998 because of potentially harmful interactions with other drugs.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntihypertensive Agents +31
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1GVoltage-dependent T-type calcium channel subunit alpha-1HVoltage-dependent L-type calcium channel subunit alpha-1C +8
Waktu Paruh17 to 25 hours at s…
Vol. Distribusi-
Klirens-
Genetik -
Mibenratide DB15195
small molecule | CAS: 1239011-83-6

Mibenratide is under investigation in clinical trial NCT01798745 (A Study to Assess the Pharmacokinetics and Pharmacodynamics of JNJ-54452840 in Participants With Heart Failure and Anti-beta1-adrenergic Receptor Autoantibodies).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibolerone DB11429
small molecule | CAS: 3704-09-4

Mibolerone is a potent anabolic steroid which is both higher affinity and more selective for the androgen receptor than metribolone.

Kategori:
EstranesEstrenesFused-Ring Compounds +7
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Micafungin Approved DB01141
small molecule | CAS: 235114-32-6

Micafungin is an antifungal drug. It belongs to the antifungal class of compounds known as echinocandins and exerts its effect by inhibiting the synthesis of 1,3-beta-D-glucan, an integral component of the fungal cell wall.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntifungal Agents +9
Target Protein:
1,3-beta-glucan synthase component FKS11,3-beta-glucan synthase component GSC2
Waktu Paruh14-17 hours
Vol. Distribusi* 0.39 ± 0.11 L/kg …
Klirens* 0.359 +/- 0.179 m…
Genetik -
Miconazole Approved DB01110
small molecule | CAS: 22916-47-8

Miconazole is a broad-spectrum azole antifungal with some activity against Gram-positive bacteria as well.[A203636] It is widely used to treat mucosal yeast infections, including both oral and vaginal infections; although intravenous miconazole is no longer a…

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +41
Target Protein:
Lanosterol 14-alpha demethylaseNitric oxide synthase 3Nitric oxide synthase, inducible +5
Waktu ParuhMiconazole has a te…
Vol. DistribusiA 1200 mg miconazol…
Klirens-
Genetik -
Microascus brevicaulis Approved DB10823
biotech

Microascus brevicaulis is a fungus which can provoke allergic reactions. Microascus brevicaulis extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Micronomicin Approved DB13274
small molecule | CAS: 52093-21-7

Micronomicin is an aminoglycoside antibiotic which is marketed in Japan, and sold under the brand names Sagamicin and Luxomicina.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Microsporum audouinii Approved DB10842
biotech

Microsporum audouinii is a fungus which can provoke allergic reactions. Microsporum audouinii extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Midazolam Approved DB00683
small molecule | CAS: 59467-70-8

Midazolam is a short-acting hypnotic-sedative drug with anxiolytic, muscle relaxant, anticonvulsant, sedative, hypnotic, and amnesic properties.[A173842] It belongs to a class of drugs called _benzodiazepines_. This drug is unique from others in this class du…

Kategori:
Adjuvants, AnesthesiaAnestheticsAnti-Anxiety Agents +27
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site +1
Waktu Paruh**Intravenous**: …
Vol. DistribusiFemale gender, old …
Klirens**Intramuscular** …
Genetik -
Midecamycin DB13456
small molecule | CAS: 35457-80-8

Midecamycin is a naturally occurring 16-membered macrolide[A33072] that fits under the category of acetoxy-substituted macrolide antibiotics. In this molecule, an acetoxy group is substituted on the position 9 of the 16-member ring and on position 4 of the te…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +12
Waktu ParuhThe half-life of mi…
Vol. DistribusiThe reported appare…
KlirensMidecamycin present…
Genetik -
Midodrine Approved DB00211
small molecule | CAS: 42794-76-3

An ethanolamine derivative that is an adrenergic alpha agonist. It is used as a vasoconstrictor agent in the treatment of hypotension.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +19
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor
Waktu ParuhThe metabolites dis…
Vol. Distribusi-
Klirens* Renal cl=385 mL/m…
Genetik -
Midomafetamine DB01454
small molecule | CAS: 42542-10-9

An N-substituted amphetamine analog. It is a widely abused drug classified as a hallucinogen and causes marked, long-lasting changes in brain serotonergic systems. It is commonly referred to as MDMA or ecstasy. It is a widely abused drug classified as a hallu…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +20
Target Protein:
Synaptic vesicular amine transporterSodium-dependent noradrenaline transporterSodium-dependent serotonin transporter +4
Waktu Paruh6–10 (though durati…
Vol. Distribusi-
Klirens-
Genetik -
Midostaurin Approved DB06595
small molecule | CAS: 120685-11-2

Midostaurin (as Rydapt) is a multitarget kinase inhibitor for the treatment for adult patients with newly diagnosed acute myeloid leukemia (AML) who have a specific genetic mutation called FLT3. It was initially characterized as a potential broad-spectrum ant…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +53
Target Protein:
Protein kinase C gamma typeProtein kinase C alpha typeVascular endothelial growth factor receptor 2 +4
Waktu ParuhElimination half li…
Vol. DistribusiThe Vd of midostaur…
KlirensThe clearance value…
Genetik -
Mifepristone Approved DB00834
small molecule | CAS: 84371-65-3

Mifepristone is a progestational and glucocorticoid hormone antagonist. Its inhibition of progesterone induces bleeding during the luteal phase and in early pregnancy by releasing endogenous prostaglandins from the endometrium or decidua. As a glucocorticoid …

Kategori:
Abortifacient AgentsAbortifacient Agents, SteroidalAdrenal Cortex Hormones +49
Target Protein:
Progesterone receptorGlucocorticoid receptorProstate-specific antigen +1
Waktu Paruh18 hours
Vol. Distribusi-
Klirens-
Genetik -
Migalastat Approved DB05018
small molecule | CAS: 108147-54-2

Fabry disease is a rare, progressive genetic disorder characterized by a defective GLA gene that causes a deficiency in the enzyme alpha-Galactosidase A (alpha-Gal A). This enzyme is responsible for breaking down glycosphingolipid substrate that, when deficie…

Kategori:
Alimentary Tract and MetabolismAlkaloidsAlpha-Galactosidase A (alpha-Gal A) Pharmacological Chaperones +6
Target Protein:
Alpha-galactosidase A
Waktu ParuhThe mean eliminatio…
Vol. DistribusiIn healthy voluntee…
KlirensFollowing ascending…
Genetik -
Miglitol Approved DB00491
small molecule | CAS: 72432-03-2

Miglitol inhibits the breakdown complex carbohydrates into glucose. It is primarily used in diabetes mellitus type 2 for establishing greater glycemic control by preventing the digestion of carbohydrates (such as disaccharides, oligosaccharides, and polysacch…

Kategori:
Alimentary Tract and MetabolismAlkaloidsBlood Glucose Lowering Agents +10
Target Protein:
Lysosomal alpha-glucosidaseNeutral alpha-glucosidase ABNeutral alpha-glucosidase C +1
Waktu ParuhThe elimination hal…
Vol. Distribusi* 0.18 L/kg
Klirens-
Genetik -
Miglustat Approved DB00419
small molecule | CAS: 72599-27-0

Miglustat, commonly marketed under the trade name Zavesca, is a drug used to treat Gaucher disease. It inhibits the enzyme glucosylceramide synthase, an essential enzyme for the synthesis of most glycosphingolipids. It is only used for patients who cannot be …

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnti-HIV Agents +14
Target Protein:
Ceramide glucosyltransferase
Waktu ParuhThe effective half-…
Vol. Distribusi-
Klirens-
Genetik -
Milademetan DB15257
small molecule | CAS: 1398568-47-2

Milademetan is under investigation in clinical trial NCT02319369 (Safety, Tolerability and Pharmacokinetics of Milademetan Alone and With 5-Azacitidine (AZA) in Acute Myelogenous Leukemia (AML) or High-Risk Myelodysplastic Syndrome (MDS)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Coagulation factor VIII
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milataxel DB12334
small molecule | CAS: 352425-37-7

Milataxel has been used in trials studying the treatment of Mesothelioma.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +2
Target Protein:
Tubulin beta-1 chainTubulin beta chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milatuzumab DB12943
biotech | CAS: 899796-83-9

Milatuzumab has been used in trials studying the treatment of Lupus Nephritis, Multiple Myeloma (MM), GVHD (Acute or Chronic), Myelodysplastic Syndrome, and Chronic Lymphocytic Leukemia, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 129496-10-2

Deskripsi belum tersedia.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 802539-81-7

Milciclib Maleate is under investigation in clinical trial NCT01301391 (Study of Oral PHA-848125AC in Patients With Malignant Thymoma Previously Treated With Multiple Lines of Chemotherapy).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Cyclin-dependent kinase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milk thistle Approved DB14375
biotech | CAS: 65666-07-1

Milk thistle is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
AngiospermsAsteraceaeBiological Products +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Milnacipran Approved DB04896
small molecule | CAS: 92623-85-3

Milnacipran is a selective serotonin and norepinephrine reuptake inhibitor (SNRI) and like many agents in this category was originally developed for and continues to be approved and indicated for the treatment of depression [F3928, F3934, A175786, A175951]. F…

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAgents producing tachycardia +30
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterNMDA receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThe total plasma cl…
Genetik -
Milrinone Approved DB00235
small molecule | CAS: 78415-72-2

Heart failure is a multifactorial condition that affects roughly 1-2% of the adult population. Often the result of long-term myocardial ischemia, cardiomyopathy, or other cardiac insults, heart failure results from an inability of the heart to perfuse periphe…

Kategori:
AminesAminopyridinesCardiac Stimulants Excl. Cardiac Glycosides +12
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu ParuhMilrinone administe…
Vol. DistribusiMilrinone administe…
KlirensMilrinone administe…
Genetik -
Miltefosine Approved DB09031
small molecule | CAS: 58066-85-6

Miltefosine is a broad spectrum antimicrobial, anti-leishmanial, phospholipid drug that was originally developed in the 1980s as an anti-cancer agent. It is currently the only recognized oral agent used to treat visceral, cutaneous, and mucosal forms of leish…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAminesAnti-Infective Agents +9
Target Protein:
Phospholipase A2ATP-dependent translocase ABCB1
Waktu ParuhThe primary elimina…
Vol. DistribusiRadioactivity studi…
KlirensPlasma clearance is…
Genetik -
Milvexian DB16233
small molecule | CAS: 1802425-99-5

Milvexian is under investigation in clinical trial NCT03766581 (A Study on BMS-986177 for the Prevention of a Stroke in Patients Receiving Aspirin and Clopidogrel).

Target Protein:
Coagulation factor XI
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mimopezil DB05520
small molecule | CAS: 180694-97-7

Mimopezil is an acetylcholinesterase (AChE) inhibitor that has demonstrated potential use in the treatment of Alzheimer's disease. Mimopezil is a pro-drug that is rapidly absorbed and converted into huperzine A.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mimosine DB01055
small molecule | CAS: 500-44-7

Mimosine is an antineoplastic alanine-substituted pyridine derivative isolated from _Leucena glauca_.

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +2
Target Protein:
Serine hydroxymethyltransferase, cytosolicC-C motif chemokine 2Tyrosinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minaprine Approved DB00805
small molecule | CAS: 25905-77-5

Minaprine is a psychotropic drug which has proved to be effective in the treatment of various depressive states. Like most antidepressants minaprine antagonizes behavioral despair. Minaprine is an amino-phenylpyridazine antidepressant reported to be relative…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +17
Target Protein:
Amine oxidase [flavin-containing] A5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2A +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mineral oil Approved DB11057
small molecule | CAS: 8042-47-5

Mineral oil, or paraffin oil, is a mixture of higher alkanes from a mineral source, such as petroleum. Petroleum mineral oil is manufactured from crude oils by vacuum distillation to produce several distillates and a residual oil that are then further refined…

Kategori:
Alimentary Tract and MetabolismBasic Ointments and ProtectantsDermatologicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minigastrin DB19196
biotech | CAS: 101212-63-9

Minigastrin is under investigation in clinical trial NCT06155994 (68ga-dota-mgs5 PET/CT in Patients With Advanced Neuroendocrine Tumours).

Kategori:
Amino Acids, Peptides, and ProteinsGastrointestinal HormonesHormones +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Minnelide DB17309
small molecule | CAS: 1254702-87-8

Deskripsi belum tersedia.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +6
Target Protein:
Heat shock 70 kDa protein 1BHeat shock 70 kDa protein 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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