Hasil Filter

14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (14063)

Halaman 179 / 282
Methyldopa Approved DB00968
small molecule | CAS: 555-30-6

Methyldopa, or ?-methyldopa, is a centrally acting sympatholytic agent and an antihypertensive agent.[A231784] It is an analog of DOPA (3,4?hydroxyphenylanine), and it is a prodrug, meaning that the drug requires biotransformation to an active metabolite for …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +28
Target Protein:
D(2) dopamine receptorAromatic-L-amino-acid decarboxylaseAlpha-2A adrenergic receptor
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensThe renal clearance…
Genetik -
Methylene blue Approved DB09241
small molecule | CAS: 61-73-4

Methylene blue is an oxidation-reduction agent. The intravenous form of methylene blue is approved by the FDA for the treatment of pediatric and adult patients with acquired methemoglobinemia. Historically, it has been widely used in Africa to treat malaria, …

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +51
Target Protein:
Guanylate cyclase soluble subunit alpha-2Nitric oxide synthase 1
Waktu Paruh5–6.5 hours (after …
Vol. Distribusi10 mg/kg (in rats).
Klirens3.0 ± 0.7 L/min.
Genetik -
small molecule | CAS: 82801-81-8

Deskripsi belum tersedia.

Kategori:
Adrenergic AgentsAminesAmphetamines +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylergometrine Approved DB00353
small molecule | CAS: 113-42-8

A homolog of ergonovine containing one more CH2 group. (Merck Index, 11th ed)

Kategori:
Agents that produce hypertensionAlkaloidsCytochrome P-450 CYP3A Inhibitors +14
Target Protein:
D(1A) dopamine receptor5-hydroxytryptamine receptor 2B
Waktu Paruh3.39 hours
Vol. Distribusi* 56.1 ± 0 L
Klirens-
Genetik -
small molecule | CAS: 624-78-2

Deskripsi belum tersedia.

Target Protein:
Myoglobin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 105-41-9

Deskripsi belum tersedia.

Kategori:
5-alpha Reductase InhibitorsAndrostanesAndrostanols +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylinositol DB12969
small molecule | CAS: 10284-63-6

Methylinositol has been used in trials studying the treatment of Dementia and Alzheimer's Disease.

Kategori:
AlcoholsCarbohydratesSugar Alcohols
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2682-20-4

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsCompounds used in a research, industrial, or household settingDisinfectants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylliberine DB17930
small molecule | CAS: 51168-26-4

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 516-05-2

A malonic acid derivative which is a vital intermediate in the metabolism of fat and protein. Abnormalities in methylmalonic acid metabolism lead to methylmalonic aciduria. This metabolic disease is attributed to a block in the enzymatic conversion of methylm…

Kategori:
Acids, AcyclicDicarboxylic AcidsMalonates
Target Protein:
Methylmalonyl-CoA carboxyltransferase 12S subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1115-84-0

Methylmethionine chloride may be useful in helping the healing of gastric ulcers. In Japan, it is used as an over the counter product for gastrointestinal health support. It is also called "Vitamin U", but it is not a true vitamin.

Kategori:
Alimentary Tract and MetabolismDrugs for Acid Related DisordersDrugs for Peptic Ulcer and Gastro-Oesophageal Reflux Disease (Gord)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylnaltrexone Approved DB06800
small molecule | CAS: 916055-93-1

Methylnaltrexone is a pheriphally-acting ?-opioid antagonist that acts on the gastrointestinal tract to decrease opioid-induced constipation without producing analgesic effects or withdrawal symptoms. It is also a weak CYP2D6 inhibitor. FDA approved in 2008.

Kategori:
Alimentary Tract and MetabolismAlkaloidsAmines +16
Target Protein:
Mu-type opioid receptorMelanocortin receptor 4Kappa-type opioid receptor
Waktu Paruhterminal: 8.89 ± 2.…
Vol. DistribusiVolume of distribut…
Klirens10.5 ± 1.5 ml/min/k…
Genetik -
Methylone DB19192
small molecule | CAS: 186028-79-5

Methylone is under investigation in clinical trial NCT05741710 (A Study to Assess the use of Methylone in the Treatment of PTSD).

Kategori:
AminesAmphetaminesCentral Nervous System Stimulants +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylparaben Approved DB14212
small molecule | CAS: 99-76-3

Methylparaben is used in allergenic testing.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +10
Target Protein:
Transient receptor potential cation channel subfamily A member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylphenidate Approved DB00422
small molecule | CAS: 113-45-1

Methylphenidate is a central nervous system stimulant used most commonly in the treatment of Attention-Deficit/Hyperactivity Disorder (ADHD) and for narcolepsy. Also known as the marketed products Ritalin, Concerta, or Biphentin, methylphenidate is used with …

Kategori:
Acids, CarbocyclicAgents that produce hypertensionAgents that reduce seizure threshold +17
Target Protein:
Sodium-dependent dopamine transporter5-hydroxytryptamine receptor 1ASodium-dependent noradrenaline transporter
Waktu ParuhConcerta: The half-…
Vol. DistribusiConcerta: Plasma me…
KlirensThe apparent mean s…
Genetik -
Methylphenobarbital Approved DB00849
small molecule | CAS: 115-38-8

A barbiturate that is metabolized to phenobarbital. It has been used for similar purposes, especially in epilepsy, but there is no evidence mephobarbital offers any advantage over phenobarbital.

Kategori:
Anticholinergic AgentsAnticonvulsantsBarbiturates +20
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-2Gamma-aminobutyric acid receptor subunit alpha-3Gamma-aminobutyric acid receptor subunit alpha-4 +8
Waktu Paruh34 (range 11-67) ho…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 4206-94-4

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicCholinesterase Inhibitors +3
Target Protein:
AcetylcholinesteraseCholinesteraseEsterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylprednisolone Approved DB00959
small molecule | CAS: 83-43-2

Methylprednisolone is a [prednisolone] derivative glucocorticoid with higher potency than [prednisone].[A188811] It was first described in the literature in the late 1950s.[A188811,A188814] Methylprednisolone was granted FDA approval on 24 October 1957.[L1…

Kategori:
Adrenal Cortex HormonesAdrenalsAnti-Acne Preparations +50
Target Protein:
Glucocorticoid receptorAnnexin A1
Waktu ParuhMethylprednisolone …
Vol. DistribusiThe average volume …
KlirensThe average plasma …
Genetik -
small molecule | CAS: 2921-57-5

A water-soluble ester of methylprednisolone used for cardiac, allergic, and hypoxic emergencies.

Kategori:
Adrenal Cortex HormonesAdrenalsAnti-Inflammatory Agents +21
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methylprednisone Approved DB12952
small molecule | CAS: 91523-05-6

Methylprednisone has been used in trials studying the treatment of Leukemia, Rheumatoid Arthritis, Renal Transplantation, Kidney Transplantation, and Acute Lymphocytic Leukemia, among others.

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 CYP3A4 Substrates (strength unknown) +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10605-24-0

Deskripsi belum tersedia.

Kategori:
Antianginal AgentsCardiac TherapyOrganic Nitrates +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1119361-12-4

Methylsamidorphan is under investigation in clinical trial NCT01418092 (ALK37-007: Evaluation of Safety and Efficacy of ALKS 37 (RDC-1036) in Adults With Opioid-induced Constipation (OIC)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 26046-90-2

Methylselenocysteine has been used in trials studying the prevention of Prostate Carcinoma and No Evidence of Disease.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAmino Acids, Sulfur +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methyltestosterone Approved DB06710
small molecule | CAS: 58-18-4

A synthetic anabolic steroid used for treating men with testosterone deficiency or similar androgen replacement therapies. Also, has antineoplastic properties and so has been used secondarily in women with advanced breast cancer. Methyltestosterone is a sched…

Kategori:
3-Oxoandrosten (4) DerivativesAnabolic AgentsAndrogens +20
Target Protein:
Androgen receptorEstrogen receptor
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 342-69-8

An analog of inosine with a methylthio group replacing the hydroxyl group in the 6-position.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +6
Target Protein:
Purine nucleoside phosphorylase DeoD-type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7060-82-4

Deskripsi belum tersedia.

Kategori:
Oxidation-Reduction ActivityOxidation-Reduction AgentSerotonergic Drugs Shown to Increase Risk of Serotonin Syndrome
Target Protein:
AcetylcholinesteraseTranscriptional regulator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 56-04-2

Deskripsi belum tersedia.

Kategori:
Antithyroid agentsHormone AntagonistsHormones, Hormone Substitutes, and Hormone Antagonists +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Lysozyme C
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 59322-44-0

Deskripsi belum tersedia.

Target Protein:
Trans-sialidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methyprylon Approved DB01107
small molecule | CAS: 125-64-4

Methyprylon is a sedative of the piperidinedione derivative family that was previously used for the treatment of insomnia. However, with the introduction of newer drugs with fewer side effects, such as benzodiazepines, the clinical use of methyprylon is now l…

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +3
Target Protein:
GABA(A) ReceptorGamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh6-16 hours
Vol. Distribusi-
Klirens-
Genetik -
Methysergide Approved DB00247
small molecule | CAS: 361-37-5

An ergot derivative that is a congener of lysergic acid diethylamide. It antagonizes the effects of serotonin in blood vessels and gastrointestinal smooth muscle, but has few of the properties of other ergot alkaloids. Methysergide is used prophylactically i…

Kategori:
Agents that produce hypertensionAlkaloidsAnalgesics +20
Target Protein:
5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metiamide DB08805
small molecule | CAS: 34839-70-8

Metiamide is an H-2 receptor antagonist derived from burimamide. It was an intermediate product on the path to developing cimetidine.

Kategori:
Acid ReducersAmidesAnti-Ulcer Agents +8
Target Protein:
Histamine H2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meticillin Approved DB01603
small molecule | CAS: 61-32-5

One of the penicillins which is resistant to penicillinase but susceptible to a penicillin-binding protein. It is inactivated by gastric acid so administered by injection.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
MecA PBP2' (penicillin binding protein 2')Penicillin-binding protein 2aPenicillin-binding protein 1b +3
Waktu Paruh25-60 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meticrane Approved DB13284
small molecule | CAS: 1084-65-7

Meticrane is a diuretic medication. It has been marketed in Japan under the trade name Arresten and is used to lower blood pressure [L5647].

Kategori:
DiureticsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metipranolol Approved DB01214
small molecule | CAS: 22664-55-7

A beta-adrenergic antagonist effective for both beta-1 and beta-2 receptors. It is used as an antiarrhythmic, antihypertensive, and antiglaucoma agent.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metixene Approved DB00340
small molecule | CAS: 4969-02-2

Metixene (or methixene) is a anticholinergic used as an antiparkinsonian agent.

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +6
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metizoline DB13614
small molecule | CAS: 17692-22-7

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoclopramide Approved DB01233
small molecule | CAS: 364-62-5

Diabetic gastroparesis is a condition that causes frequent nausea and vomiting, which has a negative impact on quality of life and poses a significant burden on the healthcare system.[A184934] Metoclopramide is a dopamine antagonist used to treat nausea and v…

Kategori:
Acids, CarbocyclicAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +35
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3AMuscarinic acetylcholine receptor M1 +1
Gen Terkait:
KCNH2 ADRA1D CYP2D6 +4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik 7 Varian
Metocurine Approved DB01336
small molecule | CAS: 5152-30-7

Dimethyltubocurarinium (INN) or metocurine (USAN), also known as dimethyltubocurarine, is a non-depolarizing muscle relaxant. Patients on chronic anticonvulsant drugs are relatively resistant to metocurine. [A2393]

Kategori:
Agents producing tachycardiaAlkaloidsAmines +18
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metolazone Approved DB00524
small molecule | CAS: 17560-51-9

A quinazoline-sulfonamide that is considered a thiazide-like diuretic which is long-acting so useful in chronic renal failure. It also tends to lower blood pressure and increase potassium loss.

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +21
Target Protein:
Solute carrier family 12 member 3
Waktu ParuhApproximately 14 ho…
Vol. Distribusi-
Klirens-
Genetik -
Metoprolol Approved DB00264
small molecule | CAS: 51384-51-1

Metoprolol is a selective beta-1 blocker commonly employed as the succinate and tartrate derivatives depending if the formulation is designed to be of immediate release or extended release.[A175159, L5530] The possibility of the generation of these formulatio…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta adrenergic receptor
Gen Terkait:
ADRB1 CYP2D6 ADRB1
Waktu ParuhThe immediate relea…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik 3 Varian
Metoserpate DB11530
small molecule | CAS: 1178-28-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIndole Alkaloids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metreleptin Approved DB09046
biotech | CAS: 186018-45-1

Metreleptin, a recombinant analog of the human hormone leptin, is an orphan drug used to treat complications of leptin deficiency in people with lipodystrophy. Lipodystrophies include a range of disorders characterized by the reduction, absence, or altered di…

Kategori:
AdipokinesAlimentary Tract and MetabolismAmino Acids and Derivatives +11
Target Protein:
Leptin receptor
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing intraveno…
KlirensThe clearance of me…
Genetik -
Metribolone DB02998
small molecule | CAS: 965-93-5

A synthetic non-aromatizable androgen and anabolic steroid. It binds strongly to the androgen receptor and has therefore also been used as an affinity label for this receptor in the prostate and in prostatic tumors.

Kategori:
EstranesEstrenesFused-Ring Compounds +1
Target Protein:
Progesterone receptorAndrogen receptorNuclear receptor coactivator 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrifonate DB11473
small molecule | CAS: 52-68-6

Metrifonate or trichlorfon is an irreversible organophosphate acetylcholinesterase inhibitor. It is a prodrug which is activated non-enzymatically into 2,2-dichlorovinyl dimethyl phosphate.

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizamide DB01578
small molecule | CAS: 31112-62-6

Metrizamide is a solute for density gradient centrifugation offering higher maximum solution density without the problems of increased viscosity. It is also used as a resorbable, non-ionic contrast medium.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizoic acid Approved DB09346
small molecule | CAS: 1949-45-7

Metrizoic acid is a molecule used as a contrast medium. It present a higher risk of allergic reactions due to its high osmolality. Its approval has been discontinued by the FDA. One study in 1976 demonstrated that metrizoic acid, when used for cardiac angiog…

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metronidazole Approved DB00916
small molecule | CAS: 443-48-1

Metronidazole is a commonly used antibiotic, belonging to the nitroimidazole class of antibiotics.[L3754] It is frequently used to treat gastrointestinal infections as well as trichomoniasis and giardiasis, and amebiasis which are parasitic infections.[A18103…

Kategori:
Agents that reduce seizure thresholdAlimentary Tract and MetabolismAnti-Bacterial Agents +38
Target Protein:
Oxygen-insensitive NADPH nitroreductaseAnaerobic bacterial DNAProtozoal DNA
Waktu ParuhThe elimination hal…
Vol. DistribusiMetronidazole is wi…
KlirensDose adjustments ma…
Genetik -
small molecule | CAS: 13182-89-3

Deskripsi belum tersedia.

Kategori:
ImidazolesNitro CompoundsNitroimidazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 8901–8950 dari 14063
Sebelumnya Halaman 179 / 282 Berikutnya