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6694

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3751 (56.0%)
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Halaman 18 / 134
Afamitresgene autoleucel Approved DB18592
biotech

Afamitresgene autoleucel is a melanoma-associated antigen A4 (MAGE-A4)-directed genetically modified autologous T cell immunotherapy product consisting of CD4 and CD8 positive T cells transduced with a self-inactivating lentiviral vector (LV) expressing an af…

Kategori:
Autologous Cellular Immunotherapy
Waktu Paruh-
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Afasevikumab DB14798
biotech | CAS: 1589503-30-9

Afasevikumab is under investigation in clinical trial NCT01480310 (Study to Investigate the Safety, Pharmacokinetics, and Immunogenicity of Subcutaneous MCAF5352A in Healthy Volunteers).

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Affitope AD01 DB06086
biotech

Affitope AD01 is an investigational drug developed for immunization to treat Alzheimer's Disease. AD01 is a short peptide (7 amino acids in length) that induces Aß-targeting antibodies, therefore lowering Aß aggregates.

Target Protein:
Amyloid-beta precursor protein
Waktu Paruh-
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Afimetoran DB16580
small molecule | CAS: 2171019-55-7

Afimetoran is an immunomodulator and an antagonist of toll-like receptors 7 and 8.[L32018, L32023] It is also is under investigation in clinical trial NCT04269356 (Study to Assess the Way the Body Absorbs, Distributes, Breaks Down and Eliminates Radioactive B…

Target Protein:
Toll-like receptor 7Toll-like receptor 8
Waktu Paruh-
Vol. Distribusi-
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Aflibercept Approved DB08885
biotech | CAS: 862111-32-8

Aflibercept is a recombinant protein composed of the binding domains of two human vascular endothelial growth factor (VEGF) receptors, VEGFR1 and VEGFR2, fused with the Fc region of human immunoglobulin gamma 1 (IgG1).[A261130] Structurally, Aflibercept is a …

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +16
Target Protein:
Vascular endothelial growth factor A, long formPlacenta growth factorVascular endothelial growth factor B
Waktu ParuhFor the intravitrea…
Vol. DistribusiThe volume of distr…
KlirensFollowing an hour o…
Genetik -
AG-858 DB05502
biotech

AG-858 (autologous heat-shock protein 70 peptide vaccine) is a recombinant cancer vaccine made with tumor-derived heat shock protein 70 (HSP70) peptide complexes. HSP70 associates with antigenic peptides, transporting them into antigen presenting cells (APC)…

Waktu Paruh-
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AG0301-COVID19 DB15856
biotech

AG0301-COVID19 is a vaccine candidate developed by AnGes Inc. and Osaka University. The candidate is a plasmid DNA vaccine developed using an intradermal gene transfer method targeting the SARS-CoV-2 spike protein. The gene transfer method increases the effic…

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AG0302-COVID19 DB16435
biotech

Sponsored by Anges, Inc. in Japan, the AG0302-COVID19 is a DNA-based vaccine that recently completed Phase I/II trials (NCT04527081)[A226813, L30548].

Waktu Paruh-
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AGA2115 DB17840
biotech

AGA2115 is a humanized bispecific antibody neutralizing both sclerostin and Dickkopf-1. Developed by Angitia Biopharmaceuticals, AGA2115 is being investigated for the treatment of osteogenesis imperfect.[L46646]

Waktu Paruh-
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Agatolimod DB15018
biotech | CAS: 207623-20-9

Agatolimod is under investigation in clinical trial NCT00471471 (Vaccine Therapy in Treating Patients With Recurrent Stage III or Stage IV Melanoma That Cannot Be Removed by Surgery).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
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AGF-94 DB18023
small molecule | CAS: 136784-51-5

Deskripsi belum tersedia.

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AGIL-FA DB16973
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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biotech

Agkistrodon piscivorus antivenin is derived and purified immunoglobulin fragments obtained from other domestic animals such as sheep previously immunized with Agkistrodon piscivorus (_Cottonmouth_ or _Water Moccasin snake_). The final purified antivenin produ…

Kategori:
AntiveninsPassively Acquired ImmunityVenom Neutralization
Target Protein:
Group 10 secretory phospholipase A2
Waktu Paruh12 to 23 hours [FDA…
Vol. Distribusi-
KlirensSystemic clearance …
Genetik -
Agmatine DB08838
small molecule | CAS: 306-60-5

Agmantine is a natural metabolite of the amino acid arginine. It is formed when arginine is decarboxylated by the enzyme arginine decarboxylase and is found naturally in ragweed pollen, ergot fungi, octopus muscle, herring sperm, sponges, and the mammalian br…

Kategori:
Agents causing hyperkalemiaAmidinesAntiarrhythmic agents +12
Target Protein:
Alpha-2C adrenergic receptorNischarinAcetylcholine receptor subunit alpha +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Agomelatine Approved DB06594
small molecule | CAS: 138112-76-2

Agomelatine is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-HT2C) receptors, tested in an animal model of depression. Agomelatine was developed in Europe by Servier Labo…

Kategori:
AcetatesAcids, AcyclicAmides +15
Target Protein:
5-hydroxytryptamine receptor 2CMelatonin receptor type 1AMelatonin receptor type 1B
Waktu Paruh<2 hours
Vol. Distribusi-
Klirens-
Genetik -
AGRO100 DB04998
biotech | CAS: 301636-59-9

AGRO100 is an oligonucleotide that functions as an aptamer and binds to nucleolin, a protein found intranuclear in all cells, but uniquely expressed on the surface of tumor cells. Such binding leads to internalization of the complex, and a strong anti-prolife…

Kategori:
Aptamers, NucleotideNucleic Acids, Nucleotides, and NucleosidesNucleotides +2
Target Protein:
NF-kappa-B essential modulator
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Agrostis gigantea top Approved DB14757
biotech

Agrostis gigantea top is the flowering part of the Agrostis gigantea plant. Agrostis gigantea top is mainly used in allergenic testing.

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AGS-16C3F DB17551
biotech

AGS 16C3F is an intravenously administered, anti-ectonucleotide pyrophosphatase/phosphodiesterase 3 (ENPP3) antibody-drug conjugate. AGS-16C3F is under investigation in clinical trial NCT02639182 (A Study of AGS-16C3F vs. Axitinib in Metastatic Renal Cell Car…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
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AGTC-401 DB18432
biotech

AGTC-401 is a recombinant adeno-associated virus vector expressing the cyclic nucleotide gated channel beta subunit (rAAV-CNGB3).

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AGTC-402 DB18433
biotech

AGTC-402 is a recombinant adeno-associated virus vector expressing the cyclic nucleotide gated channel alpha subunit (CNGA3).

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Genetik -
biotech | CAS: 2417550-70-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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AIT-034 DB06106
small molecule | CAS: 138117-48-3

AIT-034 is a distinct chemical analog of hypoxanthine and pyrollidone that has been demonstrated in animal studies to enhance memory and to reverse memory deficits in severely impaired animals that do not respond to Neotrofin. AIT-034 does not induce the prod…

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Aklavine DB19070
small molecule | CAS: 66676-88-8

Aklavine is under investigation in clinical trial NCT03026842 (Decitabine Versus Conventional Chemotherapy for Maintenance Therapy of Acute Myeloid Leukemia With T(8;21)).

Kategori:
Adjuvants, ImmunologicAminoglycoside AntibacterialsAnthracyclines +7
Waktu Paruh-
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Genetik -
biotech

Ala-geninthiocin is a novel thiopeptide antibacterial compound derived from marine _Streptomyces_ species.[A192840] It has exhibited potent _in vitro_ activity against gram-positive bacteria including _Staphylococcus aureus_, _Bacillus subtilis_, _Mycobacteri…

Kategori:
Anti-Bacterial Agents
Waktu Paruh-
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Alamifovir DB06368
small molecule | CAS: 193681-12-8

Alamifovir is an antiviral agent specific for HBV.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Alanine DB00160
small molecule | CAS: 56-41-7

Alanine is a non-essential amino acid that occurs in high levels in its free state in plasma. It is produced from pyruvate by transamination. It is involved in sugar and acid metabolism, increases immunity, and provides energy for muscle tissue, brain, and th…

Kategori:
AlanineAmino AcidsAmino Acids, Peptides, and Proteins +3
Target Protein:
4-aminobutyrate aminotransferase, mitochondrialAlanine--glyoxylate aminotransferaseAlanine aminotransferase 1 +10
Waktu Paruh-
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Alanosine DB05540
small molecule | CAS: 5854-93-3

An amino acid analogue and antibiotic derived from the bacterium Streptomyces alanosinicus with antimetabolite and potential antineoplastic activities.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntibiotics, Antineoplastic +4
Target Protein:
Aspartate carbamoyltransferase catalytic subunitAdenylosuccinate synthetase isozyme 2Adenylosuccinate synthetase isozyme 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 39537-23-0

Alanyl Glutamine is under investigation in clinical trial NCT00338221 (Clinical Trial of Alanyl-Glutamine or Glycine in Children With Persistent Diarrhea or Malnutrition).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +4
Waktu Paruh-
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Alaproclate DB13233
small molecule | CAS: 60719-82-6

Alaproclate was developed as one of the first selective serotonin reuptake inhibitor (SSRI) antidepressants by Astra AB (now AstraZeneca) in the 1970s. Development was discontinued due to concerns over hepatotoxicity observed in animal studies. Alaproclate ha…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntidepressive Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Alatrofloxacin Approved DB09335
small molecule | CAS: 146961-76-4

Alatrofloxacin is a fluoroquinolone antibiotic developed by Pfizer, delivered as a mesylate salt. It was withdrawn from the U.S. market in 2001.

Kategori:
4-QuinolonesAnti-Infective AgentsEnzyme Inhibitors +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Albaconazole DB12073
small molecule | CAS: 187949-02-6

Albaconazole has been used in trials studying the basic science of Onychomycosis.

Kategori:
Anti-Infective AgentsAntifungal AgentsAzole Antifungals +3
Waktu Paruh-
Vol. Distribusi-
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Albendazole Approved DB00518
small molecule | CAS: 54965-21-8

A benzimidazole broad-spectrum anthelmintic structurally related to mebendazole that is effective against many diseases. (From Martindale, The Extra Pharmacopoeia, 30th ed, p38)

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +23
Target Protein:
Tubulin beta-2 chainTubulin alpha-1A chainTubulin beta-4B chain +1
Waktu ParuhTerminal eliminatio…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 472960-22-8

Albumin-interferon alpha (Albuferon) is a novel, long-acting form of interferon alpha. Recombinant interferon alpha is approved for the treatment of hepatitis C, hepatitis B, and a broad range of cancers. Human Genome Sciences modified interferon alpha to imp…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +10
Waktu Paruh-
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Albumin human Approved DB00062
biotech | CAS: 9048-46-8

Human serum albumin is the primary protein present in human blood plasma. The main function of albumin is to maintain the oncotic pressure of blood [A33706]. It binds to water, cations (such as Ca2+, Na+ and K+), fatty acids, hormones, bilirubin, thyroxine (T…

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood and Blood Forming Organs +13
Target Protein:
Nitric oxide
Waktu Paruh-
Vol. DistribusiAlbumin is distribu…
Klirens-
Genetik -
Albusomatropin DB12950
biotech | CAS: 1613273-96-3

Albusomatropin has been used in trials studying the treatment of Growth Hormone-Deficiency and Growth Hormone Deficiency.

Kategori:
AlbuminsAmino Acids, Peptides, and ProteinsBlood Proteins +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Albuterol Approved DB01001
small molecule | CAS: 18559-94-9

Salbutamol (Albuterol [USAN]) is a short-acting, selective beta2-adrenergic receptor agonist used in the treatment of asthma and COPD. It is 29 times more selective for beta2 receptors than beta1 receptors giving it higher specificity for pulmonary beta recep…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +27
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik -
Alcaftadine Approved DB06766
small molecule | CAS: 147084-10-4

Alcaftadine is a H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis. This drug was approved in July 2010.

Kategori:
Decongestants and AntiallergicsDrugs that are Mainly Renally ExcretedHeterocyclic Compounds, Fused-Ring +8
Target Protein:
Histamine H1 receptor
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Alclofenac Approved DB13167
small molecule | CAS: 22131-79-9

Alclofenac is a non-steroidal anti-inflammatory drug. It was withdrawn from the market in the United Kingdom in 1979.

Kategori:
Acetic Acid Derivatives and Related SubstancesAcids, CarbocyclicAgents causing hyperkalemia +14
Target Protein:
Prostaglandin G/H synthase 2
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe volume of distr…
KlirensFor oral dose of 50…
Genetik -
Aldesleukin Approved DB00041
biotech | CAS: 110942-02-4

Aldesleukin, a lymphokine, is produced by recombinant DNA technology using a genetically engineered E. coli strain containing an analog of the human interleukin-2 gene. Genetic engineering techniques were used to modify the human IL-2 gene, and the resulting …

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAnti-HIV Agents +26
Target Protein:
Interleukin-2 receptor subunit betaInterleukin-2 receptor subunit alphaCytokine receptor common subunit gamma
Waktu Paruh13 min-85 min
Vol. Distribusi0.18 l/kg
Klirens-
Genetik -
Aldoxorubicin DB06013
small molecule | CAS: 1361644-26-9

Aldoxorubicin, an antineoplastic agents, is an albumin-binding prodrug of doxorubicin.

Kategori:
AnthracyclinesAntineoplastic AgentsCarbohydrates +4
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alectinib Approved DB11363
small molecule | CAS: 1256580-46-7

Alectinib is a second generation oral drug that selectively inhibits the activity of anaplastic lymphoma kinase (ALK) tyrosine kinase. It is specifically used in the treatment of non-small cell lung cancer (NSCLC) expressing the ALK-EML4 (echinoderm microtubu…

Kategori:
Anaplastic lymphoma kinase (ALK) inhibitorsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
ALK tyrosine kinase receptor
Waktu ParuhThe mean eliminatio…
Vol. Distribusi4016 L
KlirensThe apparent cleara…
Genetik -
Aleglitazar DB08915
small molecule | CAS: 475479-34-6

Aleglitazar is an investigational drug from the company Hoffmann–La Roche and is currently in a phase III clinical trial called ALECARDIO. It is being investigated for use in patients with type II diabetes to reduce their risks of cardiovascular mortality and…

Kategori:
Sulfur Compounds
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gammaNuclear receptor coactivator 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alemtuzumab Approved DB00087
biotech | CAS: 216503-57-0

Alemtuzumab is a humanized monoclonal antibody specific to lymphocyte antigens. It is a recombinant DNA-derived humanized monoclonal antibody (Campath-1H) that is directed against the 21-28 kD cell surface glycoprotein, CD52. The Campath-1H antibody is an IgG…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
CAMPATH-1 antigenLow affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +4
Waktu ParuhThe elimination hal…
Vol. DistribusiAlemtuzumab is larg…
KlirensClearance of alemtu…
Genetik -
Alendronic acid Approved DB00630
small molecule | CAS: 66376-36-1

Alendronic acid is a second generation bisphosphonate that is used for the treatment of some forms of osteoperosis and Paget's disease[FDA Label][A959,A203111]. It functions by preventing resorption of bone[FDA Label][A959].

Kategori:
Agents Causing Muscle ToxicityBisphosphonatesBone Density Conservation Agents +5
Target Protein:
Farnesyl pyrophosphate synthaseHydroxylapatiteTyrosine-protein phosphatase non-receptor type 4 +3
Waktu ParuhDue to alendronic a…
Vol. Distribusi28L[FDA Label].
Klirens71mL/min[FDA Label].
Genetik -
Alfacalcidol Approved DB01436
small molecule | CAS: 41294-56-8

Alfacalcidol, or 1-alpha-hydroxycholecalciferol or 1-alpha-hydroxyvitamin D3, is a non-endogenous analogue of [vitamin D].[A234044] It plays an essential function in calcium homeostasis and bone metabolism. Alfacaldisol is activated by the enzyme 25-hydroxyla…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCholestanes +13
Target Protein:
Vitamin D3 receptor25-hydroxyvitamin D-1 alpha hydroxylase, mitochondrialRetinoic acid receptor RXR-alpha
Waktu ParuhThe half-life of al…
Vol. Distribusi-
Klirens-
Genetik -
Alfentanil Approved DB00802
small molecule | CAS: 71195-58-9

A short-acting opioid anesthetic and analgesic derivative of fentanyl. It produces an early peak analgesic effect and fast recovery of consciousness. Alfentanil is effective as an anesthetic during surgery, for supplementation of analgesia during surgical pro…

Kategori:
Agents that produce hypertensionAnalgesicsAnesthetics +25
Target Protein:
Mu-type opioid receptor
Waktu Paruh90-111 minutes
Vol. Distribusi* 0.4 to 1 L/kg
Klirens* 5 mL/kg/min
Genetik -
biotech | CAS: 473553-86-5

Alferminogene tadenovec, Cardium’s lead product candidate, is being developed for the potential treatment of myocardial ischemia that gives rise to angina symptoms associated with coronary heart disease. Alferminogene tadenovec represents a new therapeutic cl…

Kategori:
Antianginal AgentsVasodilating Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Algenpantucel-L DB17184
biotech

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesVaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Alginic acid Approved DB13518
small molecule | CAS: 9005-32-7

Alginic acid, also referred to as algin or alginate, is a hydrophilic or anionic polysaccharide isolated from certain brown seaweed (_Phacophycae_) via alkaline extraction. It is present in cell walls of brown algae where it forms a viscous gel when binding w…

Kategori:
Acids, AcyclicAcids, AldehydicAlginates +11
Waktu ParuhThis pharmacokineti…
Vol. DistribusiThis pharmacokineti…
KlirensThis pharmacokineti…
Genetik -
Alglucerase Approved DB00088
biotech | CAS: 143003-46-7

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 49.4 to 282.1 mL/…
Klirens-
Genetik -
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