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1977

Total database: 17430
Struktur (SMILES)
1074 (54.3%)
Target
1046 (52.9%)
Genomik
39 (2.0%)
Referensi
1977 (100.0%)

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Hasil Pencarian (1977)

Halaman 18 / 40
Iluzanebart DB18275
biotech | CAS: 2733621-19-5

Deskripsi belum tersedia.

Waktu Paruh-
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Imalumab DB15558
biotech | CAS: 1430205-07-4

Imalumab is under investigation in clinical trial NCT02540356 (Phase 1/2a Two-arm Dose-escalation Study of BAX69 in Subjects With Malignant Ascites of Ovarian Cancer).

Waktu Paruh-
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Genetik -
biotech | CAS: 138660-99-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
Waktu Paruh-
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Imdusiran DB19014
biotech | CAS: 2839476-19-4

Imdusiran is under investigation in clinical trial NCT06245291 (Study of Imdusiran (AB-729) in Combination With Intermittent Dosing of Durvalumab in Subjects With Chronic HBV Infection).

Waktu Paruh-
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Imetelstat Approved DB14909
small molecule | CAS: 868169-64-6

Imetelstat is a first-in-class 18-amino acid oligonucleotide that directly and competitively inhibits human telomerase.[A263973] It is used to treat anemia in patients with myelodysplastic syndromes (MDS), a group of hematologic disorders characterized by ine…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +6
Target Protein:
Telomerase reverse transcriptaseHuman telomerase RNA component
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
Klirens-
Genetik -
IMGN632 DB17337
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Imidafenacin DB09262
small molecule | CAS: 170105-16-5

Imidafenacin is an antispasmodic agent with anticholinergic effects. It antagonizes muscarinic receptors in the bladder to reduce the frequency of urination in the treatment of overactive bladder. It is marketed in Japan under the tradenames Staybla by Ono Ph…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCytochrome P-450 CYP3A Substrates +8
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu ParuhThe half life of el…
Vol. DistribusiThe estimated volum…
KlirensThe estimated clear…
Genetik -
Imlifidase Approved DB15258
biotech | CAS: 1947415-68-0

Chronic kidney disease (CKD) is a progressive and irreversible disease that represents a significant burden for both the individual and healthcare system at large.[A225916] Currently available treatments for end-stage renal disease are limited to dialysis and…

Kategori:
Antineoplastic and Immunomodulating AgentsEndopeptidasesImmunosuppressive Agents +2
Target Protein:
IgG heavy chain
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
IMM-101 DB15850
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma[A220013,A220018,A220023]. Studies with …

Kategori:
Biological ProductsComplex MixturesMelanoma, therapy +1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
IMM101 DB15851
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma [PMID: 21930686; PMID: 30107850; PMID: …

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IMMU-114 DB18458
biotech

IMMU-114 is antibody-drug conjugate consisting of humanized anti-HLA-DR IgG4 monoclonal antibody specific for alpha-chain linked to SN-38 via a CL2A linker.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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Imsidolimab DB16658
biotech | CAS: 2102543-86-0

Imsidolimab is under investigation in clinical trial NCT03633396 (A Study to Evaluate the Efficacy and Safety of ANB019 in Subjects With Palmoplantar Pustulosis).

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Genetik -
biotech

The SARS-CoV-2 Inactivated Vaccine is a purified vaccine that contains multiple antigens from the virus and is inactivated in Vero Cells[A219758]. This vaccine specifically was developed in collaboration with the Chinese Academy of Medical Sciences, West Chin…

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INCB-057643 DB16054
small molecule | CAS: 1820889-23-3

INCB-057643 is under investigation in clinical trial NCT02959437 (Azacitidine Combined With Pembrolizumab and Epacadostat in Subjects With Advanced Solid Tumors (ECHO-206)).

Kategori:
AcidsAcids, NoncarboxylicAntineoplastic Agents +1
Waktu Paruh-
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Inclisiran Approved DB14901
biotech | CAS: 1639324-58-5

Inclisiran is a long-acting, synthetic small interfering RNA (siRNA) directed against proprotein convertase subtilisin-kexin type 9 (PCSK9), which is a serine protease that regulates plasma low-density lipoprotein cholesterol (LDL-C) levels. By binding to PCS…

Kategori:
Antisense Elements (Genetics)Compounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +16
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThere is limited in…
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAlcoholsCarbohydrates +7
Waktu Paruh-
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Indacaterol Approved DB05039
small molecule | CAS: 312753-06-3

Indacaterol is a novel, ultra-long-acting, rapid onset ?(2)-adrenoceptor agonist developed for Novartis for the once-daily management of asthma and chronic obstructive pulmonary disease. It was approved by the European Medicines Agency (EMA) on 30 November 20…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +17
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIndacaterol serum c…
Vol. DistribusiAfter intravenous i…
KlirensRenal clearance of …
Genetik -
biotech | CAS: 138955-27-8

Tumor associated glycoprotein (TAG) 72 (B72.3) monoclonal antibody conjugated with Indium 111 for radioimaging colon tumors. Satumomab Pendetide (trade name: OncoScint®) is no longer commercially available.

Kategori:
AcetatesAcids, AcyclicAmines +14
Target Protein:
Tumor-associated glycoprotein 72 (TAG-72)
Waktu Paruh0.8 hours (mammalia…
Vol. Distribusi-
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Genetik -
Indocyanine green acid form Approved DB09374
small molecule | CAS: 28782-33-4

Indocyanine Green is a water soluble, tricarbocyanine dye with a peak spectral absorption at 800 nm. The chemical name for Indocyanine Green is 1 H-Benz[e]indolium, 2-[7-[1,3-dihydro-1,1-dimethyl-3-(4-sulfobutyl)-2H-benz[e] indol-2-ylidene]-1,3,5-heptatrienyl…

Kategori:
BSEP/ABCB11 SubstratesCardiac FunctionColoring Agents +6
Waktu ParuhICG has a half-life…
Vol. DistribusiICG distribution in…
KlirensClearance of dyes w…
Genetik -
Indomethacin Approved DB00328
small molecule | CAS: 53-86-1

Indometacin, or indomethacin, is a non-steroidal anti-inflammatory drug (NSAID) with anti-inflammatory, analgesic, and antipyretic properties. NSAIDs consist of agents that are structurally unrelated; the NSAID chemical classification of indometacin is an ind…

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +49
Target Protein:
Prostaglandin G/H synthase 2Phospholipase A2, membrane associatedHuman Cyclooxygenases +8
Waktu ParuhIndometacin disposi…
Vol. DistribusiThe volume of distr…
KlirensIn a clinical pharm…
Genetik -
Indopan DB01446
small molecule | CAS: 299-26-3

Indopan (alpha-methyltryptamine) is a stimulant and psychoactive drug which produces effects similar to 3,4-methylenedioxy-N-methylamphetamine (MDMA), despite being structurally dissimilar. It was developed in the 1960's by Upjohn with the intention for use a…

Kategori:
AminesBiogenic AminesBiogenic Monoamines +3
Waktu Paruh-
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Inebilizumab Approved DB12530
biotech | CAS: 1299440-37-1

Inappropriate growth of or self-directed antibody production by B-cells is the etiological underpinning of a variety of conditions, including the multiple sclerosis-like neurological condition neuromyelitis optica spectrum disorder (NMOSD).[A214283, A214286] …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhInebilizumab exhibi…
Vol. DistribusiInebilizumab has an…
KlirensInebilizumab has an…
Genetik -
Infliximab Approved DB00065
biotech | CAS: 170277-31-3

Infliximab is a tumor necrosis factor (TNF-alpha or TNF-?) blocker and a chimeric monoclonal IgG1 antibody composed of human constant (75%) and murine variable (25%) regions [A31469]. Infliximab is produced by a recombinant cell line cultured by continuous pe…

Kategori:
Agents Causing Muscle ToxicityAgents reducing cytokine levelsAmino Acids, Peptides, and Proteins +21
Target Protein:
Tumor necrosis factor
Gen Terkait:
FCGR3A
Waktu ParuhThe median terminal…
Vol. DistribusiBased on a pharmaco…
KlirensIn patients with Cr…
Genetik 1 Varian
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

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Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

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Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

A seasonally-specific component of the influenza vaccine. The influenza vaccine, also known as the "flu shot", is a vaccine that protects against infection from the influenza viruses. Vaccines provide protection from influenza by exposing the immune system to…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1383547-60-1

Ingenol disoxate is under investigation in clinical trial NCT02120456 (Safety and Efficacy of Escalating Doses of LEO 43204 Applied Once Daily for Two Consecutive Days on Approximately 250 cm2 on Trunk and Extremities in Subjects With Actinic Keratosis).

Kategori:
Terpenes
Waktu Paruh-
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Ingenol mebutate Approved DB05013
small molecule | CAS: 75567-37-2

Ingenol mebutate was approved by the FDA in January 2012, and it is marketed under the name Picato®. Picato gel is indicated for the topical treatment of actinic keratosis. Before approval, ingenol mebutate was called PEP005 as an investigational drug. PEP005…

Kategori:
Cell Death InducerDermatologicalsIncreased Cellular Death +2
Target Protein:
Protein kinase C delta typeProtein kinase C alpha type
Waktu ParuhThere is no half-li…
Vol. DistribusiThere is no volume …
KlirensThere is no clearan…
Genetik -
INO-4800 DB15693
biotech

INO-4800 is a DNA vaccine containing the full sequence for the SARS-CoV-2 Spike (S) protein in development for immunization against COVID-19.[A214475] Early _in vitro_ studies using HEK-293T cells demonstrated that the transfection of INO-4800 results in the …

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
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Inotuzumab ozogamicin Approved DB05889
biotech | CAS: 635715-01-4

Inotuzumab ozogamicin is an antibody-drug conjugate consisting of a humanized IgG4 kappa CD22-targeting monoclonal antibody covalently attached to calicheamicin derivative, N-acetyl-gamma-calicheamicin dimethylhydrazide.[A20352] The antibody portion of the dr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntibodies +33
Target Protein:
B-cell receptor CD22
Waktu ParuhIn patients with re…
Vol. DistribusiIn humans, the tota…
KlirensThe pharmacokinetic…
Genetik -
Insulin degludec Approved DB09564
biotech | CAS: 844439-96-9

Insulin degludec is an ultra-long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes.[A18561,A18562,A18563,A18564,A174934] Insulin is typically prescribed for the management of diabetes mellitus to mimic the ac…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +13
Target Protein:
InsulinInsulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhThe half-life after…
Vol. DistribusiUsing a one-compart…
KlirensThe mean apparent c…
Genetik -
Insulin detemir Approved DB01307
biotech | CAS: 169148-63-4

Insulin detemir is a long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes.[A2358, A2359, A2360, A44] Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenou…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +13
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhAfter subcutaneous …
Vol. DistribusiInsulin detemir has…
KlirensThe apparent cleara…
Genetik -
Insulin glargine Approved DB00047
biotech | CAS: 160337-95-1

Insulin glargine is a long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insuli…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAntimetabolites +18
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
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Genetik -
Insulin icodec Approved DB16693
biotech | CAS: 1188379-43-2

Insulin icodec is an ultra long-acting basal insulin analogue. It is a re-engineered version of the ultra long-acting oral basal insulin OI338, with several modifications introduced to significantly extend the half-life.[A264093] These modifications - which c…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +10
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhThe mean half-life …
Vol. DistribusiAccording to popula…
KlirensAccording to popula…
Genetik -
Insulin lispro Approved DB00046
biotech | CAS: 133107-64-9

Insulin lispro is a rapid-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insulin, a peptid…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +14
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhAfter subcutaneous …
Vol. DistribusiWhen administered i…
KlirensWhen administered i…
Genetik -
biotech | CAS: 67763-97-7

The insulin-like growth factor II is a well-characterized neutral peptide believed to be secreted by the liver and to circulate in the blood. This factor presents effects related to growth regulation, insulin-like and mitogenic activities. To perform its biol…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Interferon alfa DB05258
biotech

Natural interferon alpha or Multiferon is obtained from the leukocyte fraction of human blood following induction with Sendai virus. Interferon alfa contains several naturally occurring IFN-? subtypes and is purified by affinity chromatography. Interferon alp…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntiviral Agents +14
Target Protein:
Interferon alpha/beta receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 142192-09-4

Interferon alfa-2c is under investigation in clinical trial NCT00485563 (A Phase II Study of EC17 (Folate-hapten Conjugate) in Patients With Progressive Metastatic Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytochrome P-450 CYP1A2 Inhibitors +8
Waktu Paruh-
Vol. Distribusi-
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Iodine Approved DB05382
small molecule | CAS: 7553-56-2

Iodine is commonly used as an antiseptic for minor cuts and abrasions, preventing infections that may result from contaminated wounds. Additionally, iodine has been studied in the treatment of fibrocystic disease and breast cancer.[A3413,A192153,A192156,A1921…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiseptics and Disinfectants +12
Target Protein:
Sodium/iodide cotransporterMicrobial proteins
Waktu Paruh-
Vol. Distribusi-
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Iodine I-125 DB14804
small molecule | CAS: 14158-31-7

Iodine I-125 is under investigation in clinical trial NCT00079417 (Neoadjuvant Carboplatin and Vincristine and Standard Local Ophthalmic Therapy in Treating Patients With Intraocular Retinoblastoma).

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Iodoform Approved DB13813
small molecule | CAS: 75-47-8

Iodoform is an organoiodine compound with the formula CHI3 and a tetrahedral molecular geometry. It is a relatively water-insoluble yellow solid that is chemically reactive in free-radical reactions [A32890]. Due to its antimicrobial properties following topi…

Kategori:
DermatologicalsHydrocarbons, HalogenatedMedicated Dressings +2
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
small molecule | CAS: 147-58-0

Iodohippuric acid is under investigation in clinical trial NCT02599844 (Impact of Pediatric Acute Renal Injury in Severe Sepsis in Young Adults).

Kategori:
Acids, CarbocyclicAmidesBenzamides and benzamide derivatives +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 949575-24-0

Iofolastat I-123 is under investigation in clinical trial NCT00992745 (A Phase I Pilot Study Comparing 123I MIP 1072 Versus 111In Capromab Pendetide in Subjects With Metastatic Prostate Cancer).

Kategori:
AmidesAmino AcidsAmino Acids, Acidic +2
Target Protein:
Glutamate carboxypeptidase 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ioforminol DB12439
small molecule | CAS: 1095110-48-7

Ioforminol has been used in trials studying the diagnostic of Cardio Renal Safety in High-risk Elderly Subjects Undergoing a Coronary CATH With or Without PCI.

Kategori:
Acids, AcyclicAcids, CarbocyclicAmides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 873438-88-1

Iopofosine I-131 (NM-404 I-131) is under investigation in clinical trial NCT01495663 (Dose Escalation Study of I-131-CLR1404 in Subjects With Cancer That Does Not Respond to Treatment or Has Returned).

Kategori:
AlcoholsBenzene DerivativesEthers +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ioxilan Approved DB09135
small molecule | CAS: 107793-72-6

Ioxilan is a tri-iodinated diagnostic contrast agent. Intravascular injection results in opacification of vessels in the path of flow of the contrast medium, permitting radiographic visualization of the internal structures of the human body until significant …

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +11
Waktu ParuhAn initial fast dis…
Vol. DistribusiIoxilan is distribu…
KlirensThe total clearance…
Genetik -
Ipafricept DB15045
biotech | CAS: 1391727-24-4

Ipafricept is under investigation in clinical trial NCT01608867 (A Dose Escalation Study of OMP-54F28 in Subjects With Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iproniazid DB04818
small molecule | CAS: 54-92-2

Withdrawn from the Canadian market in July 1964 due to interactions with food products containing tyrosine.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +18
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Irinotecan Approved DB00762
small molecule | CAS: 97682-44-5

Irinotecan is a topoisomerase inhibitor used for chemotherapy. It is a water-soluble analogue of [camptothecin], which is extracted from the Chinese tree _Camptotheca acuminate_.[A263376] The bis-piperidine side chain in the structure of irinotecan bestows en…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +29
Target Protein:
DNA topoisomerase I, mitochondrialDNA topoisomerase 1
Gen Terkait:
SLCO1B1 UGT1A1 UGT1A7 +2
Waktu ParuhAfter intravenous i…
Vol. DistribusiFollowing intraveno…
KlirensThe mean (± standar…
Genetik 5 Varian
Menampilkan 851–900 dari 1977
Sebelumnya Halaman 18 / 40 Berikutnya